| |
Remark |
G Protein-coupled receptors
|
Rhodopsin family
|
Acetylcholine (muscarinic)
|
Adrenaline
|
Dopamine
|
Histamine
|
Serotonin
|
Tachykinin / neurokinin
|
Ghrelin
|
Orexin
|
Neuropeptide Y
|
Opioid
|
mu-opioid receptor [HSA:4988] [KO:K04215]
|
Trimebutine [DG:DG00031]
|
Naloxegol [DG:DG00078]
|
Diphenoxylate [DG:DG00090]
|
Loperamide [DG:DG00092]
|
D08144 Loperamide (INN)
D00729 Loperamide hydrochloride (JAN/USP)
D07113 Loperamide oxide (INN)
|
Agonist
Agonist
Agonist
|
Fentanyl [DG:DG00791]
|
Alfentanil [DG:DG00792]
|
Sufentanil [DG:DG00793]
|
Remifentanil [DG:DG00795]
|
Morphine [DG:DG00810]
|
Hydromorphone [DG:DG00811]
|
Oxycodone [DG:DG00813]
|
Dihydrocodeine [DG:DG00814]
|
Pethidine [DG:DG00816]
|
Dextropropoxyphene [DG:DG00818]
|
Pentazocine [DG:DG00819]
|
Buprenorphine [DG:DG00820]
|
Butorphanol [DG:DG00821]
|
Nalbuphine [DG:DG00822]
|
Tilidine [DG:DG00823]
|
Tramadol [DG:DG00824]
|
Meptazinol [DG:DG00825]
|
Tapentadol [DG:DG00826]
|
Naltrexone [DG:DG00997]
|
Nalmefene [DG:DG00998]
|
Methadone [DG:DG00999]
|
Levomethadone [DG:DG01002]
|
Diamorphine [DG:DG01003]
|
Ethylmorphine [DG:DG01074]
|
Hydrocodone [DG:DG01075]
|
Codeine [DG:DG01076]
|
Nalorphine [DG:DG01151]
|
Naloxone [DG:DG01155]
|
Diprenorphine [DG:DG01273]
|
Carfentanil [DG:DG01339]
|
Eptazocine [DG:DG01340]
|
Levorphanol [DG:DG01341]
|
Naldemedine [DG:DG01342]
|
Oxymorphone [DG:DG01343]
|
Benzhydrocodone [DG:DG01850]
|
Axelopran [DG:DG01857]
|
Acetyldihydrocodeine
|
Alvimopan
|
Bevenopran
|
Brifentanil
|
Cebranopadol
|
Cyclazocine
|
Dezocine
|
Difenoxin
|
Eluxadoline
|
Etorphine
|
Levacetylmethadol
|
Levallorphan
|
Levomethadyl
|
Lofentanil
|
Methylnaltrexone bromide
|
Methadyl
|
Methylsamidorphan [DG:DG01830]
|
Mirfentanil
|
Ocfentanil
|
Propoxyphene
|
Quadazocine
|
Trimeperidine
|
kappa-opioid receptor [HSA:4986] [KO:K04214]
|
delta-opioid receptor [HSA:4985] [KO:K04213]
|
sigma1-opioid receptor [HSA:10280]
|
Angiotensin
|
Bradykinin
|
Endothelin
|
Lutropin-choriogonadotropic hormone
|
Follicle stimulating hormone
|
Oxytocin
|
Vasopressin
|
Melanocortin
|
Gonadotropin-releasing hormone
|
Somatostatin
|
Thyrotropin-releasing hormone
|
Cholecystokinin
|
Motilin
|
Thrombin
|
Purine / pyrimidine
|
Adenosine
|
Prostaglandin
|
Prostacyclin
|
Leukotriene
|
Thromboxane
|
Sphingolipid
|
Free fatty acid
|
Cannabinoid
|
Platelet activating factor
|
Melatonin
|
Cysteinyl leukotriene
|
Secretin receptor family
|
Metabotropic glutamate receptor family
|
Others
|
|
|
Cytokine receptors
|
|
|
Nuclear receptors
|
|
|
Ion channels
|
|
|
Transporters
|
|
|
Enzymes
|
|
|
Protein kinases
|
|
|
Cytokines
|
|
|
Others
|