| alpha1-Adrenergic receptor antagonist |
| Prazosin |
| Prazosin (INN) |
| Prazosin hydrochloride (JP17/USP) <JP/US> |
| Indoramin |
| Indoramin (USAN/INN) |
| Indoramin hydrochloride (USAN) |
| Trimazosin |
| Trimazosin (INN) |
| Trimazosin hydrochloride (USAN) |
| Doxazosin |
| Doxazosin (INN) |
| Doxazosin mesylate (USP); Doxazosin mesilate (JP17) <JP/US> |
| Urapidil |
| Urapidil (JP17/INN) <JP> |
| Urapidil hydrochloride |
| Ketanserin |
| Ketanserin (USAN/INN) |
| Ketanserin tartrate |
| Phentolamine |
| Phentolamine (INN) |
| Phentolamine mesylate (USP); Phentolamine mesilate (JAN/INN) <JP/US> |
| Tolazoline |
| Tolazoline (INN) |
| Tolazoline hydrochloride (JAN/USP) |
| Nicergoline |
| Nicergoline (JP17/USAN/INN) <JP> |
| Nicergoline tartrate |
| Phenoxybenzamine |
| Phenoxybenzamine (INN) |
| Phenoxybenzamine hydrochloride (USP) <US> |
| Moxisylyte |
| Moxisylyte (INN) |
| Moxisylyte hydrochloride (JAN) |
| Ifenprodil |
| Ifenprodil (INN) |
| Ifenprodil tartrate (JP17) <JP> |
| Labetalol |
| Labetalol (INN) <US> |
| Labetalol hydrochloride (JP17/USP) <JP/US> |
| Carvedilol |
| Carvedilol (JP17/USP/INN) <JP/US> |
| Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN) <US> |
| Alfuzosin |
| Alfuzosin (INN) |
| Alfuzosin hydrochloride (JAN/USAN) <US> |
| Tamsulosin |
| Tamsulosin (INN) |
| Tamsulosin hydrochloride (JP17/USP) <JP/US> |
| Terazosin |
| Terazosin (INN) |
| Terazosin hydrochloride (USP); Terazosin hydrochloride hydrate (JAN) <JP/US> |
| Terazosin hydrochloride anhydrous <US> |
| Silodosin (JP17/INN) <JP/US> |
| Levomepromazine |
| Methotrimeprazine (USP); Levomepromazine (USAN/INN) |
| Levomepromazine hydrochloride (JAN/USAN) <JP> |
| Levomepromazine maleate (JP17/USAN) <JP> |
| Pimozide (JP17/USP/INN) <JP/US> |
| Clozapine (JAN/USP/INN) <JP/US> |
| Olanzapine |
| Olanzapine (JAN/USP/INN) <JP/US> |
| Olanzapine pamoate (USAN) <US> |
| Sertindole (USAN/INN) |
| Quetiapine |
| Quetiapine (INN) |
| Quetiapine fumarate (JP17/USP) <JP/US> |
| Asenapine |
| Asenapine (INN) <US> |
| Asenapine maleate (JAN/USAN) <JP/US> |
| Risperidone (JP17/USP/INN) <JP/US> |
| Mianserin |
| Mianserin (INN) |
| Mianserin hydrochloride (JAN/USAN) <JP> |
| Setiptiline |
| Setiptiline (INN) |
| Setiptiline maleate (JAN) <JP> |
| Amosulalol |
| Amosulalol (INN) |
| Amosulalol hydrochloride (JP17) <JP> |
| Arotinolol |
| Arotinolol (INN) |
| Arotinolol hydrochloride (JP17) <JP> |
| Naftopidil (JP17/INN) <JP> |
| Bunazosin |
| Bunazosin (INN) |
| Bunazosin hydrochloride (JP17) <JP> |
| Medroxalol |
| Medroxalol (USAN/INN) |
| Medroxalol hydrochloride (USAN) |
| Fiduxosin hydrochloride (USAN) |
| Pegoxel 7 stearate (USAN) |
| alpha2-Adrenergic receptor antagonist |
| Phentolamine |
| Phentolamine (INN) |
| Phentolamine mesylate (USP); Phentolamine mesilate (JAN/INN) <JP/US> |
| Tolazoline |
| Tolazoline (INN) |
| Tolazoline hydrochloride (JAN/USP) |
| Phenoxybenzamine |
| Phenoxybenzamine (INN) |
| Phenoxybenzamine hydrochloride (USP) <US> |
| Yohimbin |
| Yohimbine (DCF) |
| Yohimbine hydrochloride (USP) |
| Piribedil (INN) |
| Chlorpromazine |
| Chlorpromazine (USP/INN) |
| Chlorpromazine hydrochloride (JP17/USP) <JP/US> |
| Chlorpromazine hibenzate (JAN) |
| Chlorpromazine phenolphthalinate (JAN) <JP> |
| Chlorpromazine tannate (JAN) |
| Levomepromazine |
| Methotrimeprazine (USP); Levomepromazine (USAN/INN) |
| Levomepromazine hydrochloride (JAN/USAN) <JP> |
| Levomepromazine maleate (JP17/USAN) <JP> |
| Asenapine |
| Asenapine (INN) <US> |
| Asenapine maleate (JAN/USAN) <JP/US> |
| Mianserin |
| Mianserin (INN) |
| Mianserin hydrochloride (JAN/USAN) <JP> |
| Mirtazapine |
| Mirtazapine (JAN/USP/INN) <JP/US> |
| Mirtazapine hydrate (JAN) |
| Setiptiline |
| Setiptiline (INN) |
| Setiptiline maleate (JAN) <JP> |
| Sunepitron hydrochloride (USAN) |
| Aptazapine maleate (USAN) |
| Atipamezole (USAN/INN) |
| Delequamine hydrochloride (USAN) |
| Fluparoxan hydrochloride (USAN) |
| Imiloxan hydrochloride (USAN) |