C00989 |
4-Hydroxybutanoic acid; 4-Hydroxybutanoate; 4-Hydroxybutyric acid |
(P) unclassified |
C06807 |
Acetophenazine |
(P) unclassified |
C07521 |
Thiopental |
(P) unclassified |
C17723 |
Metabutethamine |
(P) unclassified |
D00033 |
Phenol (JP18/USP); Liquefied phenol (JP18); Phenol for disinfection (JP18); Phenol, liquefied; Paoscle (TN); Phenol (TN); Liquefied phenol (TN); Phenol for disinfection (TN) |
(P) unclassified |
D00102 |
Nitrous oxide (JP18/USP); Nitrous oxide (TN) |
(P) unclassified |
D00110 |
Cocaine (USP); Cocaine (TN) |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
D00241 |
Baclofen (JP18/USP/INN); Kemstro (TN); Lioresal (TN) |
(P) unclassified |
D00250 |
Capsaicin (JAN/USP); Zostrix (TN) |
(P) unclassified |
D00270 |
Chlorpromazine (USP/INN); Thorazine (TN) |
(P) unclassified |
D00292 |
Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00293 |
Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 / Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 |
D00358 |
Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) |
(P) Enzyme: CYP1A2 CYP3A4 |
D00373 |
Thioridazine (USP/INN); Mellaril-S (TN) |
(P) unclassified |
D00390 |
Triflupromazine (USP/INN); Vesprin (TN) |
(P) unclassified |
D00403 |
Methotrimeprazine (USP); Levomepromazine (USAN/INN); Levoprome (TN) |
(P) unclassified |
D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
D00430 |
Secobarbital (USP/INN); Seconal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 |
D00474 |
Primidone (JP18/USP/INN); Mysoline (TN) |
(P) unclassified |
D00479 |
Prochlorperazine maleate (JP18/USP); Compazine (TN) |
(P) unclassified |
D00493 |
Prochlorperazine (JAN/USP/INN); Compro (TN) |
(P) unclassified |
D00498 |
Pentazocine (JP18/USP/INN); Fortral (TN) |
(P) unclassified |
D00499 |
Pentobarbital (USP/INN); Nembutal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00500 |
Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00503 |
Perphenazine (JP18/USP/INN); Trilafon (TN) |
(P) unclassified |
D00506 |
Phenobarbital (JP18/USP/INN); Luminal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00512 |
Phenytoin (JP18/USP/INN); Dilantin (TN) |
(P) unclassified |
D00542 |
Halothane (JP18/USP/INN); Fluothane (TN) |
(P) Enzyme: CYP3A4 |
D00543 |
Enflurane (JP18/USP/INN); Ethrane (TN) |
(P) unclassified |
D00544 |
Methoxyflurane (USP/INN); Penthrane (TN) |
(P) Enzyme: CYP3A4 |
D00545 |
Isoflurane (JP18/USP/INN); Forane (TN) |
(P) unclassified |
D00546 |
Desflurane (JAN/USP/INN); Suprane (TN) |
(P) unclassified |
D00547 |
Sevoflurane (JP18/USAN/INN); Ultane (TN) |
(P) unclassified |
D00548 |
Etomidate (USP/INN); Amidate (TN) |
(P) Target: GABRA1 |
D00549 |
Propofol (JAN/USP/INN); Diprivan (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 / Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00551 |
Tetracaine (USP/INN); Amethocaine; Amethocaine (TN) |
(P) unclassified |
D00552 |
Benzocaine (USP/INN); Ethyl aminobenzoate (JP18); Parathesin (TN) |
(P) unclassified |
D00553 |
Prilocaine (USP/INN); Propitocaine (JAN) |
(P) unclassified |
D00555 |
Amobarbital (JP18/INN); Isomytal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00578 |
Voriconazole (JP18/USP/INN); Vfend (TN) |
(P) unclassified |
D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) Enzyme: CYP3A4 |
D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 |
D00698 |
Aprobarbital (INN); Alurate (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00699 |
Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00711 |
Ketamine hydrochloride (JP18/USP); Ketalar (TN) |
(P) unclassified |
D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) Target: GABRA1 |
D00713 |
Thiamylal sodium (JP18); Surital (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00714 |
Thiopental sodium (JP18/USP/INN); Pentothal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D00732 |
Chloroprocaine hydrochloride (USP); Clorotekal (TN); Iheezo (TN); Nesacaine (TN) |
(P) unclassified |
D00733 |
Dibucaine (USP); Cinchocaine (INN); Nupercaine (TN) |
(P) unclassified |
D00735 |
Dyclonine hydrochloride (USP); Dyclone (TN); Dyclopro (TN) |
(P) unclassified |
D00737 |
Etidocaine hydrochloride; Duranest (TN) |
(P) unclassified |
D00738 |
Mepivacaine hydrochloride (JP18/USP); Carbocaine (TN); Polocaine (TN); Scandonest plain (TN) |
(P) unclassified |
D00740 |
Procaine hydrochloride (JP18/USP); Novocain (TN) |
(P) unclassified |
D00741 |
Tetracaine hydrochloride (JP18/USP); Protocaine hydrochloride (TN) |
(P) unclassified |
D00788 |
Acetophenazine maleate (USAN); Tindal (TN) |
(P) unclassified |
D00789 |
Chlorpromazine hydrochloride (JP18/USP); Sonazine (TN) |
(P) unclassified |
D00791 |
Fluphenazine hydrochloride (JAN/USP); Prolixin (TN) |
(P) unclassified |
D00792 |
Fluphenazine enanthate (JP18/USP); Prolixin enanthate (TN) |
(P) unclassified |
D00793 |
Fluphenazine decanoate (JAN/USP); Prolixin decanoate (TN) |
(P) unclassified |
D00795 |
Mesoridazine besylate (USP); Serentil (TN) |
(P) unclassified |
D00797 |
Promazine hydrochloride (USP); Sparine (TN) |
(P) unclassified |
D00798 |
Thioridazine hydrochloride (JP18/USP); Mellaril (TN) |
(P) unclassified |
D00799 |
Trifluoperazine hydrochloride (JAN/USP); Stelazine (TN) |
(P) unclassified |
D00800 |
Triflupromazine hydrochloride (JAN/USP); Vesprin (TN) |
(P) unclassified |
D00824 |
Fluvoxamine maleate (JP18/USP); Luvox (TN) |
(P) CYP inhibition: CYP1A2 CYP3A4 |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
D00835 |
Alfentanil hydrochloride (USP); Alfenta (TN) |
(P) unclassified |
D00845 |
Sufentanil citrate (USP); Dsuvia (TN); Sufenta (TN) |
(P) unclassified |
D00961 |
Bicalutamide (JP18/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
D01071 |
Hexobarbital (JAN/INN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D01130 |
Thiethylperazine maleate (JAN/USP); Norzine (TN) |
(P) unclassified |
D01152 |
Oxethazaine (JP18/USAN); Oxetacaine (INN); Strocain (TN) |
(P) unclassified |
D01177 |
Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) |
(P) unclassified |
D01243 |
Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 / Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D01280 |
Warfarin potassium (JP18); Athrombin-K (TN) |
(P) unclassified |
D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
D01310 |
Secobarbital sodium (JAN/USP); Seconal sodium (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D01355 |
Tramadol hydrochloride (JP18/USP); Ultram (TN) |
(P) Enzyme: CYP3A4 |
D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D01399 |
Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 |
D01412 |
Perazine maleate (JAN) |
(P) unclassified |
D01447 |
Thioproperazine mesilate (JAN); Thioproperazine mesylate |
(P) unclassified |
D01448 |
Trifluoperazine maleate (JAN); Trifluoperazine (TN) |
(P) unclassified |
D01450 |
Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) |
(P) Enzyme: CYP3A4 |
D01485 |
Propericiazine (JAN); Periciazine; Neuleptil (TN) |
(P) unclassified |
D01520 |
Levomepromazine hydrochloride (JAN/USAN); Nozinan (TN) |
(P) unclassified |
D01740 |
Barbital (JP18/INN); Barbital (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D01768 |
Benoxinate hydrochloride (USP); Oxybuprocaine hydrochloride (JP18); Benoxil (TN) |
(P) unclassified |
D01772 |
Ether (JP18/USP); Diethyl ether |
(P) unclassified |
D01860 |
Perazine dimalonate (JAN) |
(P) unclassified |
D01878 |
Tolycaine hydrochloride (JAN) |
(P) unclassified |
D01967 |
p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN); Diethylaminoethyl p-butylaminobenzoate hydrochloride (JAN); Calvital liquid (TN); T cain (TN) |
(P) unclassified |
D02022 |
Prochlorperazine mesilate (JAN); Prochlorperazine dimethanesulfonate; Novamin (TN) |
(P) unclassified |
D02037 |
Perphenazine maleate (JP18); PZC (TN) |
(P) unclassified |
D02086 |
Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
D02098 |
Proparacaine hydrochloride (USP); Alcaine (TN); Ophthetic (TN) |
(P) unclassified |
D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
D02163 |
Fluphenazine maleate (JAN); Flumezin (TN) |
(P) unclassified |
D02182 |
Cocaine hydrochloride (JP18/USP); Cocaine hydrochloride (TN) |
(P) unclassified |
D02220 |
Dibucaine hydrochloride (JP18/USP); Nupercaine hydrochloride (TN); Percamin (TN) |
(P) unclassified |
D02227 |
Pentazocine hydrochloride (JAN/USP); Sosegon (TN); Talacen (TN) |
(P) unclassified |
D02248 |
Levomepromazine maleate (JP18/USAN); Hirnamin (TN) |
(P) unclassified |
D02252 |
Amobarbital sodium (JAN/USP); Amytal sodium (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D02253 |
Pentobarbital calcium (JP18); Ravona (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D02354 |
Thiethylperazine (USAN/INN) |
(P) unclassified |
D02372 |
Perospirone hydrochloride hydrate (JAN); Lullan (TN) |
(P) unclassified |
D02456 |
Aminobenzoic acid (USP); p-Aminobenzoic acid; RVPaba lipstick (TN) |
(P) unclassified |
D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
D02604 |
Acepromazine maleate (USP) |
(P) unclassified |
D02605 |
Methoxypromazine maleate |
(P) unclassified |
D02607 |
Mepazine acetate |
(P) unclassified |
D02608 |
Perazine fendizoate (JAN) |
(P) unclassified |
D02609 |
Prochlorperazine edisylate (USP); Compazine syrup (TN) |
(P) unclassified |
D02610 |
Thiethylperazine malate (JAN); Torecan (TN) |
(P) unclassified |
D02611 |
Phenoperidine (INN) |
(P) unclassified |
D02618 |
Butobarbital (BAN); Butethal; Neonal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D02642 |
Butaperazine (USAN) |
(P) unclassified |
D02643 |
Butaperazine maleate (USAN) |
(P) unclassified |
D02644 |
Carphenazine maleate (USAN); Proketazine (TN) |
(P) unclassified |
D02653 |
Cyclophenazine hydrochloride (USAN) |
(P) unclassified |
D02671 |
Mesoridazine (USAN/INN); Lidanar (TN) |
(P) unclassified |
D02679 |
Piperacetazine (USAN/INN); Quide (TN) |
(P) unclassified |
D02680 |
Pipotiazine palmitate (USAN); Piportil depot (TN) |
(P) unclassified |
D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
D02732 |
Pranlukast hydrate (JP18); Onon (TN) |
(P) Enzyme: CYP3A4 |
D02812 |
Aliflurane (USAN/INN) |
(P) unclassified |
D02817 |
Allobarbital (USAN/INN) |
(P) unclassified |
D02906 |
Aminobenzoate potassium (USP); Potaba (TN) |
(P) unclassified |
D02907 |
Aminobenzoate sodium (USP); Sodium aminobenzoate |
(P) unclassified |
D02941 |
Anileridine (USP/INN) |
(P) unclassified |
D02942 |
Anileridine hydrochloride (USP); Leritine (TN) |
(P) unclassified |
D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02991 |
Articaine hydrochloride (JAN/USP) |
(P) unclassified |
D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
D03180 |
Butabarbital (USP); Secbutabarbital (BAN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D03182 |
Butalbital (USP/INN); Sandoptal (TN) |
(P) unclassified |
D03274 |
Chlorpromazine hibenzate (JAN); Contomin (TN) |
(P) unclassified |
D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 |
D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP inhibition: CYP1A2 / CYP induction: CYP3A4 |
D03719 |
Dexivacaine (USAN/INN) |
(P) unclassified |
D03841 |
Nitrous oxide and oxygen; Anesoxyn (TN) |
(P) unclassified |
D03852 |
Droperidol and fentanyl citrate; Innovar (TN) |
(P) Enzyme: CYP3A4 |
D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 |
D04034 |
Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) |
(P) unclassified |
D04038 |
Perphenazine fendizoate (JAN); PZC (TN) |
(P) unclassified |
D04048 |
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
D04077 |
Eterobarb (USAN/INN); Antilon (TN) |
(P) unclassified |
D04088 |
Ethyl chloride (USP) |
(P) unclassified |
D04095 |
Etidocaine (USAN/INN) |
(P) unclassified |
D04237 |
Fluroxene (USAN); Fluoromar (TN) |
(P) unclassified |
D04257 |
Fospropofol disodium (USAN); Aquavan (TN); Lusedra (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
D04965 |
Perphenazine hydrochloride; Perphenazine dihydrochloride; PZC intramuscular injection (TN) |
(P) unclassified |
D04985 |
Methohexital (USP/INN) |
(P) Target: GABRA1 |
D05177 |
Nitisinone (JAN/USAN/INN); Orfadin (TN) |
(P) unclassified |
D05208 |
Norflurane (USAN/INN) |
(P) unclassified |
D05626 |
Propanidid (USAN/INN); Epontol (TN) |
(P) unclassified |
D05665 |
Pyrrocaine (USAN/INN) |
(P) unclassified |
D05743 |
Rodocaine (USAN) |
(P) unclassified |
D05745 |
Roflurane (USAN/INN) |
(P) unclassified |
D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
D05866 |
Sodium oxybate (USAN); Sodium gammahydroxybutyrate; Xyrem (TN) |
(P) unclassified |
D05938 |
Sufentanil (USAN/INN) |
(P) unclassified |
D06055 |
Teflurane (USAN/INN) |
(P) unclassified |
D06106 |
Thiamylal |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D06405 |
Nalfurafine hydrochloride (JAN/USAN) |
(P) Enzyme: CYP3A4 |
D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 |
D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 |
D06534 |
Phenolated water (JP18); Phenolated water for disinfection (JP18); Phenol hydrate; Phenol water (TN); Phenolated water for disinfection (TN) |
(P) unclassified |
D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D06887 |
Talbutal (INN); Lotusate (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D07065 |
Acepromazine (INN); Concentrat vo34 (TN) |
(P) unclassified |
D07122 |
Alfentanil (INN); Rapifen (TN) |
(P) unclassified |
D07282 |
Alfaxalone (INN) |
(P) unclassified |
D07284 |
Butanilicaine (INN) |
(P) unclassified |
D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D07307 |
Cyamemazine (INN); Tercian (TN) |
(P) unclassified |
D07308 |
Chlorproethazine (INN) |
(P) unclassified |
D07321 |
Vinylbital (INN); Vinylbitone |
(P) unclassified |
D07322 |
Vinbarbital (INN) |
(P) unclassified |
D07323 |
Cyclobarbital (INN); Ciclobarbital (TN) |
(P) unclassified |
D07324 |
Proxibarbal (INN); Centralgol (TN) |
(P) unclassified |
D07468 |
Articaine (INN); Carticaine |
(P) unclassified |
D07523 |
Betaine (JAN); Cystadane (TN) |
(P) unclassified |
D07552 |
Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) |
(P) Enzyme: CYP3A4 |
D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
D07678 |
Chloroprocaine (INN) |
(P) unclassified |
D07685 |
Chlorproethazine hydrochloride; Neuriplege (TN) |
(P) unclassified |
D07756 |
Cyamemazine tartrate; Tercian (TN) |
(P) unclassified |
D07757 |
Cyclobarbital calcium (BAN); Phanodorn calcium (TN) |
(P) unclassified |
D07865 |
Dixyrazine; Esucos (TN) |
(P) unclassified |
D07881 |
Dyclonine (INN) |
(P) unclassified |
D07977 |
Fluphenazine (INN); Moditen (TN) |
(P) unclassified |
D08098 |
Ketamine (INN); Tekam (TN) |
(P) unclassified |
D08116 |
Levobupivacaine (INN); Novabupi (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
D08127 |
Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
D08181 |
Mepivacaine (INN); Carboplyin Dental (TN) |
(P) unclassified |
D08311 |
Oxetacaine hydrochloride; Emoren (TN) |
(P) unclassified |
D08319 |
Oxybuprocaine (INN); Monofree oxybuprocaine (TN) |
(P) unclassified |
D08341 |
Perphenazine decanoate; Trilafon dekanoat (TN) |
(P) unclassified |
D08342 |
Perphenazine enantate; Perphenazine enanthate; Trilafon (TN) |
(P) unclassified |
D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ |
D08385 |
Pipotiazine (INN); Piportil (TN) |
(P) unclassified |
D08422 |
Procaine (INN); Solution of novocain (TN) |
(P) unclassified |
D08430 |
Promazine (INN); Combelen [veterinary] (TN) |
(P) unclassified |
D08448 |
Proxymetacaine (INN); Proparacaine |
(P) unclassified |
D08473 |
Remifentanil (INN); Ultiva (TN) |
(P) unclassified |
D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
D08490 |
Ropivacaine (INN); Naropin (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
D08585 |
Thioproperazine (INN) |
(P) unclassified |
D08636 |
Trifluoperazine (INN); Apo-trifluoperazine (TN) |
(P) unclassified |
D08640 |
Trimecaine (INN); Mesidicain; Mesocain |
(P) unclassified |
D08641 |
Trimecaine hydrochloride; Mesocain (TN) |
(P) unclassified |
D09216 |
Thiopropazate (INN) |
(P) unclassified |
D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(P) Enzyme: CYP3A4 |
D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 |
D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
D09819 |
Chlorpromazine tannate (JAN) |
(P) unclassified |
D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP inhibition: CYP1A2 / CYP induction: CYP3A4 |
D09999 |
Tramadol hydrochloride and acetaminophen; Tramcet (TN) |
(P) Enzyme: CYP3A4 |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 |
D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 |
D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
D10811 |
Fentanyl hydrochloride (JAN); Ionsys (TN) |
(P) Enzyme: CYP3A4 |
D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) Enzyme: CYP3A4 |
D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 |
D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
D11027 |
Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) |
(P) unclassified |
D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11062 |
Osilodrostat phosphate (JAN/USAN); Isturisa (TN) |
(P) Enzyme: CYP3A4 |
D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
D11404 |
Asciminib hydrochloride (JAN/USAN); Scemblix (TN) |
(P) Enzyme: CYP3A4 |
D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
D11708 |
Givosiran sodium (JAN); Givlaari (TN) |
(P) unclassified |
D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 |
D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) CYP inhibition: CYP1A2 |
D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |