Drug interactions with metabolizing enzymes and transporters

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 CYP inhbitors
   CYP1A2 [HSA:1544]
   CYP2A6 [HSA:1548]
   CYP2B6 [HSA:1555]
   CYP2C8 [HSA:1558]
   CYP2C9 [HSA:1559]
     Amiodarone [DG:DG00204]
Moderate (in vivo)
     Benzbromarone
     Bucolome
     Capecitabine
Weak (in vivo)
     Carmofur
     Cimetidine [DG:DG00017]
     Choline fenofibrate
     Cotrimoxazole
Weak (in vivo)
     Croconazole
     Ciclosporin
     Delavirdine [DG:DG00662]
     Diosmin
     Disulfiram
     Doxifluridine
     Lovastatin
     Fenofibrate
     Etravirine
Weak (in vivo)
     Fluconazole [DG:DG00371]
Moderate (in vivo)
     Fluorouracil [DG:DG00687]
     Fluvastatin [DG:DG00354]
Weak (in vivo)
     Fluvoxamine [DG:DG00946]
Weak (in vivo)
     Isoconazole [DG:DG00365]
     Isoniazid [DG:DG00642]
     Lanoconazole
       D01092  Lanoconazole (JAN/INN)
 
     Leflunomide
     Miconazole [DG:DG00004]
Moderate (in vivo)
     Metronidazole
Weak (in vivo)
     Neticonazole
     Oxandrolone
Moderate (in vivo)
     Oxiconazole [DG:DG00367]
     Phenylbutazone [DG:DG00745]
     Probenecid
     Sertraline [DG:DG00945]
     Sulconazole [DG:DG00366]
     Sulfinpyrazone
Weak (in vivo)
     Stiripentol
     Sulfamethoxazole
     Sulfaphenazole
     Teniposide
     Tegafur
     Tigecycline
     Tienilic acid
     Voriconazole
Weak (in vivo)
     Zafirlukast
Weak (in vivo)
   CYP2C19 [HSA:1557]
   CYP2D6 [HSA:1565]
   CYP3A4 [HSA:1576]
   CYP3A5 [HSA:1577]
   CYP3A7 [HSA:1551]
   CYP3A [HSA:1576 1577 1551]
   CYP17 [HSA:1586]
 
 CYP inducers
 
 CYP substrates
 
 Transporter inhibitors
 
 Transporter inducers
 
 Transporter substrates

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According to FDA Guidance on Drug Interactions
Last updated: August 19, 2016

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