CYP inhbitors
CYP inducers
CYP substrates
Transporter inhibitors
Transporter inducers
Transporter substrates
ABCB1 [HSA:5243]
Aliskiren [DG:DG00352]
FDA
Ambrisentan
Apixaban
Berberine [DG:DG01773]
Cetirizine [DG:DG01107]
Citalopram [DG:DG00943]
Colchicine
Ciclosporin
Dabigatran etexilate
Digoxin
Digitoxin
Doxorubicin [DG:DG00696]
Edoxaban [DG:DG01398]
Everolimus
Fexofenadine [DG:DG01117]
Glyburide
Imatinib [DG:DG00710]
Indacaterol [DG:DG01057]
Irinotecan [DG:DG00726]
Lapatinib [DG:DG00715]
Loperamide [DG:DG00092]
D08144 Loperamide (INN) D00729 Loperamide hydrochloride (JAN/USP) D07113 Loperamide oxide (INN)
Maraviroc
Mianserin [DG:DG00951]
Nilotinib [DG:DG00716]
Paclitaxel
Paroxetine [DG:DG00944]
Posaconazole
Quinidine [DG:DG00192]
Ranolazine [DG:DG00247]
Rivaroxaban
Saquinavir [DG:DG00653]
Saxagliptin [DG:DG00119]
Sirolimus
Sitagliptin [DG:DG00118]
Talinolol
Tolvaptan
Topotecan [DG:DG00725]
Verapamil [DG:DG00329]
Vinblastine [DG:DG00689]
ABCB4 [HSA:5244]
ABCB11 [HSA:8647]
ABCC2 [HSA:1244]
ABCC3 [HSA:8714]
ABCC4 [HSA:10257]
ABCG2 [HSA:9429]
OAT1 [HSA:9356]
OAT2 [HSA:10864]
OAT3 [HSA:9376]
SLC15A1 [HSA:6564]
SCL15A2 [HSA:6565]
SLCO1A2 [HSA:6579]
SLCO1B1 [HSA:10599]
SLCO1B3 [HSA:28234]
SLCO2B1 [HSA:11309]
SLC22A1 [HSA:6580]
SLC22A2 [HSA:6582]
SLC22A3 [HSA:6581]
SLC28A2 [HSA:9153]
SLC28A3 [HSA:64078]
SLC29A1 [HSA:2030]
SLC29A2 [HSA:3177]
MATE1 [HSA:55244]
MATE2 [HSA:146802]