KEGG   DRUG: Nipocalimab
Entry
D11666                      Drug                                   
Name
Nipocalimab (USAN);
Nipocalimab (genetical recombination) (JAN)
Formula
C6266H9722N1670O1992S46
Exact mass
141707.7937
Mol weight
141795.31
Sequence
(Heavy chain)
EVQLLESGGG LVQPGGSLRL SCAASGFTFS TYAMGWVRQA PGKGLEWVSS IGASGSQTRY
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCARLA IGDSYWGQGT MVTVSSASTK
GPSVFPLAPS SKSTSGGTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTQTYICN VNHKPSNTKV DKKVEPKSCD KTHTCPPCPA PELLGGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP REEQYASTYR
VVSVLTVLHQ DWLNGKEYKC KVSNKALPAP IEKTISKAKG QPREPQVYTL PPSREEMTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPG
(Light chain)
QSALTQPASV SGSPGQSITI SCTGTGSDVG SYNLVSWYQQ HPGKAPKLMI YGDSERPSGV
SNRFSGSKSG NTASLTISGL QAEDEADYYC SSYAGSGIYV FGTGTKVTVL GQPKAAPSVT
LFPPSSEELQ ANKATLVCLI SDFYPGAVTV AWKADSSPVK AGVETTTPSK QSNNKYAASS
YLSLTPEQWK SHKSYSCQVT HEGSTVEKTV APTECS
(disulfide bridge: H22-H96, H143-H199, H219-L215, H225-H'225, H228-H'228, H260-H320, H366-H424, H'22-H'96, H'143-H'199, H'219-L'215, H'260-H'320, H'366-H'424, L22-L90, L138-L197, L'22-L'90, L'138-L'197)
  Type
Peptide
Efficacy
Autoimmune disease treatment, Anti-Fc receptor antibody
  Type
Monoclonal antibody
Comment
Treatment of diseases mediated by pathogenic IgG autoantibodies and alloantibodies
Target
FCGRT [HSA:2217] [KO:K24019]
Brite
Target-based classification of drugs [BR:br08310]
 Not elsewhere classified
  Organismal systems
   Immune system
    FCGRT
     D11666  Nipocalimab (USAN)
Other DBs
CAS: 2211985-36-1
PubChem: 405226533
LinkDB

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