KEGG   DRUG: Narsoplimab
Entry
D11531                      Drug                                   
Name
Narsoplimab (USAN)
Formula
C6340H9876N1680O1996S48
Exact mass
143018.9533
Mol weight
143107.52
Sequence
(Heavy chain)
QVTLKESGPV LVKPTETLTL TCTVSGFSLS RGKMGVSWIR QPPGKALEWL AHIFSSDEKS
YRTSLKSRLT ISKDTSKNQV VLTMTNMDPV DTATYYCARI RRGGIDYWGQ GTLVTVSSAS
TKGPSVFPLA PCSRSTSEST AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTKTYT CNVDHKPSNT KVDKRVESKY GPPCPPCPAP EFLGGPSVFL
FPPKPKDTLM ISRTPEVTCV VVDVSQEDPE VQFNWYVDGV EVHNAKTKPR EEQFNSTYRV
VSVLTVLHQD WLNGKEYKCK VSNKGLPSSI EKTISKAKGQ PREPQVYTLP PSQEEMTKNQ
VSLTCLVKGF YPSDIAVEWE SNGQPENNYK TTPPVLDSDG SFFLYSRLTV DKSRWQEGNV
FSCSVMHEAL HNHYTQKSLS LSLGK
(Light chain)
QPVLTQPPSL SVSPGQTASI TCSGEKLGDK YAYWYQQKPG QSPVLVMYQD KQRPSGIPER
FSGSNSGNTA TLTISGTQAM DEADYYCQAW DSSTAVFGGG TKLTVLGQPK AAPSVTLFPP
SSEELQANKA TLVCLISDFY PGAVTVAWKA DSSPVKAGVE TTTPSKQSNN KYAASSYLSL
TPEQWKSHRS YSCQVTHEGS TVEKTVAPTE CS
(Disulfide bridge: H22-H97, H132-L211, H145-H201, H224-H'224, H227-H'227, H259-H319, H365-H423, H'22-H'97, H'132-L'211, H'145-H'201, H'259-H'319, H'365-H'423, L22-L87, L134-L193, L'22-L'87, L'134-L'193)
  Type
Peptide
Efficacy
Anti-inflammatory, Immunomodulator, Anti-mannan-binding lectin serine protease antibody
  Type
Monoclonal antibody
Comment
Treatment of immunoglobulin A nephropathy
Target
MASP2 [HSA:10747] [KO:K03993]
  Pathway
hsa04610  Complement and coagulation cascades
Brite
Target-based classification of drugs [BR:br08310]
 Peptidases and inhibitors
  Serine peptidases
   Chymotrypsin family
    MASP2
     D11531  Narsoplimab (USAN)
Other DBs
CAS: 2108782-45-0
PubChem: 384585507
LinkDB

» Japanese version   » Back

DBGET integrated database retrieval system