Drug interactions with metabolizing enzymes and transporters

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 CYP inhbitors
 
 CYP inducers
 
 CYP substrates
 
 Transporter inhibitors
 
 Transporter inducers
 
 Transporter substrates
   ABCB1 [HSA:5243]
     Aliskiren [DG:DG00352]
FDA
     Ambrisentan
FDA
     Apixaban
     Berberine [DG:DG01773]
     Cetirizine [DG:DG01107]
     Citalopram [DG:DG00943]
     Colchicine
FDA
     Ciclosporin
     Dabigatran etexilate
FDA
     Digoxin
FDA
     Digitoxin
     Doxorubicin [DG:DG00696]
     Edoxaban [DG:DG01398]
     Everolimus
FDA
     Fexofenadine [DG:DG01117]
FDA
     Glyburide
     Imatinib [DG:DG00710]
FDA
     Indacaterol [DG:DG01057]
     Irinotecan [DG:DG00726]
     Lapatinib [DG:DG00715]
FDA
     Loperamide [DG:DG00092]
       D08144  Loperamide (INN)
       D00729  Loperamide hydrochloride (JAN/USP)
       D07113  Loperamide oxide (INN)
 
 
 
     Maraviroc
FDA
     Mianserin [DG:DG00951]
     Nilotinib [DG:DG00716]
FDA
     Paclitaxel
     Paroxetine [DG:DG00944]
     Posaconazole
FDA
     Quinidine  [DG:DG00192]
     Ranolazine [DG:DG00247]
FDA
     Rivaroxaban
     Saquinavir [DG:DG00653]
     Saxagliptin [DG:DG00119]
FDA
     Sirolimus
FDA
     Sitagliptin [DG:DG00118]
FDA
     Talinolol
FDA
     Tolvaptan
FDA
     Topotecan [DG:DG00725]
FDA
     Verapamil [DG:DG00329]
     Vinblastine [DG:DG00689]
   ABCB4 [HSA:5244]
   ABCB11 [HSA:8647]
   ABCC2 [HSA:1244]
   ABCC3 [HSA:8714]
   ABCC4 [HSA:10257]
   ABCG2 [HSA:9429]
   OAT1 [HSA:9356]
   OAT2 [HSA:10864]
   OAT3 [HSA:9376]
   SLC15A1 [HSA:6564]
   SCL15A2 [HSA:6565]
   SLCO1A2 [HSA:6579]
   SLCO1B1 [HSA:10599]
   SLCO1B3 [HSA:28234]
   SLCO2B1 [HSA:11309]
   SLC22A1 [HSA:6580]
   SLC22A2 [HSA:6582]
   SLC22A3 [HSA:6581]
   SLC28A2 [HSA:9153]
   SLC28A3 [HSA:64078]
   SLC29A1 [HSA:2030]
   SLC29A2 [HSA:3177]
   MATE1 [HSA:55244]
   MATE2 [HSA:146802]

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According to FDA Guidance on Drug Interactions
Last updated: August 19, 2016

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