KEGG   DRUG: Turigrobart
Entry
D13226                      Drug                                   
Name
Turigrobart (USAN)
Formula
C6350H9828N1688O2000S40
Exact mass
143010.8054
Mol weight
143098.76
Sequence
(Heavy chain)
QVQLQESGPG LVKPSETLSL TCTVSGGSIS SYYWSWIRQP AGKGLEWIGR IYPSGNTNYN
PSLKSRVTIS VDTSKNQFSL KLSSVTAADT AVYYCARGGL VMDVWGQGTL VTVSSASTKG
PSVFPLAPCS RSTSESTAAL GCLVKDYFPE PVTVSWNSGA LTSGVHTFPA VLQSSGLYSL
SSVVTVPSSS LGTKTYTCNV DHKPSNTKVD KRVESKYGPP CPPCPAPEAA GGPSVFLFPP
KPKDTLMISR TPEVTCVVVD VSQEDPEVQF NWYVDGVEVH NAKTKPREEQ FNSTYRVVSV
LTVLHQDWLN GKEYKCKVSN KGLPSSIEKT ISKAKGQPRE PQVYTLPPSQ EEMTKNQVSL
TCLVKGFYPS DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSRLTVDKS RWQEGNVFSC
SVMHEALHNH YTQKSLSLSL G
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCRASQSVE FSYLAWYQQK PGQAPRLLIY GASSRATGIP
DRFSGSGSGT DFTLTISRLE PEDFAVYYCH QYGTNPFTFG QGTKVEIKRT VAAPSVFIFP
PSDEQLKSGT ASVVCLLNNF YPREAKVQWK VDNALQSGNS QESVTEQDSK DSTYSLSSTL
TLSKADYEKH KVYACEVTHQ GLSSPVTKSF NRGEC
(Disulfide bridge: H22-H95, H129-L215, H142-H198, H221-H'221, H224-H'224, H256-H316, H362-H420, H'22-H'95, H'129-L'215, H'142-H'198, H'256-H'316, H'362-H'420, L23-L89, L135-L195, L'23-L'89, L'135-L'195)
  Type
Peptide
Efficacy
Pain relief (neuropathic)
  Type
Monoclonal antibody
Comment
Treatment of chronic pain
Target
EREG [HSA:2069] [KO:K09784]
  Pathway
hsa04010  MAPK signaling pathway
hsa04151  PI3K-Akt signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Signaling molecules and receptors
  Cytokines
   Growth factors (RTK-binding)
    EREG
     D13226  Turigrobart (USAN)
Other DBs
CAS: 3047668-82-3
PubChem: 522705674
LinkDB

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