C07051 |
Indinavir |
(P) unclassified |
C07521 |
Thiopental |
(P) unclassified |
D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) |
(P) Enzyme: CYP3A4 |
D00125 |
Etoposide (JP18/USP/INN); Vepesid (TN) |
(P) unclassified |
D00140 |
Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) |
(P) unclassified |
D00168 |
Cytarabine (JP18/USP/INN); ARA-C; Depocyt (TN) |
(P) unclassified |
D00184 |
Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00208 |
Mitomycin (USP/INN); Mitomycin C (JP18); MMC; Jelmyto (TN); Mitomycin (TN); Muamycin (TN) |
(P) unclassified |
D00210 |
Norfloxacin (JP18/USP/INN); Noroxin (TN) |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(CI,P) CYP induction: CYP3A4 |
D00214 |
Dactinomycin (USP); Actinomycin D (JP18); Cosmegen (TN) |
(P) unclassified |
D00251 |
Captopril (JP18/USP/INN); Apopril (TN); Capoten (TN) |
(P) unclassified |
D00252 |
Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00275 |
Cisplatin (JP18/USP/INN); Platinol (TN) |
(P) unclassified |
D00276 |
Clarithromycin (JP18/USP/INN); Biaxin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00282 |
Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) |
(P) CYP inhibition: CYP3A4 |
D00287 |
Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) |
(P) Enzyme: CYP3A4 |
D00288 |
Dacarbazine (JAN/USP/INN); DTIC-Dome (TN) |
(P) unclassified |
D00292 |
Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00293 |
Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 |
D00295 |
Cimetidine (JP18/USP/INN); Tagamet (TN) |
(P) CYP inhibition: CYP3A4 |
D00322 |
Fluconazole (JP18/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
D00323 |
Flucytosine (JP18/USP/INN); Ancobon (TN) |
(P) unclassified |
D00326 |
Fluoxetine (USAN/INN); Fluoxetine (TN) |
(P) unclassified |
D00341 |
Hydroxyurea (USP); Hydroxycarbamide (JAN/INN); Droxia (TN); Hydrea (TN); Siklos (TN) |
(P) unclassified |
D00343 |
Ifosfamide (JAN/USP/INN); Ifex (TN) |
(P) Enzyme: CYP3A4 |
D00350 |
Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00351 |
Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00362 |
Lisinopril (USP); Lisinopril hydrate (JP18); Lisinopril dihydrate; Prinivil (TN); Zestril (TN) |
(P) unclassified |
D00383 |
Trandolapril (JAN/USP/INN); Mavik (TN) |
(P) unclassified |
D00395 |
Troglitazone (JAN/USAN/INN); Rezulin (TN) |
(P) unclassified |
D00416 |
Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) |
(P) unclassified |
D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
D00421 |
Ramipril (USP/INN); Altace (TN) |
(P) unclassified |
D00422 |
Ranitidine (USAN/INN); Ranitidine (TN) |
(P) unclassified |
D00424 |
Rifabutin (JAN/USP/INN); Mycobutin (TN) |
(P) Enzyme: CYP3A4 |
D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
D00430 |
Secobarbital (USP/INN); Seconal (TN) |
(P) unclassified |
D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 |
D00459 |
Quinapril hydrochloride (JP18/USP); Accupril (TN) |
(P) unclassified |
D00474 |
Primidone (JP18/USP/INN); Mysoline (TN) |
(P) unclassified |
D00491 |
Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) |
(P) Enzyme: CYP3A4 |
D00499 |
Pentobarbital (USP/INN); Nembutal (TN) |
(P) unclassified |
D00500 |
Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) |
(P) unclassified |
D00506 |
Phenobarbital (JP18/USP/INN); Luminal (TN) |
(P) unclassified |
D00512 |
Phenytoin (JP18/USP/INN); Dilantin (TN) |
(P) unclassified |
D00533 |
Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) |
(P) unclassified |
D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 |
D00554 |
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00555 |
Amobarbital (JP18/INN); Isomytal (TN) |
(P) unclassified |
D00578 |
Voriconazole (JP18/USP/INN); Vfend (TN) |
(P) unclassified |
D00584 |
Fluorouracil (JP18/USP/INN); 5-FU (TN); Adrucil (TN); Carac (TN); Fluoroplex (TN) |
(P) unclassified |
D00585 |
Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) |
(P) Enzyme: CYP3A4 |
D00619 |
Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00620 |
Benazepril hydrochloride (JAN/USP); Lotensin (TN) |
(P) unclassified |
D00621 |
Enalapril maleate (JP18/USP); Renivace (TN); Vasotec (TN) |
(P) unclassified |
D00622 |
Fosinopril sodium (USP); Monopril (TN) |
(P) unclassified |
D00623 |
Moexipril hydrochloride (USP); Univasc (TN) |
(P) unclassified |
D00624 |
Perindopril erbumine (JAN/USP); Aceon (TN) |
(P) unclassified |
D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 |
D00673 |
Ranitidine hydrochloride (JP18/USP); Zantac (TN) |
(P) unclassified |
D00698 |
Aprobarbital (INN); Alurate (TN) |
(P) unclassified |
D00699 |
Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) |
(P) unclassified |
D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) unclassified |
D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
D00707 |
Fomepizole (JAN/USAN/INN); Antizol (TN) |
(P) CYP inhibition: CYP3A4 |
D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) unclassified |
D00713 |
Thiamylal sodium (JP18); Surital (TN) |
(P) unclassified |
D00714 |
Thiopental sodium (JP18/USP/INN); Pentothal (TN) |
(P) unclassified |
D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Enzyme: CYP3A4 / Target: MTOR / CYP inhibition: CYP3A4 |
D00780 |
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00823 |
Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) |
(P) unclassified |
D00824 |
Fluvoxamine maleate (JP18/USP); Luvox (TN) |
(P) CYP inhibition: CYP3A4 |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
D00851 |
Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) |
(P) unclassified |
D00854 |
Quinupristin and dalfopristin; Synercid (TN) |
(P) CYP inhibition: CYP3A4 |
D00879 |
Rifapentine (USAN/INN); Priftin (TN) |
(P) CYP induction: CYP3A4 |
D00882 |
Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) |
(P) unclassified |
D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) Enzyme: CYP3A4 |
D00895 |
Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) |
(P) unclassified |
D00896 |
Efavirenz (JAN/USP/INN); Sustiva (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00960 |
Anastrozole (JP18/USP/INN); Arimidex (TN) |
(P) CYP inhibition: CYP3A4 |
D00961 |
Bicalutamide (JP18/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
D00975 |
Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01059 |
Nimustine hydrochloride (JAN); Nidran (TN) |
(P) unclassified |
D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
D01068 |
Vinblastine sulfate (JP18/USP); Exal (TN); Velban (TN) |
(P) Enzyme: CYP3A4 |
D01069 |
Cilazapril (USAN); Cilazapril hydrate (JP18); Inhibace (TN) |
(P) unclassified |
D01071 |
Hexobarbital (JAN/INN) |
(P) unclassified |
D01078 |
Telithromycin (JAN/USAN/INN); Ketek (TN) |
(P) unclassified |
D01119 |
Temocapril hydrochloride (JP18/USAN); Acecol (TN) |
(P) unclassified |
D01155 |
Gemcitabine hydrochloride (JAN/USP); Gemzar (TN) |
(P) unclassified |
D01211 |
Leucovorin calcium (USP); Calcium folinate (JP18); Uzel (TN); Wellcovorin (TN) |
(P) unclassified |
D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01235 |
Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01236 |
Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 |
D01264 |
Daunorubicin hydrochloride (JP18/USP); Cerubidine (TN) |
(P) unclassified |
D01275 |
Doxorubicin hydrochloride (JP18/USP); Adriacin (TN); Adriamycin (TN); Doxil (TN); Rubex (TN) |
(P) unclassified |
D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
D01280 |
Warfarin potassium (JP18); Athrombin-K (TN) |
(P) unclassified |
D01309 |
Doxifluridine (JP18/INN); Furtulon (TN) |
(P) unclassified |
D01310 |
Secobarbital sodium (JAN/USP); Seconal sodium (TN) |
(P) unclassified |
D01322 |
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01339 |
Midecamycin (JP18/INN); Medemycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01361 |
Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) |
(P) unclassified |
D01363 |
Carboplatin (JP18/USP/INN); Paraplatin (TN) |
(P) unclassified |
D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) unclassified |
D01404 |
Sobuzoxane (JAN); Perazolin (TN) |
(P) unclassified |
D01416 |
Nedaplatin (JAN/INN); Aqupla (TN) |
(P) unclassified |
D01425 |
Lopinavir (JAN/USP/INN) |
(P) unclassified |
D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
D01510 |
Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01549 |
Imidapril hydrochloride (JP18); Tanatril (TN) |
(P) unclassified |
D01615 |
Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01632 |
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01633 |
Enocitabine (JAN/INN); Sunrabin (TN) |
(P) unclassified |
D01636 |
Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01667 |
Delapril hydrochloride (JAN/USAN); Adecut (TN) |
(P) unclassified |
D01740 |
Barbital (JP18/INN); Barbital (TN) |
(P) unclassified |
D01747 |
Idarubicin hydrochloride (JP18/USP); Idamycin (TN) |
(P) unclassified |
D01760 |
Ranimustine (JAN/INN); Cymerin (TN) |
(P) unclassified |
D01769 |
Vindesine sulfate (JAN/USAN); Fildesin (TN) |
(P) unclassified |
D01790 |
Oxaliplatin (JAN/USP/INN); Eloxatin (TN) |
(P) unclassified |
D01832 |
Modafinil (JAN/USP/INN); Provigil (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01900 |
Alacepril (JP18/INN); Cetapril (TN) |
(P) unclassified |
D01907 |
Fludarabine phosphate (JAN/USP); Fludara (TN) |
(P) unclassified |
D01911 |
Aclarubicin hydrochloride (JP18); Aclacinon (TN) |
(P) unclassified |
D01935 |
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) |
(P) Enzyme: CYP3A4 |
D01948 |
Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01980 |
Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) |
(P) CYP inhibition: CYP3A4 |
D02009 |
Erythromycin lactobionate (JP18/USP); Erythrocin (TN) |
(P) unclassified |
D02063 |
Peplomycin sulfate (JP18/USAN); Pepleo (TN) |
(P) unclassified |
D02096 |
Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) |
(P) CYP induction: CYP3A4 |
D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
D02126 |
Primaquine phosphate (JAN/USP); Primaquine (TN) |
(P) unclassified |
D02131 |
Tegafur and uracil; Uftoral (TN) |
(P) unclassified |
D02165 |
Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) |
(P) Enzyme: CYP3A4 |
D02166 |
Mitoxantrone hydrochloride (JAN/USP); Novantron (TN) |
(P) unclassified |
D02168 |
Topotecan hydrochloride (USAN); Nogitecan hydrochloride (JAN); Hycamtin (TN); Potactasol (TN) |
(P) unclassified |
D02174 |
Dexamethasone acetate (JAN/USP); Decadronal (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02177 |
Bleomycin sulfate (JP18/USP); Blenoxane (TN) |
(P) unclassified |
D02184 |
Erythromycin stearate (JP18/USP); Bristamycin (TN) |
(P) unclassified |
D02197 |
Vincristine sulfate (JP18/USP); VCR; Marqibo (TN); Oncovin (TN); Vincasar (TN); Vincrex (TN) |
(P) unclassified |
D02214 |
Epirubicin hydrochloride (JP18/USP); EPI; Ellence (TN) |
(P) unclassified |
D02252 |
Amobarbital sodium (JAN/USP); Amytal sodium (TN) |
(P) unclassified |
D02253 |
Pentobarbital calcium (JP18); Ravona (TN) |
(P) unclassified |
D02356 |
Verapamil (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02372 |
Perospirone hydrochloride hydrate (JAN); Lullan (TN) |
(P) unclassified |
D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) unclassified |
D02523 |
Erythromycin acistrate (USAN); Erasis (TN) |
(P) unclassified |
D02524 |
Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) |
(P) unclassified |
D02525 |
Erythromycin propionate (USAN) |
(P) unclassified |
D02537 |
Dronedarone (INN) |
(P) unclassified |
D02554 |
Rifaximin (JAN/USAN/INN); Xifaxan (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) CYP inhibition: CYP3A4 |
D02556 |
Ravuconazole (prop.INN) |
(P) unclassified |
D02591 |
Dexamethasone acefurate (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02592 |
Dexamethasone beloxil (USAN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02618 |
Butobarbital (BAN); Butethal; Neonal (TN) |
(P) unclassified |
D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
D02732 |
Pranlukast hydrate (JP18); Onon (TN) |
(P) Enzyme: CYP3A4 |
D02817 |
Allobarbital (USAN/INN) |
(P) unclassified |
D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D03046 |
Cytarabine ocfosfate hydrate (JAN); Cytarabine ocfosphate hydrate; Fosteabine sodium monohydrate; Starasid (TN) |
(P) unclassified |
D03077 |
Benazeprilat (USAN/INN) |
(P) unclassified |
D03098 |
Berythromycin (USAN/INN); Erythromycin B |
(P) unclassified |
D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
D03165 |
Bromocriptine (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03180 |
Butabarbital (USP); Secbutabarbital (BAN) |
(P) unclassified |
D03182 |
Butalbital (USP/INN); Sandoptal (TN) |
(P) unclassified |
D03229 |
Bleomycin hydrochloride (JP18); BLM; Bleo (TN) |
(P) unclassified |
D03230 |
Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) |
(P) unclassified |
D03250 |
Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) |
(P) unclassified |
D03440 |
Ceronapril (USAN/INN) |
(P) unclassified |
D03503 |
Cimetidine hydrochloride (USP); Cimetidine hydrochloride (TN) |
(P) CYP inhibition: CYP3A4 |
D03656 |
Darunavir (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 |
D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
D03752 |
Quinapril (INN) |
(P) unclassified |
D03753 |
Perindopril (USAN/INN) |
(P) unclassified |
D03756 |
Indolapril hydrochloride (USAN) |
(P) unclassified |
D03758 |
Libenzapril (USAN/INN) |
(P) unclassified |
D03760 |
Pentopril (USAN/INN) |
(P) unclassified |
D03763 |
Pivopril (USAN/INN) |
(P) unclassified |
D03765 |
Spirapril hydrochloride (USAN); Renormax (TN) |
(P) unclassified |
D03767 |
Zofenopril calcium (USAN); Zoprace (TN) |
(P) unclassified |
D03769 |
Enalaprilat (USP); Enalaprilat dihydrate; Vasotec (TN) |
(P) unclassified |
D03772 |
Fosinoprilat (USAN/INN) |
(P) unclassified |
D03773 |
Quinaprilat (USAN/INN) |
(P) unclassified |
D03775 |
Spiraprilat (USAN/INN) |
(P) unclassified |
D03776 |
Zofenoprilat arginine (USAN) |
(P) unclassified |
D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03846 |
Dimethyl fumarate (JAN/USAN); Tecfidera (TN) |
(P) unclassified |
D03914 |
Dronedarone hydrochloride (USP); Multaq (TN) |
(P) unclassified |
D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 |
D04054 |
Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate |
(P) unclassified |
D04059 |
Mepenzolate bromide and phenobarbital; Trancolon P (TN) |
(P) unclassified |
D04077 |
Eterobarb (USAN/INN); Antilon (TN) |
(P) unclassified |
D04112 |
Etravirine (JAN/USAN/INN); Intelence (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D04187 |
Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) |
(P) unclassified |
D04307 |
Proxyphylline, ephedrine hydrochloride and phenobarbital; Asthmolysin D (TN) |
(P) unclassified |
D04475 |
Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) |
(P) unclassified |
D04477 |
Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) |
(P) unclassified |
D04536 |
Influenza virus vaccine (USP); FluShield (TN); Fluarix quadrivalent (TN) |
(P) unclassified |
D04539 |
Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) |
(P) unclassified |
D04540 |
Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) |
(P) unclassified |
D04547 |
Insulin, isophane (USP); Isophane insulin human (genetical recombination) injectable aqueous suspension (JP18); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) |
(P) unclassified |
D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(P) unclassified |
D04866 |
Freeze-dried live attenuated measles vaccine (JP18) |
(CI) unclassified |
D04985 |
Methohexital (USP/INN) |
(P) unclassified |
D05024 |
Mibefradil dihydrochloride (USAN); Posicor (TN) |
(P) unclassified |
D05152 |
Netupitant (USAN/INN) |
(P) unclassified |
D05182 |
Influenza HA vaccine (JP18) |
(P) unclassified |
D05351 |
Josamycin propionate (JP18); Josamy (TN) |
(P) CYP inhibition: CYP3A4 |
D05544 |
Live oral polimyelitis vaccine (JAN); Poliovirus vaccine live oral; Orimune (TN) |
(CI) unclassified |
D05699 |
Ranitidine bismuth citrate (USAN); Tritec (TN) |
(P) unclassified |
D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D05932 |
Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) |
(P) unclassified |
D06076 |
Teprotide (USAN/INN) |
(P) unclassified |
D06106 |
Thiamylal |
(P) unclassified |
D06399 |
Tegafur, gimeracil and oteracil potassium; Ts-1 (TN); Teysuno (TN) |
(P) unclassified |
D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 |
D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 |
D06466 |
Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) |
(CI) unclassified |
D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06503 |
Pemetrexed sodium hydrate (JAN); Pemetrexed disodium heptahydrate; Alimta (TN) |
(P) unclassified |
D06512 |
Freeze-dried live attenuated rubella vaccine (JP18) |
(CI) unclassified |
D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D06887 |
Talbutal (INN); Lotusate (TN) |
(P) unclassified |
D07073 |
Dexamethasone cipecilate (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07085 |
Bendamustine hydrochloride (JAN/USAN); Treanda (TN); Ribomustin (TN) |
(P) unclassified |
D07100 |
Amrubicin hydrochloride (JAN/USAN); Calsed (TN) |
(P) unclassified |
D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) unclassified |
D07321 |
Vinylbital (INN); Vinylbitone |
(P) unclassified |
D07322 |
Vinbarbital (INN) |
(P) unclassified |
D07323 |
Cyclobarbital (INN); Ciclobarbital (TN) |
(P) unclassified |
D07324 |
Proxibarbal (INN); Centralgol (TN) |
(P) unclassified |
D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
D07499 |
Benazepril (INN); Benazepril Sandoz (TN); Forteekor [veterinary] (TN) |
(P) unclassified |
D07538 |
Bosentan (INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
D07699 |
Cilazapril (INN); Inhibace (TN) |
(P) unclassified |
D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07748 |
Conivaptan (INN) |
(P) unclassified |
D07757 |
Cyclobarbital calcium (BAN); Phanodorn calcium (TN) |
(P) unclassified |
D07781 |
Delapril (INN); Delaket (TN) |
(P) unclassified |
D07782 |
Delavirdine (INN) |
(P) unclassified |
D07796 |
Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07797 |
Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07798 |
Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07799 |
Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07800 |
Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07801 |
Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07802 |
Dexamethasone phosphate; Decadron-phosphate (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07866 |
Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) |
(P) Enzyme: CYP3A4 |
D07892 |
Enalapril (INN); Enalapril (TN) |
(P) unclassified |
D07909 |
Erythromycin thiocyanate; Erythrocin (TN) |
(P) unclassified |
D07910 |
Erythromycin stinoprate (INN); Erysec (TN) |
(P) unclassified |
D07928 |
Ethinylestradiol propanesulfonate; Turisteron (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07984 |
Fluvoxamine (INN) |
(P) CYP inhibition: CYP3A4 |
D07992 |
Fosinopril (INN); Monopril (TN) |
(P) unclassified |
D07993 |
Fosphenytoin (INN) |
(P) CYP induction: CYP3A4 |
D08068 |
Imidapril (INN); Hipertene (TN) |
(P) unclassified |
D08080 |
Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP18); Insulin Humacart (TN) |
(P) unclassified |
D08131 |
Lisinopril (INN); Zestril (TN) |
(P) unclassified |
D08195 |
Methadone (BAN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08217 |
Mibefradil (INN) |
(P) unclassified |
D08225 |
Moexipril (INN) |
(P) unclassified |
D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08287 |
Norfloxacin nicotinate; Quinabic soluble powder (TN) [veterinary] |
(P) unclassified |
D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) unclassified |
D08386 |
Pirarubicin hydrochloride; Pinorubin (TN); Therarubicin (TN) |
(P) unclassified |
D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
D08529 |
Spirapril (INN) |
(P) unclassified |
D08566 |
Temocapril (INN) |
(P) unclassified |
D08616 |
Teneligliptin (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08688 |
Zofenopril (INN); Zofenil (TN) |
(P) unclassified |
D08774 |
Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08837 |
Aclidinium bromide (JAN/USAN/INN); Tudorza pressair (TN); Eklira genuair (TN) |
(P) CYP inhibition: CYP3A4 |
D08876 |
Boceprevir (INN/USAN); Victrelis (TN) |
(P) unclassified |
D08914 |
Eribulin mesylate (USAN); Eribulin mesilate (JAN); Halaven (TN) |
(P) Enzyme: CYP3A4 |
D09012 |
Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(P) unclassified |
D09197 |
Valsartan and hydrochlorothiazide (JP18); Co-dio (TN) |
(P) unclassified |
D09215 |
Eslicarbazepine (USAN/INN) |
(P) CYP induction: CYP3A4 |
D09347 |
Fostamatinib (USAN) |
(P) Enzyme: CYP3A4 |
D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) Enzyme: CYP3A4 |
D09394 |
Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) |
(P) CYP inhibition: CYP3A4 |
D09612 |
Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) |
(P) CYP induction: CYP3A4 |
D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(P) Enzyme: CYP3A4 |
D09725 |
Emulsified influenza HA vaccine (A/H1N1); Arepanrix (H1N1) (TN) |
(P) unclassified |
D09727 |
Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) |
(P) unclassified |
D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 |
D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
D09881 |
Cobicistat (JAN/USAN/INN); Tybost (TN) |
(P) Enzyme-Target: CYP3A4 |
D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
D10064 |
Dabrafenib (USAN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10065 |
Daclatasvir (USAN) |
(P) Enzyme: CYP3A4 |
D10081 |
Simeprevir (JAN/USAN) |
(P) unclassified |
D10093 |
Asunaprevir (JAN/USAN); Sunvepra (TN) |
(P) CYP induction: CYP3A4 |
D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10105 |
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) |
(P) Enzyme: CYP3A4 |
D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
D10246 |
Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 |
D10469 |
Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) |
(P) unclassified |
D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10526 |
Trifluridine and tipiracil hydrochloride; Lonsurf (TN) |
(P) unclassified |
D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
D10570 |
Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) |
(P) unclassified |
D10582 |
Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) |
(P) CYP inhibition: CYP3A4 |
D10596 |
Pemetrexed sodium hemipentahydrate (JAN); Pemetrexed disodium hemipentahydrate; Pemetrexed accord (TN) |
(P) unclassified |
D10639 |
Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) |
(P) unclassified |
D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
D10644 |
Isavuconazonium (USAN) |
(P) unclassified |
D10745 |
Ombitasvir, paritaprevir and ritonavir; Technivie (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10753 |
Atazanavir and cobicistat; Evotaz (TN) |
(P) Enzyme: CYP3A4 |
D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
D10756 |
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) |
(P) unclassified |
D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 |
D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
D10882 |
Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) |
(P) CYP induction: CYP3A4 |
D10895 |
Fosaprepitant (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 |
D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
D11034 |
Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) |
(P) unclassified |
D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11072 |
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) |
(P) unclassified |
D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
D11390 |
Daunorubicin and cytarabine; Vyxeos (TN) |
(P) unclassified |
D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
D11521 |
Lamivudine, nevirapine and zidovudine |
(P) unclassified |
D11565 |
Grazoprevir (USAN/INN); Grazoprevir anhydrous |
(P) unclassified |
D11567 |
Insulin degludec and liraglutide; Xultophy (TN) |
(P) unclassified |
D11580 |
Perindopril arginine |
(P) unclassified |
D11661 |
Bendamustine hydrochloride hydrate (JAN); Bendamustine hydrochloride monohydrate; Treakisym (TN) |
(P) unclassified |
D11673 |
Berotralstat (USAN/INN) |
(P) CYP inhibition: CYP3A4 |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 |
D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
D11858 |
Omeprazole magnesium, amoxicillin and rifabutin; Talicia (TN) |
(P) unclassified |
D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
D11968 |
Teneligliptin hydrobromide (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
D12015 |
St. John's wort; SJW |
(P) unclassified |
D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) Enzyme: CYP3A4 |
D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(P) unclassified |
D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |
D12619 |
Ensitrelvir (USAN/INN) |
(P) unclassified |
D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |