+E Drug
#
Target-based Classification of Drugs
!
AG Protein-coupled receptors
B Rhodopsin family
C Acetylcholine (muscarinic)
D CHRM [HSA:1128 1129 1131 1132 1133] [KO:K04129 K04130 K04131 K04132 K04133]
E D08389 Pirenzepine (INN)
E D01297 Pirenzepine hydrochloride (USAN)
E D05276 Pirenzepine hydrochloride hydrate (JP18) <JP>
E D08160 Mebeverine (INN)
E D04868 Mebeverine hydrochloride (USAN)
E D07821 Dihexyverine (INN)
E D03824 Dihexyverine hydrochloride (USAN)
E D07079 Difemerine (INN)
E D08382 Piperidolate (INN)
E D01165 Piperidolate hydrochloride (JAN) <JP>
E D03088 Benzilonium bromide (USAN/INN)
E D07081 Penthienate bromide (NF XIII)
E D00481 Propantheline bromide (JP18/USP/INN) <JP>
E D07083 Otilonium bromide (INN)
E D00721 Methanthelinium bromide (INN)
E D05535 Poldine methylsulfate (USAN)
E D00720 Mepenzolate bromide (JP18/INN) <JP>
E D01532 Bevonium methylsulfate (JAN)
E D07084 Pipenzolate bromide (INN)
E D01201 Tiemonium iodide (JAN/INN)
E D01377 Prifinium bromide (JAN/INN)
E D02535 Timepidium bromide hydrate (JP18) <JP>
E D07070 Fenpiverinium bromide (INN)
E D01538 Valethamate bromide (JAN)
E D00113 Atropine (USP)
E D02069 Atropine sulfate (JP18/USP) <JP/US>
E D00147 Hyoscyamine (USP)
E D00719 Hyoscyamine sulfate (USP)
E D01648 Hyoscyamine methylbromide (JAN)
E D04479 Hyoscyamine hydrobromide (USP)
E D01451 Scopolamine butylbromide (JP18) <JP>
E D01077 Methylatropine nitrate (USAN)
E D03814 Atropine methylbromide (JAN)
E D01976 N-Methylscopolamine methylsulfate (JAN) <JP>
E D07951 Fentonium bromide (INN)
E D07099 Cimetropium bromide (JAN/INN)
E D02070 Homatropine methylbromide (USP)
E D00138 Scopolamine (INN) <US>
E D02071 Scopolamine hydrobromide (USP) <JP>
E D10939 Glycopyrronium tosylate (USAN) <JP/US>
E D00465 Oxybutynin (USAN/INN) <US>
E D00722 Oxybutynin chloride (USP) <JP/US>
E D08441 Propiverine (INN)
E D01007 Propiverine hydrochloride (JP18) <JP>
E D00765 Rocuronium bromide (JAN/USP/INN) <JP/US>
E D08418 Pridinol (INN)
E D02064 Pridinol mesilate (JAN) <JP>
E D08419 Pridinol hydrochloride
E D08638 Trihexyphenidyl (INN)
E D00787 Trihexyphenidyl hydrochloride (JP18/USP) <JP/US>
E D00779 Biperiden (JAN/USP/INN)
E D02246 Biperiden hydrochloride (JP18/USP) <JP>
E D02247 Biperiden lactate (JAN/USP) <JP>
E D08209 Metixene (INN)
E D01871 Methixene hydrochloride (USAN)
E D08425 Procyclidine (INN)
E D00782 Procyclidine hydrochloride (USP)
E D08426 Profenamine (INN)
E D01118 Profenamine hydrochloride (JAN)
E D03276 Profenamine hibenzate (JAN)
E D03711 Dexetimide (USAN/INN)
E D07804 Dexetimide hydrochloride
E D07301 Phenglutarimide (INN)
E D08157 Mazaticol (INN)
E D03264 Mazaticol hydrochloride hydrate (JAN) <JP>
E D07302 Bornaprine (INN)
E D07303 Tropatepine (INN)
E D08653 Tropatepine hydrochloride
E D07511 Benzatropine (INN)
E D00778 Benztropine mesylate (USP) <US>
E D04087 Ethybenztropine (USAN)
E D00270 Chlorpromazine (USP/INN)
E D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
E D03274 Chlorpromazine hibenzate (JAN)
E D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
E D09819 Chlorpromazine tannate (JAN)
E D00524 Carbachol (JAN/USP/INN) <US>
E D01000 Bethanechol chloride (JP18/USP) <JP/US>
E D07349 Choline alfoscerate (INN)
E D02212 Ipratropium bromide (USP) <JP/US>
E D01946 Oxitropium bromide (JAN/INN)
E D08837 Aclidinium bromide (JAN/USAN/INN) <JP/US>
E D10181 Umeclidinium bromide (JAN/USAN) <JP/US>
E D00999 Acetylcholine chloride (JP18/USP/INN) <JP/US>
E D07759 Cyclopentolate (INN)
E D01002 Cyclopentolate hydrochloride (JP18/USP) <JP/US>
E D01004 Homatropine hydrobromide (JP18/USP)
E D00397 Tropicamide (JP18/USP/INN) <JP/US>
E D04970 Methacholine chloride (JAN/USP/INN) <JP/US>
E D00232 Anisotropine methylbromide (USAN)
E D00715 Methscopolamine bromide (USP) <US>
E D00716 Clidinium bromide (USP/INN)
E D01175 Carpronium chloride (JAN/INN) <JP>
E D01231 Piroheptine hydrochloride (JAN) <JP>
E D01315 Methylbenactyzium bromide (JP18/INN)
E D01318 Diphenidol hydrochloride (USAN) <JP>
E D01359 Etomidoline (JAN/INN)
E D01463 Diponium bromide (JAN/INN)
E D01491 Butropium bromide (JP18/INN) <JP>
E D01521 Pipethanate hydrochloride (JAN)
E D01600 Diphenylpiperidinomethyldioxolan iodide (JAN)
E D01815 Oxapium iodide (JP18/INN)
E D01955 Aclatonium napadisilate (JAN)
E D01987 Pipethanate ethobromide (JAN)
E D02417 Flutropium bromide (JAN)
E D02603 Diethazine hydrochloride
E D03011 Atropine oxide hydrochloride (USAN)
E D03076 Benapryzine hydrochloride (USAN)
E D03087 Benzetimide hydrochloride (USAN)
E D03858 Diphenidol (USAN/INN)
E D03859 Diphenidol pamoate (USAN)
E D03970 Elantrine (USAN)
E D03979 Elucaine (USAN)
E D04116 Eucatropine hydrochloride (USP XXXII)
E D04434 Heteronium bromide (USAN/INN)
E D05012 Metoquizine (USAN/INN)
E D05035 Milameline hydrochloride (USAN)
E D05360 Parapenzolate bromide (USAN/INN)
E D05418 Pentapiperium methylsulfate (USAN)
E D05452 Phencarbamide (USAN)
E D05628 Propenzolate hydrochloride (USAN)
E D05703 Rapacuronium bromide (USAN/INN)
E D06015 Tazomeline citrate (USAN)
E D06061 Tematropium methylsulfate (USAN)
E D06175 Tofenacin hydrochloride (USAN)
E D06192 Toquizine (USAN)
E D06217 Triampyzine sulfate (USAN)
E D07477 Atropine oxide (INN)
E D07513 Benzetimide (INN)
E D07823 Diethazine (INN)
E D08384 Pipethanate (INN)
E D08395 Piroheptine (INN)
E D08595 Tiemonium methylsulfate
E D09402 Darotropium bromide (USAN/INN)
E D09752 Carpronium chloride hydrate (JAN) <JP>
E D10180 Umeclidinium (USAN)
E D10545 Batefenterol (USAN)
E D10546 Batefenterol succinate (USAN)
E D11383 Blarcamesine (USAN)
E D11549 Blarcamesine hydrochloride (USAN)
D CHRM1 [HSA:1128] [KO:K04129]
E D08325 Oxyphencyclimine (INN)
E D01006 Oxyphencyclimine hydrochloride (JAN)
E D07820 Dicycloverine (INN)
E D00717 Dicyclomine hydrochloride (JAN/USP) <US>
E D06877 Oxyphenonium bromide (INN)
E D00723 Tridihexethyl chloride (BAN)
E D06273 Imidafenacin (JAN/INN) <JP>
E D02750 Aceclidine (USAN/INN)
E D02876 Alvameline maleate (USAN)
E D04057 Esoxybutynin chloride (USAN)
E D05779 Sabcomeline hydrochloride (USAN)
E D06000 Talsaclidine fumarate (USAN)
E D06330 Xanomeline (USAN)
E D06331 Xanomeline tartrate (USAN)
E D11098 Telenzepine hydrochloride hydrate (JAN)
D CHRM2 [HSA:1129] [KO:K04130]
E D08325 Oxyphencyclimine (INN)
E D01006 Oxyphencyclimine hydrochloride (JAN)
E D07820 Dicycloverine (INN)
E D00717 Dicyclomine hydrochloride (JAN/USP) <US>
E D00723 Tridihexethyl chloride (BAN)
E D07853 Dimetindene (INN)
E D01103 Trospium chloride (JAN/USP/INN) <US>
E D07226 Fesoterodine (INN)
E D08923 Fesoterodine fumarate (JAN/USAN) <JP/US>
E D02292 Gallamine triethiodide (USP)
E D00525 Pilocarpine (JAN/USP)
E D02200 Pilocarpine hydrochloride (JP18/USP) <JP/US>
E D05478 Pilocarpine nitrate (USP)
E D08376 Pilocarpine borate
E D02876 Alvameline maleate (USAN)
E D04057 Esoxybutynin chloride (USAN)
D CHRM3 [HSA:1131] [KO:K04131]
E D08325 Oxyphencyclimine (INN)
E D01006 Oxyphencyclimine hydrochloride (JAN)
E D07078 Rociverine (INN)
E D07820 Dicycloverine (INN)
E D00717 Dicyclomine hydrochloride (JAN/USP) <US>
E D00540 Glycopyrrolate (USP) <JP/US>
E D00723 Tridihexethyl chloride (BAN)
E D01005 Isopropamide iodide (JAN/USP/INN)
E D01003 Hexocyclium metilsulfate (INN)
E D06878 Diphemanil metilsulfate (INN)
E D00193 Dexpanthenol (USP/INN) <JP>
E D10938 Glycopyrronium (USAN)
E D00646 Tolterodine (USAN/INN)
E D01148 Tolterodine tartrate (JAN/USP) <JP/US>
E D08522 Solifenacin (INN)
E D01269 Solifenacin succinate (JAN/USAN/INN) <JP/US>
E D01103 Trospium chloride (JAN/USP/INN) <US>
E D03654 Darifenacin (USAN/INN)
E D01699 Darifenacin hydrobromide (JAN/USAN) <US>
E D07226 Fesoterodine (INN)
E D08923 Fesoterodine fumarate (JAN/USAN) <JP/US>
E D10853 Desfesoterodine (INN)
E D06273 Imidafenacin (JAN/INN) <JP>
E D00525 Pilocarpine (JAN/USP)
E D02200 Pilocarpine hydrochloride (JP18/USP) <JP/US>
E D05478 Pilocarpine nitrate (USP)
E D08376 Pilocarpine borate
E D07667 Cevimeline (INN)
E D00661 Cevimeline hydrochloride (USAN) <JP/US>
E D01929 Tiotropium bromide hydrate (JAN) <JP/US>
E D10978 Revefenacin (USAN/INN) <US>
E D01875 Tiquizium bromide (JAN/INN) <JP>
E D02876 Alvameline maleate (USAN)
E D04057 Esoxybutynin chloride (USAN)
E D10989 Sofpironium bromide (JAN/USAN/INN) <JP>
E D11900 Navafenterol (USAN)
E D11901 Navafenterol saccharinate (USAN)
D CHRM4 [HSA:1132] [KO:K04132]
E D06330 Xanomeline (USAN)
E D06331 Xanomeline tartrate (USAN)
E D12468 Emraclidine (USAN/INN)
C Adrenaline
D ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
E D00095 Epinephrine (USP/INN) <JP/US>
E D00996 Epinephrine hydrochloride (JAN)
E D02149 Epinephrine bitartrate (JAN/USP)
E D02774 Adrenalone (USAN/INN)
E D07560 Adrenalone hydrochloride
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D07931 Etilefrine (INN)
E D01573 Etilefrine hydrochloride (JP18) <JP>
E D00076 Noradrenaline (JP18) <JP>
E D05206 Norepinephrine bitartrate (USP) <US>
E D08284 Norepinephrine hydrochoride
E D09794 Norepinephrine hydrochloride (JAN)
E D08286 Norfenefrine (INN)
E D01405 Norfenefrine hydrochloride (JAN)
E D08365 Phenylephrine (INN)
E D00511 Phenylephrine hydrochloride (JP18/USP) <JP/US>
E D08366 Phenylephrine tartrate
E D08966 Phenylephrine bitartrate (USP)
E D08192 Metaraminol (INN)
E D01019 Metaraminol bitartrate (JAN/USP)
E D08201 Methoxamine (BAN)
E D01020 Methoxamine hydrochloride (JAN)
E D08220 Midodrine (INN)
E D01307 Midodrine hydrochloride (JAN/USP) <JP/US>
E D00124 Ephedrine (USP)
E D01386 Ephedrine hydrochloride (JP18/USP) <JP/US>
E D04018 Ephedrine sulfate (USP) <US>
E D01277 Droxidopa (JP18/USAN/INN) <JP/US>
E D08411 Prazosin (INN)
E D00609 Prazosin hydrochloride (JP18/USP) <JP/US>
E D04531 Indoramin (USAN/INN)
E D04532 Indoramin hydrochloride (USAN)
E D08212 Trimazosin (INN)
E D06234 Trimazosin hydrochloride (USAN)
E D07874 Doxazosin (INN)
E D00608 Doxazosin mesylate (USP) <JP/US>
E D01333 Urapidil (JP18/INN) <JP>
E D08662 Urapidil hydrochloride
E D08362 Phentolamine (INN)
E D00509 Phentolamine mesylate (USP) <JP/US>
E D08614 Tolazoline (INN)
E D00997 Tolazoline hydrochloride (JAN/USP)
E D02268 Ergoloid mesylates (USP)
E D01290 Nicergoline (JP18/USAN/INN) <JP>
E D08271 Nicergoline tartrate
E D07834 Dihydroergocristine (BAN)
E D07833 Dihydroergocristine mesilate (BAN)
E D08358 Phenoxybenzamine (INN)
E D00507 Phenoxybenzamine hydrochloride (USP) <US>
E D08239 Moxisylyte (INN)
E D01571 Moxisylyte hydrochloride (JAN)
E D08064 Ifenprodil (INN)
E D01445 Ifenprodil tartrate (JP18) <JP>
E D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
E D08106 Labetalol (INN)
E D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
E D00255 Carvedilol (JP18/USP/INN) <JP/US>
E D03415 Carvedilol phosphate (USAN) <US>
E D08207 Methylergometrine (INN)
E D00680 Methylergonovine maleate (USP) <JP/US>
E D07906 Ergotamine (INN)
E D07905 Ergometrine (INN)
E D01163 Ergonovine maleate (USP)
E D08560 Tamsulosin (INN)
E D01024 Tamsulosin hydrochloride (JP18/USP) <JP/US>
E D08569 Terazosin (INN)
E D00610 Terazosin hydrochloride (USP) <JP/US>
E D11585 Terazosin hydrochloride anhydrous <US>
E D00679 Ergotamine tartrate (JP18/USP) <US>
E D01485 Propericiazine (JAN) <JP>
E D00308 Droperidol (JP18/USP/INN) <JP/US>
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D08257 Nefazodone (INN)
E D00819 Nefazodone hydrochloride (USP) <US>
E D08578 Tetryzoline (INN)
E D00756 Tetrahydrozoline nitrate (JAN)
E D01023 Tetrahydrozoline hydrochloride (JAN/USP)
E D08684 Xylometazoline (INN)
E D00757 Xylometazoline hydrochloride (USP)
E D08253 Naphazoline (INN)
E D00743 Naphazoline hydrochloride (JP18/USP)
E D01021 Naphazoline nitrate (JP18) <JP>
E D08624 Tramazoline (INN)
E D01347 Tramazoline hydrochloride (JAN/USAN) <JP>
E D08368 Phenylpropanolamine (INN)
E D01224 Phenylpropanolamine hydrochloride (JAN/USP)
E D05466 Phenylpropanolamine polistirex (USAN)
E D08449 Pseudoephedrine (INN)
E D00485 Pseudoephedrine hydrochloride (USP)
E D05648 Pseudoephedrine polistirex (USAN)
E D05649 Pseudoephedrine sulfate (USP)
E D02349 Dipivefrin (USAN)
E D01017 Dipivefrin hydrochloride (USP) <JP>
E D08115 Levobunolol (INN)
E D01025 Levobunolol hydrochloride (JAN/USP) <JP/US>
E D07775 Dapiprazole (INN)
E D03648 Dapiprazole hydrochloride (USAN) <US>
E D00607 Guanadrel sulfate (USAN)
E D01171 Monatepil maleate (JAN/USAN)
E D01444 Bunitrolol hydrochloride (JAN)
E D01469 Amosulalol hydrochloride (JP18) <JP>
E D01674 Naftopidil (JP18/INN) <JP>
E D01691 Nipradilol (JAN/INN) <JP>
E D01830 Arotinolol hydrochloride (JP18) <JP>
E D01887 Bunazosin hydrochloride (JP18) <JP>
E D01952 L-Methylephedrine hydrochloride (JAN)
E D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
E D02568 Flesinoxan (INN)
E D02901 Amidephrine mesylate (USAN)
E D03887 Domazoline fumarate (USAN)
E D04026 Epinephryl borate (USP)
E D05228 Octodrine (USAN/INN)
E D05395 Pelanserin hydrochloride (USAN)
E D05637 Propylhexedrine (USP/INN)
E D05688 Racepinephrine (USP/INN)
E D05689 Racepinephrine hydrochloride (USP)
E D07451 Amosulalol (INN)
E D07465 Arotinolol (INN)
E D07550 Bunazosin (INN)
E D08029 Guanadrel (INN)
E D08206 Methylephedrine (BAN)
E D08444 Propylhexedrine hydrochloride
E D08982 Racephedrine Hydrochloride (USAN)
E D09842 dl-Methylephedrine saccharinate (JAN)
D ADRA1A [HSA:148] [KO:K04135]
E D07097 Isometheptene mucate (USP)
E D08322 Oxymetazoline (INN)
E D01022 Oxymetazoline hydrochloride (JAN/USP) <US>
E D07124 Alfuzosin (INN)
E D01692 Alfuzosin hydrochloride (JAN/USAN) <US>
E D01965 Silodosin (JP18/INN) <JP/US>
E D04184 Fiduxosin hydrochloride (USAN)
E D06380 Zolertine hydrochloride (USAN)
E D06394 Dabuzalgron hydrochloride (USAN)
E D09784 Garomefrine hydrochloride (JAN)
D ADRA1D [HSA:146] [KO:K04137]
E D06380 Zolertine hydrochloride (USAN)
D ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
E D00095 Epinephrine (USP/INN) <JP/US>
E D00996 Epinephrine hydrochloride (JAN)
E D02149 Epinephrine bitartrate (JAN/USP)
E D07931 Etilefrine (INN)
E D01573 Etilefrine hydrochloride (JP18) <JP>
E D00076 Noradrenaline (JP18) <JP>
E D05206 Norepinephrine bitartrate (USP) <US>
E D08284 Norepinephrine hydrochoride
E D09794 Norepinephrine hydrochloride (JAN)
E D08192 Metaraminol (INN)
E D01019 Metaraminol bitartrate (JAN/USP)
E D00124 Ephedrine (USP)
E D01386 Ephedrine hydrochloride (JP18/USP) <JP/US>
E D04018 Ephedrine sulfate (USP) <US>
E D01277 Droxidopa (JP18/USAN/INN) <JP/US>
E D08205 Methyldopa (INN)
E D00405 Methyldopa (USP) <JP/US>
E D00281 Clonidine (JAN/USP/INN) <US>
E D00604 Clonidine hydrochloride (JP18/USP) <JP/US>
E D05087 Moxonidine (USAN/INN)
E D08482 Rilmenidine (INN)
E D01603 Bethanidine sulfate (JAN/USAN)
E D08362 Phentolamine (INN)
E D00509 Phentolamine mesylate (USP) <JP/US>
E D08614 Tolazoline (INN)
E D00997 Tolazoline hydrochloride (JAN/USP)
E D02268 Ergoloid mesylates (USP)
E D07834 Dihydroergocristine (BAN)
E D07833 Dihydroergocristine mesilate (BAN)
E D08358 Phenoxybenzamine (INN)
E D00507 Phenoxybenzamine hydrochloride (USP) <US>
E D07540 Brimonidine (INN)
E D02076 Brimonidine tartrate (JAN/USAN) <JP/US>
E D08207 Methylergometrine (INN)
E D00680 Methylergonovine maleate (USP) <JP/US>
E D07905 Ergometrine (INN)
E D01163 Ergonovine maleate (USP)
E D08685 Yohimbine (DCF)
E D06671 Yohimbine hydrochloride (USP)
E D08611 Tizanidine (INN)
E D00776 Tizanidine hydrochloride (JP18/USP) <JP/US>
E D00270 Chlorpromazine (USP/INN)
E D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
E D03274 Chlorpromazine hibenzate (JAN)
E D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
E D09819 Chlorpromazine tannate (JAN)
E D00283 Clozapine (JAN/USP/INN) <JP/US>
E D00514 Dexmedetomidine (USAN/INN)
E D01205 Dexmedetomidine hydrochloride (JAN/USP) <JP/US>
E D08216 Mianserin (INN)
E D01358 Mianserin hydrochloride (JAN/USAN) <JP>
E D00563 Mirtazapine (JAN/USP/INN) <JP/US>
E D11056 Mirtazapine hydrate (JAN)
E D08141 Lofexidine (INN)
E D04765 Lofexidine hydrochloride (USAN) <US>
E D08684 Xylometazoline (INN)
E D00757 Xylometazoline hydrochloride (USP)
E D08624 Tramazoline (INN)
E D01347 Tramazoline hydrochloride (JAN/USAN) <JP>
E D08368 Phenylpropanolamine (INN)
E D01224 Phenylpropanolamine hydrochloride (JAN/USP)
E D05466 Phenylpropanolamine polistirex (USAN)
E D08449 Pseudoephedrine (INN)
E D00485 Pseudoephedrine hydrochloride (USP)
E D05648 Pseudoephedrine polistirex (USAN)
E D05649 Pseudoephedrine sulfate (USP)
E D02349 Dipivefrin (USAN)
E D01017 Dipivefrin hydrochloride (USP) <JP>
E D07461 Apraclonidine (INN)
E D01008 Apraclonidine hydrochloride (JAN/USP) <JP/US>
E D00605 Guanabenz acetate (JP18/USP) <JP>
E D00607 Guanadrel sulfate (USAN)
E D01952 L-Methylephedrine hydrochloride (JAN)
E D02034 Setiptiline maleate (JAN) <JP>
E D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
E D02388 Levonordefrin (USP)
E D02407 Lidamidine hydrochloride (USAN)
E D02569 Sunepitron hydrochloride (USAN)
E D02972 Aptazapine maleate (USAN)
E D03002 Atipamezole (USAN/INN)
E D03672 Delequamine hydrochloride (USAN)
E D03702 Detomidine hydrochloride (USAN)
E D03887 Domazoline fumarate (USAN)
E D04026 Epinephryl borate (USP)
E D04124 Fadolmidine hydrochloride (USAN)
E D04223 Fluparoxan hydrochloride (USAN)
E D04375 Guanabenz (USAN/INN)
E D04883 Medetomidine hydrochloride (USAN)
E D05119 Napamezole hydrochloride (USAN)
E D05228 Octodrine (USAN/INN)
E D05637 Propylhexedrine (USP/INN)
E D05688 Racepinephrine (USP/INN)
E D05689 Racepinephrine hydrochloride (USP)
E D06344 Xylazine hydrochloride (USP)
E D07795 Detomidine (INN)
E D08029 Guanadrel (INN)
E D08126 Lidamidine (INN)
E D08165 Medetomidine (INN)
E D08206 Methylephedrine (BAN)
E D08444 Propylhexedrine hydrochloride
E D08487 Romifidine (INN)
E D08511 Setiptiline (INN)
E D08683 Xylazine (USP/INN)
E D08982 Racephedrine Hydrochloride (USAN)
E D09842 dl-Methylephedrine saccharinate (JAN)
E D11320 Vatinoxan (USAN)
E D11321 Vatinoxan hydrochloride (USAN)
D ADRA2A [HSA:150] [KO:K04138]
E D08031 Guanfacine (INN)
E D00606 Guanfacine hydrochloride (JAN/USP) <JP/US>
E D00560 Pimozide (JP18/USP/INN) <US>
D ADRA2B [HSA:151] [KO:K04139]
E D04514 Imiloxan hydrochloride (USAN)
D ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
E D00095 Epinephrine (USP/INN) <JP/US>
E D00996 Epinephrine hydrochloride (JAN)
E D02149 Epinephrine bitartrate (JAN/USP)
E D07931 Etilefrine (INN)
E D01573 Etilefrine hydrochloride (JP18) <JP>
E D08090 Isoprenaline (INN)
E D01390 Isoproterenol hydrochloride (USP) <JP/US>
E D02066 Isoproterenol sulfate (USP)
E D02150 l-Isoprenaline hydrochloride (JP18) <JP>
E D00076 Noradrenaline (JP18) <JP>
E D05206 Norepinephrine bitartrate (USP) <US>
E D08284 Norepinephrine hydrochoride
E D09794 Norepinephrine hydrochloride (JAN)
E D02976 Arbutamine hydrochloride (USAN)
E D00124 Ephedrine (USP)
E D01386 Ephedrine hydrochloride (JP18/USP) <JP/US>
E D04018 Ephedrine sulfate (USP) <US>
E D01277 Droxidopa (JP18/USAN/INN) <JP/US>
E D07156 Alprenolol (INN)
E D01182 Alprenolol hydrochloride (JP18/USAN)
E D08318 Oxprenolol (INN)
E D01806 Oxprenolol hydrochloride (JP18/USP)
E D00513 Pindolol (JP18/USP/INN) <JP/US>
E D08443 Propranolol (INN)
E D00483 Propranolol hydrochloride (JP18/USP) <JP/US>
E D07181 Mepindolol (INN)
E D07624 Carteolol (INN)
E D00599 Carteolol hydrochloride (JP18/USP) <JP/US>
E D07182 Tertatolol (INN)
E D08572 Tertatolol hydrochloride
E D07537 Bopindolol (INN)
E D01794 Bopindolol malonate (JAN)
E D07590 Bupranolol (INN)
E D01454 Bupranolol hydrochloride (JP18)
E D08074 Penbutolol (INN)
E D00602 Penbutolol sulfate (JP18/USP)
E D07183 Cloranolol (INN)
E D07184 Talinolol (INN)
E D08368 Phenylpropanolamine (INN)
E D01224 Phenylpropanolamine hydrochloride (JAN/USP)
E D05466 Phenylpropanolamine polistirex (USAN)
E D08449 Pseudoephedrine (INN)
E D00485 Pseudoephedrine hydrochloride (USP)
E D05648 Pseudoephedrine polistirex (USAN)
E D05649 Pseudoephedrine sulfate (USP)
E D02349 Dipivefrin (USAN)
E D01017 Dipivefrin hydrochloride (USP) <JP>
E D08115 Levobunolol (INN)
E D01025 Levobunolol hydrochloride (JAN/USP) <JP/US>
E D02374 Metipranolol (USAN/INN)
E D02081 Metipranolol hydrochloride
E D07496 Befunolol (INN)
E D01512 Befunolol hydrochloride (JAN)
E D01444 Bunitrolol hydrochloride (JAN)
E D01504 Bufetolol hydrochloride (JP18) <JP>
E D01691 Nipradilol (JAN/INN) <JP>
E D01795 Tilisolol hydrochloride (JAN)
E D01906 Dilevalol hydrochloride (JAN/USAN)
E D01952 L-Methylephedrine hydrochloride (JAN)
E D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
E D02765 Adaprolol maleate (USAN)
E D02834 Alprenoxime hydrochloride (USAN)
E D03502 Cimaterol (USAN/INN)
E D03729 Dexpropranolol hydrochloride (USAN)
E D03759 Diacetolol hydrochloride (USAN)
E D04026 Epinephryl borate (USP)
E D04120 Exaprolol hydrochloride (USAN)
E D04190 Flestolol sulfate (USAN)
E D04888 Medroxalol (USAN/INN)
E D04889 Medroxalol hydrochloride (USAN)
E D05228 Octodrine (USAN/INN)
E D05345 Pamatolol sulfate (USAN)
E D05688 Racepinephrine (USP/INN)
E D05689 Racepinephrine hydrochloride (USP)
E D06014 Tazolol hydrochloride (USAN)
E D06162 Tiprenolol hydrochloride (USAN)
E D06176 Tolamolol (USAN/INN)
E D08206 Methylephedrine (BAN)
E D08598 Tilisolol (INN)
E D08982 Racephedrine Hydrochloride (USAN)
E D09842 dl-Methylephedrine saccharinate (JAN)
E D09843 Beradilol monoethyl maleate (JAN)
D ADRB1 [HSA:153] [KO:K04141]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D03879 Dobutamine (USAN/INN)
E D00632 Dobutamine hydrochloride (JP18/USP) <JP/US>
E D03880 Dobutamine lactobionate (USAN)
E D03881 Dobutamine tartrate (USAN)
E D06328 Xamoterol (USAN)
E D06329 Xamoterol fumarate (USAN)
E D08600 Timolol (INN)
E D00378 Timolol (USAN) <US>
E D00603 Timolol maleate (JP18/USP) <JP/US>
E D08525 Sotalol (INN)
E D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
E D00432 Nadolol (JP18/USP/INN) <JP/US>
E D05587 Practolol (USAN)
E D02358 Metoprolol (USAN/INN)
E D00601 Metoprolol tartrate (JP18/USP) <JP/US>
E D00635 Metoprolol succinate (USP) <US>
E D05011 Metoprolol fumarate (USP)
E D00235 Atenolol (JP18/USP/INN) <JP/US>
E D02338 Acebutolol (USAN/INN)
E D00597 Acebutolol hydrochloride (JP18/USP) <US>
E D07526 Betaxolol (INN)
E D00598 Betaxolol hydrochloride (JP18/USP) <JP/US>
E D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
E D02342 Bisoprolol (JAN/USAN/INN) <JP>
E D00634 Bisoprolol fumarate (JP18/USP) <JP/US>
E D07660 Celiprolol (INN)
E D01741 Celiprolol hydrochloride (JAN/USAN) <JP>
E D07916 Esmolol (INN)
E D00644 Esmolol hydrochloride (JAN/USP) <JP/US>
E D06646 Epanolol (USAN/INN)
E D01471 Esatenolol (JAN/INN)
E D05127 Nebivolol (USAN/INN)
E D06622 Nebivolol hydrochloride (USAN) <US>
E D01847 Landiolol hydrochloride (JAN/USAN) <JP>
E D12410 Landiolol (USAN/INN)
E D08106 Labetalol (INN)
E D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
E D00255 Carvedilol (JP18/USP/INN) <JP/US>
E D03415 Carvedilol phosphate (USAN) <US>
E D01469 Amosulalol hydrochloride (JP18) <JP>
E D01492 Bucumolol hydrochloride (JP18)
E D01830 Arotinolol hydrochloride (JP18) <JP>
E D01903 Docarpamine (JAN/INN) <JP>
E D01958 Indenolol hydrochloride (JP18)
E D02389 Primidolol (USAN/INN)
E D02614 Denopamine (JAN/INN) <JP>
E D03177 Bunolol hydrochloride (USAN)
E D03195 Butopamine (USAN/INN)
E D03449 Cetamolol hydrochloride (USAN)
E D03490 Cicloprolol hydrochloride (USAN)
E D04708 Levdobutamine lactobionate (USAN)
E D04710 Levobetaxolol hydrochloride (USAN)
E D07451 Amosulalol (INN)
E D07465 Arotinolol (INN)
E D08078 Indenolol (INN)
D ADRB2 [HSA:154] [KO:K04142]
E D03891 Dopexamine (USAN/INN)
E D03892 Dopexamine hydrochloride (USAN)
E D08092 Isoxsuprine (INN)
E D01748 Isoxsuprine hydrochloride (JP18/USP) <JP>
E D08093 Isoxsuprine lactate
E D08600 Timolol (INN)
E D00378 Timolol (USAN) <US>
E D00603 Timolol maleate (JP18/USP) <JP/US>
E D08525 Sotalol (INN)
E D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
E D00432 Nadolol (JP18/USP/INN) <JP/US>
E D08106 Labetalol (INN)
E D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
E D00255 Carvedilol (JP18/USP/INN) <JP/US>
E D03415 Carvedilol phosphate (USAN) <US>
E D02359 Ritodrine (USAN/INN)
E D01263 Ritodrine hydrochloride (JP18/USP) <JP>
E D04157 Fenoterol (USAN/INN)
E D01428 Fenoterol hydrobromide (JAN) <JP>
E D08300 Orciprenaline (INN)
E D00685 Metaproterenol sulfate (USP)
E D04954 Metaproterenol polistirex (USAN)
E D02147 Albuterol (USP)
E D00683 Albuterol sulfate (USP) <JP/US>
E D08570 Terbutaline (INN)
E D00688 Terbutaline sulfate (JP18/USP) <JP/US>
E D05730 Rimiterol hydrobromide (USAN)
E D08039 Hexoprenaline (INN)
E D02396 Hexoprenaline sulfate (USAN)
E D04625 Isoetharine (USP)
E D02093 Isoetharine hydrochloride (USP)
E D04626 Isoetharine mesylate (USP)
E D08387 Pirbuterol (INN)
E D00686 Pirbuterol acetate (USAN)
E D01349 Pirbuterol hydrochloride (JAN/USAN)
E D08629 Tretoquinol (INN)
E D01978 Trimetoquinol hydrochloride
E D05037 Trimetoquinol hydrochloride hydrate (JP18) <JP>
E D03402 Carbuterol hydrochloride (USAN)
E D02151 Tulobuterol (JP18/INN) <JP>
E D01362 Tulobuterol hydrochloride (JP18) <JP>
E D05792 Salmeterol (USAN/INN)
E D00687 Salmeterol xinafoate (JAN/USP) <JP/US>
E D07990 Formoterol (INN)
E D01373 Formoterol fumarate (USP) <US>
E D05277 Formoterol fumarate hydrate (JP18) <JP/US>
E D07713 Clenbuterol (INN)
E D01360 Clenbuterol hydrochloride (JAN/USP) <JP>
E D08474 Reproterol (INN)
E D05718 Reproterol hydrochloride (USAN)
E D08424 Procaterol (INN)
E D02404 Procaterol hydrochloride (USAN)
E D05366 Procaterol hydrochloride hydrate (JP18) <JP>
E D07534 Bitolterol (INN)
E D00684 Bitolterol mesylate (USAN)
E D09318 Indacaterol (USAN/INN)
E D09319 Indacaterol maleate (JAN/USAN) <JP>
E D11009 Indacaterol acetate (JAN)
E D10145 Olodaterol (USAN/INN)
E D10020 Olodaterol hydrochloride (JAN/USAN) <US>
E D01635 Methoxyphenamine hydrochloride (JAN)
E D07377 Bambuterol (INN)
E D07489 Bambuterol hydrochloride
E D01469 Amosulalol hydrochloride (JP18) <JP>
E D01492 Bucumolol hydrochloride (JP18)
E D01589 Mabuterol hydrochloride (JAN)
E D01830 Arotinolol hydrochloride (JP18) <JP>
E D01835 Clorprenaline hydrochloride (JAN/USAN)
E D01958 Indenolol hydrochloride (JP18)
E D02281 Levalbuterol hydrochloride (USP) <US>
E D02981 Arformoterol tartrate (USAN) <US>
E D03170 Bucindolol hydrochloride (USAN)
E D03177 Bunolol hydrochloride (USAN)
E D03198 Butoxamine hydrochloride (USAN)
E D03587 Colterol mesylate (USAN)
E D04072 Etafedrine hydrochloride (USAN)
E D04701 Levalbuterol sulfate (USAN)
E D04703 Levalbuterol tartrate (USAN) <US>
E D04953 Metalol hydrochloride (USAN)
E D05476 Picumeterol fumarate (USAN)
E D05691 Ractopamine hydrochloride (USP)
E D05832 Sibenadet hydrochloride (USAN)
E D05902 Soterenol hydrochloride (USAN)
E D06374 Zinterol hydrochloride (USAN)
E D06562 Bedoradrine sulfate (USAN)
E D07451 Amosulalol (INN)
E D07463 Arformoterol (INN)
E D07465 Arotinolol (INN)
E D07608 Carazolol (INN)
E D08078 Indenolol (INN)
E D08124 Levosalbutamol (INN)
E D08945 Milveterol hydrochloride (USAN)
E D09696 Vilanterol (USAN)
E D09697 Vilanterol trifenatate (JAN/USAN)
E D10219 Abediterol (USAN/INN)
E D10220 Abediterol napadisylate (USAN)
E D10545 Batefenterol (USAN)
E D10546 Batefenterol succinate (USAN)
E D11900 Navafenterol (USAN)
E D11901 Navafenterol saccharinate (USAN)
D ADRB3 [HSA:155] [KO:K04143]
E D09535 Mirabegron (USAN/JAN) <JP/US>
E D02702 Talibegron hydrochloride (USAN)
E D05879 Solabegron hydrochloride (USAN)
E D08850 Amibegron (USAN/INN)
E D08851 Amibegron hydrochloride (USAN)
E D09344 Fasobegron (INN)
E D09732 Ritobegron ethyl hydrochloride (JAN)
E D10433 Vibegron (JAN/USAN) <JP/US>
C Dopamine
D DRD [HSA:1812 1813 1814 1815 1816] [KO:K04144 K04145 K04146 K04147 K05840]
E D07870 Dopamine (INN)
E D00633 Dopamine hydrochloride (JP18/USP) <JP/US>
E D03891 Dopexamine (USAN/INN)
E D03892 Dopexamine hydrochloride (USAN)
E D00059 Levodopa (JP18/USP/INN) <JP/US>
E D02676 Oxiperomide (USAN/INN)
E D04097 Etilevodopa (USAN/INN)
E D09886 Dexpramipexole (USAN/INN)
E D09887 Dexpramipexole dihydrochloride (USAN)
E D11839 Foslevodopa (JAN/USAN/INN)
D DRD1 [HSA:1812] [KO:K04144]
E D04488 Ibopamine (USAN/INN)
E D08057 Ibopamine hydrochloride
E D07946 Fenoldopam (INN)
E D00613 Fenoldopam mesylate (USP) <US>
E D07460 Apomorphine (BAN)
E D02004 Apomorphine hydrochloride (USP) <JP/US>
E D08339 Pergolide (INN)
E D00502 Pergolide mesylate (USP) <JP>
E D07065 Acepromazine (INN)
E D02604 Acepromazine maleate (USP)
E D00788 Acetophenazine maleate (USAN)
E D08385 Pipotiazine (INN)
E D02680 Pipotiazine palmitate (USAN)
E D01044 Flupentixol (INN)
E D02236 Flupentixol dihydrochloride (JAN)
E D07976 Flupentixol decanoate
E D02613 Clopenthixol (USAN)
E D00790 Chlorprothixene (JAN/USAN/INN)
E D02162 Chlorprothixene hydrochloride (JAN)
E D07686 Chlorprothixene acetate
E D07687 Chlorprothixene citrate
E D03556 Zuclopenthixol (INN)
E D08691 Zuclopenthixol acetate
E D08692 Zuclopenthixol decanoate
E D08693 Zuclopenthixol dihydrochloride
E D01903 Docarpamine (JAN/INN) <JP>
E D02641 Butaclamol hydrochloride (USAN)
E D02644 Carphenazine maleate (USAN)
E D02775 Adrogolide hydrochloride (USAN)
E D03494 Ciladopa hydrochloride (USAN)
E D03937 Ecopipam hydrochloride (USAN)
E D10329 Zicronapine (USAN/INN)
E D10495 Zicronapine succinate (USAN)
E D11431 Tavapadon (USAN)
E D11822 Mevidalen hydroxybenzoate (USAN)
E D11826 Mevidalen (USAN)
D DRD2 [HSA:1813] [KO:K04145]
E D00726 Metoclopramide (JP18/INN) <JP>
E D02213 Metoclopramide hydrochloride (JAN) <JP>
E D05008 Metoclopramide hydrochloride (USP) <US>
E D01745 Domperidone (JP18/USAN/INN) <JP>
E D07868 Domperidone maleate
E D07101 Bromopride (INN)
E D07102 Alizapride (INN)
E D07563 Alizapride hydrochloride
E D03534 Clebopride (USAN)
E D01742 Clebopride malate (JP18)
E D08094 Itopride (INN)
E D02729 Itopride hydrochloride (JAN) <JP>
E D05010 Metopimazine (USAN/INN)
E D04488 Ibopamine (USAN/INN)
E D08057 Ibopamine hydrochloride
E D03165 Bromocriptine (USAN/INN)
E D00780 Bromocriptine mesylate (USP) <JP/US>
E D08132 Lisuride (INN)
E D01462 Lisuride maleate (JAN)
E D00987 Cabergoline (JP18/USP/INN) <JP/US>
E D07217 Quinagolide (INN/BAN)
E D08457 Quinagolide hydrochloride (BAN)
E D01348 Terguride (JAN/INN)
E D07460 Apomorphine (BAN)
E D02004 Apomorphine hydrochloride (USP) <JP/US>
E D08339 Pergolide (INN)
E D00502 Pergolide mesylate (USP) <JP>
E D07836 Dihydroergocryptine mesilate
E D08489 Ropinirole (USAN/INN)
E D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
E D05575 Pramipexole (USAN/INN)
E D00559 Pramipexole dihydrochloride (USP) <JP/US>
E D07305 Piribedil (INN)
E D05768 Rotigotine (JAN/USAN/INN) <JP/US>
E D00270 Chlorpromazine (USP/INN)
E D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
E D03274 Chlorpromazine hibenzate (JAN)
E D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
E D09819 Chlorpromazine tannate (JAN)
E D00403 Methotrimeprazine (USP)
E D01520 Levomepromazine hydrochloride (JAN/USAN) <JP>
E D02248 Levomepromazine maleate (JP18/USAN) <JP>
E D08430 Promazine (INN)
E D00797 Promazine hydrochloride (USP)
E D07065 Acepromazine (INN)
E D02604 Acepromazine maleate (USP)
E D00390 Triflupromazine (USP/INN)
E D00800 Triflupromazine hydrochloride (JAN/USP)
E D07977 Fluphenazine (INN)
E D00791 Fluphenazine hydrochloride (JAN/USP) <US>
E D00792 Fluphenazine enanthate (JP18/USP)
E D00793 Fluphenazine decanoate (JAN/USP) <JP/US>
E D02163 Fluphenazine maleate (JAN) <JP>
E D00503 Perphenazine (JP18/USP/INN) <JP/US>
E D02037 Perphenazine maleate (JP18) <JP>
E D04038 Perphenazine fendizoate (JAN) <JP>
E D04965 Perphenazine hydrochloride <JP>
E D08341 Perphenazine decanoate
E D08342 Perphenazine enantate
E D00493 Prochlorperazine (JAN/USP/INN) <US>
E D00479 Prochlorperazine maleate (JP18/USP) <JP/US>
E D02022 Prochlorperazine mesilate (JAN) <JP>
E D02609 Prochlorperazine edisylate (USP) <US>
E D08636 Trifluoperazine (INN)
E D00799 Trifluoperazine hydrochloride (JAN/USP) <US>
E D01448 Trifluoperazine maleate (JAN)
E D00788 Acetophenazine maleate (USAN)
E D08585 Thioproperazine (INN)
E D01447 Thioproperazine mesilate (JAN)
E D01412 Perazine maleate (JAN)
E D01860 Perazine dimalonate (JAN)
E D02608 Perazine fendizoate (JAN)
E D01485 Propericiazine (JAN) <JP>
E D00373 Thioridazine (USP/INN)
E D00798 Thioridazine hydrochloride (JP18/USP) <US>
E D02671 Mesoridazine (USAN/INN)
E D00795 Mesoridazine besylate (USP)
E D08385 Pipotiazine (INN)
E D02680 Pipotiazine palmitate (USAN)
E D00136 Haloperidol (JP18/USP/INN) <JP/US>
E D01898 Haloperidol decanoate (JAN/USP) <JP/US>
E D08035 Haloperidol lactate <US>
E D02625 Trifluperidol (USAN/INN)
E D08637 Trifluperidol hydrochloride
E D07309 Melperone (INN)
E D08172 Melperone hydrochloride
E D02623 Moperone (INN)
E D01105 Moperone hydrochloride (JAN)
E D02622 Pipamperone (USAN/INN)
E D01482 Pipamperone hydrochloride (JAN) <JP>
E D01101 Bromperidol (JAN/USAN/INN) <JP>
E D02626 Bromperidol decanoate (USAN)
E D02627 Benperidol (USAN/INN)
E D00308 Droperidol (JP18/USP/INN) <JP/US>
E D11169 Lumateperone (USAN/INN)
E D11170 Lumateperone tosylate (USAN) <US>
E D08226 Molindone (INN)
E D00796 Molindone hydrochloride (USP) <US>
E D00561 Sertindole (USAN/INN)
E D08687 Ziprasidone (INN)
E D01939 Ziprasidone hydrochloride (USP) <US>
E D02100 Ziprasidone mesylate (USAN) <US>
E D04820 Lurasidone hydrochloride (JAN/USAN) <JP/US>
E D01044 Flupentixol (INN)
E D02236 Flupentixol dihydrochloride (JAN)
E D07976 Flupentixol decanoate
E D02613 Clopenthixol (USAN)
E D00790 Chlorprothixene (JAN/USAN/INN)
E D02162 Chlorprothixene hydrochloride (JAN)
E D07686 Chlorprothixene acetate
E D07687 Chlorprothixene citrate
E D00374 Thiothixene (USP) <US>
E D02612 Thiothixene hydrochloride (USP)
E D03556 Zuclopenthixol (INN)
E D08691 Zuclopenthixol acetate
E D08692 Zuclopenthixol decanoate
E D08693 Zuclopenthixol dihydrochloride
E D00560 Pimozide (JP18/USP/INN) <US>
E D02340 Loxapine (USAN/INN) <US>
E D00794 Loxapine succinate (USP) <US>
E D08148 Loxapine hydrochloride
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D08456 Quetiapine (INN)
E D00458 Quetiapine fumarate (JP18/USP) <JP/US>
E D11769 Asenapine (INN) <US>
E D02995 Asenapine maleate (JAN/USAN) <JP/US>
E D01226 Sulpiride (JP18/USAN/INN) <JP>
E D08549 Sultopride (INN)
E D02208 Sultopride hydrochloride (JAN) <JP>
E D08590 Tiapride (INN)
E D01522 Tiapride hydrochloride (JP18) <JP>
E D02682 Remoxipride (USAN)
E D02683 Remoxipride hydrochloride (USAN)
E D07310 Amisulpride (INN) <US>
E D07312 Levosulpiride (INN)
E D00426 Risperidone (JP18/USP/INN) <JP/US>
E D08235 Mosapramine (INN)
E D01548 Mosapramine hydrochloride (JAN) <JP>
E D01321 Zotepine (JAN/INN) <JP>
E D01164 Aripiprazole (JAN/USP/INN) <JP/US>
E D10355 Aripiprazole cavoxil (USAN)
E D10364 Aripiprazole lauroxil (USAN) <US>
E D10516 Aripiprazole hydrate (JAN) <JP/US>
E D05339 Paliperidone (JAN/USP/INN) <JP/US>
E D05340 Paliperidone palmitate (JAN/USAN) <JP/US>
E D02666 Iloperidone (USAN/INN) <US>
E D09997 Cariprazine (USAN/INN)
E D09876 Cariprazine hydrochloride (JAN/USAN) <US>
E D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
E D07593 Buspirone (INN)
E D00702 Buspirone hydrochloride (USP) <US>
E D08297 Opipramol (INN)
E D01477 Opipramol hydrochloride (JAN/USAN)
E D02354 Thiethylperazine (USAN/INN)
E D01130 Thiethylperazine maleate (JAN/USP)
E D02610 Thiethylperazine malate (JAN)
E D01051 Spiperone (JAN/USAN) <JP>
E D01176 Blonanserin (JAN/INN) <JP>
E D01468 Nemonapride (JAN/INN) <JP>
E D01505 Talipexole hydrochloride (JAN)
E D02035 Timiperone (JAN) <JP>
E D02371 Clocapramine hydrochloride hydrate (JP18) <JP>
E D02372 Perospirone hydrochloride hydrate (JAN) <JP>
E D02605 Methoxypromazine maleate
E D02634 Alentemol hydrobromide (USAN)
E D02641 Butaclamol hydrochloride (USAN)
E D02644 Carphenazine maleate (USAN)
E D02645 Carvotroline hydrochloride (USAN)
E D02670 Mazapertine succinate (USAN)
E D02675 Ocaperidone (USAN)
E D02681 Piquindone hydrochloride (USAN)
E D02688 Tiospirone hydrochloride (USAN)
E D03214 Aplindore fumarate (USAN)
E D03494 Ciladopa hydrochloride (USAN)
E D04693 Lergotrile (USAN/INN)
E D04694 Lergotrile mesylate (USAN)
E D05124 Naxagolide hydrochloride (USAN)
E D05677 Quinelorane hydrochloride (USAN)
E D05682 Quinpirole hydrochloride (USAN)
E D05690 Raclopride C11 (USAN)
E D05804 Sarizotan hydrochloride (USAN)
E D05832 Sibenadet hydrochloride (USAN)
E D06566 Bifeprunox (USAN/INN)
E D06567 Bifeprunox mesylate (USAN)
E D07718 Clocapramine (INN)
E D07835 Dihydroergocryptine
E D08558 Talipexole (INN)
E D09366 Pardoprunox hydrochloride (USAN)
E D09397 Pardoprunox (USAN/INN)
E D09953 Pridopidine (USAN/INN)
E D09954 Pridopidine hydrochloride (USAN)
E D10329 Zicronapine (USAN/INN)
E D10495 Zicronapine succinate (USAN)
E D11982 Trazpiroben (USAN/INN)
D DRD3 [HSA:1814] [KO:K04146]
E D08132 Lisuride (INN)
E D01462 Lisuride maleate (JAN)
E D08489 Ropinirole (USAN/INN)
E D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
E D05575 Pramipexole (USAN/INN)
E D00559 Pramipexole dihydrochloride (USP) <JP/US>
E D07305 Piribedil (INN)
E D00374 Thiothixene (USP) <US>
E D02612 Thiothixene hydrochloride (USP)
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D07310 Amisulpride (INN) <US>
E D01164 Aripiprazole (JAN/USP/INN) <JP/US>
E D10355 Aripiprazole cavoxil (USAN)
E D10364 Aripiprazole lauroxil (USAN) <US>
E D10516 Aripiprazole hydrate (JAN) <JP/US>
E D07316 Captodiame (BAN)
E D01176 Blonanserin (JAN/INN) <JP>
E D03214 Aplindore fumarate (USAN)
E D05682 Quinpirole hydrochloride (USAN)
E D09366 Pardoprunox hydrochloride (USAN)
E D09397 Pardoprunox (USAN/INN)
E D11982 Trazpiroben (USAN/INN)
D DRD4 [HSA:1815] [KO:K04147]
E D08132 Lisuride (INN)
E D01462 Lisuride maleate (JAN)
E D08489 Ropinirole (USAN/INN)
E D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
E D05575 Pramipexole (USAN/INN)
E D00559 Pramipexole dihydrochloride (USP) <JP/US>
E D00283 Clozapine (JAN/USP/INN) <JP/US>
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D02656 Fananserin (USAN/INN)
E D05891 Sonepiprazole mesylate (USAN)
D DRD5 [HSA:1816] [KO:K05840]
E D03937 Ecopipam hydrochloride (USAN)
E D11431 Tavapadon (USAN)
C Histamine
D HRH1 [HSA:3269] [KO:K04149]
E D08587 Thonzylamine (INN)
E D01801 Thonzylamine hydrochloride (JAN/USAN)
E D08183 Mepyramine (INN)
E D05660 Pyrilamine maleate (USP)
E D07194 Thenalidine (INN)
E D08645 Tripelennamine (INN)
E D02091 Tripelennamine hydrochloride (USP)
E D06246 Tripelennamine citrate
E D07195 Chloropyramine (INN)
E D07679 Chloropyramine hydrochloride
E D00494 Promethazine (JAN/INN)
E D00480 Promethazine hydrochloride (JP18/USP) <JP/US>
E D01242 Promethazine teoclate (JAN/INN)
E D03290 Promethazine methylenedisalicylate (JAN) <JP>
E D08432 Promethazine maleate
E D08768 Promethazine hibenzate <JP>
E D07196 Tolpropamine (INN)
E D07853 Dimetindene (INN)
E D01343 Dimethindene maleate (USAN)
E D03535 Clemastine (USAN)
E D00666 Clemastine fumarate (JP18/USP) <JP/US>
E D07197 Bamipine (INN)
E D07492 Bamipine dihydrochloride
E D07493 Bamipine lactate
E D08355 Pheniramine (INN)
E D01174 Pheniramine maleate (JAN/USP)
E D08091 Isothipendyl (INN)
E D01143 Isothipendyl hydrochloride (JAN)
E D00300 Diphenhydramine (JP18/INN) <JP>
E D00669 Diphenhydramine hydrochloride (JP18/USP) <JP/US>
E D02419 Diphenhydramine salicylate (JAN)
E D03285 Diphenhydramine tannate (JP18)
E D03360 Diphenhydramine laurylsulfate (JAN) <JP>
E D03854 Diphenhydramine citrate (USP)
E D07198 Chlorphenoxamine (INN)
E D07684 Chlorphenoxamine hydrochloride
E D07875 Doxepin (INN)
E D00814 Doxepin hydrochloride (USP) <US>
E D00774 Orphenadrine citrate (USP) <US>
E D07854 Dimetotiazine (INN)
E D01902 Fonazine mesylate (USAN) <JP>
E D02599 Orphenadrine hydrochloride
E D00270 Chlorpromazine (USP/INN)
E D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
E D03274 Chlorpromazine hibenzate (JAN)
E D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
E D09819 Chlorpromazine tannate (JAN)
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D08054 Hydroxyzine (INN)
E D00672 Hydroxyzine hydrochloride (JP18/USP) <JP/US>
E D01096 Hydroxyzine pamoate (JP18/USP) <JP/US>
E D08297 Opipramol (INN)
E D01477 Opipramol hydrochloride (JAN/USAN)
E D08216 Mianserin (INN)
E D01358 Mianserin hydrochloride (JAN/USAN) <JP>
E D07522 Betahistine (INN)
E D01592 Betahistine mesilate (JP18) <JP>
E D03102 Betahistine hydrochloride (USP)
E D01295 Cinnarizine (JAN/USAN/INN)
E D07734 Cinnarizine dihydrochloride
E D08117 Levocabastine (INN)
E D01717 Levocabastine hydrochloride (JAN/USP) <JP>
E D07483 Azelastine (INN)
E D00659 Azelastine hydrochloride (JP18/USP) <JP/US>
E D07458 Antazoline (INN)
E D02950 Antazoline phosphate (USP)
E D07459 Antazoline hydrochloride
E D08293 Olopatadine (INN)
E D01192 Olopatadine hydrochloride (JP18/USP) <JP/US>
E D03166 Bromodiphenhydramine hydrochloride (USP)
E D07862 Diphenylpyraline (INN)
E D01172 Diphenylpyraline hydrochloride (JAN)
E D01627 Diphenylpyraline teoclate (JAN)
E D07617 Carbinoxamine (INN)
E D01336 Carbinoxamine maleate (JAN/USP) <US>
E D09808 Carbinoxamine diphenyldisulfonate (JAN)
E D07878 Doxylamine (INN)
E D02327 Doxylamine succinate (USP)
E D00520 Dimenhydrinate (JP18/USP/INN) <JP/US>
E D07543 Brompheniramine (INN)
E D00663 Brompheniramine maleate (USP)
E D07803 Dexchlorpheniramine (INN)
E D00668 Dexchlorpheniramine maleate (USP) <JP/US>
E D07398 Chlorphenamine (INN)
E D00665 Chlorpheniramine maleate (JP18/USP) <JP>
E D03475 Chlorpheniramine polistirex (USAN)
E D03704 Dexbrompheniramine maleate (USP)
E D07400 Histapyrrodine (INN)
E D07125 Alimemazine (INN)
E D02245 Trimeprazine tartrate (USP) <JP>
E D04979 Methdilazine (INN)
E D04980 Methdilazine hydrochloride (USP)
E D01324 Mequitazine (JP18/INN) <JP>
E D07401 Oxomemazine (INN)
E D07547 Buclizine (INN)
E D02089 Buclizine hydrochloride (USAN)
E D03621 Cyclizine (INN)
E D02090 Cyclizine lactate (BAN)
E D03622 Cyclizine hydrochloride (USP)
E D08163 Meclozine (BAN)
E D01317 Meclizine hydrochloride (JAN/USP) <US>
E D07662 Cetirizine (INN)
E D00664 Cetirizine hydrochloride (JP18/USP) <JP/US>
E D07402 Levocetirizine (USAN/INN)
E D08118 Levocetirizine dihydrochloride (USP) <JP/US>
E D07765 Cyproheptadine (INN)
E D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
E D08353 Phenindamine (INN)
E D02148 Phenindamine tartrate (USAN)
E D08648 Triprolidine (INN)
E D01782 Triprolidine hydrochloride (USP)
E D07403 Pyrrobutamine (BAN)
E D07482 Azatadine (INN)
E D00662 Azatadine maleate (USP)
E D00234 Astemizole (JAN/USP/INN)
E D00521 Terfenadine (JAN/USAN/INN)
E D00364 Loratadine (JAN/USP/INN) <JP/US>
E D08161 Mebhydrolin (INN)
E D01786 Mebhydrolin napadisilate (JAN)
E D07404 Deptropine (INN)
E D07790 Deptropine citrate
E D08105 Ketotifen (INN)
E D01332 Ketotifen fumarate (JP18/USAN) <JP/US>
E D02760 Acrivastine (USAN/INN)
E D01478 Ebastine (JP18/USAN/INN) <JP>
E D07406 Pimethixene (INN)
E D07900 Epinastine (INN)
E D01713 Epinastine hydrochloride (JAN) <JP/US>
E D01117 Mizolastine (JAN/INN)
E D07958 Fexofenadine (INN)
E D00671 Fexofenadine hydrochloride (JP18/USP) <JP/US>
E D03693 Desloratadine (JAN/USP/INN) <JP/US>
E D07407 Rupatadine (INN)
E D08497 Rupatadine fumarate (JAN) <JP>
E D09570 Bilastine (JAN/INN) <JP>
E D10230 Quifenadine (INN)
E D10510 Sequifenadine
E D07890 Emedastine (INN)
E D02249 Emedastine difumarate (JP18/USP) <JP>
E D06552 Alcaftadine (JAN/USAN/INN) <US>
E D04445 Histamine phosphate (USP) <US>
E D01460 Homochlorcyclizine hydrochloride (JP18) <JP>
E D01654 Bepotastine besylate (USAN) <JP/US>
E D01701 Difeterol hydrochloride (JAN)
E D02067 Diphenylimidazole (JAN)
E D03056 Barmastine (USAN/INN)
E D03491 Cidoxepin hydrochloride (USAN)
E D03568 Closiramine aceturate (USAN)
E D03620 Cycliramine maleate (USAN)
E D03893 Dorastine hydrochloride (USAN)
E D03963 Efletirizine dihydrochloride (USAN)
E D04055 Esmirtazapine maleate (USAN)
E D04494 Icotidine (USAN)
E D05196 Noberastine (USAN/INN)
E D05664 Pyroxamine maleate (USAN)
E D05742 Rocastine hydrochloride (USAN)
E D05769 Rotoxamine (USAN/INN)
E D06012 Tazifylline hydrochloride (USAN)
E D06021 Tecastemizole (USAN/INN)
E D06063 Temelastine (USAN/INN)
E D06084 Tesmilifene hydrochloride (USAN)
E D06376 Zolamine hydrochloride (USAN)
E D07532 Bisulepin
E D07533 Bisulepin hydrochloride
E D07860 Dioxopromethazine hydrochloride
E D07889 Embramine (INN)
E D08040 Histamine (DCF) <US>
E D08041 Homochlorcyclizine (INN)
E D08305 Orphenadrine (INN)
E D08967 Phenyltoloxamine citrate (USP)
E D09705 Bepotastine (USAN/INN)
E D09747 Difeterol phosphate (JAN)
E D09748 Difeterol (JAN/INN)
E D09838 Broizine (JAN)
D HRH2 [HSA:3274] [KO:K04150]
E D00295 Cimetidine (JP18/USP/INN) <JP/US>
E D03503 Cimetidine hydrochloride (USP) <US>
E D00422 Ranitidine (USAN/INN)
E D00673 Ranitidine hydrochloride (JP18/USP) <JP/US>
E D00318 Famotidine (JP18/USP/INN) <JP/US>
E D00440 Nizatidine (JP18/USP/INN) <JP/US>
E D07072 Niperotidine (INN)
E D08494 Roxatidine (INN)
E D01467 Roxatidine acetate hydrochloride (JP18/USAN) <JP>
E D08495 Roxatidine acetate (BAN)
E D05699 Ranitidine bismuth citrate (USAN)
E D01131 Lafutidine (JP18/INN) <JP>
E D00721 Methanthelinium bromide (INN)
E D01187 Betazole hydrochloride (JAN)
E D04445 Histamine phosphate (USP) <US>
E D01193 Osutidine (JAN/INN)
E D01698 Dalcotidine (JAN/INN)
E D01861 Pibutidine hydrochloride (JAN)
E D03889 Donetidine (USAN)
E D04098 Etintidine hydrochloride (USAN)
E D04494 Icotidine (USAN)
E D04517 Impromidine hydrochloride (USAN)
E D04680 Lavoltidine succinate (USAN)
E D04794 Lupitidine hydrochloride (USAN)
E D05004 Metiamide (USAN/INN)
E D05306 Oxmetidine hydrochloride (USAN)
E D05307 Oxmetidine mesylate (USAN)
E D05939 Sufotidine (USAN/INN)
E D06157 Tiotidine (USAN/INN)
E D06355 Zaltidine hydrochloride (USAN)
E D08040 Histamine (DCF) <US>
D HRH3 [HSA:11255] [KO:K04151]
E D07522 Betahistine (INN)
E D01592 Betahistine mesilate (JP18) <JP>
E D03102 Betahistine hydrochloride (USP)
E D10749 Pitolisant (USAN/INN)
E D11490 Pitolisant hydrochloride (USAN) <US>
E D04445 Histamine phosphate (USP) <US>
E D03518 Cipralisant maleate (USAN)
E D08040 Histamine (DCF) <US>
E D09870 Bavisant (USAN/INN)
E D09871 Bavisant dihydrochloride (USAN)
E D10128 Irdabisant (USAN)
E D10129 Irdabisant hydrochloride (USAN)
D HRH4 [HSA:59340] [KO:K04152]
E D08040 Histamine (DCF) <US>
E D10735 Toreforant (USAN/INN)
E D10736 Toreforant tartrate (USAN)
E D11819 Adriforant (USAN/INN)
C Serotonin
D HTR1 [HSA:3350 3351 3352 3354 3355] [KO:K04153]
E D07700 Cinitapride (INN)
E D07701 Cinitapride tartrate
E D05523 Pizotyline (USAN)
E D08397 Pizotifen malate
E D01321 Zotepine (JAN/INN) <JP>
E D07765 Cyproheptadine (INN)
E D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
E D04533 Indorenate hydrochloride (USAN)
D HTR1A [HSA:3350] [KO:K04153]
E D07906 Ergotamine (INN)
E D02577 Flibanserin (USAN/INN) <US>
E D00679 Ergotamine tartrate (JP18/USP) <US>
E D02357 Methysergide (USAN/INN)
E D00681 Methysergide maleate (USP)
E D08385 Pipotiazine (INN)
E D02680 Pipotiazine palmitate (USAN)
E D02995 Asenapine maleate (JAN/USAN) <JP/US>
E D01164 Aripiprazole (JAN/USP/INN) <JP/US>
E D10355 Aripiprazole cavoxil (USAN)
E D10364 Aripiprazole lauroxil (USAN) <US>
E D10516 Aripiprazole hydrate (JAN) <JP/US>
E D09997 Cariprazine (USAN/INN)
E D09876 Cariprazine hydrochloride (JAN/USAN) <US>
E D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
E D07593 Buspirone (INN)
E D00702 Buspirone hydrochloride (USP) <US>
E D04314 Gepirone hydrochloride (USAN)
E D09698 Vilazodone (USAN/INN)
E D09699 Vilazodone hydrochloride (USAN) <US>
E D10184 Vortioxetine (USAN)
E D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
E D12544 Vortioxetine hemihydrobromide (USAN)
E D06327 Xaliproden (USAN)
E D01537 Xaliproden hydrochloride (JAN)
E D01992 Tandospirone citrate (JAN/USAN) <JP>
E D02568 Flesinoxan (INN)
E D02569 Sunepitron hydrochloride (USAN)
E D02576 Eptapirone (INN)
E D02688 Tiospirone hydrochloride (USAN)
E D02767 Adatanserin hydrochloride (USAN)
E D03121 Binospirone mesylate (USAN)
E D04611 Ipsapirone hydrochloride (USAN)
E D04683 Lecozotan hydrochloride (USAN)
E D05804 Sarizotan hydrochloride (USAN)
E D06354 Zalospirone hydrochloride (USAN)
E D06566 Bifeprunox (USAN/INN)
E D06567 Bifeprunox mesylate (USAN)
E D08561 Tandospirone (INN)
E D09358 Naluzotan (USAN/INN)
E D09359 Naluzotan hydrochloride (USAN)
E D09366 Pardoprunox hydrochloride (USAN)
E D09397 Pardoprunox (USAN/INN)
E D12474 Ulotaront (USAN/INN)
E D12475 Ulotaront hydrochloride (USAN)
D HTR1B [HSA:3351] [KO:K04153]
E D07906 Ergotamine (INN)
E D07837 Dihydroergotamine (INN)
E D02211 Dihydroergotamine mesylate (USP) <US>
E D07838 Dihydroergotamine tartrate
E D00679 Ergotamine tartrate (JP18/USP) <US>
E D00451 Sumatriptan (JAN/USP/INN) <JP/US>
E D00676 Sumatriptan succinate (JAN/USP) <JP/US>
E D08255 Naratriptan (INN)
E D00674 Naratriptan hydrochloride (JAN/USP) <JP/US>
E D00415 Zolmitriptan (JAN/USP/INN) <JP/US>
E D08485 Rizatriptan (INN)
E D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
E D05740 Rizatriptan sulfate (USAN)
E D02824 Almotriptan (USAN)
E D02825 Almotriptan malate (USP) <US>
E D07887 Eletriptan (INN)
E D01973 Eletriptan hydrobromide (JAN/USAN) <JP/US>
E D11617 Eletriptan hydrobromide monohydrate <US>
E D07997 Frovatriptan (INN)
E D04264 Frovatriptan succinate (USAN) <US>
E D02826 Alniditan dihydrochloride (USAN)
E D03014 Avitriptan fumarate (USAN)
E D03982 Elzasonan citrate (USAN)
E D03983 Elzasonan hydrochloride (USAN)
D HTR1D [HSA:3352] [KO:K04153]
E D07945 Fenfluramine (INN)
E D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
E D07906 Ergotamine (INN)
E D07837 Dihydroergotamine (INN)
E D02211 Dihydroergotamine mesylate (USP) <US>
E D07838 Dihydroergotamine tartrate
E D00679 Ergotamine tartrate (JP18/USP) <US>
E D00451 Sumatriptan (JAN/USP/INN) <JP/US>
E D00676 Sumatriptan succinate (JAN/USP) <JP/US>
E D08255 Naratriptan (INN)
E D00674 Naratriptan hydrochloride (JAN/USP) <JP/US>
E D00415 Zolmitriptan (JAN/USP/INN) <JP/US>
E D08485 Rizatriptan (INN)
E D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
E D05740 Rizatriptan sulfate (USAN)
E D02824 Almotriptan (USAN)
E D02825 Almotriptan malate (USP) <US>
E D07887 Eletriptan (INN)
E D01973 Eletriptan hydrobromide (JAN/USAN) <JP/US>
E D11617 Eletriptan hydrobromide monohydrate <US>
E D07997 Frovatriptan (INN)
E D04264 Frovatriptan succinate (USAN) <US>
E D02826 Alniditan dihydrochloride (USAN)
E D03014 Avitriptan fumarate (USAN)
E D03982 Elzasonan citrate (USAN)
E D03983 Elzasonan hydrochloride (USAN)
D HTR1F [HSA:3355] [KO:K04153]
E D10338 Lasmiditan (USAN/INN)
E D10424 Lasmiditan succinate (JAN/USAN) <JP/US>
D HTR2 [HSA:3356 3357 3358] [KO:K04157]
E D07700 Cinitapride (INN)
E D07701 Cinitapride tartrate
E D02577 Flibanserin (USAN/INN) <US>
E D02357 Methysergide (USAN/INN)
E D00681 Methysergide maleate (USP)
E D05523 Pizotyline (USAN)
E D08397 Pizotifen malate
E D07854 Dimetotiazine (INN)
E D01902 Fonazine mesylate (USAN) <JP>
E D00270 Chlorpromazine (USP/INN)
E D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
E D03274 Chlorpromazine hibenzate (JAN)
E D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
E D09819 Chlorpromazine tannate (JAN)
E D01485 Propericiazine (JAN) <JP>
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D02666 Iloperidone (USAN/INN) <US>
E D08297 Opipramol (INN)
E D01477 Opipramol hydrochloride (JAN/USAN)
E D08626 Trazodone (INN)
E D00820 Trazodone hydrochloride (JAN/USP) <JP/US>
E D00563 Mirtazapine (JAN/USP/INN) <JP/US>
E D11056 Mirtazapine hydrate (JAN)
E D07765 Cyproheptadine (INN)
E D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
E D02675 Ocaperidone (USAN)
E D02686 Setoperone (USAN/INN)
E D02688 Tiospirone hydrochloride (USAN)
E D02767 Adatanserin hydrochloride (USAN)
E D04320 Glemanserin (USAN/INN)
E D05015 Metrenperone (USAN/INN)
E D05395 Pelanserin hydrochloride (USAN)
E D05829 Sergolexole maleate (USAN)
E D06253 Tropanserin hydrochloride (USAN)
E D06343 Xylamidine tosylate (USAN)
D HTR2A [HSA:3356] [KO:K04157]
E D00274 Cisapride (USP/INN)
E D02092 Cisapride (JAN)
E D07945 Fenfluramine (INN)
E D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
E D02363 Ketanserin (USAN/INN)
E D08099 Ketanserin tartrate
E D08244 Naftidrofuryl (INN)
E D05107 Nafronyl oxalate (USAN)
E D07307 Cyamemazine (INN)
E D07756 Cyamemazine tartrate
E D02671 Mesoridazine (USAN/INN)
E D00795 Mesoridazine besylate (USP)
E D08385 Pipotiazine (INN)
E D02680 Pipotiazine palmitate (USAN)
E D11169 Lumateperone (USAN/INN)
E D11170 Lumateperone tosylate (USAN) <US>
E D00561 Sertindole (USAN/INN)
E D08687 Ziprasidone (INN)
E D01939 Ziprasidone hydrochloride (USP) <US>
E D02100 Ziprasidone mesylate (USAN) <US>
E D04820 Lurasidone hydrochloride (JAN/USAN) <JP/US>
E D02340 Loxapine (USAN/INN) <US>
E D00794 Loxapine succinate (USP) <US>
E D08148 Loxapine hydrochloride
E D00283 Clozapine (JAN/USP/INN) <JP/US>
E D08456 Quetiapine (INN)
E D00458 Quetiapine fumarate (JP18/USP) <JP/US>
E D11769 Asenapine (INN) <US>
E D02995 Asenapine maleate (JAN/USAN) <JP/US>
E D00426 Risperidone (JP18/USP/INN) <JP/US>
E D08235 Mosapramine (INN)
E D01548 Mosapramine hydrochloride (JAN) <JP>
E D01164 Aripiprazole (JAN/USP/INN) <JP/US>
E D10355 Aripiprazole cavoxil (USAN)
E D10364 Aripiprazole lauroxil (USAN) <US>
E D10516 Aripiprazole hydrate (JAN) <JP/US>
E D05339 Paliperidone (JAN/USP/INN) <JP/US>
E D05340 Paliperidone palmitate (JAN/USAN) <JP/US>
E D09997 Cariprazine (USAN/INN)
E D09876 Cariprazine hydrochloride (JAN/USAN) <US>
E D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
E D08969 Pimavanserin tartrate (USAN) <US>
E D08216 Mianserin (INN)
E D01358 Mianserin hydrochloride (JAN/USAN) <JP>
E D08257 Nefazodone (INN)
E D00819 Nefazodone hydrochloride (USP) <US>
E D01176 Blonanserin (JAN/INN) <JP>
E D01624 Sarpogrelate hydrochloride (JP18) <JP>
E D02372 Perospirone hydrochloride hydrate (JAN) <JP>
E D02656 Fananserin (USAN/INN)
E D02836 Altanserin tartrate (USAN)
E D02893 Amesergide (USAN/INN)
E D03005 Atiprosin maleate (USAN)
E D04055 Esmirtazapine maleate (USAN)
E D04788 Lubazodone hydrochloride (USAN)
E D05738 Ritanserin (USAN/INN)
E D06632 Pruvanserin (USAN/INN)
E D06633 Pruvanserin hydrochloride (USAN)
E D08508 Sarpogrelate (INN)
E D09645 Nelotanserin (USAN/INN)
E D09976 Temanogrel (USAN/INN)
E D09977 Temanogrel hydrochloride (USAN)
E D10006 Eplivanserin (USAN/INN)
E D10329 Zicronapine (USAN/INN)
E D10495 Zicronapine succinate (USAN)
D HTR2C [HSA:3358] [KO:K04157]
E D07945 Fenfluramine (INN)
E D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
E D06613 Lorcaserin hydrochloride (USAN)
E D11566 Lorcaserin hydrochloride hemihydrate
E D07307 Cyamemazine (INN)
E D07756 Cyamemazine tartrate
E D00283 Clozapine (JAN/USP/INN) <JP/US>
E D02995 Asenapine maleate (JAN/USAN) <JP/US>
E D08969 Pimavanserin tartrate (USAN) <US>
E D07316 Captodiame (BAN)
E D08216 Mianserin (INN)
E D01358 Mianserin hydrochloride (JAN/USAN) <JP>
E D08257 Nefazodone (INN)
E D00819 Nefazodone hydrochloride (USP) <US>
E D02578 Agomelatine (INN)
E D02893 Amesergide (USAN/INN)
E D05738 Ritanserin (USAN/INN)
E D06660 Vabicaserin hydrochloride (USAN)
E D10170 Tedatioxetine (USAN)
E D10171 Tedatioxetine hydrobromide (USAN)
E D10710 Idalopirdine (USAN/INN)
D HTR4 [HSA:3360] [KO:K04160]
E D00274 Cisapride (USP/INN)
E D02092 Cisapride (JAN)
E D07700 Cinitapride (INN)
E D07701 Cinitapride tartrate
E D08236 Mosapride (INN)
E D01994 Mosapride citrate hydrate (JP18) <JP>
E D09205 Prucalopride (USAN/INN)
E D10152 Prucalopride succinate (USAN) <US>
E D06056 Tegaserod (USAN/INN)
E D02730 Tegaserod maleate (USAN)
E D01838 Fabesetron hydrochloride (JAN)
E D05471 Piboserod hydrochloride (USAN)
E D05941 Sulamserod hydrochloride (USAN)
E D06396 Renzapride (INN)
E D09693 Velusetrag (USAN/INN)
E D09694 Velusetrag hydrochloride (USAN)
E D09933 Naronapride (USAN/INN)
E D09934 Naronapride dihydrochloride (USAN)
E D11220 Relenopride (USAN/INN)
E D11221 Relenopride hydrochloride (USAN)
E D12157 Felcisetrag (USAN/INN)
D HTR6 [HSA:3362] [KO:K04162]
E D00454 Olanzapine (JAN/USP/INN) <JP/US>
E D06623 Olanzapine pamoate (USAN) <US>
E D02995 Asenapine maleate (JAN/USAN) <JP/US>
E D02688 Tiospirone hydrochloride (USAN)
E D10099 Cerlapirdine (USAN)
E D10100 Cerlapirdine hydrochloride (USAN)
E D10710 Idalopirdine (USAN/INN)
E D10747 Idalopirdine hydrochloride (JAN)
D HTR7 [HSA:3363] [KO:K04163]
E D02357 Methysergide (USAN/INN)
E D00681 Methysergide maleate (USP)
E D02995 Asenapine maleate (JAN/USAN) <JP/US>
C Trace amine
D TAAR [HSA:134864 9287 9038 319100 83551 134860] [KO:K05051]
E D11830 Ralmitaront (USAN/INN)
D TAAR1 [HSA:134864] [KO:K05051]
E D12474 Ulotaront (USAN/INN)
E D12475 Ulotaront hydrochloride (USAN)
C Angiotensin
D AGTR1 [HSA:185] [KO:K04166]
E D02939 Angiotensin amide (USAN)
E D00150 Angiotensin II (INN)
E D02014 Angiotensin II (USAN)
E D11142 Angiotensin II acetate (USAN) <US>
E D08146 Losartan (INN)
E D00357 Losartan potassium (JP18/USP) <JP/US>
E D04040 Eprosartan (USAN/INN)
E D02082 Eprosartan mesylate (USAN)
E D00400 Valsartan (JP18/USP/INN) <JP/US>
E D00523 Irbesartan (JP18/USP/INN) <JP/US>
E D06010 Tasosartan (USAN/INN)
E D00522 Candesartan (USAN/INN)
E D00626 Candesartan cilexetil (JP18/USP) <JP/US>
E D00627 Telmisartan (JP18/USP/INN) <JP/US>
E D01204 Olmesartan medoxomil (JP18/USP) <JP/US>
E D08067 Azilsartan medoxomil (USAN)
E D08865 Azilsartan kamedoxomil (USAN) <US>
E D10556 Fimasartan (INN)
E D01922 Pratosartan (JAN/INN)
E D04126 Saralasin acetate (USAN)
E D04243 Forasartan (USAN/INN)
E D05246 Olmesartan (USAN/INN)
E D05801 Saprisartan potassium (USAN)
E D08864 Azilsartan (JAN/USAN/INN) <JP>
E D11776 Sparsentan (USAN/INN) <US>
D AGTR2 [HSA:186] [KO:K04167]
E D02939 Angiotensin amide (USAN)
E D00150 Angiotensin II (INN)
E D02014 Angiotensin II (USAN)
E D11142 Angiotensin II acetate (USAN) <US>
E D04126 Saralasin acetate (USAN)
C Bradykinin
D BDKRB2 [HSA:624] [KO:K03916]
E D04492 Icatibant acetate (JAN/USAN) <JP/US>
E D03677 Deltibant (USAN/INN)
E D08937 Labradimil (INN/USAN)
C Cholecystokinin
D CCKAR [HSA:886] [KO:K04194]
E D03442 Ceruletide (USAN/INN)
E D03443 Ceruletide diethylamine (USAN)
E D01113 Loxiglumide (JAN/INN)
E D01858 Panazepide (JAN)
E D02693 Devazepide (USAN/INN)
E D02710 Tarazepide (INN)
D CCKBR [HSA:887] [KO:K04195]
E D01818 Proglumide (JP18/USAN/INN)
E D01631 Pentagastrin (JAN/USAN/INN)
E D01858 Panazepide (JAN)
C Endothelin
D EDNR [HSA:1909 1910] [KO:K04197 K04198]
E D07538 Bosentan (INN)
E D01227 Bosentan (USAN) <JP/US>
E D10135 Macitentan (JAN/USAN) <JP/US>
E D11441 Aprocitentan (USAN/INN)
E D11974 Centhaquine (USAN)
E D11975 Centhaquine citrate (USAN)
D EDNRA [HSA:1909] [KO:K04197]
E D07077 Ambrisentan (JAN/INN) <JP/US>
E D07171 Sitaxentan (USAN/INN)
E D08517 Sitaxentan sodium (USAN)
E D03009 Atrasentan hydrochloride (USAN)
E D03953 Edonentan (USAN)
E D04128 Fandosentan potassium (USAN)
E D07682 Clazosentan sodium (JAN) <JP>
E D07741 Zibotentan (JAN/USAN/INN)
E D11664 Clazosentan (USAN/INN)
E D11776 Sparsentan (USAN/INN) <US>
D EDNRB [HSA:1910] [KO:K04198]
E D11964 Sovatelitide (USAN)
C Follicle stimulating hormone
D FSHR [HSA:2492] [KO:K04247]
E D06457 Gonadotropin, chorionic (USP) <JP/US>
E D02692 Menotropins (USAN) <JP>
E D06459 Purified human menopausal gonadotrophin (JAN) <JP>
E D05258 Serum gonadotrophin (JAN)
E D06269 Urofollitropin (USAN/INN)
E D04429 Follitropin alfa (genetical recombination) (JAN) <JP/US>
E D04430 Follitropin beta (genetical recombination) (JAN)
E D08895 Corifollitropin alfa (INN/USAN)
E D06400 Follitropin delta (USAN) <JP/US>
C Ghrelin
D GHSR [HSA:2693] [KO:K04284]
E D10563 Macimorelin (USAN)
E D10562 Macimorelin acetate (USAN) <US>
E D02040 Pralmorelin dihydrochloride (USAN) <JP>
E D03373 Capromorelin tartrate (USAN)
E D05734 Rismorelin porcine (USAN)
E D08856 Anamorelin hydrochloride (JAN/USAN) <JP>
E D09981 Ulimorelin (USAN/INN)
E D09982 Ulimorelin hydrochloride (USAN)
E D10660 Relamorelin (USAN/INN)
C Gonadotropin-releasing hormone
D GNRHR [HSA:2798] [KO:K04280]
E D08027 Gonadorelin (INN)
E D00988 Gonadorelin hydrochloride (USP)
E D03267 Gonadorelin diacetate (JP18) <JP>
E D04361 Gonadorelin acetate (USP)
E D08241 Nafarelin (INN)
E D00990 Nafarelin acetate (USAN) <JP/US>
E D08010 Ganirelix (INN)
E D04302 Ganirelix acetate (JAN/USAN) <JP/US>
E D07665 Cetrorelix (INN)
E D01685 Cetrorelix acetate (JAN/USAN) <JP/US>
E D09335 Elagolix (USAN/INN)
E D09336 Elagolix sodium (USAN) <US>
E D11608 Linzagolix (USAN/INN)
E D11609 Linzagolix choline (USAN)
E D07259 Buserelin (INN)
E D01831 Buserelin acetate (JAN/USAN) <JP>
E D08113 Leuprorelin (INN)
E D00989 Leuprolide acetate (USP) <JP/US>
E D12337 Leuprolide mesylate <US>
E D04405 Goserelin (USAN/INN)
E D00573 Goserelin acetate (JAN/USP) <JP/US>
E D06247 Triptorelin (USAN/INN)
E D06248 Triptorelin pamoate (USAN) <US>
E D08649 Triptorelin acetate
E D02369 Histrelin (USAN/INN)
E D02116 Histrelin acetate <US>
E D02738 Abarelix (USAN/INN)
E D08901 Degarelix (INN/USAN)
E D08635 Degarelix acetate (USAN)
E D09400 Degarelix acetate (JAN) <JP/US>
E D10888 Relugolix (JAN/USAN/INN) <JP/US>
E D04644 Iturelix (USAN/INN)
E D04823 Lutrelin acetate (USAN)
E D05599 Prazarelix acetate (USAN)
E D07957 Fertirelin (INN)
E D11351 Opigolix (USAN/INN)
C Lutropin-choriogonadotropic hormone
D LHCGR [HSA:3973] [KO:K04248]
E D06457 Gonadotropin, chorionic (USP) <JP/US>
E D02692 Menotropins (USAN) <JP>
E D06459 Purified human menopausal gonadotrophin (JAN) <JP>
E D05258 Serum gonadotrophin (JAN)
E D04824 Lutropin alfa (USAN/INN)
E D03478 Choriogonadotropin alfa (USAN/INN) <JP/US>
C Melanocortin
D MC1R [HSA:4157] [KO:K04199]
E D10511 Afamelanotide (USAN/INN)
E D11334 Afamelanotide acetate (USAN) <US>
E D06569 Bremelanotide (USAN/INN)
E D11629 Bremelanotide acetate (USAN) <US>
E D12148 Dersimelagon phosphate (USAN)
D MC2R [HSA:4158] [KO:K04200]
E D00146 Corticotropin (USP/INN) <US>
E D03593 Corticotropin zinc hydroxide
E D06544 Corticotropin, repository (USP)
E D00284 Cosyntropin (USP) <US>
E D02105 Tetracosactide acetate (JAN) <JP>
E D07417 Alsactide (INN)
E D05827 Seractide acetate (USAN)
E D09801 Giractide acetate (JAN)
E D09937 Giractide (INN)
D MC4R [HSA:4160] [KO:K04202]
E D11927 Setmelanotide (USAN/INN)
E D11928 Setmelanotide acetate <US>
E D11929 Setmelanotide hydrochloride (USAN)
E D06569 Bremelanotide (USAN/INN)
E D11629 Bremelanotide acetate (USAN) <US>
C Motilin
D MLNR [HSA:2862] [KO:K05266]
E D02801 Alemcinal (USAN/INN)
E D03216 Atilmotin (USAN/INN)
E D04497 Idremcinal (USAN/INN)
E D05053 Mitemcinal fumarate (USAN)
E D10330 Camicinal (USAN/INN)
C Neuropeptide Y
D NPY5R [HSA:4889] [KO:K04207]
E D08026 Velneperit (USAN/INN)
C Opioid
D OPRM1 [HSA:4988] [KO:K04215]
E D08639 Trimebutine (INN)
E D01500 Trimebutine maleate (JP18) <JP>
E D06618 Methylnaltrexone bromide (JAN/USAN) <US>
E D02878 Alvimopan (USAN) <US>
E D10479 Naloxegol (USAN/INN)
E D10375 Naloxegol oxalate (USAN) <US>
E D08249 Naloxone (INN)
E D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
E D11620 Naloxone hydrochloride dihydrate <US>
E D10188 Naldemedine (USAN/INN)
E D10478 Naldemedine tosylate (JAN/USAN) <JP/US>
E D07861 Diphenoxylate (INN)
E D03860 Diphenoxylate hydrochloride (USP)
E D08144 Loperamide (INN)
E D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
E D03809 Difenoxin (USAN/INN)
E D11583 Difenoxin hydrochloride
E D07113 Loperamide oxide (INN)
E D10403 Eluxadoline (USAN) <US>
E D00320 Fentanyl (JAN/USP/INN) <JP/US>
E D01399 Fentanyl citrate (JP18/USP) <JP/US>
E D10811 Fentanyl hydrochloride (JAN)
E D07122 Alfentanil (INN)
E D00835 Alfentanil hydrochloride (USP) <US>
E D05938 Sufentanil (USAN/INN)
E D00845 Sufentanil citrate (USP) <US>
E D02941 Anileridine (USP/INN)
E D02942 Anileridine hydrochloride (USP)
E D08473 Remifentanil (INN)
E D01177 Remifentanil hydrochloride (JAN/USAN) <JP/US>
E D08233 Morphine (BAN)
E D00842 Morphine sulfate (USP) <JP/US>
E D02271 Morphine hydrochloride hydrate (JP18) <JP>
E D08234 Morphine tartrate
E D08047 Hydromorphone (INN)
E D00839 Hydromorphone hydrochloride (JAN/USP) <JP/US>
E D07285 Nicomorphine (INN)
E D08273 Nicomorphine hydrochloride
E D05312 Oxycodone (USAN/INN) <US>
E D00847 Oxycodone hydrochloride (USP) <US>
E D03783 Oxycodone terephthalate (USP)
E D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
E D07831 Dihydrocodeine (INN)
E D01481 Dihydrocodeine phosphate (JP18) <JP>
E D03825 Dihydrocodeine bitartrate (USP)
E D07832 Dihydrocodeine thiocyanate
E D08323 Oxymorphone (INN)
E D00844 Oxymorphone hydrochloride (USP) <US>
E D08100 Ketobemidone (INN)
E D08101 Ketobemidone hydrochloride
E D08343 Pethidine (INN)
E D01383 Meperidine hydrochloride (USP) <JP/US>
E D07809 Dextropropoxyphene (INN)
E D00482 Propoxyphene hydrochloride (USAN) <US>
E D05632 Propoxyphene napsylate (USAN)
E D00498 Pentazocine (JP18/USP/INN) <JP>
E D02111 Pentazocine lactate (USP)
E D02227 Pentazocine hydrochloride (JAN/USP) <JP>
E D07132 Buprenorphine (JAN/INN) <JP/US>
E D00836 Buprenorphine hydrochloride (JP18/USP) <JP/US>
E D03197 Butorphanol (USAN/INN)
E D00837 Butorphanol tartrate (JAN/USP) <US>
E D08246 Nalbuphine (INN)
E D00843 Nalbuphine hydrochloride (USAN) <US>
E D08597 Tilidine (INN)
E D06147 Tilidine hydrochloride (USAN)
E D08623 Tramadol (INN)
E D01355 Tramadol hydrochloride (JP18/USP) <JP/US>
E D00838 Dezocine (USAN)
E D08182 Meptazinol (INN)
E D04924 Meptazinol hydrochloride (USAN)
E D06007 Tapentadol (USAN/INN)
E D10199 Tapentadol hydrochloride (JAN) <JP/US>
E D11214 Oliceridine (USAN/INN)
E D05113 Naltrexone (USAN/INN) <US>
E D02095 Naltrexone hydrochloride (USP) <US>
E D05111 Nalmefene (USAN/INN)
E D02104 Nalmefene hydrochloride <US>
E D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
E D08195 Methadone (BAN)
E D02102 Methadone hydrochloride (JAN/USP) <JP/US>
E D04716 Levomethadyl acetate (USAN)
E D00840 Levomethadyl acetate hydrochloride (USAN)
E D08121 Levomethadone (INN)
E D08122 Levomethadone hydrochloride
E D07286 Diamorphine (BAN)
E D07810 Diacetylmorphine hydrochloride
E D07929 Ethylmorphine (BAN)
E D02205 Ethylmorphine hydrochloride hydrate (JP18)
E D08045 Hydrocodone (INN)
E D03725 Hydrocodone bitartrate (USP) <US>
E D04461 Hydrocodone polistirex (USAN)
E D08046 Hydrocodone hydrochloride
E D00195 Codeine (USP)
E D02101 Codeine phosphate (USP) <JP>
E D03579 Codeine polistirex (USAN)
E D03580 Codeine sulfate (USP) <US>
E D07740 Codeine hydrochloride
E D07385 Pholcodine (INN)
E D07557 O-Acetyldihydrocodeine hydrochloride
E D08247 Nalorphine (INN)
E D08248 Nalorphine hydrochloride (USP)
E D00841 Levorphanol tartrate (USP) <US>
E D01435 Ethoheptazine citrate (JAN)
E D02238 Levallorphan tartrate (JP18) <JP>
E D03156 Brifentanil hydrochloride (USAN)
E D03405 Carfentanil citrate (USAN)
E D03618 Cyclazocine (USAN/INN)
E D04764 Lofentanil oxalate (USAN)
E D04973 Methadyl acetate (USAN)
E D05048 Mirfentanil hydrochloride (USAN)
E D05217 Ocfentanil hydrochloride (USAN)
E D05631 Propiram fumarate (USAN)
E D05667 Quadazocine mesylate (USAN)
E D06189 Tonazocine mesylate (USAN)
E D06208 Trefentanil hydrochloride (USAN)
E D06268 Trimeperidine (INN)
E D06342 Xorphanol mesylate (USAN)
E D07620 Carfentanil (INN)
E D07863 Diprenorphine (INN)
E D07864 Diprenorphine hydrochloride
E D07937 Etorphine (INN)
E D08123 Levorphanol (INN)
E D10162 Samidorphan (USAN)
E D10163 Samidorphan l-malate (USAN)
E D10349 Bevenopran (USAN/INN)
E D10371 Methylsamidorphan (USAN)
E D10436 Cebranopadol (USAN/INN)
E D10612 Benzhydrocodone (USAN/INN)
E D10648 Methylsamidorphan chloride (USAN/INN)
E D10690 Axelopran sulfate (USAN)
E D10692 Benzhydrocodone hydrochloride (USAN)
E D10740 Axelopran (USAN/INN)
E D11291 Asalhydromorphone (USAN)
E D11292 Asalhydromorphone hydrochloride (USAN)
E D11424 Oxycodegol (USAN)
E D11425 Oxycodegol phosphate (USAN)
D OPRK1 [HSA:4986] [KO:K04214]
E D08639 Trimebutine (INN)
E D01500 Trimebutine maleate (JP18) <JP>
E D08249 Naloxone (INN)
E D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
E D11620 Naloxone hydrochloride dihydrate <US>
E D08144 Loperamide (INN)
E D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
E D07113 Loperamide oxide (INN)
E D10403 Eluxadoline (USAN) <US>
E D05312 Oxycodone (USAN/INN) <US>
E D00847 Oxycodone hydrochloride (USP) <US>
E D03783 Oxycodone terephthalate (USP)
E D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
E D08100 Ketobemidone (INN)
E D08101 Ketobemidone hydrochloride
E D00498 Pentazocine (JP18/USP/INN) <JP>
E D02111 Pentazocine lactate (USP)
E D02227 Pentazocine hydrochloride (JAN/USP) <JP>
E D07132 Buprenorphine (JAN/INN) <JP/US>
E D00836 Buprenorphine hydrochloride (JP18/USP) <JP/US>
E D03197 Butorphanol (USAN/INN)
E D00837 Butorphanol tartrate (JAN/USP) <US>
E D08246 Nalbuphine (INN)
E D00843 Nalbuphine hydrochloride (USAN) <US>
E D00838 Dezocine (USAN)
E D05113 Naltrexone (USAN/INN) <US>
E D02095 Naltrexone hydrochloride (USP) <US>
E D05111 Nalmefene (USAN/INN)
E D02104 Nalmefene hydrochloride <US>
E D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
E D08247 Nalorphine (INN)
E D08248 Nalorphine hydrochloride (USP)
E D06405 Nalfurafine hydrochloride (JAN/USAN) <JP>
E D11111 Difelikefalin (USAN/INN)
E D10890 Difelikefalin acetate (JAN) <US>
E D01879 Eptazocine hydrobromide (JAN)
E D02238 Levallorphan tartrate (JP18) <JP>
E D03618 Cyclazocine (USAN/INN)
E D04649 Ketazocine (USAN/INN)
E D05299 Oxilorphan (USAN/INN)
E D05646 Proxorphan tartrate (USAN)
E D05667 Quadazocine mesylate (USAN)
E D05907 Spiradoline mesylate (USAN)
E D06189 Tonazocine mesylate (USAN)
E D06342 Xorphanol mesylate (USAN)
E D06395 Enadoline hydrochloride (USAN)
E D07863 Diprenorphine (INN)
E D07864 Diprenorphine hydrochloride
E D07904 Eptazocine (INN)
E D07937 Etorphine (INN)
E D11831 Aticaprant (USAN/INN)
D OPRD1 [HSA:4985] [KO:K04213]
E D08249 Naloxone (INN)
E D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
E D11620 Naloxone hydrochloride dihydrate <US>
E D08144 Loperamide (INN)
E D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
E D07113 Loperamide oxide (INN)
E D10403 Eluxadoline (USAN) <US>
E D05312 Oxycodone (USAN/INN) <US>
E D00847 Oxycodone hydrochloride (USP) <US>
E D03783 Oxycodone terephthalate (USP)
E D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
E D08100 Ketobemidone (INN)
E D08101 Ketobemidone hydrochloride
E D08246 Nalbuphine (INN)
E D00843 Nalbuphine hydrochloride (USAN) <US>
E D05113 Naltrexone (USAN/INN) <US>
E D02095 Naltrexone hydrochloride (USP) <US>
E D05111 Nalmefene (USAN/INN)
E D02104 Nalmefene hydrochloride <US>
E D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
E D02238 Levallorphan tartrate (JP18) <JP>
E D05007 Metkephamid acetate (USAN)
E D05667 Quadazocine mesylate (USAN)
E D06189 Tonazocine mesylate (USAN)
E D06342 Xorphanol mesylate (USAN)
E D07937 Etorphine (INN)
D OPRL1 [HSA:4987] [KO:K04216]
E D10436 Cebranopadol (USAN/INN)
C Orexin
D HCRTR [HSA:3061 3062] [KO:K04238 K04239]
E D10082 Suvorexant (JAN/USAN) <JP/US>
E D11022 Lemborexant (JAN/USAN/INN) <JP/US>
E D09964 Almorexant (INN)
E D10345 Filorexant (USAN)
E D11886 Daridorexant (USAN/INN)
E D11887 Daridorexant hydrochloride (JAN/USAN) <US>
D HCRTR2 [HSA:3062] [KO:K04239]
E D11269 Seltorexant (USAN/INN)
C Oxytocin
D OXTR [HSA:5021] [KO:K04229]
E D03008 Atosiban (USAN/INN)
E D07475 Atosiban acetate
E D07228 Demoxytocin (INN)
E D00089 Oxytocin (JP18/USP/INN) <JP/US>
E D07229 Carbetocin (USAN/INN/BAN)
E D08986 Retosiban (USAN)
E D09797 Cargutocin (INN/JAN)
E D10117 Epelsiban (USAN)
E D10118 Epelsiban besylate (USAN)
C Relaxin
D RXFP1 [HSA:59350] [KO:K04306]
E D10488 Serelaxin (USAN/INN)
C Somatostatin
D SSTR [HSA:6751 6752 6753 6754 6755] [KO:K04217 K04218 K04219 K04220 K04221]
E D07431 Somatostatin (INN)
E D05812 Seglitide acetate (USAN)
E D11192 Veldoreotide (USAN/INN)
D SSTR1 [HSA:6751] [KO:K04217]
E D10147 Pasireotide (USAN)
E D10497 Pasireotide diaspartate <US>
E D10566 Pasireotide pamoate (JAN) <JP/US>
D SSTR2 [HSA:6752] [KO:K04218]
E D00442 Octreotide (USAN/INN)
E D02250 Octreotide acetate (JAN) <JP>
E D05230 Octreotide pamoate (USAN)
E D06495 Octreotide acetate (USP) <US>
E D04666 Lanreotide acetate (JAN/USAN) <JP/US>
E D06281 Vapreotide (USAN/INN)
E D09988 Vapreotide acetate (USAN)
E D10147 Pasireotide (USAN)
E D10497 Pasireotide diaspartate <US>
E D10566 Pasireotide pamoate (JAN) <JP/US>
E D02108 Indium In 111 pentetreotide (USP) <JP/US>
E D11651 Edotreotide gallium Ga-68 <US>
E D11882 Copper Cu 64 dotatate <US>
E D11033 Lutetium (177Lu) oxodotreotide (INN) <JP/US>
E D11204 Octreotide hydrochloride (USAN)
E D11845 Tidutamab (USAN/INN)
E D12431 Lutetium Lu177 edotreotide (USAN)
E D12477 Paltusotine (USAN/INN)
E D12478 Paltusotine hydrochloride (USAN)
D SSTR3 [HSA:6753] [KO:K04219]
E D10147 Pasireotide (USAN)
E D10497 Pasireotide diaspartate <US>
E D10566 Pasireotide pamoate (JAN) <JP/US>
E D02108 Indium In 111 pentetreotide (USP) <JP/US>
D SSTR5 [HSA:6755] [KO:K04221]
E D04666 Lanreotide acetate (JAN/USAN) <JP/US>
E D06281 Vapreotide (USAN/INN)
E D09988 Vapreotide acetate (USAN)
E D10147 Pasireotide (USAN)
E D10497 Pasireotide diaspartate <US>
E D10566 Pasireotide pamoate (JAN) <JP/US>
E D02108 Indium In 111 pentetreotide (USP) <JP/US>
C Tachykinin
D TACR1 (NK1R) [HSA:6869] [KO:K04222]
E D02968 Aprepitant (JAN/USP/INN) <JP/US>
E D10895 Fosaprepitant (INN)
E D06597 Fosaprepitant dimeglumine (USAN) <JP/US>
E D06574 Casopitant mesylate (USAN)
E D10742 Rolapitant (USAN/INN)
E D08988 Rolapitant hydrochloride (USAN) <US>
E D03221 Befetupitant (USAN/INN)
E D04122 Ezlopitant (USAN/INN)
E D04860 Maropitant citrate (USAN)
E D05152 Netupitant (USAN/INN)
E D06293 Vestipitant mesylate (USAN)
E D06317 Vofopitant dihydrochloride (USAN)
E D09378 Serlopitant (USAN)
E D09650 Orvepitant (USAN/INN)
E D09651 Orvepitant maleate (USAN)
E D10391 Telmapitant (USAN)
E D11065 Fosnetupitant (USAN/INN)
E D11370 Fosnetupitant chloride hydrochloride (JAN/USAN) <JP>
E D11728 Tradipitant (USAN/INN)
E D12123 Elinzanetant (USAN/INN)
D TACR3 (NK3R) [HSA:6870] [KO:K04224]
E D11976 Fezolinetant (USAN)
E D05996 Talnetant hydrochloride (USAN)
E D11345 Pavinetant (USAN/INN)
E D12123 Elinzanetant (USAN/INN)
C Thrombin
D F2R (PAR1) [HSA:2149] [KO:K03914]
E D09765 Vorapaxar (USAN/INN)
E D09766 Vorapaxar sulfate (JAN/USAN) <US>
E D09866 Atopaxar (USAN)
E D09867 Atopaxar hydrobromide (USAN)
C Thyrotropin-releasing hormone
D TRHR [HSA:7201] [KO:K04282]
E D06120 Thyrotropin alfa (USAN/INN) <JP/US>
E D00176 Protirelin (JP18/USAN/INN) <JP>
E D02007 Protirelin tartrate hydrate (JP18) <JP>
E D01925 Taltirelin hydrate (JP18) <JP>
E D02588 Montirelin (INN)
E D09845 Montirelin hydrate (JAN)
E D10594 Rovatirelin hydrate (JAN)
C Vasopressin
D AVPR1 [HSA:552 553] [KO:K04226 K04227]
E D00101 Vasopressin (JP18/USP) <JP/US>
E D09820 Vasopressin tannate (JAN)
E D02983 Argipressin tannate (USAN)
E D00366 Lypressin (USAN/INN)
E D06672 Terlipressin (USAN/INN)
E D08571 Terlipressin acetate (JAN) <US>
E D07227 Ornipressin (INN)
D AVPR1A [HSA:552] [KO:K04226]
E D07748 Conivaptan (INN)
E D01236 Conivaptan hydrochloride (JAN/USAN)
E D04137 Felypressin (USAN/INN)
E D11476 Balovaptan (USAN/INN)
D AVPR2 [HSA:554] [KO:K04228]
E D01213 Tolvaptan (JAN/USAN/INN) <JP/US>
E D11659 Tolvaptan sodium phosphate (JAN) <JP>
E D07748 Conivaptan (INN)
E D01236 Conivaptan hydrochloride (JAN/USAN)
E D00101 Vasopressin (JP18/USP) <JP/US>
E D09820 Vasopressin tannate (JAN)
E D02983 Argipressin tannate (USAN)
E D00291 Desmopressin (INN)
E D02235 Desmopressin acetate (USP) <JP/US>
E D00366 Lypressin (USAN/INN)
E D06672 Terlipressin (USAN/INN)
E D08571 Terlipressin acetate (JAN) <US>
E D07227 Ornipressin (INN)
E D01855 Mozavaptane hydrochloride (JAN)
E D04752 Lixivaptan (USAN/INN)
C Purine / pyrimidine
D P2RY12 [HSA:64805] [KO:K04298]
E D07729 Clopidogrel (USP/INN)
E D00769 Clopidogrel bisulfate (USP) <JP/US>
E D10823 Clopidogrel hydrochloride
E D10824 Clopidogrel besilate
E D08594 Ticlopidine (INN)
E D01028 Ticlopidine hydrochloride (JP18/USP) <JP>
E D05597 Prasugrel hydrochloride (JAN/USAN) <JP/US>
E D09017 Ticagrelor (JAN/USAN/INN) <JP/US>
E D03359 Cangrelor (USAN/INN)
E D03361 Cangrelor tetrasodium (USAN) <US>
E D08983 Regrelor disodium (USAN)
E D09607 Elinogrel (USAN/INN)
E D09608 Elinogrel potassium (USAN)
C Adenosine
D ADORA [HSA:134 135 136 140] [KO:K04265 K04266 K04267 K04268]
E D00045 Adenosine (JAN/USP) <JP/US>
E D02300 Adenosine triphosphate disodium hydrate (JAN) <JP>
E D02769 Adenosine phosphate (USAN/INN)
E D08646 Triphosadenine (DCF)
E D08647 Triphosadenine disodium salt
D ADORA1 [HSA:134] [KO:K04265]
E D00528 Caffeine (USP) <JP>
E D01453 Caffeine hydrate (JP18) <JP>
E D07603 Caffeine citrate (USP) <US>
E D00691 Dyphylline (USP) <JP>
E D02017 Oxtriphylline (USP)
E D01771 Proxyphylline (JAN/INN) <JP>
E D00371 Theophylline (JP18) <JP/US>
E D01712 Theophylline sodium acetate (JAN)
E D06103 Theophylline (USP)
E D06104 Theophylline sodium glycinate (USP)
E D00227 Aminophylline (USP/INN)
E D05429 Aminophylline hydrate (JP18) <JP>
E D11630 Aminophylline dihydrate <US>
E D07491 Bamifylline (INN)
E D03051 Bamifylline hydrochloride (USAN)
E D02964 Apaxifylline (USAN/INN)
E D04006 Enprofylline (USAN/INN)
E D05125 Naxifylline (USAN/INN)
E D05818 Selodenoson (USAN/INN)
E D06019 Tecadenoson (USAN/INN)
E D08989 Rolofylline (USAN)
E D09684 Tonapofylline (USAN/INN)
E D10493 Trabodenoson (USAN/INN)
D ADORA2 [HSA:135 136] [KO:K04266 K04267]
E D01771 Proxyphylline (JAN/INN) <JP>
E D04006 Enprofylline (USAN/INN)
E D12369 Etrumadenant (USAN/INN)
D ADORA2A [HSA:135] [KO:K04266]
E D12568 Regadenoson (INN) <US>
E D05711 Regadenoson (USAN) <US>
E D00528 Caffeine (USP) <JP>
E D01453 Caffeine hydrate (JP18) <JP>
E D07603 Caffeine citrate (USP) <US>
E D04641 Istradefylline (JAN/USAN/INN) <JP/US>
E D02017 Oxtriphylline (USP)
E D03898 Doxofylline (USAN/INN)
E D03120 Binodenoson (USAN/INN)
E D03212 Apadenoson (USAN)
E D09003 Sonedenoson (USAN)
E D09717 Preladenant (USAN/INN)
E D09991 Vipadenant (USAN/INN)
E D10174 Tozadenant (USAN)
E D10362 Evodenoson (USAN)
E D11547 Ciforadenant (USAN)
E D11978 Inupadenant (USAN)
E D11979 Inupadenant hydrochloride (USAN)
D ADORA2B [HSA:136] [KO:K04267]
E D00691 Dyphylline (USP) <JP>
E D00371 Theophylline (JP18) <JP/US>
E D01712 Theophylline sodium acetate (JAN)
E D06103 Theophylline (USP)
E D06104 Theophylline sodium glycinate (USP)
E D00227 Aminophylline (USP/INN)
E D05429 Aminophylline hydrate (JP18) <JP>
E D11630 Aminophylline dihydrate <US>
D ADORA3 [HSA:140] [KO:K04268]
E D10971 Piclidenoson (USAN/INN)
E D11128 Namodenoson (USAN/INN)
C Cysteinyl leukotriene
D CYSLTR1 [HSA:10800] [KO:K04322]
E D00411 Zafirlukast (JAN/USAN/INN) <US>
E D08408 Pranlukast (INN)
E D02732 Pranlukast hydrate (JP18) <JP>
E D08229 Montelukast (INN)
E D00529 Montelukast sodium (JP18/USP) <JP/US>
E D01385 Ibudilast (JP18/INN) <JP>
E D02384 Verlukast (USAN/INN)
E D02739 Ablukast (USAN/INN)
E D02741 Ablukast sodium (USAN)
E D02846 Cinalukast (USAN/INN)
E D02848 Pobilukast edamine (USAN)
E D02849 Ritolukast (USAN/INN)
E D02850 Sulukast (USAN/INN)
E D02851 Tomelukast (USAN/INN)
E D06659 Tipelukast (USAN)
C Free fatty acid
D FFAR1 [HSA:2864] [KO:K04325]
E D10336 Fasiglifam (USAN/INN)
E D10567 Fasiglifam hydrate (JAN)
C Leukotriene
D LTB4R [HSA:1241 56413] [KO:K04296 K04297]
E D04074 Etalocib (USAN)
E D05085 Moxilubant maleate (USAN)
E D06140 Ticolubant (USAN/INN)
C Prostaglandin
D PTGDR [HSA:5729] [KO:K04332]
E D01128 Ramatroban (JAN/INN) <JP>
E D08940 Laropiprant (INN/USAN)
E D09990 Vidupiprant (USAN/INN)
E D10326 Setipiprant (USAN/INN)
E D10631 Fevipiprant (JAN/USAN/INN)
D PTGER1 [HSA:5731] [KO:K04258]
E D00180 Alprostadil (JP18/USP/INN) <JP/US>
E D02705 Alprostadil alfadex (JP18) <JP>
E D02073 Gemeprost (JAN/USAN/INN) <JP>
E D01869 Ornoprostil (JAN/INN)
E D02722 Limaprost (INN)
E D02723 Ecraprost (USAN/INN)
E D02860 Limaprost alfadex (JP18) <JP>
E D03999 Enisoprost (USAN/INN)
D PTGER2 [HSA:5732] [KO:K04259]
E D00419 Misoprostol (JAN/USP/INN) <JP/US>
E D01891 Enprostil (JAN/USAN/INN)
E D00079 Dinoprostone (JAN/USP/INN) <JP/US>
E D03269 Dinoprostone betadex (JAN)
E D02725 Sulprostone (USAN/INN)
E D10965 Omidenepag (USAN/INN)
E D10966 Omidenepag isopropyl (JAN) <JP/US>
E D02726 Meteneprost (USAN/INN)
E D02975 Arbaprostil (USAN/INN)
E D03187 Butaprost (USAN/INN)
E D05732 Rioprostil (USAN/INN)
E D06240 Trimoprostil (USAN/INN)
E D09613 Evatanepag (USAN/INN)
E D09614 Evatanepag sodium (USAN)
E D09968 Taprenepag (USAN/INN)
E D09969 Taprenepag isopropyl (USAN)
D PTGER3 [HSA:5733] [KO:K04260]
E D00419 Misoprostol (JAN/USP/INN) <JP/US>
E D01891 Enprostil (JAN/USAN/INN)
D PTGER4 [HSA:5734] [KO:K04261]
E D00419 Misoprostol (JAN/USP/INN) <JP/US>
E D10638 Grapiprant (USAN/INN)
D PTGFR [HSA:5737] [KO:K04262]
E D00081 Dinoprost (JP18/USAN/INN) <JP>
E D01352 Dinoprost tromethamine (JAN/USP)
E D02343 Carboprost (USAN/INN)
E D00682 Carboprost tromethamine (USP) <US>
E D03399 Carboprost methyl (USAN)
E D00356 Latanoprost (JAN/USP/INN) <JP/US>
E D08661 Unoprostone (INN)
E D01452 Isopropyl unoprostone (JAN) <JP>
E D02724 Bimatoprost (JAN/USAN/INN) <JP/US>
E D01964 Travoprost (JAN/USP/INN) <JP/US>
E D06274 Tafluprost (JAN/USAN/INN) <JP/US>
E D10441 Latanoprostene bunod (USAN/INN) <US>
E D02719 Rosaprostol (INN)
E D02727 Cloprostenol sodium (USP)
E D05642 Prostalene (USAN)
E D07730 Cloprostenol (INN)
E D07932 Etiproston (INN)
E D08591 Tiaprost (INN)
C Prostacyclin
D PTGIR [HSA:5739] [KO:K04263]
E D00106 Epoprostenol (USAN/INN)
E D01337 Epoprostenol sodium (JAN/USAN) <JP/US>
E D02721 Iloprost (USAN/INN) <JP/US>
E D08065 Iloprost tromethamine
E D02720 Beraprost (USAN)
E D01551 Beraprost sodium (JP18/USAN) <JP>
E D06213 Treprostinil (JAN/USAN/INN) <JP/US>
E D08628 Treprostinil monosodium salt
E D10430 Treprostinil diolamine (USAN) <US>
E D12005 Treprostinil palmitil (USAN/INN)
E D09994 Selexipag (JAN/USAN/INN) <JP/US>
E D01385 Ibudilast (JP18/INN) <JP>
E D01188 Pimilprost (JAN/INN)
E D02048 Clinprost (JAN/INN)
E D03522 Ciprostene calcium (USAN)
E D10628 Esuberaprost (USAN/INN)
E D10703 Esuberaprost sodium (USAN)
E D10725 Ralinepag (USAN/INN)
E D11446 Esuberaprost potassium (USAN)
C Sphingolipid
D S1PR [HSA:1901 9294 1903 8698 53637] [KO:K04288 K04292 K04290 K04293 K04295]
E D10968 Ozanimod (USAN/INN)
E D10967 Ozanimod hydrochloride (JAN/USAN) <US>
E D10904 Amiselimod hydrochloride (USAN)
E D10905 Amiselimod (USAN/INN)
E D10930 Etrasimod (USAN)
D S1PR1 [HSA:1901] [KO:K04288]
E D10001 Fingolimod (INN)
E D04187 Fingolimod hydrochloride (JAN/USAN) <JP/US>
E D11460 Siponimod (USAN/INN)
E D11072 Siponimod fumarate (USAN) <JP/US>
E D11215 Ponesimod (USAN/INN) <US>
E D11283 Cenerimod (USAN/INN)
E D12376 Udifitimod (USAN)
E D12377 Udifitimod hydrochloride (USAN)
E D12549 Fingolimod lauryl sulfate <US>
D S1PR5 [HSA:53637] [KO:K04295]
E D11460 Siponimod (USAN/INN)
E D11072 Siponimod fumarate (USAN) <JP/US>
C Thromboxane
D TBXA2R [HSA:6915] [KO:K04264]
E D07140 Picotamide (BAN)
E D01896 Cilostazol (JP18/USP/INN) <JP/US>
E D01123 Seratrodast (JAN/USAN/INN) <JP>
E D01128 Ramatroban (JAN/INN) <JP>
E D03642 Daltroban (USAN/INN)
E D04500 Ifetroban (USAN/INN)
E D04501 Ifetroban sodium (USAN)
E D05727 Ridogrel (USAN/INN)
E D05970 Sulotroban (USAN/INN)
E D06077 Terbogrel (USAN/INN)
E D06280 Vapiprost hydrochloride (JAN/USAN)
E D09774 Imitrodast sodium (JAN)
E D09824 Domitroban calcium hydrate (JAN)
C Cannabinoid
D CNR [HSA:1268 1269] [KO:K04277 K04278]
E D00306 Dronabinol (USP/INN) <US>
E D05099 Nabilone (USAN/INN) <US>
E D10915 Cannabidiol (USAN/INN) <US>
E D12305 Onternabez (USAN)
D CNR1 [HSA:1268] [KO:K04277]
E D05731 Rimonabant (JAN/USAN/INN)
E D04717 Levonantradol hydrochloride (USAN)
E D05117 Nantradol hydrochloride (USAN)
E D09009 Taranabant (USAN/INN)
E D09349 Ibipinabant (USAN/INN)
E D09362 Otenabant (USAN/INN)
E D09363 Otenabant hydrochloride (USAN)
E D11435 Nimacimab (USAN)
D CNR2 [HSA:1269] [KO:K04278]
E D11312 Lenabasum (USAN/INN)
E D11429 Olorinab (USAN)
E D12511 Vicasinabin (USAN/INN)
C Melatonin
D MTNR1 [HSA:4543 4544] [KO:K04285 K04286]
E D08170 Melatonin (JAN) <JP>
E D02689 Ramelteon (JAN/USAN/INN) <JP/US>
E D09388 Tasimelteon (USAN/INN) <US>
E D02578 Agomelatine (INN)
C Platelet activating factor
D PTAFR [HSA:5724] [KO:K04279]
E D07407 Rupatadine (INN)
E D08497 Rupatadine fumarate (JAN) <JP>
E D01652 Apafant (JAN/USAN/INN)
E D02590 Israpafant (JAN/INN)
E D04724 Lexipafant (USAN/INN)
C R-spondin
D LGR5 [HSA:8549] [KO:K04308]
E D12416 Petosemtamab (USAN/INN)
B Secretin receptor family
C Calcitonin
D CALCR [HSA:799] [KO:K04576]
E D00249 Calcitonin salmon (JP18/USP/INN) <US>
E D03287 Elcatonin (JP18/INN) <JP>
E D09600 Davalintide (USAN/INN)
E D09601 Davalintide acetate (USAN)
E D09771 Avicatonin (JAN/INN)
D CALCRL [HSA:10203] [KO:K04577]
E D10928 Erenumab (USAN/INN) <JP/US>
E D10673 Ubrogepant (USAN/INN) <US>
E D10662 Rimegepant (USAN/INN)
E D10663 Rimegepant sulfate (USAN) <US>
E D11313 Atogepant (USAN) <US>
E D09391 Telcagepant (USAN)
E D09392 Telcagepant potassium (USAN)
E D09600 Davalintide (USAN/INN)
E D09601 Davalintide acetate (USAN)
E D11898 Zavegepant (USAN)
E D11899 Zavegepant hydrochloride (USAN)
C Parathyroid hormone
D PTH1R [HSA:5745] [KO:K04585]
E D06078 Teriparatide (USP/INN) <JP/US>
E D03358 Teriparatide acetate (JAN) <JP>
E D06546 Teriparatide acetate (USAN)
E D05364 Parathyroid hormone (human) (USAN) <US>
E D10885 Abaloparatide (USAN/INN) <US>
E D11563 Abaloparatide acetate (JAN) <JP>
E D12395 Palopegteriparatide (USAN/INN)
D PTH2R [HSA:5746] [KO:K04586]
E D05364 Parathyroid hormone (human) (USAN) <US>
C Corticotropin-releasing hormone
D CRHR [HSA:1394 1395] [KO:K04578 K04579]
E D03905 Corticorelin (human) (JAN) <JP>
E D03591 Corticorelin acetate (USAN)
E D03592 Corticorelin ovine triflutate (USAN)
D CRHR1 [HSA:1394] [KO:K04578]
E D09610 Emicerfont (USAN/INN)
E D09695 Verucerfont (USAN/INN)
E D10022 Pexacerfont (USAN/INN)
E D12366 Crinecerfont (USAN)
C Growth hormone-releasing hormone
D GHRHR [HSA:2692] [KO:K04584]
E D08509 Sermorelin (INN)
E D02117 Sermorelin acetate (USAN)
E D06655 Tesamorelin (USAN)
E D09015 Tesamorelin acetate (USAN) <US>
E D08523 Somatorelin (INN)
E D03326 Somatorelin acetate (JAN)
E D04491 Ibutamoren mesylate (USAN)
C Glucagon
D GLP1R [HSA:2740] [KO:K04581]
E D11034 Insulin glargine and lixisenatide <JP/US>
E D11567 Insulin degludec and liraglutide <JP/US>
E D04121 Exenatide (JAN/USAN/INN) <JP/US>
E D06404 Liraglutide (USAN/INN) <JP/US>
E D09729 Lixisenatide (JAN/USAN/INN) <JP/US>
E D08843 Albiglutide (USAN)
E D09889 Dulaglutide (USAN/INN) <JP/US>
E D10025 Semaglutide (USAN/INN) <JP/US>
E D11924 Beinaglutide (INN)
E D11360 Tirzepatide (JAN/USAN) <JP/US>
E D09723 Taspoglutide (USAN/INN)
E D10970 Pegapamodutide (USAN)
E D11418 Avexitide (USAN)
E D11419 Avexitide acetate (USAN)
E D11910 Danuglipron (USAN)
E D11911 Danuglipron tromethamine (USAN)
E D11947 Efpeglenatide (USAN/INN)
E D12225 Mazdutide (USAN)
E D12341 Vurolenatide (USAN)
E D12430 Retatrutide (USAN)
E D12529 Orforglipron calcium (USAN)
E D12536 Orforglipron (USAN)
E D12555 Lotiglipron (USAN)
D GLP2R [HSA:9340] [KO:K04582]
E D06053 Teduglutide (USAN/INN) <JP/US>
E D11337 Glepaglutide (USAN)
D GCGR [HSA:2642] [KO:K04583]
E D00116 Glucagon (genetical recombination) (JP18) <JP/US>
E D02118 Glucagon hydrochloride <US>
E D11359 Dasiglucagon (USAN)
E D12314 Dasiglucagon hydrochloride <US>
E D11230 Crotedumab (USAN/INN)
E D11614 Volagidemab (USAN)
E D12225 Mazdutide (USAN)
E D12430 Retatrutide (USAN)
C Gastric inhibitory polypeptide
D GIPR [HSA:2696] [KO:K04580]
E D11360 Tirzepatide (JAN/USAN) <JP/US>
E D12430 Retatrutide (USAN)
C Secretin
D SCTR [HSA:6344] [KO:K04588]
E D02021 Secretin (JAN/USAN/INN) <US>
B Metabotropic glutamate receptor family
C Glutamate (metabotropic)
D GRM2 [HSA:2912] [KO:K04605]
E D03966 Eglumetad (USAN)
E D08908 Eglumegad (INN)
E D09008 Talaglumetad hydrochloride (USAN)
E D09949 Pomaglumetad methionil (USAN)
E D10896 Pomaglumetad methionil (INN)
D GRM3 [HSA:2913] [KO:K04606]
E D09008 Talaglumetad hydrochloride (USAN)
E D09949 Pomaglumetad methionil (USAN)
E D10896 Pomaglumetad methionil (INN)
D GRM5 [HSA:2915] [KO:K04604]
E D04155 Fenobam (USAN)
C GABA (metabotropic)
D GABBR [HSA:2550 9568] [KO:K04615]
E D00241 Baclofen (JP18/USP/INN) <JP/US>
E D00058 gamma-Aminobutyric acid (JAN) <JP>
E D05621 Progabide (USAN/INN)
E D08861 Arbaclofen placarbil (USAN/INN)
E D09791 Arbaclofen (USAN)
E D12240 Valiloxybate (USAN)
C Chemoreception
D TAS1R2 [HSA:80834] [KO:K04625]
E D02381 Aspartame (NF/INN)
E D08836 Acesulfame potassium (NF)
E D08862 Aspartame acesulfame (NF)
D TAS1R3 [HSA:83756] [KO:K04626]
E D02381 Aspartame (NF/INN)
E D08836 Acesulfame potassium (NF)
E D08862 Aspartame acesulfame (NF)
C Calcium-sensing
D CASR [HSA:846] [KO:K04612]
E D03504 Cinacalcet (USAN)
E D03505 Cinacalcet hydrochloride (JAN/USAN) <JP/US>
E D10676 Etelcalcetide (USAN/INN)
E D10677 Etelcalcetide hydrochloride (JAN/USAN) <JP/US>
E D06020 Tecalcet hydrochloride (USAN)
E D08991 Ronacaleret hydrochloride (USAN)
E D11063 Evocalcet (JAN/INN) <JP>
E D11564 Upacicalcet sodium hydrate (JAN) <JP>
C Orphan GPRC5
D GPRC5D [HSA:55507] [KO:K04621]
E D12180 Talquetamab (USAN/INN)
B Frizzled / Smoothened family
C Frizzled
D FZD7 [HSA:8324] [KO:K02432]
E D10410 Vantictumab (USAN)
D FZD8 [HSA:8325] [KO:K02375]
E D11758 Ipafricept (USAN/INN)
C Smoothened
D SMO [HSA:6608] [KO:K06226]
E D09992 Vismodegib (USAN/INN) <US>
E D10119 Sonidegib (USAN/INN)
E D10729 Sonidegib phosphate (USAN) <US>
E D10636 Glasdegib (USAN/INN)
E D11107 Glasdegib maleate (JAN) <US>
E D10324 Patidegib (USAN)
E D10325 Patidegib hydrochloride (USAN)
E D10671 Taladegib (USAN/INN)
B Others
C Vomeronasal pheromone
D V1R [HSA:57191 317701 317702 317703 317705] [KO:K04614]
E D12524 Fasedienol (USAN/INN)
#
AIon channels
B Ligand-gated ion channels
C Acetylcholine (nicotinic)
D CHRN [HSA:1134 1135 1136 1137 1138 8973 1139 55584 57053 1140 1141 1142 1143 1144 1145 1146] [KO:K04803 K04804 K04805 K04806 K04807 K04808 K04809 K04810 K04811 K04812 K04813 K04814 K04815 K04816 K04817 K04818]
E D00611 Mecamylamine hydrochloride (USP) <US>
E D03365 Nicotine (USP) <JP/US>
E D05156 Nicotine bitartrate (USAN)
E D05157 Nicotine polacrilex (USP)
E D07770 Cytisinicline (USAN)
E D00999 Acetylcholine chloride (JP18/USP/INN) <JP/US>
E D02202 Lobeline hydrochloride (JAN)
E D02364 Lobeline (INN)
E D08138 Lobeline sulfate
D CHRN (muscle type) [HSA:1134 1140 1144 1145 1146] [KO:K04803 K04812 K04816 K04817 K04818]
E D00766 Succinylcholine chloride (USP) <US>
E D02275 Suxamethonium chloride hydrate (JP18) <JP>
E D00761 Metocurine iodide (USAN)
E D04303 Gantacurium chloride (USAN/INN)
D CHRN (neuronal type) [HSA:1135 1136 1137 1138 8973 1139 55584 57053 1141 1142 1143] [KO:K04804 K04805 K04806 K04807 K04808 K04809 K04810 K04811 K04813 K04814 K04815]
E D02207 Tubocurarine chloride (USP)
E D08655 Tubocurarine chloride (INN)
E D07272 Dimethyltubocurarine (BAN)
E D00492 Pancuronium bromide (JP18/USP/INN) <US>
E D00767 Vecuronium bromide (JAN/USP/INN) <JP/US>
E D00758 Atracurium besylate (USP) <US>
E D00764 Pipecuronium bromide (JAN/USAN/INN)
E D00760 Doxacurium chloride (USAN/INN)
E D07273 Fazadinium bromide (INN)
E D00765 Rocuronium bromide (JAN/USP/INN) <JP/US>
E D00763 Mivacurium chloride (USAN/INN)
E D00759 Cisatracurium besylate (USP) <US>
E D02204 Hexamethonium bromide (JAN/INN)
D CHRNA7 [HSA:1139] [KO:K04809]
E D10613 Bradanicline (USAN/INN)
E D10626 Encenicline (USAN/INN)
E D10693 Bradanicline hydrochloride (USAN)
E D10702 Encenicline hydrochloride (USAN)
E D10789 Encenicline hydrochloride hydrate (JAN)
D CHRNA10 [HSA:57053] [KO:K04811]
E D00612 Trimetaphan camsilate (JAN/INN)
D CHRNA3/CHRNB4 [HSA:1136 1143] [KO:K04805 K04815]
E D06016 Tebanicline tosylate (USAN)
D CHRNA4/CHRNB2 [HSA:1137 1141] [KO:K04806 K04813]
E D08669 Varenicline (INN)
E D06282 Varenicline tartrate (JAN/USAN) <JP/US>
E D02839 Altinicline maleate (USAN)
E D06016 Tebanicline tosylate (USAN)
E D08935 Ispronicline (INN/USAN)
E D08987 Rivanicline galactarate (USAN)
E D09367 Pozanicline (USAN)
E D09368 Pozanicline tartrate (USAN)
E D09382 Sofinicline (USAN)
E D09383 Sofinicline benzenesulfonate (USAN)
E D10111 Dexmecamylamine (USAN)
E D10112 Dexmecamylamine hydrochloride (USAN)
C Serotonin
D HTR3 [HSA:3359 9177 170572 200909 285242] [KO:K04819]
E D07129 Alosetron (INN)
E D02829 Alosetron hydrochloride (USAN) <US>
E D03495 Cilansetron (USAN/INN)
E D03496 Cilansetron hydrochloride (USAN)
E D00456 Ondansetron (JAN/USP/INN) <US>
E D00678 Ondansetron hydrochloride hydrate (JAN/USP) <JP/US>
E D02130 Tropisetron (INN)
E D02041 Tropisetron hydrochloride (JAN)
E D07867 Dolasetron (INN)
E D00725 Dolasetron mesylate (USP)
E D07175 Palonosetron (INN)
E D05343 Palonosetron hydrochloride (JAN/USP) <JP/US>
E D00283 Clozapine (JAN/USP/INN) <JP/US>
E D08216 Mianserin (INN)
E D01358 Mianserin hydrochloride (JAN/USAN) <JP>
E D00563 Mirtazapine (JAN/USP/INN) <JP/US>
E D11056 Mirtazapine hydrate (JAN)
E D10184 Vortioxetine (USAN)
E D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
E D12544 Vortioxetine hemihydrobromide (USAN)
E D01613 Azasetron hydrochloride (JAN)
E D01838 Fabesetron hydrochloride (JAN)
E D02016 Ramosetron hydrochloride (JAN) <JP>
E D02632 Indisetron hydrochloride (JAN)
E D03060 Batanopride hydrochloride (USAN)
E D03073 Bemesetron (USAN/INN)
E D03662 Dazopride fumarate (USAN)
E D04294 Galdansetron hydrochloride (USAN)
E D04642 Itasetron (USAN/INN)
E D04821 Lurosetron mesylate (USAN)
E D05050 Mirisetron maleate (USAN)
E D05348 Pancopride (USAN/INN)
E D05685 Quipazine maleate (USAN)
E D06253 Tropanserin hydrochloride (USAN)
E D06353 Zacopride hydrochloride (USAN)
E D06358 Zatosetron maleate (USAN)
E D06396 Renzapride (INN)
E D07481 Azasetron (INN)
E D08466 Ramosetron (INN)
E D09749 Itasetron hydrochloride hydrate (JAN)
E D10170 Tedatioxetine (USAN)
E D10171 Tedatioxetine hydrobromide (USAN)
D HTR3A [HSA:3359] [KO:K04819]
E D00274 Cisapride (USP/INN)
E D02092 Cisapride (JAN)
D HTR3B [HSA:9177] [KO:K04819]
E D04370 Granisetron (JAN/USAN/INN) <US>
E D00677 Granisetron hydrochloride (JAN/USP) <JP/US>
C GABA (ionotropic)
D GABR [HSA:2554 2555 2556 2557 2558 2559 2560 2561 2562 2563 2564 2565 2566 2567 2568 55879] [KO:K05175 K05181 K05184 K05185 K05186 K05189 K05192]
E D01071 Hexobarbital (JAN/INN)
E D00714 Thiopental sodium (JP18/USP/INN) <JP>
E D00549 Propofol (JAN/USP/INN) <JP/US>
E D04257 Fospropofol disodium (USAN)
E D00700 Mephobarbital (JAN/USP)
E D00506 Phenobarbital (JP18/USP/INN) <JP>
E D00701 Phenobarbital sodium (JAN/USP/INN) <JP/US>
E D08356 Phenobarbital diethylamine
E D07298 Barbexaclone (INN)
E D01382 Metharbital (JAN/INN)
E D00280 Clonazepam (JP18/USP/INN) <JP/US>
E D00058 gamma-Aminobutyric acid (JAN) <JP>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D04300 Ganaxolone (USAN/INN) <US>
E D00293 Diazepam (JP18/USP/INN) <JP/US>
E D00267 Chlordiazepoxide (JP18/USP/INN) <JP>
E D00693 Chlordiazepoxide hydrochloride (JAN/USP) <US>
E D01292 Medazepam (JP18/INN) <JP>
E D04882 Medazepam hydrochloride (USAN)
E D00464 Oxazepam (JAN/USP/INN) <US>
E D00694 Clorazepate dipotassium (JP18/USP) <JP/US>
E D03562 Clorazepate monopotassium (USAN)
E D00365 Lorazepam (JP18/USP/INN) <JP/US>
E D02770 Adinazolam (USAN/INN)
E D02771 Adinazolam mesylate (USAN)
E D01245 Bromazepam (JP18/USAN/INN) <JP>
E D01253 Clobazam (JAN/USAN/INN) <JP/US>
E D04650 Ketazolam (USAN/INN)
E D00470 Prazepam (JP18/USAN/INN)
E D00225 Alprazolam (JP18/USP/INN) <JP/US>
E D00338 Halazepam (USAN/INN)
E D08283 Nordazepam (INN)
E D01354 Fludiazepam (JP18/INN) <JP>
E D01293 Ethyl loflazepate (JP18/INN) <JP>
E D01514 Etizolam (JP18/INN) <JP>
E D01328 Clotiazepam (JP18/INN) <JP>
E D01268 Cloxazolam (JP18/INN) <JP>
E D01254 Tofisopam (JP18/INN) <JP>
E D01316 Mexazolam (JAN/INN) <JP>
E D00376 Meprobamate (JAN/USP/INN) <US>
E D00499 Pentobarbital (USP/INN)
E D00500 Pentobarbital sodium (JAN/USP) <US>
E D02253 Pentobarbital calcium (JP18) <JP>
E D00555 Amobarbital (JP18/INN) <JP>
E D02252 Amobarbital sodium (JAN/USP)
E D02618 Butobarbital (BAN)
E D01740 Barbital (JP18/INN)
E D00698 Aprobarbital (INN)
E D00430 Secobarbital (USP/INN)
E D01310 Secobarbital sodium (JAN/USP) <JP>
E D06887 Talbutal (INN)
E D00329 Flurazepam (JAN/INN)
E D00695 Flurazepam hydrochloride (USP)
E D01408 Flurazepam hydrochloride (JP18) <JP>
E D00531 Nitrazepam (JP18/USAN/INN) <JP>
E D01230 Flunitrazepam (JP18/USAN/INN) <JP>
E D00311 Estazolam (JP18/USP/INN) <JP/US>
E D00387 Triazolam (JP18/USP/INN) <JP/US>
E D01657 Lormetazepam (JAN/USAN/INN) <JP>
E D00370 Temazepam (USP/INN) <US>
E D00550 Midazolam (JAN/USP/INN) <JP/US>
E D00696 Midazolam hydrochloride (USAN) <US>
E D05028 Midazolam maleate (USAN)
E D01744 Brotizolam (JP18/USAN/INN) <JP>
E D00457 Quazepam (JAN/USP/INN) <JP/US>
E D07326 Loprazolam (INN)
E D08145 Loprazolam mesilate
E D07328 Cinolazepam (INN)
E D11788 Remimazolam (USAN/INN)
E D10194 Remimazolam besylate (USAN) <JP/US>
E D01593 Nimetazepam (JAN/INN)
E D00532 Glutethimide (JAN/INN)
E D01372 Zopiclone (JP18/INN) <JP>
E D08690 Zolpidem (INN)
E D00706 Zolpidem tartrate (JP18/USP) <JP/US>
E D02624 Eszopiclone (JAN/USP/INN) <JP/US>
E D11149 Brexanolone (USAN/INN) <US>
E D00697 Flumazenil (JAN/USP/INN) <JP/US>
E D00699 Butabarbital sodium (USP)
E D00713 Thiamylal sodium (JP18) <JP>
E D01278 Oxazolam (JP18/INN) <JP>
E D01279 Flutoprazepam (JP18/INN) <JP>
E D01286 Flutazolam (JAN/INN) <JP>
E D01564 Rilmazafone hydrochloride hydrate (JP18) <JP>
E D01758 Haloxazolam (JP18/INN) <JP>
E D02283 Iomazenil (123I) (JAN/INN) <JP>
E D02594 Abecarnil (INN)
E D02616 Pagoclone (USAN/INN)
E D02617 Ocinaplon (USAN/INN)
E D02640 Indiplon (USAN/INN)
E D02833 Alpidem (USAN/INN)
E D03155 Bretazenil (USAN/INN)
E D03180 Butabarbital (USP)
E D03737 Dextofisopam (USAN/INN)
E D04282 Gaboxadol (USAN/INN)
E D04721 Levotofisopam (USAN/INN)
E D05346 Panadiplon (USAN/INN)
E D05378 Pazinaclone (USAN/INN)
E D05980 Suritozole (USAN/INN)
E D06106 Thiamylal
E D07784 Delorazepam (INN)
E D08481 Rilmazafone (INN)
E D08507 Sarmazenil (INN)
E D08840 Adipiplon (USAN)
E D12146 Darigabat (USAN)
E D12449 Cipepofol (USAN)
D GABRA1 [HSA:2554] [KO:K05175]
E D04985 Methohexital (USP/INN)
E D00712 Methohexital sodium (USP) <US>
E D00548 Etomidate (USP/INN) <US>
E D05621 Progabide (USAN/INN)
E D01150 Methyprylon (JAN/INN)
E D00530 Zaleplon (JAN/USP/INN) <US>
E D07330 Clomethiazole (INN)
E D07725 Clomethiazole edisilate
D GABRA5 [HSA:2558] [KO:K05175]
E D12382 Alogabat (USAN)
C Glycine
D GLRA1 [HSA:2741] [KO:K05193]
E D10470 Strychnine nitrate
C Glutamate (ionotropic), non-NMDA
D GRIA [HSA:2890 2891 2892 2893] [KO:K05197 K05198 K05199 K05200]
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D08964 Perampanel (USAN)
E D10780 Perampanel hydrate (JAN) <JP/US>
E D00775 Riluzole (JAN/USP/INN) <JP/US>
E D02696 Talampanel (INN)
E D04131 Farampator (USAN/INN)
E D06656 Tezampanel (USAN)
E D09035 Zonampanel (INN/USAN)
E D09931 Mibampator (USAN/INN)
E D10107 Dasolampanel (USAN)
E D10108 Dasolampanel etibutil (USAN)
E D10109 Dasolampanel etibutil tosylate (USAN)
E D11414 Troriluzole (USAN)
E D11415 Troriluzole hydrochloride (USAN)
E D12239 Pesampator (USAN)
D GRIK [HSA:2897 2898 2899 2900 2901] [KO:K05201 K05202 K05203 K05204 K05205]
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00775 Riluzole (JAN/USP/INN) <JP/US>
E D06656 Tezampanel (USAN)
E D10107 Dasolampanel (USAN)
E D10108 Dasolampanel etibutil (USAN)
E D10109 Dasolampanel etibutil tosylate (USAN)
E D11414 Troriluzole (USAN)
E D11415 Troriluzole hydrochloride (USAN)
C Glutamate (ionotropic), NMDA
D GRIN (NMDAR) [HSA:2902 2903 2904 2905 2906 116443 116444] [KO:K05208 K05209 K05210 K05211 K05212 K05213 K05214]
E D00774 Orphenadrine citrate (USP) <US>
E D00536 Felbamate (USPINN) <US>
E D02599 Orphenadrine hydrochloride
E D08305 Orphenadrine (INN)
D GRIN (NMDAR) [HSA:2902 2903 2904 2905 2906] [KO:K05208 K05209 K05210 K05211 K05212]
E D08098 Ketamine (INN)
E D00711 Ketamine hydrochloride (JP18/USP) <JP/US>
E D07283 Esketamine (USAN/INN)
E D10627 Esketamine hydrochloride (JAN/USAN) <US>
E D07441 Amantadine (INN)
E D00777 Amantadine hydrochloride (JP18/USP) <JP/US>
E D07306 Budipine (INN)
E D07589 Budipine hydrochloride
E D08174 Memantine (INN)
E D04905 Memantine hydrochloride (JAN/USP) <JP/US>
E D07058 Acamprosate (INN)
E D02780 Acamprosate calcium (JAN/USAN) <JP/US>
E D08195 Methadone (BAN)
E D02102 Methadone hydrochloride (JAN/USP) <JP/US>
E D08121 Levomethadone (INN)
E D08122 Levomethadone hydrochloride
E D00775 Riluzole (JAN/USP/INN) <JP/US>
E D03742 Dextromethorphan (USP)
E D00848 Dextromethorphan hydrobromide (USP) <JP>
E D03744 Dextromethorphan polistirex (USAN)
E D02410 Selfotel (USAN/INN)
E D02973 Aptiganel hydrochloride (USAN)
E D03679 Delucemine hydrochloride (USAN)
E D03746 Dextrorphan hydrochloride (USAN)
E D03878 Dizocilpine maleate (USAN)
E D04308 Gavestinel (USAN/INN)
E D04728 Licostinel (USAN/INN)
E D05447 Perzinfotel (USAN/INN)
E D05453 Phencyclidine hydrochloride (USAN)
E D05714 Remacemide hydrochloride (USAN)
E D06146 Tiletamine hydrochloride (USP)
E D08596 Tiletamine (INN)
E D09917 Latrepirdine (USAN/INN)
E D09918 Latrepirdine dihydrochloride (USAN)
E D11299 Apimostinel (USAN)
E D11414 Troriluzole (USAN)
E D11415 Troriluzole hydrochloride (USAN)
E D12214 Esmethadone (USAN)
E D12215 Esmethadone hydrochloride (USAN)
E D12553 Nevadistinel (USAN)
E D12554 Risevistinel (USAN)
D GRIN2B (NMDAR2B) [HSA:2904] [KO:K05210]
E D03100 Besonprodil (USAN)
E D05145 Neramexane mesylate (USAN)
E D06204 Traxoprodil mesylate (USAN)
E D11340 Rislenemdaz (USAN)
C Epithelial sodium channel (SCNN)
D SCNN1 [HSA:6337 6338 6339 6340] [KO:K04824 K04825 K04826 K04827]
E D12346 Idrevloride (USAN)
D SCNN1 [HSA:6337 6338 6340] [KO:K04824 K04825 K04827]
E D07447 Amiloride (INN)
E D00649 Amiloride hydrochloride (USP) <US>
E D00386 Triamterene (JP18/USP/INN) <JP/US>
C ATP-gated cation channel (P2X)
D P2RX3 [HSA:5024] [KO:K05217]
E D11349 Gefapixant (USAN/INN)
E D11693 Gefapixant citrate (JAN/USAN) <JP>
E D12323 Eliapixant (USAN/INN)
E D12355 Sivopixant (JAN/INN)
D P2RX7 [HSA:5027] [KO:K05220]
E D10799 Brilliant blue G (JAN) <US>
D P2RY2 [HSA:5029] [KO:K04269]
E D03685 Denufosol tetrasodium (USAN)
E D03864 Diquafosol tetrasodium (USAN) <JP>
B Voltage-gated ion channels
C Sodium channels
D SCN1A [HSA:6323] [KO:K04833]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN2A [HSA:6326] [KO:K04834]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN3A [HSA:6328] [KO:K04836]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D07299 Lacosamide (JAN/USAN/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN4A [HSA:6329] [KO:K04837]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN5A [HSA:6331] [KO:K04838]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D05077 Moricizine (USAN)
E D02087 Moricizine hydrochloride (USP)
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D06665 Vernakalant hydrochloride (USAN)
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN8A [HSA:6334] [KO:K04840]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN9A [HSA:6335] [KO:K04841]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D07299 Lacosamide (JAN/USAN/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
E D11156 Funapide (USAN/INN)
E D11179 Vixotrigine (USAN/INN)
E D11180 Vixotrigine hydrochloride (USAN)
D SCN10A [HSA:6336] [KO:K04842]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D04095 Etidocaine (USAN/INN)
E D00737 Etidocaine hydrochloride
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D07299 Lacosamide (JAN/USAN/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
D SCN11A [HSA:11280] [KO:K04843]
E D08458 Quinidine (BAN)
E D00642 Quinidine gluconate (USP) <US>
E D00643 Quinidine polygalacturonate
E D02272 Quinidine sulfate (USP) <JP/US>
E D08459 Quinidine phenylethylbarbiturate
E D08421 Procainamide (INN)
E D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
E D00303 Disopyramide (JP18/USAN/INN) <JP>
E D00637 Disopyramide phosphate (JAN/USP) <JP/US>
E D01041 Sparteine (INN)
E D02239 Sparteine sulfate (JAN/USAN)
E D00199 Ajmaline (JP18)
E D04774 Lorajmine hydrochloride (USAN)
E D00358 Lidocaine (JP18/USP/INN) <JP/US>
E D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
E D08127 Lidocaine hydrochloride monohydrate <JP/US>
E D08215 Mexiletine (INN)
E D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
E D06172 Tocainide (USAN/INN)
E D02088 Tocainide hydrochloride (USP)
E D02969 Aprindine (USAN/INN)
E D01326 Aprindine hydrochloride (JP18/USAN) <JP>
E D08435 Propafenone (INN)
E D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
E D07962 Flecainide (INN)
E D00638 Flecainide acetate (JP18/USP) <JP/US>
E D07894 Encainide (INN)
E D03991 Encainide hydrochloride (USAN)
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03492 Cifenline (USAN)
E D01455 Cifenline succinate (USAN) <JP>
E D00551 Tetracaine (USP/INN)
E D00741 Tetracaine hydrochloride (JP18/USP) <JP/US>
E D00552 Benzocaine (USP/INN) <JP>
E D00733 Dibucaine (USP)
E D02220 Dibucaine hydrochloride (JP18/USP)
E D08422 Procaine (INN)
E D00740 Procaine hydrochloride (JP18/USP) <JP>
E D01152 Oxethazaine (JP18/USAN) <JP>
E D08311 Oxetacaine hydrochloride
E D08407 Pramocaine (INN)
E D00739 Pramoxine hydrochloride (USP)
E D02456 Aminobenzoic acid (USP)
E D02906 Aminobenzoate potassium (USP)
E D02907 Aminobenzoate sodium (USP)
E D08319 Oxybuprocaine (INN)
E D01768 Benoxinate hydrochloride (USP) <JP>
E D07678 Chloroprocaine (INN)
E D00732 Chloroprocaine hydrochloride (USP) <US>
E D07552 Bupivacaine (USAN/INN) <US>
E D01450 Bupivacaine hydrochloride (USP) <JP/US>
E D08181 Mepivacaine (INN)
E D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
E D00553 Prilocaine (USP/INN)
E D01243 Prilocaine hydrochloride (USP) <US>
E D07468 Articaine (INN)
E D02991 Articaine hydrochloride (JAN/USP)
E D08490 Ropivacaine (INN)
E D04048 Ropivacaine hydrochloride (USP) <JP/US>
E D08116 Levobupivacaine (INN)
E D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00512 Phenytoin (JP18/USP/INN) <JP/US>
E D02103 Phenytoin sodium (USP) <JP/US>
E D00375 Mephenytoin (USP/INN)
E D07993 Fosphenytoin (INN)
E D02096 Fosphenytoin sodium (USP) <US>
E D07595 Fosphenytoin sodium hydrate (JAN) <JP>
E D00252 Carbamazepine (JP18/USP/INN) <JP/US>
E D00533 Oxcarbazepine (JAN/USP/INN) <US>
E D05775 Rufinamide (JAN/USP/INN) <JP/US>
E D09215 Eslicarbazepine (USAN/INN)
E D09612 Eslicarbazepine acetate (USAN) <US>
E D00354 Lamotrigine (JAN/USP/INN) <JP/US>
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D11150 Cenobamate (USAN/INN) <US>
E D08448 Proxymetacaine (INN)
E D02098 Proparacaine hydrochloride (USP) <US>
E D01519 Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
E D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
E D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
E D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
E D02762 Actisomide (USAN/INN)
E D04521 Indecainide hydrochloride (USAN)
E D05708 Recainam hydrochloride (USAN)
E D05709 Recainam tosylate (USAN)
E D06203 Transcainide (USAN/INN)
E D06517 Pirmenol hydrochloride (USAN)
E D08377 Pilsicainide (INN)
E D08394 Pirmenol (INN)
E D09833 Levosemotiadil fumarate (JAN)
E D11155 Eleclazine (USAN/INN)
C Calcium channels
D CACNA1-T [HSA:8911 8912 8913] [KO:K04856 K04855 K04854]
E D08217 Mibefradil (INN)
E D05024 Mibefradil dihydrochloride (USAN)
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D00539 Ethosuximide (JP18/USP/INN) <JP/US>
E D00404 Methsuximide (USP) <US>
E D00399 Valproic acid (USP) <US>
E D00304 Divalproex sodium (USP) <US>
E D00710 Valproate sodium (USAN) <JP/US>
E D08667 Calcium valproate
E D00538 Zonisamide (JP18/USP/INN) <JP/US>
E D02630 Penfluridol (USAN/INN)
E D07971 Flunarizine (INN)
E D01303 Flunarizine hydrochloride (JAN/USAN)
E D02633 Lomerizine hydrochloride (JAN) <JP>
E D12061 Suvecaltamide (USAN)
E D12062 Suvecaltamide hydrocloride (USAN)
D CACNA1B [HSA:774] [KO:K04849]
E D01173 Cilnidipine (JP18/INN) <JP>
E D06363 Ziconotide (USAN/INN)
E D08686 Ziconotide acetate <US>
D CACNA1-L [HSA:775 776 778 779] [KO:K04850 K04851 K04853 K04857]
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D07845 Diltiazem (INN)
E D00616 Diltiazem hydrochloride (JP18/USP) <JP/US>
E D03830 Diltiazem malate (USAN)
E D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
E D07450 Amlodipine (USP/INN)
E D00615 Amlodipine besylate (USP) <JP/US>
E D02914 Amlodipine maleate (USAN)
E D11881 Amlodipine benzoate <US>
E D00319 Felodipine (JP18/USP/INN) <JP/US>
E D00349 Isradipine (USP/INN) <US>
E D08270 Nicardipine (INN)
E D00617 Nicardipine hydrochloride (JP18/USAN) <JP/US>
E D00437 Nifedipine (JP18/USP/INN) <JP/US>
E D00438 Nimodipine (USP/INN) <US>
E D00618 Nisoldipine (JAN/USAN/INN) <US>
E D00629 Nitrendipine (JP18/USAN/INN) <JP>
E D04657 Lacidipine (USAN/INN)
E D01908 Nilvadipine (JP18/USAN/INN) <JP>
E D08155 Manidipine (INN)
E D01553 Manidipine hydrochloride (JP18) <JP>
E D07494 Barnidipine (INN)
E D01104 Barnidipine hydrochloride (JAN) <JP>
E D08111 Lercanidipine (INN)
E D01849 Lercanidipine hydrochloride (JAN/USAN)
E D01173 Cilnidipine (JP18/INN) <JP>
E D07509 Benidipine (INN)
E D02045 Benidipine hydrochloride (JP18) <JP>
E D08892 Clevidipine (USAN/INN) <US>
E D08941 Levamlodipine malate (USAN)
E D11723 Levamlodipine maleate (USAN) <US>
E D08217 Mibefradil (INN)
E D05024 Mibefradil dihydrochloride (USAN)
E D02356 Verapamil (USAN/INN)
E D00619 Verapamil hydrochloride (JP18/USP) <JP/US>
E D08009 Gallopamil (INN)
E D01969 Gallopamil hydrochloride (JAN)
E D07185 Fendiline (INN)
E D07943 Fendiline hydrochloride
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D08340 Perhexiline (INN)
E D05442 Perhexiline maleate (USAN)
E D08441 Propiverine (INN)
E D01007 Propiverine hydrochloride (JP18) <JP>
E D00495 Paramethadione (INN)
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D01145 Azelnidipine (JP18/INN) <JP>
E D01151 Lemildipine (JAN/INN)
E D01171 Monatepil maleate (JAN/USAN)
E D01562 Aranidipine (JAN/INN) <JP>
E D01604 Efonidipine hydrochloride ethanolate (JAN) <JP>
E D01933 Vatanidipine hydrochloride (JAN)
E D03067 Belfosdil (USAN/INN)
E D03536 Clentiazem maleate (JAN/USAN)
E D03655 Darodipine (USAN/INN)
E D04193 Flordipine (USAN/INN)
E D04260 Fostedil (USAN/INN)
E D06129 Tiapamil hydrochloride (USAN)
E D07886 Efonidipine (INN)
E D09789 Kirenidipine hydrochloride (JAN)
E D09833 Levosemotiadil fumarate (JAN)
E D10932 Etripamil (USAN/INN)
E D11102 Tamolarizine hydrochloride (JAN)
D CACNA1S [HSA:779] [KO:K04857]
E D07094 Pinaverium bromide (INN)
D CACNA2D [HSA:781 9254 55799 93589] [KO:K04858 K04859 K04860 K04861]
E D00332 Gabapentin (JAN/USP/INN) <JP/US>
E D09539 Gabapentin enacarbil (JAN/USAN/INN) <JP/US>
E D02716 Pregabalin (JAN/USAN/INN) <JP/US>
D CACNA2D1 [HSA:781] [KO:K04858]
E D11203 Mirogabalin (USAN/INN)
E D10790 Mirogabalin besylate (USAN) <JP>
D CACNA2D2 [HSA:9254] [KO:K04859]
E D11203 Mirogabalin (USAN/INN)
E D10790 Mirogabalin besylate (USAN) <JP>
C Potassium channels
D KCNA [HSA:3736 3737 3738 3739 3741 3742 3743 3744] [KO:K04874 K04875 K04876 K04877 K04878 K04879 K04880 K04881]
E D10228 Amifampridine (USAN/INN)
E D10689 Amifampridine phosphate (JAN/USAN) <US>
E D04127 Dalfampridine (USAN) <US>
D KCNA1 [HSA:3736] [KO:K04874]
E D06652 Tedisamil (USAN)
E D06653 Tedisamil sesquifumarate (USAN)
D KCNA5 [HSA:3741] [KO:K04878]
E D06665 Vernakalant hydrochloride (USAN)
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
D KCNB [HSA:3745 9312] [KO:K04885 K04886]
E D10228 Amifampridine (USAN/INN)
E D10689 Amifampridine phosphate (JAN/USAN) <US>
E D04127 Dalfampridine (USAN) <US>
D KCNC [HSA:3746 3747 3748 3749] [KO:K04887 K04888 K04889 K04890]
E D10228 Amifampridine (USAN/INN)
E D10689 Amifampridine phosphate (JAN/USAN) <US>
E D04127 Dalfampridine (USAN) <US>
D KCND [HSA:3750 3751 3752] [KO:K04891 K04892 K04893]
E D10228 Amifampridine (USAN/INN)
E D10689 Amifampridine phosphate (JAN/USAN) <US>
E D04127 Dalfampridine (USAN) <US>
E D00730 Butamben (USP)
E D03547 Clofilium phosphate (USAN/INN)
D KCND3 [HSA:3752] [KO:K04893]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D06665 Vernakalant hydrochloride (USAN)
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D01856 Nifekalant hydrochloride (JAN) <JP>
D KCNH1 [HSA:3756] [KO:K04904]
E D03547 Clofilium phosphate (USAN/INN)
D KCNH2 [HSA:3757] [KO:K04905]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D00647 Dofetilide (JAN/USP/INN) <US>
E D08060 Ibutilide (INN)
E D00648 Ibutilide fumarate (USP) <US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D08525 Sotalol (INN)
E D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D00521 Terfenadine (JAN/USAN/INN)
E D01856 Nifekalant hydrochloride (JAN) <JP>
E D03037 Azimilide dihydrochloride (USAN)
E D03547 Clofilium phosphate (USAN/INN)
E D03732 Dexsotalol hydrochloride (USAN)
E D04955 Sematilide hydrochloride (USAN)
E D06206 Trecetilide fumarate (USAN)
E D09757 Terikalant (INN)
E D09758 Ambasilide (INN)
E D09759 Trecetilide (INN)
D KCNQ [HSA:3784 3785 3786 9132 56479] [KO:K04926 K04927 K04928 K04929 K04930]
E D09569 Ezogabine (USAN)
E D04192 Flindokalner (USAN/INN)
D KCNQ1 [HSA:3784] [KO:K04926]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D03037 Azimilide dihydrochloride (USAN)
E D09757 Terikalant (INN)
E D09758 Ambasilide (INN)
D KCNMB1 [HSA:3779] [KO:K04937]
E D04192 Flindokalner (USAN/INN)
D KCNN4 [HSA:3783] [KO:K04945]
E D06640 Senicapoc (USAN)
D KCNT2 (SLICK) [HSA:343450] [KO:K04947]
E D03547 Clofilium phosphate (USAN/INN)
C Inward rectifier channels (Kir)
D KCNJ1 [HSA:3758] [KO:K04995]
E D01603 Bethanidine sulfate (JAN/USAN)
D KCNJ3 [HSA:3760] [KO:K04997]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
D KCNJ5 [HSA:3762] [KO:K04999]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D02537 Dronedarone (INN)
E D03914 Dronedarone hydrochloride (USP) <US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
D KCNJ8 [HSA:3764] [KO:K05001]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
D KCNJ11 [HSA:3767] [KO:K05004]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D03914 Dronedarone hydrochloride (USP) <US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
D KCNJ12 [HSA:3768] [KO:K05005]
E D02910 Amiodarone (USAN/INN)
E D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D01856 Nifekalant hydrochloride (JAN) <JP>
E D09757 Terikalant (INN)
C Ryanodine receptors (RYR)
D RYR [HSA:6261 6262 6263] [KO:K04961 K04962 K04963]
E D10304 Aladorian (USAN/INN)
E D10305 Aladorian sodium (USAN)
C Transient receptor potential channels
D TRPA1 [HSA:8989] [KO:K04984]
E D00064 l-Menthol (JP18) <JP>
E D04849 dl-Menthol (JP18)
E D04918 Menthol (USP)
D TRPC5 [HSA:7224] [KO:K04968]
E D01705 Clemizole hydrochloride (JAN)
E D02013 Clemizole undecylate (JAN)
D TRPM8 [HSA:79054] [KO:K04983]
E D00064 l-Menthol (JP18) <JP>
E D04849 dl-Menthol (JP18)
E D04918 Menthol (USP)
D TRPV1 [HSA:7442] [KO:K05222]
E D00250 Capsaicin (JAN/USP) <US>
E D06388 Zucapsaicin (USAN/INN)
E D05249 Olvanil (USAN)
E D08282 Nonivamide (INN)
E D10370 Mavatrep (USAN)
B Other ion channels
C Chloride channel
D CLCN2 [HSA:1181] [KO:K05011]
E D04790 Lubiprostone (JAN/USAN/INN) <JP/US>
D CLCA [HSA:1179 9635 22802] [KO:K05027 K05028 K05030]
E D03605 Crofelemer (USAN) <US>
E D08275 Niflumic acid (INN)
C Hyperpolarization-activated ion channel
D HCN [HSA:348980 610 57657 10021] [KO:K04954 K04955 K04956 K04957]
E D07165 Ivabradine (USAN/INN)
E D08095 Ivabradine hydrochloride (JAN/USAN) <JP/US>
#
ANuclear receptors
B Thyroid hormone like receptors
C Thyroid hormone receptor (THR)
D NR1A (THR) [HSA:7067 7068] [KO:K05547 K08362]
E D03750 Dextrothyroxine sodium (USAN)
E D07214 Tiratricol (INN)
E D11113 Levothyroxine sodium (INN) <US>
E D01010 Levothyroxine sodium (USP) <JP/US>
E D01011 Liothyronine sodium (JP18/USP) <JP/US>
E D01012 Dried thyroid (JP18)
E D06482 Thyroid (USP)
E D08125 Levothyroxine (BAN)
E D08128 Liothyronine (INN)
E D08129 Liothyronine hydrochloride
D NR1A2 (THRB) [HSA:7068] [KO:K08362]
E D09381 Sobetirome (USAN)
E D11602 Resmetirom (USAN/INN)
C Retinoic acid receptor (RAR)
D NR1B (RAR) [HSA:5914 5915 5916] [KO:K08527 K08528 K08529]
E D06543 Vitamin A (USP) <JP>
E D00164 Retinol palmitate (JP18) <JP/US>
E D01621 Retinol acetate (JP18)
E D08477 Retinol propionate
E D01132 Tazarotene (JAN/USAN/INN) <US>
E D00316 Etretinate (JAN/USAN/INN) <JP>
E D02754 Acitretin (USP/INN) <US>
E D00094 Tretinoin (JAN/USP/INN) <JP/US>
E D01516 Tretinoin tocoferil (JAN) <JP>
E D00348 Isotretinoin (JAN/USP) <US>
E D04636 Isotretinoin anisatil (USAN)
E D02815 Alitretinoin (USAN) <US>
E D04162 Fenretinide (USAN/INN)
D NR1B1 (RARA) [HSA:5914] [KO:K08527]
E D01418 Tamibarotene (JAN/USAN/INN) <JP>
D NR1B2 (RARB) [HSA:5915] [KO:K08528]
E D01112 Adapalene (JAN/USP/INN) <JP/US>
D NR1B3 (RARG) [HSA:5916] [KO:K08529]
E D01112 Adapalene (JAN/USP/INN) <JP/US>
E D11225 Trifarotene (USAN/INN) <US>
E D09365 Palovarotene (JAN/USAN/INN)
D PML-RARA [HSA:5371 5914] [KO:K10054 K08527]
E D00094 Tretinoin (JAN/USP/INN) <JP/US>
E D02106 Arsenic trioxide (JP18/USAN) <JP/US>
C Peroxisome proliferator-activated receptor (PPAR)
D NR1C (PPAR) [HSA:5465 5467 5468] [KO:K07294 K04504 K08530]
E D06647 Sodelglitazar (USAN)
E D09350 Indeglitazar (USAN)
D NR1C1 (PPARA) [HSA:5465] [KO:K07294]
E D12484 Carfloglitazar (INN)
E D00279 Clofibrate (JP18/USP/INN) <JP>
E D01208 Aluminum clofibrate (JAN/INN)
E D07724 Magnesium clofibrate (INN)
E D01366 Bezafibrate (JP18/USAN/INN) <JP>
E D00334 Gemfibrozil (JAN/USP/INN) <US>
E D00565 Fenofibrate (JP18/USP/INN) <JP/US>
E D03521 Ciprofibrate (USAN/INN)
E D07187 Etofibrate (INN)
E D08890 Choline fenofibrate (USAN/INN) <US>
E D01274 Tesaglitazar (JAN/USAN/INN)
E D05091 Muraglitazar (USAN/INN)
E D05397 Peliglitazar (USAN)
E D06102 Theofibrate (USAN)
E D08845 Aleglitazar (USAN)
E D08949 Naveglitazar (USAN/INN)
E D10711 Pemafibrate (JAN) <JP>
E D11208 Elafibranor (USAN)
E D11579 Fenofibric acid <US>
D NR1C3 (PPARG) [HSA:5468] [KO:K08530]
E D00395 Troglitazone (JAN/USAN/INN)
E D08491 Rosiglitazone (INN)
E D00596 Rosiglitazone maleate (JAN/USP)
E D08378 Pioglitazone (INN)
E D00945 Pioglitazone hydrochloride (JP18/USP) <JP/US>
E D11923 Lobeglitazone (INN)
E D12484 Carfloglitazar (INN)
E D01274 Tesaglitazar (JAN/USAN/INN)
E D01971 Reglitazar (JAN/INN)
E D03493 Ciglitazone (USAN/INN)
E D03653 Darglitazone sodium (USAN)
E D03941 Edaglitazone sodium (USAN)
E D03996 Englitazone sodium (USAN)
E D04132 Farglitazar (USAN/INN)
E D04411 Halofenate (USAN/INN)
E D05030 Mifobate (USAN/INN)
E D05091 Muraglitazar (USAN/INN)
E D05150 Netoglitazone (USAN/INN)
E D05397 Peliglitazar (USAN)
E D05739 Rivoglitazone (USAN/INN)
E D08845 Aleglitazar (USAN)
E D09579 Arhalofenate (USAN/INN)
E D11256 Seladelpar (USAN/INN)
E D11257 Seladelpar lysine (USAN)
E D11603 Leriglitazone (USAN/INN)
E D11604 Leriglitazone hydrochloride (USAN)
E D12242 Bocidelpar (USAN)
E D12243 Bocidelpar sulfate (USAN)
C RAR-related orphan receptor
D NR1F3 (RORC) [HSA:6097] [KO:K08534]
E D12274 Cedirogant (USAN/INN)
C Liver X receptor like receptor
D NR1H2 (LXRB) [HSA:7376] [KO:K08535]
E D12298 Abequolixron (USAN)
E D12299 Abequolixron zinc (USAN)
D NR1H3 (LXRA) [HSA:10062] [KO:K08536]
E D12298 Abequolixron (USAN)
E D12299 Abequolixron zinc (USAN)
D NR1H4 (FXR) [HSA:9971] [KO:K08537]
E D00163 Chenodiol (USAN) <JP/US>
E D00734 Ursodiol (USP) <JP/US>
E D10699 Cholic acid (JAN/USAN) <US>
E D09360 Obeticholic acid (JAN/USAN/INN) <US>
E D08277 Turofexorate isopropyl (USAN/INN)
E D11548 Tropifexor (USAN)
C Vitamin D3 like receptor
D NR1I1 (VDR) [HSA:7421] [KO:K08539]
E D00187 Ergocalciferol (JP18/USP) <US>
E D00299 Dihydrotachysterol (JAN/USP/INN)
E D01518 Alfacalcidol (JAN/INN) <JP>
E D00129 Calcitriol (JAN/USP/INN) <JP/US>
E D00188 Cholecalciferol (JP18/USP)
E D00122 Calcifediol (USP/INN) <US>
E D01125 Calcipotriene (USP) <JP/US>
E D10198 Calcipotriol hydrate (JAN) <US>
E D08554 Tacalcitol (INN)
E D01472 Tacalcitol hydrate (JP18) <JP>
E D00930 Paricalcitol (JAN/USP/INN) <US>
E D01009 Doxercalciferol (USAN/INN) <US>
E D00628 Secalciferol (JAN/USAN/INN)
E D01098 Maxacalcitol (JAN/USAN/INN) <JP>
E D01662 Falecalcitriol (JAN/INN) <JP>
E D03930 Ecalcidene (USAN/INN)
E D07578 Eldecalcitol (JAN/INN) <JP>
E D08868 Becocalcidiol (USAN/INN)
E D10565 Pefcalcitol (JAN/USAN/INN)
B Hepatocyte nuclear factor 4 like receptors
C Retinoid X receptor (RXR)
D NR2B (RXR) [HSA:6256 6257 6258] [KO:K08524 K08525 K08526]
E D00316 Etretinate (JAN/USAN/INN) <JP>
E D02754 Acitretin (USP/INN) <US>
E D02815 Alitretinoin (USAN) <US>
E D03106 Bexarotene (JAN/USAN/INN) <JP/US>
D NR2B2 (RXRB) [HSA:6257] [KO:K08525]
E D01132 Tazarotene (JAN/USAN/INN) <US>
E D01112 Adapalene (JAN/USP/INN) <JP/US>
D NR2B3 (RXRG) [HSA:6258] [KO:K08526]
E D01112 Adapalene (JAN/USP/INN) <JP/US>
B Estrogen like receptors
C Estrogen receptor
D NR3A (ESR) [HSA:2099 2100] [KO:K08550 K08551]
E D08409 Prasterone (USAN/INN) <US>
E D01616 Sodium prasterone sulfate hydrate (JP18)
E D00105 Estradiol (JAN/USP/INN) <JP/US>
E D01413 Estradiol valerate (JAN/USP/INN) <JP/US>
E D01617 Estradiol dipropionate (JAN)
E D01953 Estradiol benzoate (JP18/USP)
E D04061 Estradiol acetate (USAN) <US>
E D04063 Estradiol cypionate (USP) <US>
E D04064 Estradiol enanthate (USAN)
E D04065 Estradiol undecylate (USAN/INN)
E D07918 Estradiol hemihydrate <US>
E D07919 Estradiol 17 beta-hemisuccinate
E D00185 Estriol (JP18/USP) <JP>
E D01986 Estriol tripropionate (JAN)
E D01989 Estriol diacetate benzoate (JAN)
E D07920 Estriol succinate
E D07921 Estriol sodium succinate (BAN)
E D00269 Chlorotrianisene (INN)
E D00067 Estrone (JAN/USP/INN)
E D00312 Estrone sodium sulfate
E D00948 Estropipate (USP)
E D07221 Promestriene (INN)
E D00898 Dienestrol (USP/INN)
E D00577 Diethylstilbestrol (USP/INN)
E D00946 Diethylstilbestrol diphosphate (USP)
E D07826 Hexestrol diphosphate sodium
E D07726 Clomifene (INN)
E D00962 Clomiphene citrate (USP) <JP/US>
E D08465 Raloxifene (INN)
E D02217 Raloxifene hydrochloride (JAN/USP) <JP/US>
E D10606 Raloxifene hydrochloride hydrate (JAN) <JP>
E D03062 Bazedoxifene acetate (JAN/USAN) <JP>
E D04672 Lasofoxifene tartrate (JAN/USAN)
E D08301 Ormeloxifene (INN)
E D08559 Tamoxifen (INN)
E D00966 Tamoxifen citrate (JP18/USP) <JP/US>
E D08620 Toremifene (INN)
E D00967 Toremifene citrate (JAN/USAN) <JP/US>
E D01161 Fulvestrant (JAN/USP/INN) <JP/US>
E D11829 Fluoroestradiol F18 <US>
E D00575 Mestranol (JP18/USP/INN)
E D01265 Epitiostanol (JAN/INN)
E D01602 Mepitiostane (JP18/INN) <JP>
E D01641 Hexestrol (JAN/INN)
E D01853 Miproxifene phosphate (JAN)
E D02018 Hexestrol diacetate (JAN)
E D02758 Acolbifene hydrochloride (USAN)
E D02993 Arzoxifene hydrochloride (USAN)
E D03551 Clometherone (USAN/INN)
E D03911 Droloxifene (USAN/INN)
E D03912 Droloxifene citrate (USAN)
E D04041 Equilin (USP)
E D04071 Estrogens, esterified (USP) <US>
E D04496 Idoxifene (USAN/INN)
E D05106 Nafoxidine hydrochloride (USAN)
E D05192 Nitromifene citrate (USAN)
E D06245 Trioxifene mesylate (USAN)
E D06551 Afimoxifene (USAN/INN)
E D07121 Alfatradiol (INN)
E D07783 Delmadinone (INN)
E D08910 Enclomiphene (USAN)
E D09834 Levormeloxifene fumarate (JAN)
E D10008 Fispemifene (USAN/INN)
E D10876 Enclomiphene citrate (USAN)
E D11264 Brilanestrant (USAN/INN)
E D11513 Estetrol (USAN)
E D11514 Estetrol (JAN/USAN)
D NR3A1 (ESR1) [HSA:2099] [KO:K08550]
E D04104 Etonogestrel (USAN/INN) <US>
E D02367 Desogestrel (USAN/INN)
E D00554 Ethinyl estradiol (USP) <JP>
E D07928 Ethinylestradiol propanesulfonate
E D01639 Tibolone (JAN/USAN/INN)
E D07939 Etynodiol (INN)
E D01294 Ethynodiol diacetate (JAN/USP)
E D00289 Danazol (JP18/USP/INN) <JP/US>
E D08958 Ospemifene (INN/USAN/BAN) <US>
E D07434 Polyestradiol phosphate (INN)
E D00576 Quinestrol (USAN/INN)
E D11671 Elacestrant (USAN/INN)
E D12049 Camizestrant (USAN)
E D12145 Amcenestrant (JAN/USAN/INN)
D NR3A1* (ESR1) [HSA_VAR:2099v2] [HSA:2099] [KO:K08550]
E D11672 Elacestrant hydrochloride (USAN) <US>
D NR3A2 (ESR2) [HSA:2100] [KO:K08551]
E D06631 Prinaberel (USAN/INN)
E D09899 Erteberel (USAN/INN)
C 3-Ketosteroid receptor
D NR3C1 (GR) [HSA:2908] [KO:K05771]
E D00385 Triamcinolone (JP18/USP/INN) <JP>
E D00983 Triamcinolone acetonide (JP18/USP) <JP/US>
E D00984 Triamcinolone diacetate (JAN/USP)
E D00985 Triamcinolone hexacetonide (USP/INN)
E D06216 Triamcinolone acetonide sodium phosphate (USAN)
E D00292 Dexamethasone (JP18/USP/INN) <JP/US>
E D00975 Dexamethasone sodium phosphate (JAN/USP) <JP/US>
E D01510 Dexamethasone metasulfobenzoate sodium (JAN) <JP>
E D01615 Dexamethasone palmitate (JAN) <JP>
E D01632 Dexamethasone dipropionate (USAN) <JP>
E D01948 Dexamethasone valerate (JAN) <JP>
E D02174 Dexamethasone acetate (JAN/USP)
E D02591 Dexamethasone acefurate (USAN/INN)
E D02592 Dexamethasone beloxil (USAN)
E D07073 Dexamethasone cipecilate (JAN/INN) <JP>
E D07796 Dexamethasone 21-acetate
E D07797 Dexamethasone isonicotinate
E D07798 Dexamethasone sodium hemisulfate
E D07799 Dexamethasone 21-tebutate
E D07800 Dexamethasone 21-valerate
E D07801 Dexamethasone phenylpropionate
E D07802 Dexamethasone phosphate
E D00088 Hydrocortisone (JP18/USP/INN) <JP/US>
E D00165 Hydrocortisone acetate (JP18/USP) <US>
E D00976 Hydrocortisone cypionate
E D00977 Hydrocortisone sodium phosphate (JP18/USP) <JP>
E D00978 Hydrocortisone sodium succinate (JP18/USP) <JP/US>
E D01442 Hydrocortisone succinate (JP18)
E D01619 Hydrocortisone butyrate (JP18/USP) <JP/US>
E D01886 Hydrocortisone probutate (USAN) <JP/US>
E D02288 Hydrocortisone valerate (USP) <US>
E D04467 Hydrocortisone hemisuccinate (USP)
E D06876 Hydrocortisone aceponate (INN)
E D09796 Hydrocortisone caproate (JAN)
E D00472 Prednisolone (JP18/USP/INN) <JP/US>
E D00980 Prednisolone acetate (JP18/USP/INN) <JP/US>
E D00981 Prednisolone sodium phosphate (JP18/USP) <JP/US>
E D00982 Prednisolone tebutate (JAN/USP)
E D01239 Prednisolone sodium succinate (JP18/USP) <JP>
E D01998 Prednisolone farnesylate (JAN)
E D02156 Prednisolone hemisuccinate (USP)
E D03301 Prednisolone valerate acetate (JAN) <JP>
E D08412 Prednisolone pivalate
E D08413 Prednisolone sodium metazoate (USAN)
E D08414 Prednisolone 21-(sodium tetrahydrophthalate)
E D08415 Prednisolone steaglate (BAN)
E D00473 Prednisone (USP) <US>
E D08416 Prednisone acetate
E D00244 Betamethasone (JP18/USP/INN) <JP>
E D00972 Betamethasone sodium phosphate (JP18/USP) <JP>
E D01357 Betamethasone valerate (JP18/USP) <JP/US>
E D01402 Betamethasone acetate (JAN/USP)
E D01637 Betamethasone dipropionate (JP18/USP) <JP/US>
E D02032 Betamethasone butyrate propionate (JAN) <JP>
E D02286 Betamethasone benzoate (USP)
E D08610 Tixocortol (INN)
E D06171 Tixocortol pivalate (USAN)
E D00246 Budesonide (JP18/USP/INN) <JP/US>
E D07495 Beclometasone (INN)
E D00689 Beclomethasone dipropionate (USP) <JP/US>
E D11572 Beclomethasone dipropionate monohydrate <US>
E D01367 Fluorometholone (JP18/USP/INN) <JP/US>
E D04221 Fluorometholone acetate (USP) <US>
E D04218 Fluocortolone (USAN/INN)
E D04219 Fluocortolone caproate (USAN)
E D07973 Fluocortolone 21-pivalate
E D01825 Fluocinolone acetonide (JP18/USP/INN) <JP/US>
E D00325 Fluocinonide (JP18/USP/INN) <JP/US>
E D00407 Methylprednisolone (JP18/USP/INN) <JP/US>
E D00751 Methylprednisolone sodium succinate (JAN/USP) <JP/US>
E D00979 Methylprednisolone acetate (JAN/USP) <JP/US>
E D05000 Methylprednisolone hemisuccinate (USP)
E D05001 Methylprednisolone sodium phosphate (USAN)
E D05002 Methylprednisolone suleptanate (USAN/INN)
E D07203 Methylprednisolone aceponate (INN)
E D07717 Clobetasone (INN)
E D01273 Clobetasone butyrate (JAN/USAN) <JP>
E D04208 Flumethasone (USAN)
E D01464 Flumethasone pivalate (USP)
E D07972 Fluocortin (INN)
E D04217 Fluocortin butyl (USAN)
E D07201 Fluprednidene (INN)
E D07980 Fluprednidene acetate
E D03696 Desonide (USP/INN) <US>
E D07116 Alclometasone (INN)
E D01820 Alclometasone dipropionate (JAN/USP) <JP/US>
E D07719 Clocortolone (INN)
E D02287 Clocortolone pivalate (USP) <US>
E D03541 Clocortolone acetate (USAN)
E D04201 Flucloronide (USAN)
E D03697 Desoximetasone (USP/INN) <US>
E D03812 Diflucortolone (USAN)
E D01764 Diflucortolone valerate (JP18) <JP>
E D03813 Diflucortolone pivalate (USAN)
E D00328 Flurandrenolide (USP) <JP/US>
E D07827 Diflorasone (INN)
E D01327 Diflorasone diacetate (JP18/USP) <JP/US>
E D01387 Amcinonide (JAN/USP/INN) <JP/US>
E D07202 Halometasone (INN)
E D08227 Mometasone (INN)
E D00690 Mometasone furoate (JAN/USP) <JP/US>
E D03325 Mometasone furoate hydrate (JAN) <JP>
E D07981 Fluticasone (INN)
E D01708 Fluticasone propionate (JAN/USP) <JP/US>
E D06315 Fluticasone furoate (JAN/USAN/INN) <JP/US>
E D05601 Prednicarbate (USP/INN) <US>
E D01266 Difluprednate (JAN/USAN/INN) <JP/US>
E D08660 Ulobetasol (INN)
E D04409 Halobetasol propionate (USP) <US>
E D07715 Clobetasol (INN)
E D01272 Clobetasol propionate (JP18/USP) <JP/US>
E D01308 Halcinonide (JAN/USP/INN) <US>
E D00585 Mifepristone (JAN/USAN/INN) <US>
E D07464 Paramethasone (INN)
E D01229 Paramethasone acetate (JAN/USAN)
E D07749 Cortisone (INN)
E D00973 Cortisone acetate (JP18/USP) <JP/US>
E D07230 Prednylidene (INN)
E D05729 Rimexolone (USP/INN)
E D03671 Deflazacort (USAN/INN) <US>
E D03561 Cloprednol (USAN/INN)
E D06673 Meprednisone (USP/INN)
E D03594 Cortivazol (USAN)
E D00324 Flunisolide (JAN/USP) <US>
E D04214 Flunisolide acetate (USAN)
E D01703 Ciclesonide (JAN/USAN/INN) <JP/US>
E D02289 Medrysone (USAN)
E D04244 Formocortal (USAN/INN)
E D08147 Loteprednol (INN)
E D01689 Loteprednol etabonate (JAN/USAN) <US>
E D01434 Deprodone propionate (JAN) <JP>
E D01743 Halopredone acetate (JAN/USAN)
E D03691 Descinolone acetonide (USAN)
E D04227 Fluprednisolone (USAN/INN)
E D04228 Fluprednisolone valerate (USAN)
E D05194 Nivazol (USAN)
E D05603 Prednival (USAN)
E D05719 Resocortol butyrate (USAN)
E D06135 Ticabesone propionate (USAN)
E D06161 Tipredane (USAN)
E D06201 Tralonide (USAN/INN)
E D07814 Dichlorisone (INN)
E D07815 Dichlorisone acetate
E D07975 Flupamesone
E D08036 Halopredone (INN)
E D08429 Proligestone (INN)
E D08476 Resocortol (INN)
E D10136 Mapracorat (USAN)
E D10617 Dagrocorat (USAN/INN)
E D10634 Fosdagrocorat (USAN/INN)
E D11000 Vamorolone (USAN/INN)
E D11336 Relacorilant (USAN)
E D11665 Exicorilant (USAN/INN)
E D11667 Miricorilant (USAN/INN)
E D11937 Velsecorat (USAN/INN)
D NR3C2 (MR) [HSA:4306] [KO:K08555]
E D00443 Spironolactone (JP18/USP/INN) <JP/US>
E D01943 Canrenoate potassium (USAN) <JP>
E D03363 Canrenone (USAN)
E D01115 Eplerenone (JP18/USAN/INN) <JP/US>
E D10633 Finerenone (JAN/USAN/INN) <JP/US>
E D00386 Triamterene (JP18/USP/INN) <JP/US>
E D03917 Drospirenone (JAN/USP/INN) <US>
E D10528 Aldosterone (INN)
E D07967 Fludrocortisone (INN)
E D00986 Fludrocortisone acetate (JP18/USP) <JP/US>
E D07792 Desoxycortone (INN)
E D03698 Desoxycorticosterone acetate (USP)
E D03699 Desoxycorticosterone pivalate (USP)
E D03792 Dicirenone (USAN)
E D05020 Mexrenoate potassium (USAN)
E D05640 Prorenoate potassium (USAN/INN)
E D05912 Spiroxasone (USAN/INN)
E D10892 Esaxerenone (JAN/INN) <JP>
E D11667 Miricorilant (USAN/INN)
D NR3C3 (PGR) [HSA:5241] [KO:K08556]
E D01414 Ethylestrenol (USAN/INN)
E D00182 Norethindrone (USP) <JP/US>
E D00953 Norethindrone acetate (USP) <US>
E D08285 Norethisterone enantate
E D01580 Lynestrenol (JAN/USAN)
E D00950 Levonorgestrel (JAN/USP/INN) <JP/US>
E D05679 Quingestanol acetate (USAN)
E D08167 Megestrol (INN)
E D00952 Megestrol acetate (USP) <US>
E D08166 Medroxyprogesterone (INN)
E D00951 Medroxyprogesterone acetate (JP18/USP) <JP/US>
E D07220 Norgestrienone (INN)
E D04104 Etonogestrel (USAN/INN) <US>
E D02367 Desogestrel (USAN/INN)
E D03917 Drospirenone (JAN/USP/INN) <US>
E D09567 Ulipristal (USAN/INN)
E D09687 Ulipristal acetate (JAN/USAN) <US>
E D01159 Gestonorone caproate (JAN/USAN) <JP>
E D08052 Hydroxyprogesterone (INN)
E D00949 Hydroxyprogesterone caproate (JAN/USP/INN) <JP/US>
E D08053 Hydroxyprogesterone 17alfa-acetate
E D00066 Progesterone (JP18/USP/INN) <JP/US>
E D01217 Dydrogesterone (JP18/USP/INN) <JP>
E D04885 Medrogestone (USAN/INN)
E D07222 Nomegestrol (USAN/INN)
E D08281 Nomegestrol acetate (USAN)
E D07223 Demegestone (INN)
E D07670 Chlormadinone (INN)
E D01299 Chlormadinone acetate (JP18/USAN) <JP>
E D08431 Promegestone (INN)
E D03799 Dienogest (JAN/USAN/INN) <JP>
E D01374 Allylestrenol (JAN/INN)
E D07939 Etynodiol (INN)
E D01294 Ethynodiol diacetate (JAN/USP)
E D00289 Danazol (JP18/USP/INN) <JP/US>
E D00585 Mifepristone (JAN/USAN/INN) <US>
E D00954 Norgestrel (JP18/USP/INN)
E D02840 Altrenogest (USAN/INN)
E D02881 Amadinone acetate (USAN)
E D02996 Asoprisnil (USAN/INN)
E D04315 Gestaclone (USAN/INN)
E D04316 Gestodene (USAN/INN)
E D05003 Methynodiol diacetate (USAN)
E D05009 Metogest (USAN/INN)
E D05205 Norelgestromin (USP/INN)
E D05207 Norethynodrel (USAN)
E D05209 Norgestimate (USP/INN)
E D05308 Oxogestone phenpropionate (USAN)
E D05680 Quingestrone (USAN/INN)
E D06003 Tanaproget (USAN/INN)
E D06145 Tigestol (USAN/INN)
E D06197 Tosagestin (USAN/INN)
E D06235 Trimegestone (USAN/INN)
E D07096 Aglepristone (INN)
E D07968 Flugestone (INN)
E D08429 Proligestone (INN)
E D09571 Onapristone (INN)
E D09972 Telapristone acetate (USAN)
E D10016 Lonaprisan (USAN/INN)
E D10986 Segesterone acetate (USAN)
E D10987 Segesterone (USAN/INN)
E D11181 Vilaprisan (JAN/USAN/INN)
D NR3C4 (AR) [HSA:367] [KO:K08557]
E D07456 Androstanolone (INN)
E D00444 Stanozolol (JAN/USP/INN)
E D00389 Metandienone (INN)
E D08193 Metenolone (INN)
E D01301 Methenolone enanthate (USAN)
E D01375 Methenolone acetate (USAN) <JP>
E D00490 Oxymetholone (JP18/USP/INN)
E D05674 Quinbolone (USAN/INN)
E D08409 Prasterone (USAN/INN) <US>
E D01616 Sodium prasterone sulfate hydrate (JP18)
E D00462 Oxandrolone (JAN/USP/INN) <US>
E D07127 Norethandrolone (INN)
E D08250 Nandrolone (INN)
E D00955 Nandrolone decanoate (JAN/USP)
E D00956 Nandrolone phenpropionate (USP)
E D01476 Nandrolone cyclohexylpropionate (JAN)
E D01737 Nandrolone furylpropionate (JAN)
E D05116 Nandrolone cyclotate (USAN)
E D08251 Nandrolone laurate
E D01149 Oxabolone cipionate (JAN/INN)
E D11451 Clascoterone (USAN) <US>
E D00327 Fluoxymesterone (JAN/USP/INN)
E D00408 Methyltestosterone (JP18/USP/INN) <US>
E D00075 Testosterone (JAN/USP) <US>
E D00957 Testosterone cypionate (USP) <US>
E D00958 Testosterone enanthate (JP18/USP) <JP/US>
E D00959 Testosterone propionate (JP18/USP)
E D06085 Testosterone ketolaurate (USAN/INN)
E D06086 Testosterone phenylacetate (USAN)
E D06087 Testosterone undecanoate (USAN) <US>
E D08573 Testosterone decanoate
E D08574 Testosterone phenylpropionate
E D04947 Mesterolone (USAN/INN)
E D07670 Chlormadinone (INN)
E D01299 Chlormadinone acetate (JP18/USAN) <JP>
E D07766 Cyproterone (INN)
E D01368 Cyproterone acetate (JAN/USAN)
E D00289 Danazol (JP18/USP/INN) <JP/US>
E D00586 Flutamide (JP18/USP/INN) <JP/US>
E D00965 Nilutamide (USAN/INN) <US>
E D00961 Bicalutamide (JP18/USP/INN) <JP/US>
E D10218 Enzalutamide (JAN/USAN) <JP/US>
E D11040 Apalutamide (JAN/INN) <JP/US>
E D11045 Darolutamide (JAN/USAN/INN) <JP/US>
E D01329 Oxendolone (JAN/USAN/INN)
E D01533 Mestanolone (JAN/INN)
E D01534 Dromostanolone propionate (USAN)
E D03079 Benorterone (USAN/INN)
E D03144 Bolasterone (USAN/INN)
E D03145 Boldenone undecylenate (USAN)
E D03338 Calusterone (USAN/INN)
E D03515 Cioteronel (USAN/INN)
E D03551 Clometherone (USAN/INN)
E D03675 Delmadinone acetate (USAN)
E D05025 Mibolerone (USP/INN)
E D05174 Nisterime acetate (USAN)
E D05837 Silandrone (USAN/INN)
E D06191 Topterone (USAN/INN)
E D06211 Trenbolone acetate (USP)
E D06357 Zanoterone (USAN/INN)
E D07536 Boldenone (INN)
E D07783 Delmadinone (INN)
E D08196 Methandriol (INN)
E D08197 Methandriol dipropionate
E D08627 Trenbolone (INN)
E D10221 Enobosarm (USAN)
E D11105 Osaterone acetate (JAN)
E D11184 Ralaniten (USAN/INN)
E D11185 Ralaniten acetate (USAN)
E D12303 Deutenzalutamide (USAN)
E D12316 Bavdegalutamide (USAN)
#
AProtein kinases
B Serine/threonine kinases
C AGC group
D PRKCA [HSA:5578] [KO:K02677]
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D02970 Aprinocarsen sodium (USAN)
E D11191 Tigilanol tiglate (USAN/INN)
D PRKCB [HSA:5579] [KO:K19662]
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D04014 Enzastaurin hydrochloride (JAN/USAN)
E D05784 Safingol (USAN/INN)
E D05785 Safingol hydrochloride (USAN)
E D11191 Tigilanol tiglate (USAN/INN)
E D11935 Enzastaurin (USAN/INN)
D PRKCG [HSA:5582] [KO:K19663]
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D11191 Tigilanol tiglate (USAN/INN)
D PRKCD [HSA:5580] [KO:K06068]
E D05784 Safingol (USAN/INN)
E D05785 Safingol hydrochloride (USAN)
E D09671 Sotrastaurin (USAN/INN)
E D09718 Sotrastaurin acetate (USAN)
E D10456 Delcasertib (USAN/INN)
E D10457 Delcasertib acetate (USAN)
D PRKCE [HSA:5581] [KO:K18050]
E D05784 Safingol (USAN/INN)
E D05785 Safingol hydrochloride (USAN)
E D09671 Sotrastaurin (USAN/INN)
E D09718 Sotrastaurin acetate (USAN)
D PRKCH [HSA:5583] [KO:K18051]
E D09671 Sotrastaurin (USAN/INN)
E D09718 Sotrastaurin acetate (USAN)
D PRKCQ [HSA:5588] [KO:K18052]
E D09671 Sotrastaurin (USAN/INN)
E D09718 Sotrastaurin acetate (USAN)
D AURK [HSA:6790 9212 6795] [KO:K11481 K11479 K11480]
E D08279 Tozasertib (USAN)
E D08344 Tozasertib lactate (USAN)
E D10423 Ilorasertib (USAN)
D AURKA [HSA:6790] [KO:K11481]
E D10085 Alisertib (USAN)
E D10086 Alisertib sodium (USAN)
E D12545 Tinengotinib (USAN/INN)
D AURKB [HSA:9212] [KO:K11479]
E D12545 Tinengotinib (USAN/INN)
D AKT (PKB) [HSA:207 208 10000] [KO:K04456]
E D06221 Triciribine phosphate (USAN)
E D10381 Afuresertib (USAN)
E D10382 Afuresertib hydrochloride (USAN)
E D10641 Ipatasertib (USAN/INN)
E D10674 Uprosertib (USAN/INN)
E D11074 Ipatasertib hydrochloride (JAN)
E D11371 Capivasertib (JAN/USAN)
E D11409 Miransertib (USAN/INN)
E D11508 Miransertib mesylate (USAN)
D DMPK [HSA:1760] [KO:K08788]
E D10907 Baliforsen (USAN)
D ROCK [HSA:6093 9475] [KO:K04514 K17388]
E D07941 Fasudil (INN)
E D01840 Fasudil hydrochloride (JAN)
E D03115 Fasudil hydrochloride hydrate (JAN) <JP>
E D11030 Netarsudil (USAN/INN)
E D11031 Netarsudil mesylate (USAN) <US>
E D10463 Ripasudil hydrochloride hydrate (JAN) <JP>
E D10737 Verosudil (USAN/INN)
E D10738 Verosudil hydrochloride (USAN)
D ROCK2 [HSA:9475] [KO:K17388]
E D11815 Belumosudil (USAN)
E D11816 Belumosudil mesylate (USAN) <US>
C CAMK group
D CHEK1 [HSA:1111] [KO:K02216]
E D10397 Rabusertib (USAN/INN)
E D11206 Prexasertib (USAN/INN)
D AMPK (PRKAA) [HSA:5562 5563] [KO:K07198]
E D08351 Phenformin (BAN)
E D08352 Phenformin hydrochloride
E D04966 Metformin (USAN/INN)
E D00944 Metformin hydrochloride (JP18/USP) <JP/US>
E D00595 Buformin (USAN/INN)
E D02206 Buformin hydrochloride (JP18) <JP>
D MAPKAPK2 [HSA:9261] [KO:K04443]
E D12237 Zunsemetinib (USAN)
E D12560 Gamcemetinib (USAN)
D MKNK [HSA:8569 2872] [KO:K04372]
E D11452 Tomivosertib (USAN/INN)
E D11481 Tomivosertib hydrochloride (USAN)
E D11763 Merestinib (USAN/INN)
C CK1 group
D CSNK1E [HSA:1454] [KO:K08960]
E D11322 Umbralisib (USAN/INN)
E D11323 Umbralisib tosylate (USAN) <US>
C CMGC group
D CDK1 [HSA:983] [KO:K02087]
E D02880 Alvocidib hydrochloride (USAN)
E D09604 Dinaciclib (USAN/INN)
E D09868 Alvocidib (USAN/INN)
E D11599 Zotiraciclib (USAN)
E D11600 Zotiraciclib citrate (USAN)
D CDK2 [HSA:1017] [KO:K02206]
E D02880 Alvocidib hydrochloride (USAN)
E D09604 Dinaciclib (USAN/INN)
E D09868 Alvocidib (USAN/INN)
E D11599 Zotiraciclib (USAN)
E D11600 Zotiraciclib citrate (USAN)
D CDK4/6 [HSA:1019 1021] [KO:K02089 K02091]
E D10372 Palbociclib (JAN/USAN) <JP/US>
E D10652 Palbociclib isethionate (USAN)
E D10883 Ribociclib (USAN/INN)
E D10979 Ribociclib succinate (USAN) <US>
E D10688 Abemaciclib (JAN/USAN) <JP/US>
E D11130 Trilaciclib (USAN/INN)
E D11987 Trilaciclib dihydrochloride <US>
E D11455 Lerociclib (USAN)
D CDK4 [HSA:1019] [KO:K02089]
E D02880 Alvocidib hydrochloride (USAN)
E D09868 Alvocidib (USAN/INN)
D CDK6 [HSA:1021] [KO:K02091]
E D02880 Alvocidib hydrochloride (USAN)
E D09868 Alvocidib (USAN/INN)
D CDK7 [HSA:1022] [KO:K02202]
E D02880 Alvocidib hydrochloride (USAN)
E D09868 Alvocidib (USAN/INN)
E D11599 Zotiraciclib (USAN)
E D11600 Zotiraciclib citrate (USAN)
D CDK9 [HSA:1025] [KO:K02211]
E D09604 Dinaciclib (USAN/INN)
E D11599 Zotiraciclib (USAN)
E D11600 Zotiraciclib citrate (USAN)
E D12525 Enitociclib (USAN/INN)
D CDK5 [HSA:1020] [KO:K02090]
E D09604 Dinaciclib (USAN/INN)
D ERK [HSA:5594 5595] [KO:K04371]
E D11038 Ulixertinib (INN)
E D11285 Ravoxertinib (USAN/INN)
E D12059 Temuterkib (USAN)
E D12060 Temuterkib mesylate (USAN)
D JNK [HSA:5599 5601 5602] [KO:K04440]
E D10168 Tanzisertib (USAN)
D P38 [HSA:1432 5600 5603 6300] [KO:K04441]
E D03736 Doramapimod (USAN/INN)
E D09602 Dilmapimod (USAN/INN)
E D09603 Dilmapimod tosylate (USAN)
E D09639 Losmapimod (USAN/INN)
E D10658 Ralimetinib (USAN/INN)
E D10659 Ralimetinib mesylate (USAN)
E D10959 Neflamapimod (USAN)
D P38alpha (MAPK14) [HSA:1432] [KO:K04441]
E D08963 Pamapimod (INN/USAN)
E D09386 Talmapimod (USAN/INN)
D CLK2 [HSA:1196] [KO:K08823]
E D11588 Lorecivivint (USAN/INN)
D GSK3 [HSA:2931 2932] [KO:K08822 K03083]
E D12196 Laduviglusib (USAN)
D GSK3B [HSA:2932] [KO:K03083]
E D12304 Elraglusib (USAN)
D DYRK1A [HSA:1859] [KO:K08825]
E D11588 Lorecivivint (USAN/INN)
C STE group
D MAP2K1 (MEK1) [HSA:5604] [KO:K04368]
E D10175 Trametinib (USAN)
E D10176 Trametinib dimethyl sulfoxide (JAN/USAN) <JP/US>
E D10405 Cobimetinib (USAN/INN)
E D10615 Cobimetinib fumarate (USAN) <US>
E D10604 Binimetinib (JAN/USAN) <JP/US>
E D09666 Selumetinib (USAN/INN)
E D10024 Selumetinib sulfate (JAN/USAN) <JP/US>
E D10426 Pimasertib (USAN/INN)
E D10486 Pimasertib hydrochloride (USAN)
E D11675 Mirdametinib (USAN)
E D12473 Zapnometinib (USAN/INN)
E D12515 Avutometinib (USAN/INN)
E D12534 Avutometinib potassium (USAN)
D MAP2K2 (MEK2) [HSA:5605] [KO:K04369]
E D10175 Trametinib (USAN)
E D10176 Trametinib dimethyl sulfoxide (JAN/USAN) <JP/US>
E D10405 Cobimetinib (USAN/INN)
E D10615 Cobimetinib fumarate (USAN) <US>
E D10604 Binimetinib (JAN/USAN) <JP/US>
E D09666 Selumetinib (USAN/INN)
E D10024 Selumetinib sulfate (JAN/USAN) <JP/US>
E D10426 Pimasertib (USAN/INN)
E D10486 Pimasertib hydrochloride (USAN)
E D11675 Mirdametinib (USAN)
E D12473 Zapnometinib (USAN/INN)
E D12515 Avutometinib (USAN/INN)
E D12534 Avutometinib potassium (USAN)
D MAP3K5 (ASK1) [HSA:4217] [KO:K04426]
E D10988 Selonsertib (JAN/USAN/INN)
C TKL group
D ARAF [HSA:369] [KO:K08845]
E D12291 Tovorafenib (USAN/INN)
D BRAF [HSA:673] [KO:K04365]
E D10064 Dabrafenib (USAN)
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D11410 Lifirafenib (USAN/INN)
E D11411 Lifirafenib maleate (USAN)
E D12291 Tovorafenib (USAN/INN)
D BRAF* [HSA_VAR:673v1] [HSA:673] [KO:K04365]
E D09996 Vemurafenib (JAN/USAN/INN) <JP/US>
E D10104 Dabrafenib mesylate (USAN) <JP/US>
E D11053 Encorafenib (JAN/USAN/INN) <JP/US>
D RAF1 [HSA:5894] [KO:K04366]
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D12291 Tovorafenib (USAN/INN)
E D12515 Avutometinib (USAN/INN)
E D12534 Avutometinib potassium (USAN)
D IRAK4 [HSA:51135] [KO:K04733]
E D12167 Zimlovisertib (USAN)
E D12411 Emavusertib (USAN/INN)
E D12412 Emavusertib hydrochloride (USAN)
E D12532 Emavusertib mesylate (USAN)
E D12533 Emavusertib maleate (USAN)
E D12538 Emavusertib phosphate (USAN)
E D12539 emavusertib tosylate (USAN)
D RIPK1 [HSA:8737] [KO:K02861]
E D12352 Eclitasertib (USAN/INN)
C Other
D IKBKB [HSA:3551] [KO:K07209]
E D04050 Ertiprotafib (USAN/INN)
D PLK1 [HSA:5347] [KO:K06631]
E D10154 Rigosertib (USAN)
E D10155 Rigosertib sodium (JAN/USAN)
E D10182 Volasertib (USAN)
E D10183 Volasertib trihydrochloride (USAN)
E D11458 Onvansertib (USAN)
E D11459 Onvansertib fumarate (USAN)
D MTOR [HSA:2475] [KO:K07203]
E D06068 Temsirolimus (JAN/USAN/INN) <JP/US>
E D02714 Everolimus (JAN/USAN/INN) <JP/US>
E D08900 Ridaforolimus (JAN/USAN)
E D00753 Sirolimus (JAN/USAN/INN) <JP/US>
E D06669 Zotarolimus (USAN/INN)
E D10076 Olcorolimus (USAN)
E D10543 Apitolisib (USAN/INN)
E D10552 Dactolisib (USAN/INN)
E D10616 Dactolisib tosylate (USAN)
E D10635 Gedatolisib (USAN/INN)
E D10718 Omipalisib (USAN/INN)
E D11440 Bimiralisib (USAN/INN)
E D11501 Samotolisib (USAN)
E D11663 Onatasertib (USAN)
E D11727 Voxtalisib (USAN/INN)
E D11869 Paxalisib (USAN/INN)
D PDK [HSA:5164 5165 5166] [KO:K00898]
E D05857 Sodium dichloroacetate (USAN)
D ATR [HSA:545] [KO:K06640]
E D11148 Berzosertib (USAN/INN)
E D11787 Ceralasertib (USAN/INN)
E D12321 Camonsertib (USAN)
D WEE1 [HSA:7465] [KO:K06632]
E D11361 Adavosertib (USAN)
D BRD2 [HSA:6046] [KO:K08871]
E D10911 Birabresib (USAN/INN)
E D11131 Apabetalone (USAN/INN)
E D12006 Trotabresib (USAN)
E D12266 Pelabresib (USAN/INN)
D BRD3 [HSA:8019] [KO:K11721]
E D10911 Birabresib (USAN/INN)
E D11131 Apabetalone (USAN/INN)
E D12006 Trotabresib (USAN)
E D12266 Pelabresib (USAN/INN)
D BRD4 [HSA:23476] [KO:K11722]
E D10911 Birabresib (USAN/INN)
E D11131 Apabetalone (USAN/INN)
E D11326 Molibresib (USAN)
E D11347 Molibresib besylate (USAN)
E D11479 Mivebresib (USAN/INN)
E D12006 Trotabresib (USAN)
E D12266 Pelabresib (USAN/INN)
D BRDT [HSA:676] [KO:K11724]
E D11131 Apabetalone (USAN/INN)
E D12006 Trotabresib (USAN)
E D12266 Pelabresib (USAN/INN)
B Receptor serine/threonine kinases (RSTK)
C TGFBR1 family
D ACVR1 (ALK2) [HSA:90] [KO:K04675]
E D12547 Zilurgisertib (USAN/INN)
E D12548 Zilurgisertib fumarate (USAN)
D ACVRL1 [HSA:94] [KO:K13594]
E D10106 Dalantercept (USAN)
E D11709 Ascrinvacumab (USAN/INN)
D TGFBR1 [HSA:7046] [KO:K04674]
E D10437 Galunisertib (USAN)
C TGFBR2 family
D ACVR2A [HSA:92] [KO:K04670]
E D09670 Sotatercept (USAN/INN)
E D10620 Bimagrumab (JAN/USAN/INN)
D ACVR2B [HSA:93] [KO:K13596]
E D11701 Luspatercept (USAN/INN) <US>
E D10620 Bimagrumab (JAN/USAN/INN)
D BMPR2 [HSA:659] [KO:K04671]
E D03779 Dibotermin alfa (USAN/INN)
D TGFBR2 [HSA:7048] [KO:K04388]
E D11893 Bintrafusp alfa (USAN/INN)
B Receptor tyrosine kinases (RTK)
C EGFR family
D EGFR [HSA:1956] [KO:K04361]
E D07907 Erlotinib (INN)
E D09724 Afatinib (USAN/INN)
E D10858 Rociletinib (USAN/INN)
E D10859 Olmutinib (USAN/INN)
E D11115 Olmutinib hydrochloride (USAN)
E D09883 Dacomitinib (INN)
E D11251 Icotinib
E D12001 Mobocertinib (USAN/INN)
E D08108 Lapatinib (INN)
E D04024 Lapatinib ditosylate (USAN) <JP/US>
E D08950 Neratinib (USAN/INN)
E D10898 Neratinib maleate <US>
E D06407 Vandetanib (JAN/USAN/INN) <JP/US>
E D03455 Cetuximab (USAN/INN) <JP/US>
E D05350 Panitumumab (USAN/INN) <JP/US>
E D10018 Necitumumab (USAN/INN) <JP/US>
E D11894 Amivantamab (USAN/INN) <US>
E D04862 Masoprocol (USAN/INN)
E D03350 Canertinib dihydrochloride (USAN)
E D05399 Pelitinib (USAN/INN)
E D09660 Rindopepimut (USAN)
E D09689 Varlitinib (USAN/INN)
E D09690 Varlitinib tosylate (USAN)
E D10031 Zalutumumab (USAN/INN)
E D10439 Imgatuzumab (USAN/INN)
E D10886 Naquotinib mesylate (USAN)
E D10958 Naquotinib (USAN/INN)
E D11125 Modotuximab (USAN/INN)
E D11368 Mavelertinib (USAN/INN)
E D11410 Lifirafenib (USAN/INN)
E D11411 Lifirafenib maleate (USAN)
E D11430 Nazartinib (USAN/INN)
E D11434 Nazartinib mesylate (USAN)
E D11750 Duligotuzumab (USAN)
E D11772 Tesevatinib (USAN/INN)
E D11773 Tesevatinib tosylate (USAN)
E D11803 Cetuximab sarotalocan (USAN/INN)
E D11805 Cetuximab sarotalocan sodium (genetical recombination) (JAN) <JP>
E D11872 Serclutamab (USAN/INN)
E D11874 Serclutamab talirine (USAN/INN)
E D12229 Poziotinib (USAN/INN)
E D12230 Poziotinib hydrochloride (USAN)
E D12416 Petosemtamab (USAN/INN)
E D12457 Tuxobertinib (USAN/INN)
D EGFR* [HSA_VAR:1956v2] [HSA:1956] [KO:K04361]
E D01977 Gefitinib (JP18/USAN/INN) <JP/US>
E D04023 Erlotinib hydrochloride (JAN/USAN) <JP/US>
E D09733 Afatinib dimaleate (USAN) <JP/US>
E D10514 Dacomitinib (USAN) <JP/US>
E D11969 Mobocertinib succinate (JAN) <US>
E D11894 Amivantamab (USAN/INN) <US>
E D12506 Sunvozertinib (USAN/INN)
D EGFR* [HSA_VAR:1956v3] [HSA:1956] [KO:K04361]
E D10766 Osimertinib mesylate (USAN) <JP/US>
E D11980 Lazertinib (USAN)
E D12245 Lazertinib mesilate hydrate (JAN)
E D12258 Aumolertinib (USAN)
E D12259 Aumolertinib mesylate (USAN)
D ERBB2 (HER2, CD340) [HSA:2064] [KO:K05083]
E D09724 Afatinib (USAN/INN)
E D09733 Afatinib dimaleate (USAN) <JP/US>
E D09883 Dacomitinib (INN)
E D10514 Dacomitinib (USAN) <JP/US>
E D08108 Lapatinib (INN)
E D08950 Neratinib (USAN/INN)
E D11375 Trastuzumab duocarmazine (USAN/INN)
E D03350 Canertinib dihydrochloride (USAN)
E D04025 Mubritinib (USAN/INN)
E D06610 Lapuleucel-T (USAN)
E D09689 Varlitinib (USAN/INN)
E D09690 Varlitinib tosylate (USAN)
E D10344 Nelipepimut-S (USAN)
E D11772 Tesevatinib (USAN/INN)
E D11773 Tesevatinib tosylate (USAN)
E D11991 Zenocutuzumab (USAN/INN)
E D12011 Zanidatamab (USAN/INN)
E D12229 Poziotinib (USAN/INN)
E D12230 Poziotinib hydrochloride (USAN)
E D12236 Runimotamab (USAN)
E D12457 Tuxobertinib (USAN/INN)
D ERBB2* (HER2, CD340) [HSA_VAR:2064v1] [HSA:2064] [KO:K05083]
E D04024 Lapatinib ditosylate (USAN) <JP/US>
E D11141 Tucatinib (USAN/INN) <US>
E D12442 Tucatinib ethanolate (JAN)
E D03257 Trastuzumab (USAN/INN) <JP/US>
E D11529 Trastuzumab deruxtecan (USAN/INN) <JP/US>
E D10446 Margetuximab (USAN) <US>
D ERBB2* (HER2, CD340) [HSA_VAR:2064v1 2064v3] [HSA:2064] [KO:K05083]
E D10898 Neratinib maleate <US>
E D05446 Pertuzumab (USAN/INN) <JP/US>
E D09980 Trastuzumab emtansine (USAN/INN) <JP/US>
D ERBB3 (HER3) [HSA:2065] [KO:K05084]
E D11141 Tucatinib (USAN/INN) <US>
E D12442 Tucatinib ethanolate (JAN)
E D03350 Canertinib dihydrochloride (USAN)
E D10943 Istiratumab (USAN)
E D11239 Lumretuzumab (USAN/INN)
E D11750 Duligotuzumab (USAN)
E D11777 Seribantumab (USAN/INN)
E D11991 Zenocutuzumab (USAN/INN)
E D12184 Patritumab deruxtecan (USAN/INN)
E D12185 Patritumab (USAN/INN)
D ERBB4 (HER4) [HSA:2066] [KO:K05085]
E D09724 Afatinib (USAN/INN)
E D09733 Afatinib dimaleate (USAN) <JP/US>
E D09883 Dacomitinib (INN)
E D10514 Dacomitinib (USAN) <JP/US>
E D08950 Neratinib (USAN/INN)
E D10898 Neratinib maleate <US>
E D03350 Canertinib dihydrochloride (USAN)
E D09689 Varlitinib (USAN/INN)
E D09690 Varlitinib tosylate (USAN)
C INSR family
D INSR (CD220) [HSA:3643] [KO:K04527]
E D03230 Insulin human (USP/INN) <JP/US>
E D04548 Insulin, neutral (USAN)
E D04477 Insulin lispro (USP/INN) <JP/US>
E D04475 Insulin aspart (USP/INN) <JP/US>
E D04540 Insulin glulisine (USAN/INN) <JP/US>
E D03250 Insulin glargine (USAN/INN) <JP/US>
E D04539 Insulin detemir (USAN/INN) <JP/US>
E D09727 Insulin degludec (USAN/INN) <JP/US>
E D11034 Insulin glargine and lixisenatide <JP/US>
E D11567 Insulin degludec and liraglutide <JP/US>
E D00085 Insulin (JAN/USP)
E D04541 Insulin human, isophane (USP)
E D04542 Insulin human zinc (USP)
E D04543 Insulin human zinc, extended (USP)
E D04544 Insulin I 125 (USAN)
E D04545 Insulin I 131 (USAN)
E D04546 Insulin, dalanated (USAN)
E D04547 Insulin, isophane (USP) <JP>
E D04549 Insulin zinc, extended (USP)
E D04550 Insulin zinc, prompt (USP)
E D04551 Insulin zinc (USP)
E D05622 Proinsulin human (USAN)
E D08080 Insulin injection, biphasic isophane (BAN) <JP>
E D10473 Insulin peglispro (USAN/INN)
E D12358 Insulin icodec (USAN/INN)
D IGF1R (CD221) [HSA:3480] [KO:K05087]
E D03297 Mecasermin (USAN/INN) <JP/US>
E D04870 Mecasermin rinfabate (USAN/INN)
E D08620 Toremifene (INN)
E D00967 Toremifene citrate (JAN/USAN) <JP/US>
E D09680 Teprotumumab (USAN/INN) <US>
E D04491 Ibutamoren mesylate (USAN)
E D09328 Cixutumumab (USAN)
E D09345 Figitumumab (USAN)
E D09746 Dalotuzumab (USAN)
E D09908 Ganitumab (USAN/INN)
E D09925 Linsitinib (USAN/INN)
E D10056 Robatumumab (USAN/INN)
E D10943 Istiratumab (USAN)
D ROS1 [HSA:6098] [KO:K05088]
E D11012 Lorlatinib (JAN/USAN/INN) <JP/US>
E D11454 Repotrectinib (USAN)
E D12363 Taletrectinib (USAN/INN)
E D12364 Taletrectinib adipate (USAN)
D ROS1* [HSA_VAR:6098v1] [HSA:6098] [KO:K05088]
E D09731 Crizotinib (JAN/USAN/INN) <JP/US>
E D10926 Entrectinib (JAN/USAN/INN) <JP/US>
C PDGFR family
D PDGFR [HSA:5156 5159] [KO:K04363 K05089]
E D08953 Nilotinib (USAN/INN)
E D06413 Nilotinib hydrochloride hydrate (JAN) <JP/US>
E D12444 Nilotinib hydrochloride dihydrate (JAN)
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D06678 Motesanib (USAN)
E D08503 Toceranib (USAN)
E D08544 Toceranib phosphate (USAN)
E D09635 Linifanib (USAN/INN)
E D10102 Crenolanib (USAN)
E D10103 Crenolanib besylate (USAN)
E D10423 Ilorasertib (USAN)
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
E D12002 Seralutinib (USAN/INN)
E D12526 Catequentinib (USAN/INN)
E D12537 Catequentinib hydrochloride (USAN)
D PDGFRA [HSA:5156] [KO:K04363]
E D11353 Ripretinib (USAN) <US>
E D09939 Olaratumab (USAN/INN)
E D08947 Motesanib diphosphate (USAN)
E D10411 Tovetumab (USAN)
D PDGFRA* [HSA_VAR:5156v2] [HSA:5156] [KO:K04363]
E D11279 Avapritinib (USAN/INN) <US>
D FIP1L1-PDGFRA [HSA:5156] [KO:K04363]
E D08066 Imatinib (INN)
E D01441 Imatinib mesylate (USAN) <JP/US>
D PDGFRB [HSA:5159] [KO:K05089]
E D03065 Becaplermin (USAN/INN) <US>
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
E D10190 Tivozanib hydrochloride (USAN) <US>
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D06005 Tandutinib (USAN/INN)
E D06285 Vatalanib (USAN/INN)
E D08907 Dovitinib lactate (USAN)
E D08947 Motesanib diphosphate (USAN)
D KIT (CD117) [HSA:3815] [KO:K05091]
E D08066 Imatinib (INN)
E D01441 Imatinib mesylate (USAN) <JP/US>
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
E D08953 Nilotinib (USAN/INN)
E D06413 Nilotinib hydrochloride hydrate (JAN) <JP/US>
E D12444 Nilotinib hydrochloride dihydrate (JAN)
E D10190 Tivozanib hydrochloride (USAN) <US>
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D10229 Masitinib (INN)
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D11270 Pexidartinib (USAN/INN)
E D11271 Pexidartinib hydrochloride (JAN/USAN) <US>
E D11353 Ripretinib (USAN) <US>
E D02937 Ancestim (USAN/INN)
E D05819 Semaxanib (USAN/INN)
E D06005 Tandutinib (USAN/INN)
E D06285 Vatalanib (USAN/INN)
E D06678 Motesanib (USAN)
E D08503 Toceranib (USAN)
E D08544 Toceranib phosphate (USAN)
E D08907 Dovitinib lactate (USAN)
E D08947 Motesanib diphosphate (USAN)
E D09864 Amuvatinib (USAN/INN)
E D09865 Amuvatinib hydrochloride (USAN)
E D12175 Olverembatinib (USAN/INN)
E D12409 Barzolvolimab (USAN/INN)
E D12450 Elenestinib (USAN)
E D12526 Catequentinib (USAN/INN)
E D12537 Catequentinib hydrochloride (USAN)
E D12540 Briquilimab (USAN/INN)
D KIT* (CD117) [HSA_VAR:3815v1] [HSA:3815] [KO:K05091]
E D11279 Avapritinib (USAN/INN) <US>
E D12476 Tuspetinib (USAN)
D FLT3 (CD135) [HSA:2322] [KO:K05092]
E D11768 Pacritinib (USAN/INN) <US>
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D09955 Quizartinib (USAN/INN)
E D10709 Gilteritinib (USAN/INN)
E D04696 Lestaurtinib (USAN/INN)
E D05819 Semaxanib (USAN/INN)
E D06005 Tandutinib (USAN/INN)
E D08279 Tozasertib (USAN)
E D08344 Tozasertib lactate (USAN)
E D08907 Dovitinib lactate (USAN)
E D10102 Crenolanib (USAN)
E D10103 Crenolanib besylate (USAN)
E D11599 Zotiraciclib (USAN)
E D11600 Zotiraciclib citrate (USAN)
E D12476 Tuspetinib (USAN)
D FLT3* (CD135) [HSA_VAR:2322v1 2322v2] [HSA:2322] [KO:K05092]
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D10800 Gilteritinib fumarate (JAN/USAN) <JP/US>
D FLT3* (CD135) [HSA_VAR:2322v2] [HSA:2322] [KO:K05092]
E D09956 Quizartinib dihydrochloride (USAN) <JP>
E D11270 Pexidartinib (USAN/INN)
E D11271 Pexidartinib hydrochloride (JAN/USAN) <US>
C FGFR family
D FGFR [HSA:2260 2263 2261 2264] [KO:K04362 K05093 K05094 K05095]
E D09919 Lenvatinib (USAN/INN)
E D09920 Lenvatinib mesylate (USAN) <JP/US>
E D05716 Repifermin (USAN/INN)
E D11461 Derazantinib hydrochloride (USAN)
E D12526 Catequentinib (USAN/INN)
E D12537 Catequentinib hydrochloride (USAN)
D FGFR1 (CD331) [HSA:2260] [KO:K04362]
E D11417 Pemigatinib (JAN/USAN/INN) <JP/US>
E D11589 Infigratinib (USAN/INN)
E D11611 Infigratinib phosphate (USAN) <US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D11885 Surufatinib (USAN/INN)
E D08878 Brivanib alaninate (JAN/USAN/INN)
E D09589 Brivanib (USAN)
E D11762 Lucitanib (USAN/INN)
E D12404 Tasurgratinib (INN)
E D12405 Tasurgratinib succinate (JAN)
E D12490 Fazpilodemab (USAN/INN)
E D12545 Tinengotinib (USAN/INN)
D FGFR2 (CD332) [HSA:2263] [KO:K05093]
E D11589 Infigratinib (USAN/INN)
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D05338 Palifermin (USAN/INN) <US>
E D11762 Lucitanib (USAN/INN)
E D12404 Tasurgratinib (INN)
E D12405 Tasurgratinib succinate (JAN)
E D12455 Lirafugratinib (USAN)
E D12456 Lirafugratinib hydrochloride (USAN)
E D12545 Tinengotinib (USAN/INN)
D FGFR2* (CD332) [HSA_VAR:2263v2] [HSA:2263] [KO:K05093]
E D10927 Erdafitinib (JAN/USAN/INN) <US>
E D11417 Pemigatinib (JAN/USAN/INN) <JP/US>
E D11725 Futibatinib (JAN/USAN/INN) <US>
D FGFR2* (CD332) [HSA_VAR:2263v2 2263v1] [HSA:2263] [KO:K05093]
E D11611 Infigratinib phosphate (USAN) <US>
D FGFR3 (CD333) [HSA:2261] [KO:K05094]
E D11417 Pemigatinib (JAN/USAN/INN) <JP/US>
E D11589 Infigratinib (USAN/INN)
E D11611 Infigratinib phosphate (USAN) <US>
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D08907 Dovitinib lactate (USAN)
E D11445 Vofatamab (USAN)
E D12284 Recifercept (USAN/INN)
E D12404 Tasurgratinib (INN)
E D12405 Tasurgratinib succinate (JAN)
E D12545 Tinengotinib (USAN/INN)
D FGFR3* (CD333) [HSA_VAR:2261v2] [HSA:2261] [KO:K05094]
E D10927 Erdafitinib (JAN/USAN/INN) <US>
D FGFR4 [HSA:2264] [KO:K05095]
E D11737 Fisogatinib (USAN/INN)
C VEGFR family
D VEGFR1 (FLT1) [HSA:2321] [KO:K05096]
E D03218 Axitinib (JAN/USAN) <JP/US>
E D08881 Cediranib (USAN/INN)
E D08883 Cediranib maleate (JAN/USAN)
E D09683 Tivozanib (USAN/INN)
E D10190 Tivozanib hydrochloride (USAN) <US>
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D09919 Lenvatinib (USAN/INN)
E D09920 Lenvatinib mesylate (USAN) <JP/US>
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D11713 Selpercatinib (JAN/USAN/INN) <JP/US>
E D11885 Surufatinib (USAN/INN)
E D06285 Vatalanib (USAN/INN)
E D06678 Motesanib (USAN)
E D08907 Dovitinib lactate (USAN)
E D08947 Motesanib diphosphate (USAN)
E D09635 Linifanib (USAN/INN)
E D09926 Icrucumab (USAN/INN)
E D10423 Ilorasertib (USAN)
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
E D11762 Lucitanib (USAN/INN)
E D11977 Fruquintinib (USAN)
E D12526 Catequentinib (USAN/INN)
E D12537 Catequentinib hydrochloride (USAN)
E D12545 Tinengotinib (USAN/INN)
D VEGFR2 (KDR) [HSA:3791] [KO:K05098]
E D03218 Axitinib (JAN/USAN) <JP/US>
E D08881 Cediranib (USAN/INN)
E D08883 Cediranib maleate (JAN/USAN)
E D09683 Tivozanib (USAN/INN)
E D10190 Tivozanib hydrochloride (USAN) <US>
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
E D06407 Vandetanib (JAN/USAN/INN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D10062 Cabozantinib (USAN)
E D10095 Cabozantinib s-malate (USAN) <JP/US>
E D09919 Lenvatinib (USAN/INN)
E D09920 Lenvatinib mesylate (USAN) <JP/US>
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D05029 Midostaurin (JAN/USAN/INN) <US>
E D11885 Surufatinib (USAN/INN)
E D09371 Ramucirumab (USAN) <JP/US>
E D05819 Semaxanib (USAN/INN)
E D06285 Vatalanib (USAN/INN)
E D06678 Motesanib (USAN)
E D08503 Toceranib (USAN)
E D08544 Toceranib phosphate (USAN)
E D08878 Brivanib alaninate (JAN/USAN/INN)
E D08907 Dovitinib lactate (USAN)
E D08947 Motesanib diphosphate (USAN)
E D09589 Brivanib (USAN)
E D09618 Foretinib (USAN/INN)
E D09635 Linifanib (USAN/INN)
E D09945 Pegdinetanib (USAN/INN)
E D10224 Golvatinib (USAN)
E D10465 Golvatinib tartrate (USAN)
E D10862 Altiratinib (USAN)
E D11140 Sitravatinib (USAN/INN)
E D11288 Rivoceranib (USAN/INN)
E D11289 Rivoceranib mesylate (USAN)
E D11541 Sitravatinib malate (USAN)
E D11762 Lucitanib (USAN/INN)
E D11772 Tesevatinib (USAN/INN)
E D11773 Tesevatinib tosylate (USAN)
E D11977 Fruquintinib (USAN)
E D12526 Catequentinib (USAN/INN)
E D12537 Catequentinib hydrochloride (USAN)
E D12545 Tinengotinib (USAN/INN)
D VEGFR3 (FLT4) [HSA:2324] [KO:K05097]
E D03218 Axitinib (JAN/USAN) <JP/US>
E D08881 Cediranib (USAN/INN)
E D08883 Cediranib maleate (JAN/USAN)
E D09683 Tivozanib (USAN/INN)
E D10190 Tivozanib hydrochloride (USAN) <US>
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D09919 Lenvatinib (USAN/INN)
E D09920 Lenvatinib mesylate (USAN) <JP/US>
E D10481 Nintedanib (USAN/INN)
E D10396 Nintedanib esylate (USAN) <JP/US>
E D11713 Selpercatinib (JAN/USAN/INN) <JP/US>
E D11885 Surufatinib (USAN/INN)
E D06285 Vatalanib (USAN/INN)
E D06678 Motesanib (USAN)
E D08907 Dovitinib lactate (USAN)
E D08947 Motesanib diphosphate (USAN)
E D09635 Linifanib (USAN/INN)
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
E D11762 Lucitanib (USAN/INN)
E D11772 Tesevatinib (USAN/INN)
E D11773 Tesevatinib tosylate (USAN)
E D11977 Fruquintinib (USAN)
E D12526 Catequentinib (USAN/INN)
E D12537 Catequentinib hydrochloride (USAN)
E D12545 Tinengotinib (USAN/INN)
C MET family
D MET [HSA:4233] [KO:K05099]
E D10062 Cabozantinib (USAN)
E D10095 Cabozantinib s-malate (USAN) <JP/US>
E D10696 Capmatinib (USAN/INN)
E D11717 Tepotinib (USAN/INN)
E D11894 Amivantamab (USAN/INN) <US>
E D09618 Foretinib (USAN/INN)
E D09864 Amuvatinib (USAN/INN)
E D09865 Amuvatinib hydrochloride (USAN)
E D09941 Onartuzumab (USAN/INN)
E D10173 Tivantinib (JAN/USAN/INN)
E D10224 Golvatinib (USAN)
E D10465 Golvatinib tartrate (USAN)
E D10862 Altiratinib (USAN)
E D11136 Glesatinib (USAN/INN)
E D11139 Savolitinib (USAN/INN)
E D11140 Sitravatinib (USAN/INN)
E D11307 Telisotuzumab (USAN)
E D11344 Telisotuzumab vedotin (USAN)
E D11541 Sitravatinib malate (USAN)
E D11763 Merestinib (USAN/INN)
E D12287 Terevalefim (USAN/INN)
E D12392 Fosgonimeton (USAN)
E D12393 Fosgonimeton sodium (USAN)
E D12424 Davutamig (USAN)
E D12557 Elzovantinib (USAN/INN)
D MET* [HSA_VAR:4233v4] [HSA:4233] [KO:K05099]
E D10891 Capmatinib hydrochloride (USAN) <JP/US>
E D11073 Tepotinib hydrochloride (USAN) <JP/US>
E D12053 Vebreltinib (USAN)
D RON [HSA:4486] [KO:K05100]
E D10074 Narnatumab (USAN)
E D11763 Merestinib (USAN/INN)
C TRK family
D NTRK [HSA:4914 4915 4916] [KO:K03176 K04360 K05101]
E D11137 Larotrectinib (USAN/INN)
E D11138 Larotrectinib sulfate (JAN/USAN) <JP/US>
E D12363 Taletrectinib (USAN/INN)
E D12364 Taletrectinib adipate (USAN)
E D12432 Zurletrectinib (USAN)
D NTRK1 (TRKA) [HSA:4914] [KO:K03176]
E D11454 Repotrectinib (USAN)
E D11484 Pegcantratinib (USAN/INN)
D NTRK1* (TRKA) [HSA_VAR:4914v1] [HSA:4914] [KO:K03176]
E D10926 Entrectinib (JAN/USAN/INN) <JP/US>
D NTRK2 (TRKB) [HSA:4915] [KO:K04360]
E D10926 Entrectinib (JAN/USAN/INN) <JP/US>
D NTRK3 (TRKC) [HSA:4916] [KO:K05101]
E D10926 Entrectinib (JAN/USAN/INN) <JP/US>
E D11454 Repotrectinib (USAN)
C EPH family
D EPHA1 [HSA:2041] [KO:K05102]
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
D EPHA2 [HSA:1969] [KO:K05103]
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
D EPHB1 [HSA:2047] [KO:K05110]
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
D EPHB2 [HSA:2048] [KO:K05111]
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
D EPHB4 [HSA:2050] [KO:K05113]
E D11140 Sitravatinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
E D11772 Tesevatinib (USAN/INN)
E D11773 Tesevatinib tosylate (USAN)
C AXL family
D AXL [HSA:558] [KO:K05115]
E D10062 Cabozantinib (USAN)
E D10095 Cabozantinib s-malate (USAN) <JP/US>
E D09864 Amuvatinib (USAN/INN)
E D09865 Amuvatinib hydrochloride (USAN)
E D11140 Sitravatinib (USAN/INN)
E D11438 Bemcentinib (USAN/INN)
E D11541 Sitravatinib malate (USAN)
E D11732 Dubermatinib (USAN/INN)
E D11733 Dubermatinib tartrate (USAN)
E D11763 Merestinib (USAN/INN)
E D12219 Mecbotamab (USAN)
E D12220 Mecbotamab vedotin
E D12271 Batiraxcept (USAN)
E D12279 Mipasetamab (USAN/INN)
E D12280 Mipasetamab uzoptirine (USAN/INN)
C ALK family
D ALK (CD246) [HSA:238] [KO:K05119]
E D10542 Alectinib (USAN/INN)
E D11012 Lorlatinib (JAN/USAN/INN) <JP/US>
E D10926 Entrectinib (JAN/USAN/INN) <JP/US>
E D11346 Ensartinib (USAN)
E D11356 Ensartinib hydrochloride (USAN)
E D11454 Repotrectinib (USAN)
D EML4-ALK [HSA_VAR:238v1] [HSA:238] [KO:K05119]
E D09731 Crizotinib (JAN/USAN/INN) <JP/US>
D EML4-ALK [HSA_VAR:238v2] [HSA:238] [KO:K05119]
E D10551 Ceritinib (JAN/USAN/INN) <JP/US>
E D10450 Alectinib hydrochloride (JAN) <JP/US>
E D10866 Brigatinib (JAN/USAN) <JP/US>
E D11012 Lorlatinib (JAN/USAN/INN) <JP/US>
C TIE family
D TEK (TIE2, CD202) [HSA:7010] [KO:K05121]
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D10334 Rebastinib (USAN)
E D10399 Rebastinib Tosylate (USAN)
E D10862 Altiratinib (USAN)
E D11540 Razuprotafib (USAN)
C ROR family
D ROR2 [HSA:4920] [KO:K05123]
E D12209 Ozuriftamab (USAN)
E D12210 Ozuriftmab vedotin (USAN)
C RET family
D RET [HSA:5979] [KO:K05126]
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D08524 Sorafenib (USAN/INN)
E D06272 Sorafenib tosylate (USAN) <JP/US>
E D06407 Vandetanib (JAN/USAN/INN) <JP/US>
E D10138 Regorafenib (USAN/INN)
E D10137 Regorafenib hydrate (JAN) <JP/US>
E D09919 Lenvatinib (USAN/INN)
E D09920 Lenvatinib mesylate (USAN) <JP/US>
E D06678 Motesanib (USAN)
E D08947 Motesanib diphosphate (USAN)
E D12330 Zeteletinib (USAN)
E D12331 Zeteletinib adipate (USAN)
E D12559 Enbezotinib (USAN/INN)
D RET* [HSA_VAR:5979v1] [HSA:5979] [KO:K05126]
E D11712 Pralsetinib (USAN/INN) <US>
E D12354 Pralsetinib hydrate (JAN)
D RET* [HSA_VAR:5979v1 5979v2] [HSA:5979] [KO:K05126]
E D11713 Selpercatinib (JAN/USAN/INN) <JP/US>
C CCK family
D PTK7 [HSA:5754] [KO:K05127]
E D11118 Cofetuzumab pelidotin (USAN)
E D11119 Cofetuzumab (USAN/INN)
B Non-receptor tyrosine kinases
C SRC family
D SRC [HSA:6714] [KO:K05704]
E D11691 Tirbanibulin (USAN/INN) <US>
E D11692 Tirbanibulin mesylate (USAN)
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
E D03252 Bosutinib (USAN)
E D09728 Bosutinib hydrate (JAN) <JP/US>
E D09664 Saracatinib (USAN/INN)
E D09665 Saracatinib difumarate (USAN)
E D10423 Ilorasertib (USAN)
D FYN [HSA:2534] [KO:K05703]
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
D LYN [HSA:4067] [KO:K05854]
E D06182 Tolimidone (USAN)
E D10202 Bafetinib (USAN)
D LCK [HSA:3932] [KO:K05856]
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
D YES1 [HSA:7525] [KO:K05705]
E D03658 Dasatinib (JAN/INN) <JP>
E D06414 Dasatinib (USAN) <JP/US>
C ABL family
D ABL1 [HSA:25] [KO:K06619]
E D03252 Bosutinib (USAN)
E D09664 Saracatinib (USAN/INN)
E D09665 Saracatinib difumarate (USAN)
D BCR-ABL [HSA:25] [KO:K06619]
E D08066 Imatinib (INN)
E D03658 Dasatinib (JAN/INN) <JP>
E D08953 Nilotinib (USAN/INN)
E D09950 Ponatinib (USAN/INN)
E D11403 Asciminib (USAN/INN)
E D08279 Tozasertib (USAN)
E D08344 Tozasertib lactate (USAN)
E D10202 Bafetinib (USAN)
E D10334 Rebastinib (USAN)
E D10399 Rebastinib Tosylate (USAN)
E D11786 Vodobatinib (USAN)
D BCR-ABL [HSA_VAR:25v1] [HSA:25] [KO:K06619]
E D01441 Imatinib mesylate (USAN) <JP/US>
D BCR-ABL [HSA_VAR:25v2] [HSA:25] [KO:K06619]
E D06414 Dasatinib (USAN) <JP/US>
E D06413 Nilotinib hydrochloride hydrate (JAN) <JP/US>
E D12444 Nilotinib hydrochloride dihydrate (JAN)
E D09728 Bosutinib hydrate (JAN) <JP/US>
E D09951 Ponatinib hydrochloride (JAN/USAN) <JP/US>
E D12175 Olverembatinib (USAN/INN)
D BCR-ABL [HSA_VAR:25v1 25v2] [HSA:25] [KO:K06619]
E D11404 Asciminib hydrochloride (JAN/USAN) <JP/US>
C SYK family
D SYK [HSA:6850] [KO:K05855]
E D09347 Fostamatinib (USAN)
E D09348 Fostamatinib disodium (USAN) <JP/US>
E D11209 Entospletinib (USAN/INN)
E D11676 Gusacitinib (USAN/INN)
E D11677 Gusacitinib hydrochloride (USAN)
E D11789 Mivavotinib (USAN/INN)
E D11790 Mivavotinib citrate (USAN)
E D12476 Tuspetinib (USAN)
C JAK family
D JAK [HSA:3716 3717 3718] [KO:K11217 K04447 K11218]
E D12476 Tuspetinib (USAN)
D JAK1 [HSA:3716] [KO:K11217]
E D11400 Abrocitinib (JAN/USAN) <JP/US>
E D09959 Ruxolitinib (USAN/INN)
E D09960 Ruxolitinib phosphate (JAN/USAN) <JP/US>
E D09970 Tofacitinib (USAN)
E D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
E D10308 Baricitinib (JAN/USAN/INN) <JP/US>
E D10994 Upadacitinib (USAN/INN) <US>
E D10995 Upadacitinib tartrate (USAN)
E D11048 Upadacitinib hydrate (JAN) <JP>
E D10871 Filgotinib (USAN/INN)
E D10872 Filgotinib hydrochloride (USAN)
E D11106 Filgotinib maleate (JAN/USAN) <JP>
E D10944 Itacitinib (USAN/INN)
E D10945 Itacitinib adipate (JAN/USAN)
E D10653 Peficitinib (USAN/INN)
E D10721 Peficitinib hydrobromide (JAN/USAN) <JP>
E D10141 Oclacitinib (USAN)
E D10142 Oclacitinib maleate (USAN)
E D10315 Momelotinib (USAN/INN)
E D10358 Momelotinib dihydrochloride (USAN)
E D10728 Solcitinib (USAN/INN)
E D10889 Momelotinib hydrochloride hydrate (JAN)
E D11046 Delgocitinib (JAN/USAN) <JP>
E D11537 Brepocitinib (USAN)
E D11538 Brepocitinib tosylate (USAN)
E D11676 Gusacitinib (USAN/INN)
E D11677 Gusacitinib hydrochloride (USAN)
E D11866 Deuruxolitinib (USAN)
E D11867 Deuruxolitinib phosphate (USAN)
E D12118 Nezulcitinib (USAN)
E D12211 Ivarmacitinib (USAN)
E D12212 Ivarmacitinib sulfate (USAN)
E D12502 Golidocitinib (USAN/INN)
E D12545 Tinengotinib (USAN/INN)
D JAK2 [HSA:3717] [KO:K04447]
E D09959 Ruxolitinib (USAN/INN)
E D09960 Ruxolitinib phosphate (JAN/USAN) <JP/US>
E D10630 Fedratinib (USAN/INN)
E D11296 Fedratinib hydrochloride (USAN) <US>
E D11768 Pacritinib (USAN/INN) <US>
E D09970 Tofacitinib (USAN)
E D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
E D10308 Baricitinib (JAN/USAN/INN) <JP/US>
E D11106 Filgotinib maleate (JAN/USAN) <JP>
E D10653 Peficitinib (USAN/INN)
E D10721 Peficitinib hydrobromide (JAN/USAN) <JP>
E D10315 Momelotinib (USAN/INN)
E D10358 Momelotinib dihydrochloride (USAN)
E D10365 Gandotinib (USAN)
E D10889 Momelotinib hydrochloride hydrate (JAN)
E D11046 Delgocitinib (JAN/USAN) <JP>
E D11599 Zotiraciclib (USAN)
E D11600 Zotiraciclib citrate (USAN)
E D11676 Gusacitinib (USAN/INN)
E D11677 Gusacitinib hydrochloride (USAN)
E D11866 Deuruxolitinib (USAN)
E D11867 Deuruxolitinib phosphate (USAN)
E D12118 Nezulcitinib (USAN)
E D12545 Tinengotinib (USAN/INN)
D JAK3 [HSA:3718] [KO:K11218]
E D09970 Tofacitinib (USAN)
E D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
E D11106 Filgotinib maleate (JAN/USAN) <JP>
E D10653 Peficitinib (USAN/INN)
E D10721 Peficitinib hydrobromide (JAN/USAN) <JP>
E D10585 Decernotinib (USAN/INN)
E D11046 Delgocitinib (JAN/USAN) <JP>
E D11676 Gusacitinib (USAN/INN)
E D11677 Gusacitinib hydrochloride (USAN)
E D11970 Ritlecitinib tosilate (JAN)
E D12118 Nezulcitinib (USAN)
D TYK2 [HSA:7297] [KO:K11219]
E D09970 Tofacitinib (USAN)
E D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
E D11106 Filgotinib maleate (JAN/USAN) <JP>
E D11817 Deucravacitinib (JAN/USAN) <JP/US>
E D11046 Delgocitinib (JAN/USAN) <JP>
E D11537 Brepocitinib (USAN)
E D11538 Brepocitinib tosylate (USAN)
E D12056 Ropsacitinib (USAN)
E D12118 Nezulcitinib (USAN)
C FAK family
D PTK2B [HSA:2185] [KO:K05871]
E D10618 Defactinib (USAN/INN)
E D10619 Defactinib hydrochloride (USAN)
C Tec family
D BTK [HSA:695] [KO:K07370]
E D10223 Ibrutinib (JAN/USAN) <JP/US>
E D10893 Acalabrutinib (JAN/USAN/INN) <JP/US>
E D11720 Acalabrutinib maleate (USAN)
E D11422 Zanubrutinib (JAN/USAN/INN) <US>
E D10730 Spebrutinib (USAN/INN)
E D10731 Spebrutinib besylate (USAN)
E D11070 Tirabrutinib hydrochloride (JAN) <JP>
E D11428 Vecabrutinib (USAN/INN)
E D11457 Fenebrutinib (USAN/INN)
E D11478 Branebrutinib (USAN)
E D11502 Vecabrutinib succinate (USAN)
E D11873 Rilzabrutinib (USAN/INN)
E D12050 Pirtobrutinib (JAN/USAN) <US>
E D12052 Luxeptinib (USAN)
E D12158 Elsubrutinib (USAN/INN)
E D12160 Orelabrutinib (USAN/INN)
E D12213 Tolebrutinib (USAN/INN)
E D12285 Remibrutinib (USAN/INN)
E D12383 Edralbrutinib (USAN/INN)
E D12467 Evobrutinib (USAN/INN)
E D12489 Atuzabrutinib (USAN/INN)
E D12504 Nemtabrutinib (USAN/INN)
C InsR family
D IGF1 [HSA:3479] [KO:K05459]
E D04862 Masoprocol (USAN/INN)
D IGF2 [HSA:3481] [KO:K13769]
E D10352 Dusigitumab (USAN)
#
ACytokines and receptors
B Cytokines
C Interleukins
D IL1 [HSA:3552 3553] [KO:K04383 K04519]
E D06635 Rilonacept (USAN/INN) <US>
E D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
E D12370 Lutikizumab (INN)
D IL1A [HSA:3552] [KO:K04383]
E D11253 Bermekimab (USAN)
E D12350 Vilamakitug (USAN)
D IL1B [HSA:3553] [KO:K04519]
E D09315 Canakinumab (USAN/INN) <JP/US>
E D09911 Gevokizumab (USAN/INN)
D IL4 [HSA:3565] [KO:K05430]
E D03117 Binetrakin (USAN/INN)
E D05377 Pascolizumab (USAN/INN)
D IL5 [HSA:3567] [KO:K05428]
E D08985 Reslizumab (USAN) <US>
E D04923 Mepolizumab (USAN/INN) <JP/US>
E D12169 Depemokimab (USAN)
D IL6 [HSA:3569] [KO:K05405]
E D09669 Siltuximab (USAN/INN) <US>
E D10080 Sirukumab (USAN)
E D12487 Olokizumab (INN)
E D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
E D08976 Pomalidomide (JAN/USAN/INN) <JP/US>
D IL9 [HSA:3578] [KO:K05432]
E D09897 Enokizumab (USAN/INN)
D IL10 [HSA:3586] [KO:K05443]
E D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
D IL12 [HSA:3592 3593] [KO:K05406 K05425]
E D09214 Ustekinumab (USAN/INN) <JP/US>
E D09588 Briakinumab (USAN/INN)
E D04748 Lisofylline (USAN/INN)
E D06556 Apilimod mesylate (USAN)
D IL13 [HSA:3596] [KO:K05435]
E D09979 Tralokinumab (USAN/INN) <JP/US>
E D08857 Anrukinzumab (USAN)
E D09633 Lebrikizumab (USAN/INN)
E D11598 Romilkimab (USAN/INN)
D IL15 [HSA:3600] [KO:K05433]
E D12306 Ordesekimab (USAN)
D IL17A [HSA:3605] [KO:K05489]
E D09967 Secukinumab (USAN/INN) <JP/US>
E D10071 Ixekizumab (USAN) <JP/US>
E D11550 Bimekizumab (USAN/INN) <JP>
E D10902 Afasevikumab (USAN/INN)
E D11127 Tibulizumab (USAN/INN)
E D12278 Izokibep (USAN/INN)
D IL17F [HSA:112744] [KO:K05494]
E D11550 Bimekizumab (USAN/INN) <JP>
E D10902 Afasevikumab (USAN/INN)
D IL18 [HSA:3606] [KO:K05482]
E D04487 Iboctadekin (USAN/INN)
D IL20 [HSA:50604] [KO:K22667]
E D11756 Fletikumab (USAN/INN)
D IL22 [HSA:50616] [KO:K05445]
E D09615 Fezakinumab (USAN/INN)
E D11953 Efmarodocokin alfa (USAN/INN)
D IL23A [HSA:51561] [KO:K05426]
E D09214 Ustekinumab (USAN/INN) <JP/US>
E D09588 Briakinumab (USAN/INN)
E D10438 Guselkumab (USAN) <JP/US>
E D10400 Tildrakizumab (USAN) <JP/US>
E D11052 Risankizumab (USAN/INN) <JP/US>
E D06556 Apilimod mesylate (USAN)
E D10912 Brazikumab (USAN/INN)
E D11123 Mirikizumab (USAN/INN)
D IL33 [HSA:90865] [KO:K12967]
E D11449 Etokimab (USAN)
E D11999 Itepekimab (USAN/INN)
E D12375 Tozorakimab (USAN/INN)
C Interferons
D IFNA [HSA:3439 3440 3441 3442 3443 3444 3445 3446 3447 3448 3449 3451 3452] [KO:K05414]
E D09662 Rontalizumab (USAN/INN)
E D09668 Sifalimumab (USAN/INN)
D IFNA2 [HSA:3440] [KO:K05414]
E D12531 Nadofaragene firadenovec (USAN/INN)
D IFNB [HSA:3456] [KO:K05415]
E D12464 Dazukibart (USAN)
D IFNG [HSA:3458] [KO:K04687]
E D11120 Emapalumab (USAN/INN) <US>
E D04242 Fontolizumab (USAN/INN)
C CSF and other factors
D CSF2 [HSA:1437] [KO:K05427]
E D11121 Gimsilumab (USAN/INN)
E D11236 Lenzilumab (USAN/INN)
E D11343 Otilimab (USAN)
D PRL [HSA:5617] [KO:K05439]
E D03165 Bromocriptine (USAN/INN)
E D00780 Bromocriptine mesylate (USP) <JP/US>
E D00987 Cabergoline (JP18/USP/INN) <JP/US>
E D01348 Terguride (JAN/INN)
D TSLP [HSA:85480] [KO:K05436]
E D11771 Tezepelumab (USAN/INN) <JP/US>
C Chemokines
D CCL2 [HSA:6347] [KO:K14624]
E D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
E D03116 Bindarit (USAN/INN)
E D09877 Carlumab (USAN)
D CCL11 [HSA:6356] [KO:K16597]
E D11741 Lazucirnon (USAN)
E D11742 Lazucirnon hydrochloride (USAN)
D CXCL10 [HSA:3627] [KO:K12671]
E D10404 Eldelumab (USAN)
D CX3CL1 [HSA:6376] [KO:K05508]
E D11498 Quetmolimab (USAN)
C Tumor necrosis factors
D TNF (TNFA, TNFSF2) [HSA:7124] [KO:K03156]
E D00742 Etanercept (USAN/INN) <JP/US>
E D02598 Infliximab (USAN/INN) <JP/US>
E D07436 Afelimomab (INN)
E D02597 Adalimumab (USAN/INN) <JP/US>
E D03441 Certolizumab pegol (USAN/INN) <JP/US>
E D04358 Golimumab (USAN/INN) <JP/US>
E D11703 Opinercept (INN)
E D00754 Thalidomide (JAN/USP/INN) <JP/US>
E D04687 Lenalidomide (JAN/USAN/INN) <US>
E D09813 Lenalidomide hydrate (JAN) <JP>
E D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
E D08976 Pomalidomide (JAN/USAN/INN) <JP/US>
E D04690 Lenercept (USAN/INN)
E D05146 Nerelimomab (USAN/INN)
E D05263 Onercept (USAN/INN)
E D05393 Pegsunercept (USAN)
E D09944 Ozoralizumab (USAN) <JP>
E D10320 Placulumab (USAN/INN)
E D12420 Licaminlimab (USAN/INN)
D LTA (TNFB, TNFSF1) [HSA:4049] [KO:K05468]
E D00742 Etanercept (USAN/INN) <JP/US>
E D04690 Lenercept (USAN/INN)
E D10187 Pateclizumab (USAN)
D LTB (TNFC, TNFSF3) [HSA:4050] [KO:K03157]
E D04690 Lenercept (USAN/INN)
E D08866 Baminercept (USAN/INN)
D TNFSF4 (OX40L) [HSA:7292] [KO:K05469]
E D09943 Oxelumab (USAN/INN)
E D12550 Amlitelimab (USAN/INN)
D TNFSF5 (CD154) [HSA:959] [KO:K03161]
E D05777 Ruplizumab (USAN/INN)
E D06193 Toralizumab (USAN/INN)
E D11122 Letolizumab (USAN/INN)
D TNFSF7 (CD70) [HSA:970] [KO:K05470]
E D10341 Vorsetuzumab mafodotin (USAN/INN)
E D10342 Vorsetuzumab (USAN/INN)
D TNFSF11 (RANKL, CD254) [HSA:8600] [KO:K05473]
E D03684 Denosumab (USAN) <JP/US>
D TNFSF13 (APRIL, CD256) [HSA:8741] [KO:K05475]
E D09704 Atacicept (USAN/INN)
E D12374 Sibeprenlimab (INN)
D TNFSF13B (BAFF, CD257) [HSA:10673] [KO:K05476]
E D03068 Belimumab (USAN) <JP/US>
E D02979 Ardenermin (USAN)
E D08877 Briobacept (USAN)
E D09704 Atacicept (USAN/INN)
E D10083 Tabalumab (USAN)
E D11127 Tibulizumab (USAN/INN)
E D11907 Rozibafusp alfa (USAN/INN)
C Transforming growth factors (RSTK-binding)
D TGFB [HSA:7040 7042 7043] [KO:K13375 K13376 K13377]
E D09620 Fresolimumab (USAN/INN)
D TGFB2 [HSA:7042] [KO:K13376]
E D06563 Belagenpumatucel-L (USAN)
E D10203 Trabedersen (INN/BAN)
D MSTN [HSA:2660] [KO:K05497]
E D05917 Stamulumab (USAN)
E D10347 Ramatercept (USAN)
E D11047 Domagrozumab (USAN/INN)
E D11235 Landogrozumab (USAN/INN)
E D11242 Trevogrumab (USAN/INN)
E D11265 Taldefgrobep alfa (USAN)
E D11797 Apitegromab (USAN)
D GDF15 [HSA:9518] [KO:K05504]
E D11909 Ponsegromab (USAN)
C Growth factors (RTK-binding)
D PGF [HSA:5228] [KO:K16859]
E D09574 Aflibercept (USAN/INN) <JP/US>
E D10819 Aflibercept beta (genetical recombination) (JAN) <JP>
D VEGFA [HSA:7422] [KO:K05448]
E D06409 Bevacizumab (USAN) <JP/US>
E D09574 Aflibercept (USAN/INN) <JP/US>
E D05386 Pegaptanib sodium (JAN/USAN)
E D05697 Ranibizumab (USAN/INN) <JP/US>
E D11083 Brolucizumab (USAN/INN) <JP/US>
E D11517 Abicipar pegol (USAN/INN)
E D11516 Faricimab (USAN/INN) <JP/US>
E D08874 Bevasiranib sodium (USAN)
E D10819 Aflibercept beta (genetical recombination) (JAN) <JP>
E D11126 Navicixizumab (USAN/INN)
E D11244 Vanucizumab (USAN/INN)
E D11642 Dilpacimab (USAN/INN)
E D11890 Emvododstat (USAN)
E D12507 Tarcocimab (INN)
E D12508 Tarcocimab tedromer (INN)
D VEGFB [HSA:7423] [KO:K16858]
E D09574 Aflibercept (USAN/INN) <JP/US>
E D10819 Aflibercept beta (genetical recombination) (JAN) <JP>
D NGF [HSA:4803] [KO:K02582]
E D09387 Tanezumab (USAN/INN)
E D09907 Fulranumab (USAN/INN)
D HGF [HSA:3082] [KO:K05460]
E D09659 Rilotumumab (USAN/INN)
E D10123 Ficlatuzumab (USAN)
E D12398 Oremepermin alfa (USAN/INN)
D TGFA [HSA:7039] [KO:K08774]
E D12343 Fepixnebart (TN)
D EREG [HSA:2069] [KO:K09784]
E D12343 Fepixnebart (TN)
D ANGPT1 [HSA:284] [KO:K05465]
E D10177 Trebananib (USAN)
D ANGPT2 [HSA:285] [KO:K05466]
E D11516 Faricimab (USAN/INN) <JP/US>
E D10177 Trebananib (USAN)
E D10395 Nesvacumab (USAN)
E D11244 Vanucizumab (USAN/INN)
E D11904 Zansecimab (USAN)
D ANGPTL3 [HSA:27329] [KO:K22288]
E D11753 Evinacumab (USAN/INN) <US>
D FGF19 [HSA:9965] [KO:K22603]
E D11734 Aldafermin (USAN/INN)
D FGF21 [HSA:26291] [KO:K22429]
E D11512 Pegbelfermin (USAN)
E D11868 Efruxifermin (USAN)
E D12327 Pegozafermin (USAN)
D FGF23 [HSA:8074] [KO:K22428]
E D10913 Burosumab (USAN/INN) <JP/US>
B Cytokine receptors
C Interleukin receptors
D IL1R (CD121) [HSA:3554 7850] [KO:K04386 K04387]
E D02934 Anakinra (USAN/INN) <US>
E D11759 Isunakinra (USAN/INN)
D IL1RL1 [HSA:9173] [KO:K05171]
E D11796 Melrilimab (USAN)
E D11832 Astegolimab (USAN/INN)
D IL1RL2 (IL-36R) [HSA:8808] [KO:K05172]
E D12066 Spesolimab (USAN/INN) <JP/US>
E D11892 Imsidolimab (USAN)
D IL2RA (CD25) [HSA:3559] [KO:K05068]
E D03682 Denileukin diftitox (USAN/INN) <JP>
E D00748 Aldesleukin (USAN/INN) <US>
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D03639 Daclizumab (USAN/INN)
E D03058 Basiliximab (USAN/INN) <JP/US>
E D02743 Celmoleukin (genetical recombination) (JP18)
E D02749 Teceleukin (USAN) <JP>
E D11324 Camidanlumab (USAN)
E D11325 Camidanlumab tesirine (USAN)
E D12328 Rezpegaldesleukin (USAN)
E D12371 Nemvaleukin alfa (USAN/INN)
E D12386 Melredableukin alfa (USAN)
D IL2RB (CD122) [HSA:3560] [KO:K05069]
E D00748 Aldesleukin (USAN/INN) <US>
E D02743 Celmoleukin (genetical recombination) (JP18)
E D02749 Teceleukin (USAN) <JP>
E D11669 Bempegaldesleukin (USAN/INN)
E D12328 Rezpegaldesleukin (USAN)
D IL2RG (CD132) [HSA:3561] [KO:K05070]
E D00748 Aldesleukin (USAN/INN) <US>
E D02743 Celmoleukin (genetical recombination) (JP18)
E D02749 Teceleukin (USAN) <JP>
E D12328 Rezpegaldesleukin (USAN)
D IL3RA (CD123) [HSA:3563] [KO:K04737]
E D11358 Tagraxofusp (USAN/INN) <US>
E D03645 Daniplestim (USAN/INN)
E D04695 Leridistim (USAN/INN)
E D05036 Milodistim (USAN/INN)
E D05090 Muplestim (USAN/INN)
E D11306 Flotetuzumab (USAN/INN)
E D11841 Vibecotamab (USAN/INN)
E D12307 Pivekimab (USAN)
E D12308 Pivekimab sunirine (USAN)
D IL4R (CD124) [HSA:3566] [KO:K05071]
E D10354 Dupilumab (USAN) <JP/US>
D IL5RA (CD125) [HSA:3568] [KO:K05067]
E D09874 Benralizumab (USAN/INN) <JP/US>
D IL6R (CD126) [HSA:3570] [KO:K05055]
E D02596 Tocilizumab (USAN/INN) <JP/US>
E D10161 Sarilumab (USAN) <JP/US>
E D11079 Satralizumab (USAN/INN) <JP/US>
D IL7R (CD127) [HSA:3575] [KO:K05072]
E D12479 Lusvertikimab (USAN/INN)
D IL10R [HSA:3587 3588] [KO:K05134 K05135]
E D04505 Ilodecakin (USAN/INN)
E D11200 Pegilodecakin (USAN/INN)
D IL11RA [HSA:3590] [KO:K05056]
E D05266 Oprelvekin (USAN/INN)
D IL15RA (CD215) [HSA:3601] [KO:K05074]
E D11747 Inbakicept (USAN/INN)
D IL17RA (CD217) [HSA:23765] [KO:K05164]
E D10061 Brodalumab (USAN) <JP/US>
D IL21R (CD360) [HSA:50615] [KO:K05075]
E D09332 Denenicokin (USAN/INN)
D IL31RA [HSA:133396] [KO:K22630]
E D11080 Nemolizumab (USAN/INN) <JP>
D OSMR [HSA:9180] [KO:K05057]
E D11800 Vixarelimab (USAN)
C Interferon receptors
D IFNAR1 [HSA:3454] [KO:K05130]
E D03305 Interferon alfa (NAMALWA) (JP18) <JP>
E D03304 Interferon beta (JAN) <JP>
E D00745 Interferon alfa-2a (USAN/INN)
E D02745 Interferon alfa-2b (USAN) <US>
E D04552 Interferon alfa-n1 (USAN)
E D04554 Interferon beta-1a (USAN) <JP/US>
E D00746 Interferon beta-1b (USAN/INN) <JP/US>
E D02744 Interferon alfacon-1 (USAN/INN)
E D02748 Peginterferon alfa-2b (USAN/INN)
E D02747 Peginterferon alfa-2a (USAN/INN) <JP/US>
E D08844 Albinterferon alfa-2b (USAN)
E D10483 Peginterferon beta-1a (USAN/INN) <US>
E D11027 Ropeginterferon alfa-2b (INN) <US>
E D11082 Anifrolumab (USAN) <JP/US>
E D04553 Interferon alfa-n3 (USAN)
D IFNAR2 [HSA:3455] [KO:K05131]
E D03305 Interferon alfa (NAMALWA) (JP18) <JP>
E D03304 Interferon beta (JAN) <JP>
E D00745 Interferon alfa-2a (USAN/INN)
E D02745 Interferon alfa-2b (USAN) <US>
E D04552 Interferon alfa-n1 (USAN)
E D04554 Interferon beta-1a (USAN) <JP/US>
E D00746 Interferon beta-1b (USAN/INN) <JP/US>
E D02744 Interferon alfacon-1 (USAN/INN)
E D02748 Peginterferon alfa-2b (USAN/INN)
E D02747 Peginterferon alfa-2a (USAN/INN) <JP/US>
E D08844 Albinterferon alfa-2b (USAN)
E D10483 Peginterferon beta-1a (USAN/INN) <US>
E D11027 Ropeginterferon alfa-2b (INN) <US>
E D11082 Anifrolumab (USAN) <JP/US>
E D04553 Interferon alfa-n3 (USAN)
D IFNGR1 (CD119) [HSA:3459] [KO:K05132]
E D00747 Interferon gamma-1b (USAN/INN) <US>
E D03357 Interferon gamma-1a (genetical recombination) (JAN) <JP>
E D08805 Interferon gamma-n1 (JAN)
D IFNGR2 [HSA:3460] [KO:K05133]
E D00747 Interferon gamma-1b (USAN/INN) <US>
E D03357 Interferon gamma-1a (genetical recombination) (JAN) <JP>
E D08805 Interferon gamma-n1 (JAN)
D IFNLR1 [HSA:163702] [KO:K05140]
E D10078 Peginterferon lambda-1a (USAN)
C CSF and other factor receptors
D CSF1R (FMS, CD115) [HSA:1436] [KO:K05090]
E D08552 Sunitinib (INN)
E D06402 Sunitinib malate (JAN/USAN) <JP/US>
E D11270 Pexidartinib (USAN/INN)
E D11271 Pexidartinib hydrochloride (JAN/USAN) <US>
E D11885 Surufatinib (USAN/INN)
E D02664 Mirimostim (JAN/INN)
E D09635 Linifanib (USAN/INN)
E D11234 Emactuzumab (USAN/INN)
E D11378 Edicotinib (USAN)
E D11379 Edicotinib hydrochloride (USAN)
E D11952 Axatilimab (USAN/INN)
E D12238 Vimseltinib (USAN/INN)
E D12545 Tinengotinib (USAN/INN)
D CSF2RA (GMCSFR, CD116) [HSA:1438] [KO:K05066]
E D05066 Molgramostim (USAN/INN)
E D05803 Sargramostim (USP/INN) <US>
E D05712 Regramostim (USAN/INN)
E D09930 Mavrilimumab (USAN/INN)
D CSF3R (GCSFR, CD114) [HSA:1441] [KO:K05061]
E D03235 Filgrastim (USP/INN) <JP/US>
E D03247 Lenograstim (USAN/INN) <JP>
E D06889 Pegfilgrastim (USAN/INN) <JP/US>
E D10242 Lipegfilgrastim (USAN)
E D10310 Balugrastim (USAN/INN)
E D11026 Pegteograstim (INN)
E D11986 Efbemalenograstim alfa (USAN/INN)
E D03245 Nartograstim (genetical recombination) (JP18)
E D04695 Leridistim (USAN/INN)
E D05036 Milodistim (USAN/INN)
E D05389 Pegnartograstim (USAN/INN)
E D11188 Eflapegrastim (USAN/INN) <US>
D EPOR [HSA:2057] [KO:K05079]
E D03231 Epoetin alfa (USAN/INN) <JP/US>
E D03232 Epoetin beta (USAN/INN) <JP>
E D04032 Epoetin delta (USAN)
E D10000 Epoetin epsilon (INN)
E D10846 Epoetin theta (INN)
E D10847 Epoetin zeta (INN)
E D03651 Darbepoetin alfa (USAN/INN) <JP/US>
E D09998 Epoetin beta pegol (genetical recombination) (JAN) <JP/US>
E D09946 Peginesatide (USAN/INN)
E D09947 Peginesatide acetate (JAN/USAN)
D LEPR (CD295) [HSA:3953] [KO:K05062]
E D05014 Metreleptin (USAN/INN) <JP/US>
D GHR [HSA:2690] [KO:K05080]
E D02691 Somatropin (USP/INN) <JP/US>
E D05884 Somatrem (USAN)
E D03297 Mecasermin (USAN/INN) <JP/US>
E D04870 Mecasermin rinfabate (USAN/INN)
E D11194 Somapacitan (USAN/INN) <JP/US>
E D11486 Lonapegsomatropin (USAN/INN) <US>
E D05394 Pegvisomant (USAN/INN) <JP/US>
E D11161 Atesidorsen (USAN/INN)
E D11162 Atesidorsen sodium (USNA)
E D11193 Somavaratan (USAN/INN)
D MPL (TPOR, CD110) [HSA:4352] [KO:K05082]
E D08990 Romiplostim (USAN/INN) <JP/US>
E D03978 Eltrombopag olamine (JAN/USAN) <JP/US>
E D10476 Lusutrombopag (JAN/USAN/INN) <JP/US>
E D10306 Avatrombopag (USAN/INN)
E D10307 Avatrombopag maleate (JAN/USAN) <US>
E D09024 Totrombopag choline (USAN)
D CNTFR [HSA:1271] [KO:K05059]
E D03647 Dapiclermin (USAN/INN)
C Chemokine receptors
D CCR2 (CD192) [HSA:729230] [KO:K04177]
E D09878 Cenicriviroc (USAN/INN)
E D09879 Cenicriviroc mesylate (USAN)
E D10972 Plozalizumab (USAN/INN)
E D11997 Ilacirnon (USAN)
E D11998 Ilacirnon sodium (USAN)
D CCR4 (CD194) [HSA:1233] [KO:K04179]
E D09761 Mogamulizumab (USAN) <JP/US>
D CCR5 (CD195) [HSA:1234] [KO:K04180]
E D06670 Maraviroc (JAN/INN) <JP/US>
E D03210 Ancriviroc (USAN/INN)
E D06297 Vicriviroc maleate (USAN)
E D06557 Aplaviroc hydrochloride (USAN)
E D09878 Cenicriviroc (USAN/INN)
E D09879 Cenicriviroc mesylate (USAN)
E D11399 Leronlimab (USAN/INN)
D CCR9 (CD199) [HSA:10803] [KO:K04184]
E D10378 Vercirnon (USAN/INN)
E D10379 Vercirnon sodium (USAN)
D CXCR1 (IL8RA, CD181) [HSA:3577] [KO:K04175]
E D08984 Reparixin (USAN/INN)
E D10075 Navarixin (USAN)
E D12556 Eltrekibart (USAN)
D CXCR2 (IL8RB, CD182) [HSA:3579] [KO:K05050]
E D08984 Reparixin (USAN/INN)
E D10075 Navarixin (USAN)
E D10332 Elubrixin (USAN)
E D10387 Danirixin (USAN/INN)
E D10420 Elubrixin tosylate (USAN)
D CXCR4 (CD184) [HSA:7852] [KO:K04189]
E D08971 Plerixafor (JAN/USAN/INN) <JP/US>
E D11510 Mavorixafor (USAN)
E D12128 Balixafortide (USAN/INN)
E D12281 Motixafortide (USAN/INN)
E D12282 Motixafortide acetate (USAN)
C Tumor necrosis factor receptors
D TNFRSF1 (CD120) [HSA:7132 7133] [KO:K03158 K05141]
E D08562 Tasonermin (INN)
D TNFRSF4 (CD134, OX40) [HSA:7293] [KO:K05142]
E D11268 Vonlerolizumab (USAN/INN)
E D11301 Tavolimab (USAN/INN)
E D12543 Rocatinlimab (USAN/INN)
D TNFRSF5 (CD40) [HSA:958] [KO:K03160]
E D06071 Teneliximab (USAN/INN)
E D08896 Dacetuzumab (USAN)
E D08942 Lucatumumab (USAN)
E D11357 Bleselumab (USAN/INN)
E D11491 Selicrelumab (USAN/INN)
E D11597 Ravagalimab (USAN/INN)
E D11610 Iscalimab (USAN/INN)
E D12178 Sotigalimab (USAN)
D TNFRSF7 (CD27) [HSA:939] [KO:K05144]
E D12256 Boserolimab (USAN)
D TNFRSF8 (CD30) [HSA:943] [KO:K05145]
E D09587 Brentuximab vedotin (USAN) <JP/US>
E D04612 Iratumumab (USAN)
D TNFRSF9 (CD137) [HSA:3604] [KO:K05146]
E D09984 Urelumab (USAN/INN)
D TNFRSF10A (TRAILR1, CD261) [HSA:8797] [KO:K04722]
E D04858 Mapatumumab (USAN/INN)
D TNFRSF10B (TRAILR2, CD262) [HSA:8795] [KO:K04722]
E D06611 Lexatumumab (USAN/INN)
E D09329 Conatumumab (USAN/INN)
E D09888 Drozitumab (USAN/INN)
E D12458 Ozekibart (USAN)
D TNFRSF12A (TWEAKR, CD266) [HSA:51330] [KO:K05149]
E D09896 Enavatuzumab (USAN/INN)
D TNFRSF13C (BAFF-R, CD268) [HSA:115650] [KO:K05151]
E D12151 Ianalumab (USAN/INN)
D TNFRSF18 [HSA:8784] [KO:K05154]
E D12165 Ragifilimab (USAN/INN)
D NGFR (TNFRSF16, CD271) [HSA:4804] [KO:K02583]
E D11028 Cenegermin (INN) <US>
D TNFRSF17 (BCMA, CD269) [HSA:608] [KO:K05153]
E D11595 Belantamab mafodotin (USAN) <US>
E D12315 Ciltacabtagene autoleucel (USAN/INN) <US>
E D11556 Idecabtagene vicleucel (USAN) <US>
E D11594 Belantamab (USAN/INN)
E D11992 Pavurutamab (USAN)
E D12010 Pacanalotamab (USAN)
E D12177 Teclistamab (USAN/INN) <US>
E D12222 Linvoseltamab (USAN)
B Pattern recognition receptors
C Toll-like receptors
D TLR2 (CD282) [HSA:7097] [KO:K10159]
E D11503 Tomaralimab (USAN)
D TLR3 (CD283) [HSA:7098] [KO:K05401]
E D09661 Rintatolimod (USAN/INN)
D TLR4 (CD284) [HSA:7099] [KO:K10160]
E D06619 Mifamurtide (USAN)
E D04043 Eritoran tetrasodium (USAN)
E D09573 Eritoran sodium (JAN)
E D11668 Mosedipimod (USAN/INN)
D TLR5 [HSA:7100] [KO:K10168]
E D10368 Entolimod (USAN)
D TLR7 [HSA:51284] [KO:K05404]
E D02500 Imiquimod (JAN/USP/INN) <JP/US>
E D01666 Bropirimine (JAN/USAN/INN)
E D04619 Isatoribine (USAN)
E D04787 Loxoribine (USAN/INN)
E D11003 Vesatolimod (USAN/INN)
E D12261 Enpatoran (USAN/INN)
E D12453 Guretolimod (USAN/INN)
E D12521 Ruzotolimod (USAN/INN)
D TLR8 (CD288) [HSA:51311] [KO:K10170]
E D10716 Motolimod (USAN/INN)
E D11871 Selgantolimod (USAN/INN)
E D12261 Enpatoran (USAN/INN)
D TLR9 (CD289) [HSA:54106] [KO:K10161]
E D08841 Agatolimod (USAN)
E D08842 Agatolimod sodium (USAN)
E D11504 Tilsotolimod (USAN/INN)
E D11505 Tilsotolimod sodium (USAN)
E D12275 Cobitolimod (USAN/INN)
E D12276 Cobitolimod sodium (USAN)
C C-type lectin receptors
D CLEC4C (CD303) [HSA:170482] [KO:K06723]
E D12232 Litifilimab (USAN)
D MRC1 (CD206) [HSA:4360] [KO:K06560]
E D11543 Technetium Tc99m tilmanocept (USAN) <US>
C NOD-like receptors
D NOD2 [HSA:64127] [KO:K10165]
E D06619 Mifamurtide (USAN)
E D11385 Inarigivir soproxil (USAN)
D NLRP3 [HSA:114548] [KO:K12800]
E D12422 Selnoflast (USAN/INN)
E D12423 Selnoflast potassium (USAN)
#
ACell surface molecules and ligands
B Cell adhesion molecules: Ig superfamiy
C CD2 family
D CD2 [HSA:914] [KO:K06449]
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D05847 Siplizumab (USAN/INN)
D CD58 (LFA3) [HSA:965] [KO:K06492]
E D02800 Alefacept (USAN/INN)
D SLAMF7 (CD319) [HSA:57823] [KO:K06733]
E D09337 Elotuzumab (USAN) <JP/US>
C SIGLEC family
D CD22 (SIGLEC2) [HSA:933] [KO:K06467]
E D08933 Inotuzumab ozogamicin (USAN/INN) <JP/US>
E D09932 Moxetumomab pasudotox (USAN/INN) <US>
E D03066 Bectumomab (USAN/INN)
E D04036 Epratuzumab (USAN/INN)
E D06348 Yttrium Y 90 epratuzumab (USAN)
E D06349 Yttrium Y 90 epratuzumab tetraxetan (USAN)
D CD33 (SIGLEC3) [HSA:945] [KO:K06473]
E D03259 Gemtuzumab ozogamicin (USAN) <JP/US>
E D11294 Vadastuximab (USAN/INN)
E D11295 Vadastuximab talirine (USAN)
E D12141 Emerfetamab (USAN)
E D12152 Eluvixtamab (USAN)
D SIGLEC8 [HSA:27181] [KO:K06748]
E D11906 Lirentelimab (USAN)
C MHC
D MHC1 [HSA:3105 3106 3107 3133 3134 3135] [KO:K06751]
E D04318 Glatiramer acetate (JAN/USAN) <JP/US>
D MHC2 [HSA:3108 3109 3111 3112 3113 3115 3117 3118 3119 3122 3123 3125 3126 3127] [KO:K06752]
E D04318 Glatiramer acetate (JAN/USAN) <JP/US>
D HLA-DRB [HSA:3123 3125 3126 3127] [KO:K06752]
E D02967 Apolizumab (USAN/INN)
C CAMs
D ICAM1 (CD54) [HSA:3383] [KO:K06490]
E D02811 Alicaforsen sodium (USAN)
E D04000 Enlimomab (USAN/INN)
D NCAM1 (CD56) [HSA:4684] [KO:K06491]
E D09927 Lorvotuzumab mertansine (USAN/INN)
D CEACAM [HSA:1048 1084 1087 1088 1089 4680 634 90273] [KO:K06499]
E D04524 Indium In 111 altumomab pentetate (USAN)
E D06028 Technetium Tc 99m arcitumomab (USP)
E D02977 Arcitumomab (USAN/INN)
E D06350 Yttrium Y 90 labetuzumab (USAN)
E D06351 Yttrium Y 90 labetuzumab tetraxetan (USAN)
E D08936 Labetuzumab (INN/USAN)
E D10917 Cergutuzumab amunaleukin (USAN/INN)
E D11110 Cergutuzumab (USAN)
D EPCAM (CD326) [HSA:4072] [KO:K06737]
E D03958 Edrecolomab (USAN/INN)
E D09207 Catumaxomab (INN)
E D09027 Tucotuzumab celmoleukin (USAN/INN)
D VCAM1 [HSA:7412] [KO:K06527]
E D06570 Camobucol (USAN/INN)
E D06582 Elsibucol (USAN/INN)
E D06648 Succinobucol (USAN)
B Cell adhesion molecules: other families
C Selectins
D SEL [HSA:6401 6402 6403] [KO:K06494 K06495 K06496]
E D03114 Bimosiamose disodium (USAN)
D SELE (CD62E) [HSA:6401] [KO:K06494]
E D10487 Rivipansel (USAN/INN)
E D11310 Uproleselan sodium (USAN)
E D11332 Uproleselan (USAN/INN)
D SELP (CD62P) [HSA:6403] [KO:K06496]
E D11480 Crizanlizumab (USAN/INN) <US>
E D06194 Torapsel (USAN/INN)
E D10356 Inclacumab (USAN/INN)
C Collectins
D SFTPD [HSA:6441] [KO:K10068]
E D12333 Zelpultide alfa (USAN)
C Integrins
D ITGA4 (CD49D) [HSA:3676] [KO:K06483]
E D06886 Natalizumab (USAN/INN) <JP/US>
E D06590 Firategrast (USAN)
D ITGAL (CD11A) [HSA:3683] [KO:K05718]
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D03959 Efalizumab (USAN/INN)
E D10374 Lifitegrast (USAN/INN) <US>
E D10392 Lifitegrast sodium (USAN)
E D08993 Rovelizumab (USAN/INN)
D ITGAM (CD11B) [HSA:3684] [KO:K06461]
E D08993 Rovelizumab (USAN/INN)
E D11919 Fuzapladib sodium hydrate (JAN)
D ITGAV (CD51) [HSA:3685] [KO:K06487]
E D09631 Intetumumab (USAN/INN)
D ITGB2 (CD18) [HSA:3689] [KO:K06464]
E D08993 Rovelizumab (USAN/INN)
E D11919 Fuzapladib sodium hydrate (JAN)
D ITGB7 [HSA:3695] [KO:K06590]
E D09901 Etrolizumab (USAN/INN)
D ITGA2B/ITGB3 [HSA:3674 3690] [KO:K06476 K06493]
E D02778 Abciximab (USAN/INN)
E D06888 Eptifibatide (INN) <US>
E D08607 Tirofiban (INN)
E D01029 Tirofiban hydrochloride (USAN) <US>
E D03971 Elarofiban (USAN)
E D04659 Lamifiban (USAN/INN)
E D04660 Lamifiban hydrochloride (USAN)
E D04785 Lotrafiban hydrochloride (USAN)
E D05267 Orbofiban acetate (USAN)
E D05772 Roxifiban acetate (USAN)
E D05834 Sibrafiban (USAN/INN)
E D06335 Xemilofiban hydrochloride (USAN)
E D06649 Tadocizumab (USAN)
E D12051 Zalunfiban (USAN)
E D12163 Zalunfiban acetate (USAN)
D ITGA4/ITGB1 [HSA:3676 3688] [KO:K06483 K05719]
E D09799 Carotegrast methyl (JAN) <JP>
E D10028 Valategrast hydrochloride (USAN)
D ITGA4/ITGB7 [HSA:3676 3695] [KO:K06483 K06590]
E D08083 Vedolizumab (USAN) <JP/US>
E D09799 Carotegrast methyl (JAN) <JP>
E D10028 Valategrast hydrochloride (USAN)
E D10540 Abrilumab (USAN/INN)
D ITGA5/ITGB1 [HSA:3678 3688] [KO:K06484 K05719]
E D06319 Volociximab (USAN)
D ITGAV/ITGB3 [HSA:3685 3690] [KO:K06487 K06493]
E D09342 Etaracizumab (USAN/INN)
E D09929 Maraciclatide (USAN/INN)
D ITGAV-ITGB3/ITGB5 [HSA:3685 3690 3693] [KO:K06487 K06493 K06588]
E D03497 Cilengitide (USAN/INN)
E D09903 Fluciclatide F 18 (USAN/INN)
D ITGB2/ITGAL [HSA:3689 3683] [KO:K06464 K05718]
E D04045 Erlizumab (USAN/INN)
C CAM ligands
D CTGF [HSA:1490] [KO:K06827]
E D10969 Pamrevlumab (USAN/INN)
B Other cell surface molecules
C Immune checkpoints
D CTLA4 (CD152) [HSA:1493] [KO:K06538]
E D04603 Ipilimumab (USAN/INN) <JP/US>
E D06657 Tremelimumab (USAN/INN) <JP/US>
E D11823 Zalifrelimab (USAN/INN)
E D12186 Vudalimab (USAN)
E D12190 Cadonilimab (USAN)
E D12233 Quavonlimab (USAN/INN)
E D12317 Bavunalimab (USAN)
E D12347 Volrustomig (USAN)
E D12448 Botensilimab (USAN/INN)
D PDCD1 (PD1, CD279) [HSA:5133] [KO:K06744]
E D10316 Nivolumab (USAN/INN) <JP/US>
E D10574 Pembrolizumab (USAN) <JP>
E D11108 Cemiplimab (USAN) <JP/US>
E D11366 Dostarlimab (USAN) <US>
E D11487 Tislelizumab (USAN/INN)
E D11827 Retifanlimab (USAN)
E D10390 Pidilizumab (USAN)
E D11488 Cetrelimab (USAN/INN)
E D11605 Spartalizumab (USAN/INN)
E D11643 Budigalimab (USAN/INN)
E D11820 Balstilimab (USAN/INN)
E D11948 Pacmilimab (USAN/INN)
E D12063 Zimberelimab (USAN)
E D12119 Sintilimab (USAN/INN)
E D12186 Vudalimab (USAN)
E D12190 Cadonilimab (USAN)
E D12195 Izuralimab (USAN)
E D12198 Penpulimab (USAN)
E D12202 Toripalimab (USAN/INN)
E D12223 Rosnilimab (USAN)
E D12231 Peresolimab (USAN)
E D12332 Zeluvalimab (USAN/INN)
E D12347 Volrustomig (USAN)
D PDL1 (CD274) [HSA:29126] [KO:K06745]
E D10808 Durvalumab (USAN/INN) <JP/US>
E D10817 Avelumab (USAN) <JP/US>
E D10773 Atezolizumab (USAN/INN) <JP/US>
E D11532 Lodapolimab (USAN)
E D11747 Inbakicept (USAN/INN)
E D11893 Bintrafusp alfa (USAN/INN)
E D11946 Cosibelimab (USAN/INN)
E D12143 Pimivalimab (USAN)
E D12344 Socazolimab (USAN)
E D12349 Danburstotug (USAN)
E D12561 Enristomig (USAN)
C CD molecules
D CD3 [HSA:915 916 917] [KO:K06450 K06451 K06452]
E D09207 Catumaxomab (INN)
E D09325 Blinatumomab (USAN/INN) <JP/US>
E D12296 Tebentafusp (USAN/INN) <US>
E D05092 Muromonab-CD3 (JAN/USAN/INN)
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D06314 Visilizumab (USAN/INN)
E D08959 Otelixizumab (USAN)
E D09013 Teplizumab (USAN/INN) <US>
E D11306 Flotetuzumab (USAN/INN)
D CD3E [HSA:916] [KO:K06451]
E D11372 Duvortuxizumab (USAN)
E D11463 Mosunetuzumab (USAN/INN) <US>
E D11489 Cibisatamab (USAN/INN)
E D11534 Odronextamab (USAN)
E D11686 Plamotamab (USAN/INN)
E D11833 Glofitamab (USAN/INN)
E D11841 Vibecotamab (USAN/INN)
E D11845 Tidutamab (USAN/INN)
E D11984 Cevostamab (USAN/INN)
E D11992 Pavurutamab (USAN)
E D12007 Ubamatamab (USAN)
E D12058 Elranatamab (USAN)
E D12121 Acapatamab (USAN)
E D12177 Teclistamab (USAN/INN) <US>
E D12180 Talquetamab (USAN/INN)
E D12234 Tarlatamab (USAN)
E D12236 Runimotamab (USAN)
E D12368 Epcoritamab (USAN/INN)
E D12567 Imvotamab (USAN/INN)
D CD4 [HSA:920] [KO:K06454]
E D09575 Ibalizumab (USAN/INN) <US>
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D03420 Cedelizumab (USAN/INN)
E D05610 Priliximab (USAN/INN)
E D06356 Zanolimumab (USAN/INN)
D CD5 [HSA:921] [KO:K06455]
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D06381 Zolimomab aritox (USAN)
D CD6 (TP120) [HSA:923] [KO:K06456]
E D12426 Itolizumab (USAN/INN)
D CD7 [HSA:924] [KO:K06457]
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D CD8 [HSA:925 926] [KO:K06458 K06459]
E D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
E D10993 Tucidinostat (JAN/USAN/INN) <JP>
D CD19 [HSA:930] [KO:K06465]
E D09325 Blinatumomab (USAN/INN) <JP/US>
E D11601 Tafasitamab (USAN/INN) <US>
E D11338 Loncastuximab tesirine (USAN) <US>
E D11144 Axicabtagene ciloleucel (USAN) <US>
E D11386 Tisagenlecleucel-T (USAN) <US>
E D11880 Brexucabtagene autoleucel (USAN) <US>
E D11757 Inebilizumab (USAN/INN) <JP/US>
E D11231 Denintuzumab (USAN/INN)
E D11232 Denintuzumab mafodotin (USAN/INN)
E D11333 Loncastuximab (USAN)
E D11372 Duvortuxizumab (USAN)
E D11496 Obexelimab (USAN)
E D11990 Lisocabtagene maraleucel (USAN/INN) <US>
D CD20 [HSA:931] [KO:K06466]
E D02994 Rituximab (USAN/INN) <JP/US>
E D09314 Ofatumumab (USAN/INN) <JP/US>
E D09321 Obinutuzumab (USAN) <JP/US>
E D05218 Ocrelizumab (USAN) <US>
E D11243 Ublituximab (USAN/INN) <US>
E D08622 Tositumomab 131 iodine
E D04489 Ibritumomab tiuxetan (USAN/INN) <JP>
E D08621 Tositumomab (INN)
E D09031 Veltuzumab (USAN)
E D10482 Ocaratuzumab (USAN/INN)
E D11463 Mosunetuzumab (USAN/INN) <US>
E D11534 Odronextamab (USAN)
E D11686 Plamotamab (USAN/INN)
E D11833 Glofitamab (USAN/INN)
E D12368 Epcoritamab (USAN/INN)
E D12567 Imvotamab (USAN/INN)
D CD23 [HSA:2208] [KO:K06468]
E D06463 Lumiliximab (USAN/INN)
D CD28 [HSA:940] [KO:K06470]
E D11281 Reltecimod (USAN/INN)
E D11348 Reltecimod sodium (USAN)
E D12300 Acazicolcept (USAN)
E D12566 Nezastomig (USAN)
D CD34 [HSA:947] [KO:K06474]
E D11930 Betibeglogene autotemcel (USAN/INN) <US>
D CD37 [HSA:951] [KO:K06475]
E D12124 Lilotomab (USAN/INN)
E D12125 Lutetium (177Lu) lilotomab satetraxetan (USAN/INN)
D CD47 [HSA:961] [KO:K06266]
E D11846 Magrolimab (USAN/INN)
E D12193 Evorpacept (USAN)
E D12385 Lemzoparlimab (USAN/INN)
D CD52 [HSA:1043] [KO:K06488]
E D02802 Alemtuzumab (USAN/INN) <JP/US>
D CEACAM5 (CD66e) [HSA:1048] [KO:K06499]
E D11489 Cibisatamab (USAN/INN)
E D12309 Tusamitamab (USAN/INN)
E D12310 Tusamitamab ravtansine (USAN/INN)
D TFRC (CD71) [HSA:7037] [KO:K06503]
E D11812 Pabinafusp alfa (genetical recombination) (JAN) <JP>
E D12509 Trontinemab (USAN/INN)
D CD74 [HSA:972] [KO:K06505]
E D08944 Milatuzumab (USAN)
D CD79B [HSA:974] [KO:K06507]
E D10761 Polatuzumab vedotin (USAN) <JP/US>
D CD80 [HSA:941] [KO:K05412]
E D03203 Abatacept (USAN/INN) <JP/US>
E D03222 Belatacept (USAN/INN) <US>
E D04295 Galiximab (USAN/INN)
E D12463 Davoceticept (USAN/INN)
D LILRA4 [HSA:23547] [KO:K06512]
E D11778 Daxdilimab (USAN)
D CD86 [HSA:942] [KO:K05413]
E D03203 Abatacept (USAN/INN) <JP/US>
E D03222 Belatacept (USAN/INN) <US>
D C5AR1 (CD88) [HSA:728] [KO:K04010]
E D11093 Avacopan (JAN/USAN/INN) <JP/US>
D SEMA4 (CD100) [HSA:10507] [KO:K06521]
E D11469 Pepinemab (USAN)
D ENG (CD105) [HSA:2022] [KO:K06526]
E D11260 Carotuximab (USAN/INN)
D F3 (CD142) [HSA:2152] [KO:K03901]
E D11814 Tisotumab vedotin (USAN/INN) <US>
E D06142 Tifacogin (USAN/INN)
E D11813 Tisotumab (USAN)
D KIR2DL (CD158) [HSA:3802 3803 3804] [KO:K07981]
E D10444 Lirilumab (USAN/INN)
D ALCAM (CD166) [HSA:214] [KO:K06547]
E D11959 Praluzatamab (USAN/INN)
D SIRPA (CD172A) [HSA:140885] [KO:K06551]
E D12342 Anzurstobart (USAN)
D CD200 [HSA:4345] [KO:K06556]
E D09961 Samalizumab (USAN/INN)
D LAG3 (CD223) [HSA:3902] [KO:K06565]
E D11350 Relatlimab (USAN)
E D12156 Ieramilimab (USAN/INN)
E D12317 Bavunalimab (USAN)
E D12469 Favezelimab (INN/USAN)
E D12480 Tuparstobart (USAN)
D MUC1 (CD227) [HSA:4582] [KO:K06568]
E D06028 Technetium Tc 99m arcitumomab (USP)
E D02977 Arcitumomab (USAN/INN)
E D09700 Yttrium Y 90 clivatuzumab tetraxetan (USAN)
E D09895 Emepepimut-S (USAN)
D RHD (CD240D) [HSA:6007] [KO:K06579]
E D09663 Rozrolimupab (USAN)
D CD244 [HSA:51744] [KO:K06582]
E D10993 Tucidinostat (JAN/USAN/INN) <JP>
D BTLA (CD272) [HSA:151888] [KO:K06707]
E D12546 Venanprubart (USAN)
D ICOSLG (CD275) [HSA:23308] [KO:K06710]
E D11907 Rozibafusp alfa (USAN/INN)
D CD276 [HSA:80381] [KO:K06746]
E D11515 Omburtamab (USAN/INN)
E D11752 Enoblituzumab (USAN/INN)
E D12154 Mirzotamab (USAN/INN)
E D12517 Vobramitamab (USAN/INN)
E D12518 Voramitamab duocarmazine (USAN/INN)
D ICOS (CD278) [HSA:29851] [KO:K06713]
E D11433 Vopratelimab (USAN/INN)
E D11996 Feladilimab (USAN/INN)
E D12195 Izuralimab (USAN)
E D12300 Acazicolcept (USAN)
D NRP1 (CD304) [HSA:8829] [KO:K06724]
E D10494 Vesencumab (USAN/INN)
D KLRK1 (CD314, NKG2D) [HSA:22914] [KO:K06728]
E D12179 Tesnatilimab (USAN/INN)
D HAVCR2 (CD366) [HSA:84868] [KO:K20414]
E D12164 Sabatolimab (USAN/INN)
E D11377 Cobolimab (USAN)
E D12429 Surzebiclimab (USAN/INN)
C Other
D MUC16 (CA125) [HSA:94025] [KO:K16145]
E D05269 Oregovomab (USAN/INN)
E D11240 Sofituzumab (USAN)
E D11241 Sofituzumab vedotin (USAN/INN)
E D12007 Ubamatamab (USAN)
D TACSTD2 (TROP2) [HSA:4070] [KO:K17288]
E D10985 Sacituzumab govitecan (USAN/INN) <US>
E D12359 Datopotamab deruxtecan (USAN/INN)
E D12360 Datopotamab (USAN/INN)
D TIGIT [HSA:201633] [KO:K16350]
E D11482 Tiragolumab (USAN/INN)
E D11593 Etigilimab (USAN/INN)
E D11795 Vibostolimab (USAN)
E D12283 Ociperlimab (USAN/INN)
E D12348 Belrestotug (USAN)
E D12367 Domvanalimab (USAN/INN)
D VSIR (VISTA) [HSA:64115] [KO:K23268]
E D11474 Onvatilimab (USAN/INN)
D CLDN18 [HSA:51208] [KO:K06087]
E D11527 Zolbetuximab (USAN/INN)
D PVRL4 (NECTIN4) [HSA:81607] [KO:K06593]
E D11525 Enfortumab vedotin (USAN) <JP/US>
E D11524 Enfortumab (USAN)
#
ATransporters
B ABC transporters
C ABCC subfamily
D ABCC8 (SUR1) [HSA:6833] [KO:K05032]
E D02427 Glibornuride (USAN/INN)
E D02425 Carbutamide (INN)
E D00335 Glipizide (USP/INN) <US>
E D02430 Gliquidone (INN)
E D01599 Gliclazide (JP18/INN) <JP>
E D07117 Metahexamide (INN)
E D07118 Glisoxepide (INN)
E D00593 Glimepiride (JP18/USP/INN) <JP/US>
E D00219 Acetohexamide (JP18/USP/INN) <JP>
E D01799 Glyclopyramide (JAN/INN) <JP>
D ABCC8(SUR1)/KCNJ11(KIR6.2) [HSA:6833 3767] [KO:K05032 K05004]
E D00336 Glyburide (USP) <JP/US>
E D00271 Chlorpropamide (JP18/USP/INN) <JP>
E D00380 Tolbutamide (JP18/USP/INN)
E D06177 Tolbutamide sodium, sterile
E D00379 Tolazamide (JAN/USP/INN)
E D01356 Glymidine sodium (JAN/USAN/INN)
E D00594 Repaglinide (JAN/USP/INN) <JP/US>
E D01111 Nateglinide (JP18/USP/INN) <JP/US>
E D01854 Mitiglinide calcium hydrate (JP18) <JP>
E D01810 Nicorandil (JP18/USAN/INN) <JP>
E D00294 Diazoxide (JAN/USP/INN) <JP/US>
E D00418 Minoxidil (JAN/USP/INN) <US>
E D05482 Pinacidil (USAN)
E D02385 Levcromakalim (USAN/INN)
E D04739 Linogliride (USAN/INN)
E D04740 Linogliride fumarate (USAN)
E D05114 Naminidil (USAN/INN)
D ABCC9(SUR2)/KCNJ11(KIR6.2) [HSA:10060 3767] [KO:K05033 K05004]
E D01810 Nicorandil (JP18/USAN/INN) <JP>
E D05482 Pinacidil (USAN)
E D02385 Levcromakalim (USAN/INN)
E D05114 Naminidil (USAN/INN)
D CFTR (ABCC7) [HSA:1080] [KO:K05031]
E D03605 Crofelemer (USAN) <US>
E D09916 Ivacaftor (USAN/INN) <US>
E D10134 Lumacaftor (USAN)
E D11041 Tezacaftor (USAN/INN)
E D11402 Olacaftor (USAN)
E D11423 Deutivacaftor (USAN/INN)
E D11507 Elexacaftor (USAN)
E D11535 Bamocaftor (USAN)
E D11536 Bamocaftor potassium (USAN)
E D11682 Nesolicaftor (USAN)
E D11683 Posenacaftor (USAN)
E D11724 Galicaftor (USAN/INN)
E D12140 Navocaftor (USAN/INN)
E D12454 Icenticaftor (USAN/INN)
D CFTR* [HSA_VAR:1080v1] [HSA:1080] [KO:K05031]
E D10685 Lumacaftor and ivacaftor <US>
E D11042 Tezacaftor and ivacaftor <US>
E D11700 Elexacaftor, ivacaftor and tezacaftor <US>
C ABCD (ALD) subfamily
D ABCD1 (ALDP) [HSA:215] [KO:K05675]
E D12150 Elivaldogene autotemcel (USAN/INN) <US>
B Solute carrier family
C SLC5
D SLC5A1 (SGLT1) [HSA:6523] [KO:K14158]
E D10669 Sotagliflozin (USAN/INN)
D SLC5A2 (SGLT2) [HSA:6524] [KO:K14382]
E D08897 Dapagliflozin (USAN/INN)
E D09763 Dapagliflozin propanediol (USAN) <JP/US>
E D09592 Canagliflozin (USAN/INN) <JP/US>
E D10459 Empagliflozin (JAN/USAN/INN) <JP/US>
E D10313 Ertugliflozin (USAN/INN)
E D11043 Ertugliflozin pidolate <US>
E D10196 Ipragliflozin (INN) <US>
E D10200 Ipragliflozin L-proline (JAN) <JP>
E D10669 Sotagliflozin (USAN/INN)
E D10195 Luseogliflozin hydrate (JAN) <JP>
E D06641 Sergliflozin etabonate (USAN)
E D09978 Tofogliflozin (USAN) <JP>
E D10055 Remogliflozin etabonate (USAN/INN)
E D10865 Bexagliflozin (USAN)
C SLC6
D SLC6A1 (GAT1) [HSA:6529] [KO:K05034]
E D00332 Gabapentin (JAN/USP/INN) <JP/US>
E D09539 Gabapentin enacarbil (JAN/USAN/INN) <JP/US>
E D08588 Tiagabine (INN)
E D02097 Tiagabine hydrochloride (USP) <US>
D SLC6A2 (NAT1) [HSA:6530] [KO:K05035]
E D05458 Phentermine (USAN/INN)
E D05459 Phentermine hydrochloride (USP) <US>
E D07444 Amfepramone (INN)
E D03801 Diethylpropion hydrochloride (USP) <US>
E D00367 Mazindol (JAN/USP/INN) <JP>
E D08513 Sibutramine (INN)
E D02571 Sibutramine hydrochloride (USP)
E D01304 Amezinium metilsulfate (JAN) <JP>
E D08030 Guanethidine (INN)
E D02237 Guanethidine sulfate (USAN)
E D04382 Guanethidine monosulfate (USP)
E D07875 Doxepin (INN)
E D00814 Doxepin hydrochloride (USP) <US>
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D06007 Tapentadol (USAN/INN)
E D10199 Tapentadol hydrochloride (JAN) <JP/US>
E D07791 Desipramine (INN)
E D00812 Desipramine hydrochloride (JAN/USP) <US>
E D08070 Imipramine (INN)
E D00815 Imipramine hydrochloride (JP18/USP) <JP/US>
E D08071 Imipramine pamoate (USP) <US>
E D07727 Clomipramine (INN)
E D00811 Clomipramine hydrochloride (JP18/USP) <JP/US>
E D00394 Trimipramine (USAN/INN)
E D02408 Trimipramine maleate (JAN/USP) <JP/US>
E D08140 Lofepramine (INN)
E D01285 Lofepramine hydrochloride (JAN/USAN) <JP>
E D07448 Amitriptyline (INN)
E D00809 Amitriptyline hydrochloride (JP18/USP) <JP/US>
E D08288 Nortriptyline (INN)
E D00816 Nortriptyline hydrochloride (JP18/USP/INN) <JP/US>
E D08447 Protriptyline (INN)
E D00484 Protriptyline hydrochloride (USP) <US>
E D07872 Dosulepin (INN)
E D01546 Dothiepin hydrochloride (USAN) <JP>
E D00228 Amoxapine (JP18/USP/INN) <JP/US>
E D02566 Maprotiline (USAN)
E D00818 Maprotiline hydrochloride (JP18/USP) <JP>
E D05200 Nomifensine maleate (USAN)
E D08673 Viloxazine (INN)
E D02572 Viloxazine hydrochloride (USAN) <US>
E D07591 Bupropion (INN)
E D00817 Bupropion hydrochloride (JAN/USP) <US>
E D07938 Bupropion hydrobromide (USAN) <US>
E D08670 Venlafaxine (INN) <US>
E D00821 Venlafaxine hydrochloride (JAN/USP) <JP/US>
E D12403 Venlafaxine besylate monohydrate <US>
E D08222 Milnacipran (INN)
E D01107 Milnacipran hydrochloride (JAN/USAN) <JP/US>
E D08472 Reboxetine (INN)
E D02573 Reboxetine mesylate (USAN)
E D07880 Duloxetine (INN)
E D01179 Duloxetine hydrochloride (JAN/USP) <JP/US>
E D07793 Desvenlafaxine (INN) <US>
E D02570 Desvenlafaxine succinate (USAN) <US>
E D11619 Desvenlafaxine succinate anhydrous <US>
E D10072 Levomilnacipran (USAN/INN)
E D10133 Levomilnacipran hydrochloride (USAN) <US>
E D07445 Amfetamine (INN) <US>
E D02074 Amphetamine sulfate (USP) <US>
E D03740 Dextroamphetamine (USAN) <US>
E D02078 Dextroamphetamine sulfate (USP) <US>
E D08187 Metamfetamine (INN)
E D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
E D04999 Methylphenidate (USAN/INN) <US>
E D01296 Methylphenidate hydrochloride (JAN/USP) <JP/US>
E D07473 Atomoxetine (USP/INN)
E D02574 Atomoxetine hydrochloride (JAN/USP) <JP/US>
E D07806 Dexmethylphenidate (INN)
E D03721 Dexmethylphenidate hydrochloride (USAN) <US>
E D08130 Lisdexamfetamine (INN)
E D04747 Lisdexamfetamine dimesylate (USAN) <JP/US>
E D11315 Solriamfetol (USAN)
E D11328 Solriamfetol hydrochloride (USAN) <US>
E D02080 Phendimetrazine tartrate (USP) <US>
E D02170 Indeloxazine hydrochloride (JAN/USAN)
E D02704 Tampramine fumarate (USAN)
E D03491 Cidoxepin hydrochloride (USAN)
E D04473 Hydroxyamphetamine hydrobromide (USP)
E D04781 Lortalamine (USAN/INN)
E D05119 Napamezole hydrochloride (USAN)
E D05120 Napitane mesylate (USAN)
E D05173 Nisoxetine (USAN/INN)
E D05284 Oxaprotiline hydrochloride (USAN)
E D05454 Phenmetrazine hydrochloride (USP)
E D05663 Pyrovalerone hydrochloride (USAN)
E D05692 Radafaxine hydrochloride (USAN)
E D05997 Talopram hydrochloride (USAN)
E D06004 Tandamine hydrochloride (USAN)
E D07334 Imipraminoxide (INN)
E D07449 Amitriptylinoxide (INN)
E D07514 Benzfetamine (INN)
E D07515 Benzfetamine hydrochloride <US>
E D08072 Imipraminoxide hydrochloride
E D08077 Indeloxazine (INN)
E D08347 Phendimetrazine (INN)
E D08348 Phendimetrazine hydrochloride
E D09340 Esreboxetine (USAN/INN)
E D09341 Esreboxetine succinate (USAN)
E D09890 Edivoxetine (USAN/INN)
E D09891 Edivoxetine hydrochloride (USAN)
E D10088 Amitifadine (USAN)
E D10089 Amitifadine hydrochloride (USAN)
E D10443 Liafensine (USAN)
E D10697 Centanafadine (USAN)
E D10698 Centanafadine hydrochloride (USAN)
E D10700 Dasotraline (USAN/INN)
E D10870 Dasotraline hydrochloride (USAN)
E D11172 Midomafetamine (USAN/INN)
E D11622 Amphetamine aspartate monohydrate
E D11623 Dextroamphetamine saccharate
E D11688 Ampreloxetine (USAN/INN)
E D11689 Ampreloxetine hydrochloride (USAN)
E D11940 Toludesvenlafaxine (USAN/INN)
E D11941 Toludesvenlafaxine hydrochloride (USAN)
D SLC6A3 (DAT1) [HSA:6531] [KO:K05036]
E D05458 Phentermine (USAN/INN)
E D05459 Phentermine hydrochloride (USP) <US>
E D07444 Amfepramone (INN)
E D03801 Diethylpropion hydrochloride (USP) <US>
E D00367 Mazindol (JAN/USP/INN) <JP>
E D08513 Sibutramine (INN)
E D02571 Sibutramine hydrochloride (USP)
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D07591 Bupropion (INN)
E D00817 Bupropion hydrochloride (JAN/USP) <US>
E D07938 Bupropion hydrobromide (USAN) <US>
E D07445 Amfetamine (INN) <US>
E D02074 Amphetamine sulfate (USP) <US>
E D03740 Dextroamphetamine (USAN) <US>
E D02078 Dextroamphetamine sulfate (USP) <US>
E D08187 Metamfetamine (INN)
E D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
E D04999 Methylphenidate (USAN/INN) <US>
E D01296 Methylphenidate hydrochloride (JAN/USP) <JP/US>
E D07806 Dexmethylphenidate (INN)
E D03721 Dexmethylphenidate hydrochloride (USAN) <US>
E D08130 Lisdexamfetamine (INN)
E D04747 Lisdexamfetamine dimesylate (USAN) <JP/US>
E D03215 Armodafinil (USAN/INN) <US>
E D11315 Solriamfetol (USAN)
E D11328 Solriamfetol hydrochloride (USAN) <US>
E D10014 Ioflupane I 123 (USAN) <JP/US>
E D02897 Amfonelic acid (USAN)
E D03153 Brasofensine maleate (USAN)
E D05119 Napamezole hydrochloride (USAN)
E D05454 Phenmetrazine hydrochloride (USP)
E D05663 Pyrovalerone hydrochloride (USAN)
E D05692 Radafaxine hydrochloride (USAN)
E D07514 Benzfetamine (INN)
E D07515 Benzfetamine hydrochloride <US>
E D10088 Amitifadine (USAN)
E D10089 Amitifadine hydrochloride (USAN)
E D10697 Centanafadine (USAN)
E D10698 Centanafadine hydrochloride (USAN)
E D10700 Dasotraline (USAN/INN)
E D10870 Dasotraline hydrochloride (USAN)
E D11172 Midomafetamine (USAN/INN)
E D11622 Amphetamine aspartate monohydrate
E D11623 Dextroamphetamine saccharate
D SLC6A4 (HTT) [HSA:6532] [KO:K05037]
E D05458 Phentermine (USAN/INN)
E D05459 Phentermine hydrochloride (USP) <US>
E D07945 Fenfluramine (INN)
E D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
E D07805 Dexfenfluramine (INN)
E D03713 Dexfenfluramine hydrochloride (USAN)
E D00367 Mazindol (JAN/USP/INN) <JP>
E D08513 Sibutramine (INN)
E D02571 Sibutramine hydrochloride (USP)
E D07875 Doxepin (INN)
E D00814 Doxepin hydrochloride (USP) <US>
E D03649 Dapoxetine hydrochloride (USAN)
E D00110 Cocaine (USP)
E D02182 Cocaine hydrochloride (JP18/USP) <JP/US>
E D07791 Desipramine (INN)
E D00812 Desipramine hydrochloride (JAN/USP) <US>
E D08070 Imipramine (INN)
E D00815 Imipramine hydrochloride (JP18/USP) <JP/US>
E D08071 Imipramine pamoate (USP) <US>
E D07727 Clomipramine (INN)
E D00811 Clomipramine hydrochloride (JP18/USP) <JP/US>
E D00394 Trimipramine (USAN/INN)
E D02408 Trimipramine maleate (JAN/USP) <JP/US>
E D08140 Lofepramine (INN)
E D01285 Lofepramine hydrochloride (JAN/USAN) <JP>
E D07448 Amitriptyline (INN)
E D00809 Amitriptyline hydrochloride (JP18/USP) <JP/US>
E D08288 Nortriptyline (INN)
E D00816 Nortriptyline hydrochloride (JP18/USP/INN) <JP/US>
E D08447 Protriptyline (INN)
E D00484 Protriptyline hydrochloride (USP) <US>
E D07872 Dosulepin (INN)
E D01546 Dothiepin hydrochloride (USAN) <JP>
E D00228 Amoxapine (JP18/USP/INN) <JP/US>
E D00326 Fluoxetine (USAN/INN)
E D00823 Fluoxetine hydrochloride (JAN/USP) <US>
E D07704 Citalopram (USP/INN)
E D00822 Citalopram hydrobromide (USP) <US>
E D07705 Citalopram hydrochloride
E D02362 Paroxetine (USP/INN)
E D02260 Paroxetine hydrochloride hemihydrate (USP) <JP/US>
E D05374 Paroxetine hydrochloride (USP) <US>
E D05375 Paroxetine mesylate (USAN) <US>
E D02360 Sertraline (INN)
E D00825 Sertraline hydrochloride (JAN/USP) <JP/US>
E D02787 Alaproclate (USAN/INN)
E D07984 Fluvoxamine (INN)
E D00824 Fluvoxamine maleate (JP18/USP) <JP/US>
E D07913 Escitalopram (INN)
E D02567 Escitalopram oxalate (JAN/USP) <JP/US>
E D08626 Trazodone (INN)
E D00820 Trazodone hydrochloride (JAN/USP) <JP/US>
E D08670 Venlafaxine (INN) <US>
E D00821 Venlafaxine hydrochloride (JAN/USP) <JP/US>
E D12403 Venlafaxine besylate monohydrate <US>
E D08222 Milnacipran (INN)
E D01107 Milnacipran hydrochloride (JAN/USAN) <JP/US>
E D07880 Duloxetine (INN)
E D01179 Duloxetine hydrochloride (JAN/USP) <JP/US>
E D07793 Desvenlafaxine (INN) <US>
E D02570 Desvenlafaxine succinate (USAN) <US>
E D11619 Desvenlafaxine succinate anhydrous <US>
E D09698 Vilazodone (USAN/INN)
E D09699 Vilazodone hydrochloride (USAN) <US>
E D10184 Vortioxetine (USAN)
E D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
E D12544 Vortioxetine hemihydrobromide (USAN)
E D10072 Levomilnacipran (USAN/INN)
E D10133 Levomilnacipran hydrochloride (USAN) <US>
E D08187 Metamfetamine (INN)
E D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
E D07806 Dexmethylphenidate (INN)
E D03721 Dexmethylphenidate hydrochloride (USAN) <US>
E D02170 Indeloxazine hydrochloride (JAN/USAN)
E D03491 Cidoxepin hydrochloride (USAN)
E D04788 Lubazodone hydrochloride (USAN)
E D05491 Pirandamine hydrochloride (USAN)
E D07334 Imipraminoxide (INN)
E D07449 Amitriptylinoxide (INN)
E D08072 Imipraminoxide hydrochloride
E D08077 Indeloxazine (INN)
E D10088 Amitifadine (USAN)
E D10089 Amitifadine hydrochloride (USAN)
E D10443 Liafensine (USAN)
E D10697 Centanafadine (USAN)
E D10698 Centanafadine hydrochloride (USAN)
E D11172 Midomafetamine (USAN/INN)
E D11688 Ampreloxetine (USAN/INN)
E D11689 Ampreloxetine hydrochloride (USAN)
E D11940 Toludesvenlafaxine (USAN/INN)
E D11941 Toludesvenlafaxine hydrochloride (USAN)
D SLC6A9 (GLYT1) [HSA:6536] [KO:K05038]
E D10186 Bitopertin (JAN/USAN)
E D12527 Iclepertin (JAN/USAN/INN)
C SLC7
D SLC7A5 (LAT1) [HSA:8140] [KO:K13780]
E D12443 Nanvuranlat hydrochloride hydrate (JAN)
C SLC9
D SLC9A1 (NHE1) [HSA:6548] [KO:K05742]
E D03406 Cariporide mesylate (USAN)
E D09036 Zoniporide mesylate (INN/USAN)
D SLC9A3 (NHE3) [HSA:6550] [KO:K12040]
E D11652 Tenapanor (USAN/INN)
E D11653 Tenapanor hydrochloride (JAN/USAN) <US>
C SLC10
D SLC10A [HSA:6554 6555 8273 347051 201780 345274 84068] [KO:K14341 K14342 K14343 K14344 K14346 K14347]
E D10951 Maralixibat (USAN)
D SLC10A2 (ASBT, IBAT) [HSA:6555] [KO:K14342]
E D10952 Maralixibat chloride (USAN/INN) <US>
E D11716 Odevixibat (USAN) <US>
E D10796 Elobixibat (USAN/INN)
E D10795 Elobixibat hydrate (JAN) <JP>
E D11539 Linerixibat (JAN/USAN)
C SLC12
D SLC12A1 (NKCC2) [HSA:6557] [KO:K14425]
E D00654 Hydroflumethiazide (JAN/USP/INN)
E D00658 Trichlormethiazide (JP18/USP/INN) <JP>
E D00656 Methyclothiazide (JAN/USP/INN)
E D00461 Quinethazone (JAN/INN)
E D00272 Chlorthalidone (USP) <US>
E D00331 Furosemide (JP18/USP/INN) <JP/US>
E D07999 Sodium furosemide
E D08001 Furosemide diolamine
E D00247 Bumetanide (JP18/USP/INN) <US>
E D01634 Piretanide (JAN/USAN/INN)
E D00382 Torsemide (USP) <JP/US>
E D08619 Torasemide sodium
E D00313 Ethacrynic acid (USP) <US>
E D04079 Ethacrynate sodium (USP) <US>
E D02386 Ticrynafen (USAN)
E D05093 Muzolimine (USAN/INN)
E D04111 Etozolin (USAN/INN)
E D01323 Azosemide (JP18/USAN/INN) <JP>
E D02453 Flumethiazide (INN)
E D09772 Alilusem potassium (JAN)
D SLC12A2 (NKCC1) [HSA:6558] [KO:K10951]
E D00331 Furosemide (JP18/USP/INN) <JP/US>
E D07999 Sodium furosemide
E D08001 Furosemide diolamine
E D00247 Bumetanide (JP18/USP/INN) <US>
E D01634 Piretanide (JAN/USAN/INN)
E D00382 Torsemide (USP) <JP/US>
E D08619 Torasemide sodium
E D00313 Ethacrynic acid (USP) <US>
E D04079 Ethacrynate sodium (USP) <US>
E D02386 Ticrynafen (USAN)
E D05093 Muzolimine (USAN/INN)
E D04111 Etozolin (USAN/INN)
E D01323 Azosemide (JP18/USAN/INN) <JP>
E D09772 Alilusem potassium (JAN)
D SLC12A3 (TSC) [HSA:6559] [KO:K14426]
E D00650 Bendroflumethiazide (JAN/USP/INN)
E D00654 Hydroflumethiazide (JAN/USP/INN)
E D00340 Hydrochlorothiazide (JP18/USP/INN) <JP/US>
E D00519 Chlorothiazide (JAN/USP/INN) <US>
E D03471 Chlorothiazide sodium (USP) <US>
E D00657 Polythiazide (JAN/USAN/INN)
E D00658 Trichlormethiazide (JP18/USP/INN) <JP>
E D00656 Methyclothiazide (JAN/USP/INN)
E D00461 Quinethazone (JAN/INN)
E D00272 Chlorthalidone (USP) <US>
E D01877 Mefruside (JP18/USAN/INN) <JP>
E D00431 Metolazone (JAN/USP/INN) <US>
E D01605 Meticrane (JP18/INN)
E D00345 Indapamide (JP18/USP) <JP/US>
E D06401 Indapamide hydrate
E D00651 Benzthiazide (JAN/INN)
E D01241 Penflutizide (JAN/INN)
E D01246 Benzylhydrochlorothiazide (JAN) <JP>
E D01895 Tripamide (JAN/USAN/INN) <JP>
E D02453 Flumethiazide (INN)
D SLC12A4 [HSA:6560] [KO:K14427]
E D00247 Bumetanide (JP18/USP/INN) <US>
C SLC18
D SLC18A1 (VMAT1) [HSA:6570] [KO:K08155]
E D00197 Reserpine (JP18/USP/INN)
E D08187 Metamfetamine (INN)
E D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
E D10170 Tedatioxetine (USAN)
E D10171 Tedatioxetine hydrobromide (USAN)
D SLC18A2 (VMAT2) [HSA:6571] [KO:K08155]
E D07097 Isometheptene mucate (USP)
E D00197 Reserpine (JP18/USP/INN)
E D07445 Amfetamine (INN) <US>
E D02074 Amphetamine sulfate (USP) <US>
E D03740 Dextroamphetamine (USAN) <US>
E D02078 Dextroamphetamine sulfate (USP) <US>
E D08187 Metamfetamine (INN)
E D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
E D08575 Tetrabenazine (JAN/INN) <JP/US>
E D10675 Valbenazine (USAN/INN)
E D10999 Valbenazine tosylate (USAN) <JP/US>
E D10701 Deutetrabenazine (USAN/INN) <US>
E D07514 Benzfetamine (INN)
E D07515 Benzfetamine hydrochloride <US>
E D10170 Tedatioxetine (USAN)
E D10171 Tedatioxetine hydrobromide (USAN)
E D11172 Midomafetamine (USAN/INN)
E D11622 Amphetamine aspartate monohydrate
E D11623 Dextroamphetamine saccharate
C SLC22
D OAT4 [HSA:55867] [KO:K08207]
E D09921 Lesinurad (USAN/INN)
E D09922 Lesinurad sodium (USAN)
D URAT1 [HSA:116085] [KO:K08208]
E D01056 Benzbromarone (JP18/USAN/INN) <JP>
E D09921 Lesinurad (USAN/INN)
E D09922 Lesinurad sodium (USAN)
E D11129 Verinurad (USAN/INN)
C SLC29
D SLC29A1 (ENT1) [HSA:2030] [KO:K15014]
E D07843 Dilazep (INN)
E D02631 Dilazep dihydrochloride hydrate (JP18) <JP>
E D03906 Draflazine (USAN/INN)
C SLC34
D SLC34A2 [HSA:10568] [KO:K14683]
E D11237 Lifastuzumab (USAN)
E D11238 Lifastuzumab vedotin (USAN/INN)
C SLC40
D SLC40A1 (FPN1, IREG1) [HSA:30061] [KO:K14685]
E D12289 Vamifeport (USAN/INN)
E D12290 Vamifeport trihydrochloride (USAN)
B Major facilitator superfamily
C VNT family
D SV2 [HSA:9900 9899 22987] [KO:K06258]
E D11842 Padsevonil (JAN/USAN)
D SV2A [HSA:9900] [KO:K06258]
E D00709 Levetiracetam (JAN/USP/INN) <JP/US>
E D08879 Brivaracetam (JAN/USAN/INN) <US>
E D01914 Piracetam (JAN/USAN/INN) <JP>
E D05817 Seletracetam (USAN/INN)
B Other transporters
C Channels and pores (TC:1)
D CETP [HSA:1071] [KO:K16835]
E D05255 Omega-3-acid ethyl esters (USP) <JP/US>
E D06195 Torcetrapib (USAN/INN)
E D08855 Anacetrapib (JAN/USAN)
E D09708 Dalcetrapib (USAN/INN)
E D10121 Evacetrapib (USAN)
D XPO1 [HSA:7514] [KO:K14290]
E D11222 Selinexor (USAN/INN) <US>
E D11223 Verdinexor (USAN/INN)
E D11499 Eltanexor (USAN/INN)
C Auxiliary transport proteins (TC:8.A)
D SIGMAR1 [HSA:10280] [KO:K20719]
E D07945 Fenfluramine (INN)
E D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
E D07316 Captodiame (BAN)
E D08297 Opipramol (INN)
E D01477 Opipramol hydrochloride (JAN/USAN)
E D03742 Dextromethorphan (USP)
E D00848 Dextromethorphan hydrobromide (USP) <JP>
E D03744 Dextromethorphan polistirex (USAN)
E D02684 Rimcazole hydrochloride (USAN)
E D02688 Tiospirone hydrochloride (USAN)
E D04502 Igmesine hydrochloride (USAN)
E D11383 Blarcamesine (USAN)
E D11549 Blarcamesine hydrochloride (USAN)
D KLB [HSA:152831] [KO:K22404]
E D12490 Fazpilodemab (USAN/INN)
C Others
D TTR [HSA:7276] [KO:K20731]
E D09673 Tafamidis (JAN/USAN/INN) <JP>
E D09674 Tafamidis meglumine (JAN/USAN) <JP/US>
E D11116 Patisiran (USAN/INN)
E D10794 Patisiran sodium (JAN) <JP/US>
E D10940 Inotersen (USAN/INN)
E D10941 Inotersen sodium (USAN) <US>
E D11917 Vutrisiran (USAN/INN)
E D11916 Vutrisiran sodium (JAN) <JP/US>
E D11972 Acoramidis (USAN)
E D11973 Acoramidis hydrochloride (JAN/USAN)
D FOLR [HSA:2348 2350 2352] [KO:K13649]
E D10434 Vintafolide (USAN/INN)
E D12249 Pafolacianine (USAN)
E D12250 Pafolacianine sodium (USAN) <US>
D FOLR1 [HSA:2348] [KO:K13649]
E D09343 Farletuzumab (USAN)
E D10953 Mirvetuximab (USAN/INN)
E D10954 Mirvetuximab soravtansine (USAN/INN) <US>
E D12183 Farletuzumab ecteribulin (USAN)
D NPC1L1 [HSA:29881] [KO:K14461]
E D01966 Ezetimibe (JAN/USP/INN) <JP/US>
#
AEnzymes
B Oxidoreductases (EC1)
C Dehydrogenases [EC:1.1.1.-]
D ADH [HSA:124 125 126] [KO:K13951]
E D00707 Fomepizole (JAN/USAN/INN) <JP/US>
D AKR1B1 [HSA:231] [KO:K00011]
E D02323 Tolrestat (USAN/INN)
E D01688 Epalrestat (JP18/INN) <JP>
E D01715 Risarestat (INN)
E D01842 Fidarestat (JAN/INN)
E D02328 Zopolrestat (USAN/INN)
E D02835 Alrestatin sodium (USAN)
E D03803 Lidorestat (USAN)
E D03805 Minalrestat (USAN/INN)
E D03806 Ponalrestat (USAN/INN)
E D03807 Zenarestat (USAN/INN)
E D05893 Sorbinil (USAN/INN)
E D06403 Ranirestat (JAN/INN)
E D12384 Govorestat (USAN/INN)
E D12390 Caficrestat (USAN/INN)
D HMGCR [HSA:3156] [KO:K00021]
E D00434 Simvastatin (JP18/USP/INN) <JP/US>
E D00359 Lovastatin (USP/INN) <US>
E D08410 Pravastatin (INN)
E D00893 Pravastatin sodium (JP18/USP) <JP/US>
E D07983 Fluvastatin (INN)
E D00892 Fluvastatin sodium (JAN/USP) <JP/US>
E D07474 Atorvastatin (INN) <US>
E D00887 Atorvastatin calcium anhydorous
E D02258 Atorvastatin calcium (USP) <JP/US>
E D11095 Atorvastatin calcium propylene glycol solvate <US>
E D07661 Cerivastatin (INN)
E D00889 Cerivastatin sodium (JAN/USAN)
E D08492 Rosuvastatin (INN)
E D01915 Rosuvastatin calcium (JP18/USP) <JP/US>
E D01862 Pitavastatin calcium (JAN) <JP/US>
E D10568 Pitavastatin calcium hydrate (JP18) <JP>
E D11092 Pitavastatin magnesium <US>
E D03601 Crilvastatin (USAN/INN)
E D03643 Dalvastatin (USAN/INN)
E D03816 Tenivastatin calcium (USAN)
D IDH [HSA:3417 3418] [KO:K00031]
E D11834 Vorasidenib (USAN/INN)
E D11835 Vorasidenib citrate (USAN)
D IDH1* [HSA_VAR:3417v1] [HSA:3417] [KO:K00031]
E D11090 Ivosidenib (JAN/USAN/INN) <US>
E D12483 Olutasidenib (USAN/INN) <US>
D IDH2 [HSA:3418] [KO:K00031]
E D10901 Enasidenib (USAN/INN)
D IDH2* [HSA_VAR:3418v1] [HSA:3418] [KO:K00031]
E D11044 Enasidenib mesylate (USAN) <US>
D HSD3B [HSA:3283 3284] [KO:K00070]
E D01180 Trilostane (JAN/USAN) <JP>
E D04035 Epostane (USAN/INN)
D HSD11B1 [HSA:3290] [KO:K15680]
E D07615 Carbenoxolone (INN)
E D01899 Carbenoxolone sodium (JAN/USAN)
E D00156 Glycyrrhetinic acid (JAN) <JP>
E D02028 Diammonium glycyrrhizinate (JAN)
E D02264 Dipotassium glycyrrhizinate (JAN) <JP>
E D04987 Monoammonium glycyrrhizinate (JAN)
D IMPDH [HSA:3614 3615] [KO:K00088]
E D06130 Tiazofurin (USAN)
E D05096 Mycophenolic acid (USAN/INN)
E D00752 Mycophenolate mofetil (JAN/USP) <JP/US>
E D05094 Mycophenolate mofetil hydrochloride (USAN) <US>
E D05095 Mycophenolate sodium (USP) <US>
E D01392 Mizoribine (JP18/INN) <JP>
E D04936 Merimepodib (USAN/INN)
C Oxidases [EC:1.1.3.-]
D HAO1 [HSA:54363] [KO:K11517]
E D11925 Lumasiran (USAN/INN)
E D11926 Lumasiran sodium <US>
C Dehydrogenases [EC:1.2.1.-]
D ALDH [HSA:217 219 224] [KO:K00128]
E D00131 Disulfiram (JP18/USP/INN) <JP/US>
E D00123 Cyanamide (JP18) <JP>
D SSADH [HSA:7915] [KO:K00139]
E D00399 Valproic acid (USP) <US>
E D00304 Divalproex sodium (USP) <US>
E D00710 Valproate sodium (USAN) <JP/US>
E D08667 Calcium valproate
C Dehydrogenases [EC:1.3.-.-]
D DPYD [HSA:1806] [KO:K00207]
E D01846 Gimeracil (JAN/INN)
E D03998 Eniluracil (USAN/INN)
D SRD5A1 [HSA:6715] [KO:K12343]
E D03820 Dutasteride (JAN/USP/INN) <JP/US>
E D01134 Epristeride (JAN/USAN/INN)
E D03107 Bexlosteride (USAN/INN)
E D04498 Idronoxil (USAN/INN)
E D04646 Izonsteride (USAN/INN)
E D07121 Alfatradiol (INN)
D SRD5A2 [HSA:6716] [KO:K12344]
E D00321 Finasteride (JAN/USP/INN) <JP/US>
E D03820 Dutasteride (JAN/USP/INN) <JP/US>
E D04066 Estramustine (USAN/INN)
E D02398 Estramustine phosphate sodium (USAN)
E D06397 Estramustine phosphate sodium hydrate (JAN) <JP/US>
E D01134 Epristeride (JAN/USAN/INN)
E D04498 Idronoxil (USAN/INN)
E D04646 Izonsteride (USAN/INN)
E D07121 Alfatradiol (INN)
D SRD5A3 [HSA:79644] [KO:K12345]
E D04498 Idronoxil (USAN/INN)
D DHODH [HSA:1723] [KO:K00254]
E D00749 Leflunomide (JAN/USP/INN) <JP/US>
E D10172 Teriflunomide (USAN) <US>
E D03154 Brequinar sodium (USAN)
E D11890 Emvododstat (USAN)
C Amine oxidases [EC:1.4.3.-]
D DAO [HSA:1610] [KO:K00273]
E D11981 Luvadaxistat (USAN/INN)
D MAO [HSA:4128 4129] [KO:K00274]
E D05458 Phentermine (USAN/INN)
E D05459 Phentermine hydrochloride (USP) <US>
E D08453 Pargyline (INN)
E D02564 Pargyline hydrochloride (USAN)
E D02580 Isocarboxazid (INN) <US>
E D07337 Nialamide (INN)
E D08349 Phenelzine (BAN)
E D00505 Phenelzine sulfate (USP) <US>
E D08625 Tranylcypromine (INN)
E D00826 Tranylcypromine sulfate (USP) <US>
E D02579 Iproniazid (INN)
E D08085 Iproniazid phosphate
E D07338 Iproclozide (INN)
E D01888 Safrazine hydrochloride (JAN)
E D03239 Ladostigil tartrate (USAN)
E D03409 Caroxazone (USAN/INN)
E D04092 Etryptamine acetate (USAN)
D MAOA [HSA:4128] [KO:K00274]
E D02561 Moclobemide (USAN/INN)
E D02559 Toloxatone (INN)
E D05039 Minaprine (USAN/INN)
E D05040 Minaprine hydrochloride (USAN)
E D02560 Brofaromine (INN)
E D02563 Befloxatone (INN)
E D02581 Cimoxatone (INN)
E D03248 Clorgiline (INN)
E D08392 Pirlindole (INN)
E D08393 Pirlindole hydrochloride
D MAOB [HSA:4129] [KO:K00274]
E D03731 Selegiline (USAN/INN) <US>
E D00785 Selegiline hydrochloride (JAN/USP) <JP/US>
E D08469 Rasagiline (USAN/INN)
E D02562 Rasagiline mesylate (USAN) <JP/US>
E D10829 Rasagiline tartrate
E D10158 Safinamide (USAN/INN)
E D10191 Safinamide mesylate (USAN) <JP/US>
E D01097 Lazabemide hydrochloride (JAN/USAN)
E D03733 Mofegiline hydrochloride (USAN)
E D04681 Lazabemide (USAN/INN)
E D05033 Milacemide hydrochloride (USAN)
E D11224 Sembragiline (USAN/INN)
D AOC3 [HSA:8639] [KO:K00276]
E D08044 Hydralazine (INN)
E D04458 Hydralazine polistirex (USAN)
D AOC1 (DAO) [HSA:26] [KO:K11182]
E D05479 Pimagedine hydrochloride (USAN)
C Dihydrofolate reductase [EC:1.5.1.3]
D DHFR [HSA:1719 200895] [KO:K00287]
E D00142 Methotrexate (JP18/USP/INN) <JP/US>
E D02115 Methotrexate sodium <US>
E D07472 Pemetrexed (INN) <US>
E D03828 Pemetrexed disodium (USAN) <US>
E D06503 Pemetrexed sodium hydrate (JAN) <JP/US>
E D10596 Pemetrexed sodium hemipentahydrate (JAN) <JP/US>
E D05589 Pralatrexate (JAN/USAN/INN) <JP/US>
E D06238 Trimetrexate (USAN/INN)
E D06239 Trimetrexate glucuronate (USAN)
E D03942 Edatrexate (USAN/INN)
E D05500 Piritrexim isethionate (USAN)
E D05999 Talotrexin ammonium (USAN)
E D11352 Pemetrexed tromethamine (USAN) <US>
C NAD(P)H dehydrogenase [EC:1.6.5.2]
D NQO1 [HSA:1728] [KO:K00355]
E D08682 Warfarin (INN)
E D00564 Warfarin sodium (USP) <US>
E D01280 Warfarin potassium (JP18) <JP>
E D07064 Acenocoumarol (INN)
C Peroxidase [EC:1.11.1.-]
D TPO [HSA:7173] [KO:K00431]
E D07231 Methylthiouracil (INN)
E D00562 Propylthiouracil (JP18/USP/INN) <JP/US>
E D07519 Benzylthiouracil
E D07616 Carbimazole (INN)
E D00401 Methimazole (USP) <JP/US>
C Peroxygenase [EC:1.11.2.-]
D MPO [HSA:4353] [KO:K10789]
E D11684 Verdiperstat (USAN/INN)
C Dioxygenases [EC:1.13.11.-]
D HPD [HSA:3242] [KO:K00457]
E D05177 Nitisinone (JAN/USAN/INN) <JP/US>
D ALOX15 [HSA:246] [KO:K00460]
E D12510 Utreloxastat (USAN/INN)
D ALOX5 [HSA:240] [KO:K00461]
E D07516 Benzydamine (INN)
E D01410 Benzydamine hydrochloride (JAN/USAN)
E D07517 Benzydamine salicylate
E D03080 Benoxaprofen (USAN/INN)
E D01773 Oxatomide (JAN/USAN/INN) <JP>
E D00414 Zileuton (USP/INN) <US>
E D03010 Atreleuton (USAN/INN)
E D03652 Darbufelone mesylate (USAN)
E D03882 Docebenone (USAN/INN)
E D03990 Enazadrem phosphate (USAN)
E D04151 Fenleuton (USAN/INN)
E D04770 Lonapalene (USAN)
E D05498 Piriprost (USAN/INN)
E D05499 Piriprost potassium (USAN)
E D06017 Tebufelone (USAN/INN)
E D06075 Tepoxalin (USAN/INN)
E D09667 Setileuton (USAN/INN)
E D09850 Linazolast (JAN)
D IDO [HSA:3620 169355] [KO:K00463]
E D10640 Indoximod (USAN/INN)
D IDO1 [HSA:3620] [KO:K00463]
E D11049 Epacadostat (JAN/USAN/INN)
E D11255 Navoximod (USAN/INN)
E D11412 Linrodostat (USAN)
E D11413 Linrodostat mesylate (USAN)
C Prolyl 4-hydroxylase [EC:1.14.11.2]
D P4HA [HSA:5033 8974 283208] [KO:K00472]
E D04793 Lufironil (USAN/INN)
C HIF hydroxylase [EC:1.14.11.29]
D EGLN (HPH) [HSA:54583 112398 112399] [KO:K09592]
E D10593 Roxadustat (JAN/USAN/INN) <JP>
E D10874 Daprodustat (JAN/USAN/INN) <JP/US>
E D11078 Vadadustat (JAN/USAN/INN) <JP>
E D11273 Molidustat sodium (JAN/USAN) <JP>
E D11523 Enarodustat (JAN) <JP>
E D12122 Molidustat (USAN/INN)
C Nitic oxide synthase [EC:1.14.13.39]
D NOS [HSA:4842 4843 4846] [KO:K13240 K13241 K13242]
E D05479 Pimagedine hydrochloride (USAN)
E D09018 Tilarginine acetate (USAN)
D NOS2 [HSA:4843] [KO:K13241]
E D10386 Cindunistat (USAN/INN)
E D10419 Cindunistat hydrochloride maleate (USAN)
C Cytochrome P450 [EC:1.14.14.-]
D CYP3A [HSA:1551 1576 1577 64816] [KO:K17691 K17689 K17690 K17692]
E D09881 Cobicistat (JAN/USAN/INN) <US>
D CYP19A1 (ARO) [HSA:1588] [KO:K07434]
E D00574 Aminoglutethimide (USP/INN)
E D07260 Formestane (INN)
E D00960 Anastrozole (JP18/USP/INN) <JP/US>
E D00964 Letrozole (JAN/USP/INN) <JP/US>
E D03786 Vorozole (USAN/INN)
E D00963 Exemestane (JAN/USP/INN) <JP/US>
E D00153 Testolactone (USP/INN)
E D02451 Fadrozole hydrochloride (USAN)
E D03749 Plomestane (USAN/INN)
E D03778 Fadrozole hydrochloride hydrate (JAN)
E D03781 Liarozole fumarate (USAN)
E D03784 Liarozole hydrochloride (USAN)
E D05746 Rogletimide (USAN/INN)
E D07940 Fadrozole (INN)
D CYP17A1 [HSA:1586] [KO:K00512]
E D10950 Levoketoconazole (USAN/INN) <US>
E D00420 Mitotane (JAN/USP/INN) <JP/US>
E D09701 Abiraterone acetate (JAN/USP) <JP/US>
E D10125 Galeterone (USAN)
E D10146 Orteronel (JAN/USAN)
D CYP46A1 [HSA:10858] [KO:K07440]
E D11590 Soticlestat (USAN)
D CYP51A1 [HSA:1595] [KO:K05917]
E D03025 Azalanstat dihydrochloride (USAN)
D CYP11B1 [HSA:1584] [KO:K00497]
E D10950 Levoketoconazole (USAN/INN) <US>
E D00410 Metyrapone (JP18/USP/INN) <JP/US>
E D05019 Metyrapone tartrate (USAN)
D CYP11B2 [HSA:1585] [KO:K07433]
E D11061 Osilodrostat (USAN/INN)
E D11062 Osilodrostat phosphate (JAN/USAN) <JP/US>
D CYP11A1 [HSA:1583] [KO:K00498]
E D10950 Levoketoconazole (USAN/INN) <US>
D CYP26 [HSA:1592 56603 340665] [KO:K07437 K12664 K12665]
E D09385 Talarozole (USAN/INN)
C Other monooxygenases [EC:1.14.16.- 1.14.17.- 1.14.18.-]
D PAH* [HSA_VAR:5053v1] [HSA:5053] [KO:K00500]
E D11077 Pegvaliase (INN) <US>
D TH [HSA:7054] [KO:K00501]
E D00762 Metyrosine (USP) <JP/US>
D TPH [HSA:7166 121278] [KO:K00502]
E D09973 Telotristat (USAN/INN)
E D09974 Telotristat ethyl (USAN)
E D09975 Telotristat etiprate (USAN) <US>
D TPH1 [HSA:7166] [KO:K00502]
E D11317 Rodatristat (USAN)
E D11318 Rodatristat ethyl (USAN)
D DBH [HSA:1621] [KO:K00503]
E D03787 Nepicastat hydrochloride (USAN)
D TYR [HSA:7299] [KO:K00505]
E D00073 Hydroquinone (USP)
D HMOX [HSA:3162 3163] [KO:K00510 K21418]
E D05922 Stannsoporfin (USAN/INN)
C Prostaglandin synthase [EC:1.14.99.1]
D PTGS1 (COX1) [HSA:5742] [KO:K00509]
E D07516 Benzydamine (INN)
E D01410 Benzydamine hydrochloride (JAN/USAN)
E D07517 Benzydamine salicylate
E D00109 Aspirin (JP18/USP) <JP>
E D05181 Aspirin aluminum (JP18)
E D07579 Aspirin calcium salt
E D07580 Aspirin DL-lysine (JAN)
E D07581 Aspirin magnesium salt
E D07582 Aspirin sodium
E D07141 Indobufen (INN)
E D07421 Aloxiprin (INN)
E D07142 Triflusal (INN)
E D00141 Indomethacin (USP) <JP/US>
E D01565 Indometacin farnesil (JAN) <JP>
E D02110 Indomethacin sodium (USP) <JP/US>
E D00126 Ibuprofen (JP18/USP/INN) <JP/US>
E D01122 Ibuprofen piconol (JP18/USAN) <JP>
E D04490 Ibuprofen aluminum (USAN)
E D06606 Ibuprofen lysine (USAN) <JP/US>
E D08058 Ibuprofen arginine salt
E D08059 Ibuprofen sodium
E D09760 Ibuprofen sodium (USAN)
E D08501 Trolamine salicylate (USP)
E D07816 Diclofenac (USAN/INN) <US>
E D00903 Diclofenac potassium (USP) <US>
E D00904 Diclofenac sodium (JP18/USP) <JP/US>
E D07817 Diclofenac diethylamine
E D07818 Diclofenac hydroxyethylpyrrolidine <US>
E D07819 Diclofenac calcium
E D00118 Naproxen (JP18/USP/INN) <JP/US>
E D00970 Naproxen sodium (USP) <US>
E D10017 Naproxen etemesil (USAN)
E D00510 Phenylbutazone (JP18/USP/INN)
E D08363 Phenylbutazone calcium
E D08364 Phenylbutazone sodium
E D08324 Oxyphenbutazone (INN)
E D05319 Oxyphenbutazone hydrate
E D00120 Sulindac (JP18/USP/INN) <JP/US>
E D02355 Tolmetin (USAN/INN)
E D00158 Tolmetin sodium (JAN/USP)
E D01582 Acemetacin (JP18/INN) <JP>
E D08427 Proglumetacin (INN)
E D01765 Proglumetacin maleate (JAN) <JP>
E D08104 Ketorolac (INN)
E D00813 Ketorolac tromethamine (USP) <US>
E D01545 Aceclofenac (JAN/INN)
E D01271 Bufexamac (JAN/INN)
E D00127 Piroxicam (JP18/USP/INN) <JP/US>
E D05511 Piroxicam betadex (USAN)
E D05512 Piroxicam cinnamate (USAN)
E D05513 Piroxicam olamine (USAN)
E D01767 Tenoxicam (JAN/USAN/INN)
E D07267 Droxicam (INN)
E D01866 Lornoxicam (JAN/USAN/INN) <JP>
E D00132 Ketoprofen (JP18/USP/INN) <JP/US>
E D08102 Ketoprofen lysine
E D08103 Ketoprofen sodium
E D02350 Fenoprofen (USAN/INN)
E D00968 Fenoprofen calcium (JAN/USP) <US>
E D01344 Fenbufen (JP18/USAN/INN)
E D00330 Flurbiprofen (JP18/USP/INN) <JP/US>
E D01475 Flurbiprofen axetil (JAN) <JP>
E D02290 Flurbiprofen sodium (USP) <US>
E D10254 Esflurbiprofen (JAN)
E D01325 Tiaprofenic acid (JAN/INN)
E D00463 Oxaprozin (JP18/USP/INN) <JP/US>
E D07268 Ibuproxam (INN)
E D03715 Dexibuprofen (USAN/INN)
E D03718 Dexibuprofen lysine (USAN)
E D01513 Alminoprofen (JP18/INN)
E D07269 Dexketoprofen (INN)
E D09568 Naproxcinod (USAN/INN)
E D00151 Mefenamic acid (JP18/USP/INN) <JP/US>
E D01183 Tolfenamic acid (JAN/INN)
E D01581 Flufenamic acid (JAN/USAN/INN)
E D01823 Ufenamate (JAN/INN) <JP>
E D03254 Flufenamate aluminum (JAN) <JP>
E D02341 Meclofenamic acid (USAN/INN)
E D00169 Meclofenamate sodium (USP) <US>
E D08162 Meclofenamate sodium
E D00425 Nabumetone (JP18/USP/INN) <JP/US>
E D06072 Tenidap (USAN/INN)
E D06073 Tenidap sodium (USAN)
E D04102 Etofenamate (USAN/INN)
E D01675 Felbinac (JP18/USAN/INN) <JP>
E D01841 Felbinac ethyl (JAN)
E D08374 Piketoprofen (INN)
E D08375 Piketoprofen hydrochloride
E D08149 Loxoprofen (INN)
E D01709 Loxoprofen sodium hydrate (JP18) <JP>
E D00810 Choline salicylate (JAN/USAN/INN)
E D00566 Sodium salicylate (JP18/USP) <JP>
E D01811 Salicylamide (JAN/USP/INN)
E D00428 Salsalate (USP/INN)
E D00217 Acetaminophen (JP18/USP) <JP/US>
E D07294 Propacetamol (INN)
E D08434 Propacetamol hydrochloride
E D01578 Pranoprofen (JP18/INN) <JP>
E D05143 Nepafenac (JAN/USAN/INN) <JP/US>
E D07541 Bromfenac (INN)
E D03163 Bromfenac sodium (USAN) <JP/US>
E D00827 Magnesium salicylate (USP)
E D01090 Pamicogrel (JAN/INN)
E D01397 Ampiroxicam (JP18/INN) <JP>
E D01527 Epidihydrocholesterin (JAN)
E D01547 Zaltoprofen (JP18/INN) <JP>
E D01557 Glycol salicylate (JAN)
E D01718 Mofezolac (JAN/INN)
E D01788 Amfenac sodium (USAN)
E D03410 Carprofen (USP/INN)
E D05275 Orpanoxin (USAN/INN)
E D05451 Phenbutazone sodium glycerate (USAN)
E D05598 Pravadoline maleate (USAN)
E D05791 Salicylate meglumine (USAN)
E D06017 Tebufelone (USAN/INN)
E D06364 Zidometacin (USAN/INN)
E D07443 Amfenac (INN)
E D07453 Amtolmetin guacil (INN)
D PTGS2 (COX2) [HSA:5743] [KO:K11987]
E D07516 Benzydamine (INN)
E D01410 Benzydamine hydrochloride (JAN/USAN)
E D07517 Benzydamine salicylate
E D00109 Aspirin (JP18/USP) <JP>
E D05181 Aspirin aluminum (JP18)
E D07579 Aspirin calcium salt
E D07580 Aspirin DL-lysine (JAN)
E D07581 Aspirin magnesium salt
E D07582 Aspirin sodium
E D07141 Indobufen (INN)
E D07421 Aloxiprin (INN)
E D00141 Indomethacin (USP) <JP/US>
E D01565 Indometacin farnesil (JAN) <JP>
E D02110 Indomethacin sodium (USP) <JP/US>
E D00126 Ibuprofen (JP18/USP/INN) <JP/US>
E D01122 Ibuprofen piconol (JP18/USAN) <JP>
E D04490 Ibuprofen aluminum (USAN)
E D06606 Ibuprofen lysine (USAN) <JP/US>
E D08058 Ibuprofen arginine salt
E D08059 Ibuprofen sodium
E D09760 Ibuprofen sodium (USAN)
E D08501 Trolamine salicylate (USP)
E D07816 Diclofenac (USAN/INN) <US>
E D00903 Diclofenac potassium (USP) <US>
E D00904 Diclofenac sodium (JP18/USP) <JP/US>
E D07817 Diclofenac diethylamine
E D07818 Diclofenac hydroxyethylpyrrolidine <US>
E D07819 Diclofenac calcium
E D00118 Naproxen (JP18/USP/INN) <JP/US>
E D00970 Naproxen sodium (USP) <US>
E D10017 Naproxen etemesil (USAN)
E D00567 Celecoxib (JP18/USP/INN) <JP/US>
E D00510 Phenylbutazone (JP18/USP/INN)
E D08363 Phenylbutazone calcium
E D08364 Phenylbutazone sodium
E D08324 Oxyphenbutazone (INN)
E D05319 Oxyphenbutazone hydrate
E D00120 Sulindac (JP18/USP/INN) <JP/US>
E D02355 Tolmetin (USAN/INN)
E D00158 Tolmetin sodium (JAN/USP)
E D01252 Alclofenac (JAN/USP/INN)
E D00315 Etodolac (JP18/USP/INN) <JP/US>
E D01582 Acemetacin (JP18/INN) <JP>
E D08427 Proglumetacin (INN)
E D01765 Proglumetacin maleate (JAN) <JP>
E D08104 Ketorolac (INN)
E D00813 Ketorolac tromethamine (USP) <US>
E D01545 Aceclofenac (JAN/INN)
E D01271 Bufexamac (JAN/INN)
E D00127 Piroxicam (JP18/USP/INN) <JP/US>
E D05511 Piroxicam betadex (USAN)
E D05512 Piroxicam cinnamate (USAN)
E D05513 Piroxicam olamine (USAN)
E D01767 Tenoxicam (JAN/USAN/INN)
E D07267 Droxicam (INN)
E D01866 Lornoxicam (JAN/USAN/INN) <JP>
E D00969 Meloxicam (JAN/USP/INN) <JP/US>
E D00132 Ketoprofen (JP18/USP/INN) <JP/US>
E D08102 Ketoprofen lysine
E D08103 Ketoprofen sodium
E D02350 Fenoprofen (USAN/INN)
E D00968 Fenoprofen calcium (JAN/USP) <US>
E D01344 Fenbufen (JP18/USAN/INN)
E D00330 Flurbiprofen (JP18/USP/INN) <JP/US>
E D01475 Flurbiprofen axetil (JAN) <JP>
E D02290 Flurbiprofen sodium (USP) <US>
E D10254 Esflurbiprofen (JAN)
E D01325 Tiaprofenic acid (JAN/INN)
E D00463 Oxaprozin (JP18/USP/INN) <JP/US>
E D07268 Ibuproxam (INN)
E D03715 Dexibuprofen (USAN/INN)
E D03718 Dexibuprofen lysine (USAN)
E D01513 Alminoprofen (JP18/INN)
E D07269 Dexketoprofen (INN)
E D09568 Naproxcinod (USAN/INN)
E D00151 Mefenamic acid (JP18/USP/INN) <JP/US>
E D01183 Tolfenamic acid (JAN/INN)
E D01581 Flufenamic acid (JAN/USAN/INN)
E D01823 Ufenamate (JAN/INN) <JP>
E D03254 Flufenamate aluminum (JAN) <JP>
E D02341 Meclofenamic acid (USAN/INN)
E D00169 Meclofenamate sodium (USP) <US>
E D08162 Meclofenamate sodium
E D00568 Rofecoxib (JAN/USAN/INN)
E D02709 Valdecoxib (USAN/INN)
E D03716 Parecoxib (USAN/INN)
E D03717 Parecoxib sodium (USAN)
E D03710 Etoricoxib (USAN/INN)
E D03714 Lumiracoxib (USAN/INN)
E D10656 Polmacoxib (USAN/INN)
E D00425 Nabumetone (JP18/USP/INN) <JP/US>
E D08275 Niflumic acid (INN)
E D01049 Nimesulide (JAN/INN)
E D06072 Tenidap (USAN/INN)
E D06073 Tenidap sodium (USAN)
E D04102 Etofenamate (USAN/INN)
E D01675 Felbinac (JP18/USAN/INN) <JP>
E D01841 Felbinac ethyl (JAN)
E D08374 Piketoprofen (INN)
E D08375 Piketoprofen hydrochloride
E D08149 Loxoprofen (INN)
E D01709 Loxoprofen sodium hydrate (JP18) <JP>
E D00810 Choline salicylate (JAN/USAN/INN)
E D00566 Sodium salicylate (JP18/USP) <JP>
E D01811 Salicylamide (JAN/USP/INN)
E D00428 Salsalate (USP/INN)
E D00130 Diflunisal (JAN/USP/INN) <US>
E D00217 Acetaminophen (JP18/USP) <JP/US>
E D07294 Propacetamol (INN)
E D08434 Propacetamol hydrochloride
E D01578 Pranoprofen (JP18/INN) <JP>
E D05143 Nepafenac (JAN/USAN/INN) <JP/US>
E D07541 Bromfenac (INN)
E D03163 Bromfenac sodium (USAN) <JP/US>
E D00827 Magnesium salicylate (USP)
E D01090 Pamicogrel (JAN/INN)
E D01397 Ampiroxicam (JP18/INN) <JP>
E D01547 Zaltoprofen (JP18/INN) <JP>
E D01557 Glycol salicylate (JAN)
E D01788 Amfenac sodium (USAN)
E D01974 Tilmacoxib (JAN/USAN/INN)
E D03410 Carprofen (USP/INN)
E D03652 Darbufelone mesylate (USAN)
E D03689 Deracoxib (USAN)
E D03712 Firocoxib (USAN/INN)
E D04863 Mavacoxib (USAN)
E D05275 Orpanoxin (USAN/INN)
E D05451 Phenbutazone sodium glycerate (USAN)
E D05598 Pravadoline maleate (USAN)
E D05791 Salicylate meglumine (USAN)
E D06017 Tebufelone (USAN/INN)
E D06364 Zidometacin (USAN/INN)
E D07443 Amfenac (INN)
E D07453 Amtolmetin guacil (INN)
E D07888 Eltenac (INN)
E D08657 Apricoxib (USAN/INN)
E D11020 Diclofenac etalhyaluronate sodium (JAN) <JP>
C Histone demethylase [EC:1.14.99.66]
D KDM1A (LSD1) [HSA:23028] [KO:K11450]
E D12263 Bomedemstat (USAN/INN)
E D12264 Bomedemstat tosylate (USAN)
C Superoxide dismutase [EC:1.15.1.1]
D SOD1 [HSA:6647] [KO:K04565]
E D11811 Tofersen (JAN/USAN/INN)
C Xanthine dehydrogenase/oxidase [EC:1.17.1.4 1.17.3.2]
D XDH [HSA:7498] [KO:K00106]
E D00224 Allopurinol (JP18/USP/INN) <JP/US>
E D07564 Allopurinol sodium <US>
E D07278 Tisopurine (INN)
E D01206 Febuxostat (JAN/USAN/INN) <JP/US>
E D11081 Febuxostat hydrate (JAN) <JP/US>
E D02365 Oxypurinol (USAN)
E D02896 Amflutizole (USAN/INN)
E D09786 Topiroxostat (JAN/INN) <JP>
C Ribonucleoside-diphosphate reductase [EC:1.17.4.1]
D RRM1 [HSA:6240] [KO:K10807]
E D01370 Cladribine (JAN/USP/INN) <JP/US>
E D07966 Fludarabine (INN)
E D01907 Fludarabine phosphate (JAN/USP) <JP/US>
E D03546 Clofarabine (JAN/USAN/INN) <JP/US>
E D02368 Gemcitabine (USAN/INN)
E D01155 Gemcitabine hydrochloride (JAN/USP) <JP/US>
E D10222 Gemcitabine elaidate (USAN/INN)
E D03378 Caracemide (USAN)
E D06100 Tezacitabine (USAN)
E D12387 Fosgemcitabine palabenamide (USAN/INN)
D RRM2 [HSA:6241] [KO:K10808]
E D00341 Hydroxyurea (USP) <JP/US>
C Vitamin-K-epoxide reductase [EC:1.17.4.4]
D VKORC1 [HSA:79001] [KO:K05357]
E D03798 Dicumarol (USAN)
E D08354 Phenindione (INN)
E D08682 Warfarin (INN)
E D00564 Warfarin sodium (USP) <US>
E D01280 Warfarin potassium (JP18) <JP>
E D05457 Phenprocoumon (USAN/INN)
E D07064 Acenocoumarol (INN)
E D07131 Ethyl biscoumacetate (INN)
E D07135 Clorindione (INN)
E D07136 Diphenadione (INN)
E D07137 Tioclomarol (INN)
E D07969 Fluindione (INN)
E D07134 Flocoumafen (JAN)
E D09676 Tecarfarin (USAN/INN)
E D09677 Tecarfarin sodium (USAN)
C Thyroxine 5'-deiodinase [EC:1.21.99.4]
D DIO1 [HSA:1733] [KO:K01562]
E D00562 Propylthiouracil (JP18/USP/INN) <JP/US>
D DIO2 [HSA:1734] [KO:K17904]
E D00562 Propylthiouracil (JP18/USP/INN) <JP/US>
B Transferases (EC2)
C Methyltransferases [EC:2.1.1.-]
D COMT [HSA:1312] [KO:K00545]
E D00152 Phloroglucinol (JAN)
E D08369 Polyphloroglucinol phosphate
E D00786 Tolcapone (JAN/USP/INN) <US>
E D00781 Entacapone (JP18/USP/INN) <JP/US>
E D10825 Opicapone (JAN/USAN/INN) <JP/US>
E D01259 Flopropione (JP18/INN) <JP>
E D03241 Nitecapone (INN)
D DNMT [HSA:1786 1788 1789] [KO:K00558 K17398 K17399]
E D03021 Azacitidine (JAN/USAN/INN) <JP/US>
E D03665 Decitabine (USAN/INN) <US>
D DNMT1 [HSA:1786] [KO:K00558]
E D11740 Roducitabine (USAN)
D EZH [HSA:2145 2146] [KO:K17451 K11430]
E D11551 Valemetostat
E D11662 Valemetostat tosilate (JAN) <JP>
D EZH2 [HSA:2146] [KO:K11430]
E D11444 Tazemetostat (USAN/INN)
D EZH2* [HSA_VAR:2146v1] [HSA:2146] [KO:K11430]
E D11485 Tazemetostat hydrobromide (JAN/USAN) <JP/US>
D TYMS [HSA:7298] [KO:K00560]
E D01064 Raltitrexed (JAN/USAN/INN)
E D07472 Pemetrexed (INN) <US>
E D03828 Pemetrexed disodium (USAN) <US>
E D06503 Pemetrexed sodium hydrate (JAN) <JP/US>
E D10596 Pemetrexed sodium hemipentahydrate (JAN) <JP/US>
E D00584 Fluorouracil (JP18/USP/INN) <JP/US>
E D07974 Fluorouracil sodium salt
E D01244 Tegafur (JP18/USAN/INN) <JP>
E D01784 Carmofur (JP18/INN)
E D01223 Capecitabine (JAN/USP/INN) <JP/US>
E D04197 Floxuridine (USP/INN) <US>
E D01309 Doxifluridine (JP18/INN) <JP>
E D04964 Metesind glucuronate (USAN)
E D10803 Plevitrexed (INN)
E D11352 Pemetrexed tromethamine (USAN) <US>
E D11447 Arfolitixorin (USAN/INN)
E D12388 Fosifloxuridine nafalbenamide
C Acyltransferases [EC:2.3.1.-]
D DGAT1 [HSA:8694] [KO:K11155]
E D10657 Pradigastat sodium (USAN)
E D10664 Pradigastat (USAN)
D CPT [HSA:1374 1375 126129 1376] [KO:K08765 K19523 K19524 K08766]
E D08340 Perhexiline (INN)
E D05442 Perhexiline maleate (USAN)
D CPT1 [HSA:1374 1375 126129] [KO:K08765 K19523 K19524]
E D05292 Oxfenicine (USAN/INN)
D SOAT [HSA:6646 8435] [KO:K00637]
E D01202 Melinamide (JAN)
E D03012 Avasimibe (USAN/INN)
E D03447 Cetaben sodium (USAN)
E D03734 Eldacimibe (USAN/INN)
E D03735 Lecimibide (USAN)
D ALAS [HSA:211 212] [KO:K00643]
E D10003 Hemin (JAN) <JP/US>
D ALAS1 [HSA:211] [KO:K00643]
E D11702 Givosiran (USAN/INN)
E D11708 Givosiran sodium (JAN) <JP/US>
D LCAT [HSA:3931] [KO:K00650]
E D04268 Elastase ES <JP>
D CREBBP/EP300 [HSA:1387 2033] [KO:K04498]
E D12394 Inobrodib (USAN)
D FASN [HSA:2194] [KO:K00665]
E D12391 Denifanstat (USAN)
C gamma-Glutamyltransferase [EC:2.3.2.2]
D GGT [HSA:2678 2687 124975 2686] [KO:K18592 K00681]
E D02755 Acivicin (USAN/INN)
C E3 ubiquitin-protein ligase [EC:2.3.2.27]
D MDM2 [HSA:4193] [KO:K06643]
E D11219 Idasanutlin (USAN/INN)
E D12378 Navtemadlin (USAN/INN)
E D12399 Sulanemadlin (USAN/INN)
E D12417 Siremadlin (USAN/INN)
E D12418 Siremadlin succinate (USAN)
D MDM4 [HSA:4194] [KO:K10127]
E D12399 Sulanemadlin (USAN/INN)
C ATP citrate synthase [EC:2.3.3.8]
D ACLY (ACL) [HSA:47] [KO:K01648]
E D10691 Bempedoic acid (JAN/USAN/INN) <US>
C Hexosyltransferases [EC:2.4.1.-]
D PYG [HSA:5834 5836 5837] [KO:K00688]
E D04537 Ingliforib (USAN/INN)
D UGCG [HSA:7357] [KO:K00720]
E D05032 Miglustat (JAN/USAN/INN) <JP/US>
E D09893 Eliglustat (USAN/INN)
E D09894 Eliglustat tartrate (JAN/USAN) <JP/US>
E D11439 Lucerastat (JAN/USAN/INN)
E D11633 Venglustat (USAN/INN)
D A3GALT2 [HSA:127550] [KO:K20736]
E D10429 Tergenpumatucel-L (USAN)
C Pentosyltransferases [EC:2.4.2.-]
D PNP [HSA:4860] [KO:K03783]
E D04245 Forodesine hydrochloride (JAN/USAN) <JP>
E D05396 Peldesine (USAN)
E D06596 Forodesine (USAN/INN)
E D10431 Ulodesine (USAN)
E D10432 Ulodesine succinate (USAN)
D HPRT1 [HSA:3251] [KO:K00760]
E D04931 Mercaptopurine (INN)
E D00161 Mercaptopurine (USP) <JP/US>
E D08603 Tioguanine (INN)
E D06109 Thioguanine (USP) <US>
D NAMPT [HSA:10135] [KO:K03462]
E D09678 Teglarinad chloride (USAN/INN)
D PARP [HSA:142 10038 10039 143] [KO:K24070 K10798]
E D09692 Veliparib (JAN/USAN/INN)
D PARP1 [HSA:142] [KO:K24070]
E D09730 Olaparib (JAN/USAN/INN) <JP/US>
E D10140 Niraparib (USAN)
E D11895 Niraparib tosilate hydrate (JAN) <JP/US>
E D10079 Rucaparib (USAN/INN)
E D10157 Rucaparib phosphate (USAN)
E D10982 Rucaparib camsylate (USAN) <US>
E D10732 Talazoparib (USAN/INN)
E D10733 Talazoparib tosylate (USAN) <US>
E D11426 Pamiparib (USAN/INN)
E D09913 Iniparib (USAN/INN)
D PARP2 [HSA:10038] [KO:K10798]
E D09730 Olaparib (JAN/USAN/INN) <JP/US>
E D10140 Niraparib (USAN)
E D11895 Niraparib tosilate hydrate (JAN) <JP/US>
E D10079 Rucaparib (USAN/INN)
E D10157 Rucaparib phosphate (USAN)
E D10982 Rucaparib camsylate (USAN) <US>
E D10732 Talazoparib (USAN/INN)
E D10733 Talazoparib tosylate (USAN) <US>
E D11426 Pamiparib (USAN/INN)
D PARP3 [HSA:10039] [KO:K10798]
E D10079 Rucaparib (USAN/INN)
E D10157 Rucaparib phosphate (USAN)
E D10982 Rucaparib camsylate (USAN) <US>
E D11426 Pamiparib (USAN/INN)
D TIPARP (PARP7) [HSA:25976] [KO:K15259]
E D12408 Atamparib (USAN/INN)
C Alkyl/Aryl transferases [EC:2.5.1.-]
D FDPS [HSA:2224] [KO:K00787]
E D07281 Pamidronic acid (INN)
E D00941 Pamidronate disodium (USP) <JP/US>
E D07119 Alendronic acid (INN)
E D00939 Alendronate sodium (USP) <JP/US>
E D08056 Ibandronic acid (INN)
E D04486 Ibandronate sodium (USAN) <JP/US>
E D08484 Risedronic acid (INN)
E D00942 Risedronate sodium (USP) <US>
E D03234 Sodium risedronate hydrate (JP18) <JP/US>
E D11570 Risedronate sodium monohydrate <US>
E D08689 Zoledronic acid (INN)
E D01968 Zoledronic acid (USAN) <JP/US>
E D06378 Zoledronate disodium (USAN)
E D06379 Zoledronate trisodium (USAN)
E D10515 Zoledronic acid hemipentahydrate (JAN)
E D07123 Incadronate disodium hydrate (JAN)
E D08073 Incadronic acid (INN)
E D09198 Minodronic acid hydrate (JAN) <JP>
D GSTP1 [HSA:2950] [KO:K23790]
E D08917 Ezatiostat hydrochloride (USAN)
D FDFT1 [HSA:2222] [KO:K00801]
E D06609 Lapaquistat acetate (JAN/USAN)
D FNT [HSA:2339 2342] [KO:K05955 K05954]
E D04768 Lonafarnib (USAN/INN)
E D03720 Tipifarnib (USAN/INN)
C Aminotransferase [EC:2.6.1.-]
D ABAT [HSA:18] [KO:K13524]
E D00399 Valproic acid (USP) <US>
E D00304 Divalproex sodium (USP) <US>
E D00710 Valproate sodium (USAN) <JP/US>
E D08667 Calcium valproate
E D00535 Vigabatrin (JAN/USP/INN) <JP/US>
C Phosphotransferase [EC:2.7.1.-]
D HK [HSA:3098 3099 3101 80201] [KO:K00844]
E D07257 Lonidamine (INN)
D GCK [HSA:2645] [KO:K12407]
E D11342 Dorzagliatin (USAN)
E D08970 Piragliatin (USAN)
E D12320 Cadisegliatin (USAN)
D TK2 [HSA:7084] [KO:K00857]
E D12465 Doxecitine (USAN/INN)
E D12466 Doxribtimine (USAN/INN)
D PKLR [HSA:5313] [KO:K12406]
E D11408 Mitapivat sulfate (USAN) <US>
E D12362 Etavopivat (USAN/INN)
D PIK3C3 [HSA:5289] [KO:K00914]
E D05784 Safingol (USAN/INN)
E D05785 Safingol hydrochloride (USAN)
E D11319 Fimepinostat (USAN/INN)
D PIK3CA [HSA:5290] [KO:K00922]
E D10867 Copanlisib (USAN/INN)
E D10797 Copanlisib hydrochloride (USAN)
E D10798 Copanlisib hydrochloride hydrate (JAN) <US>
E D11869 Paxalisib (USAN/INN)
E D11942 Inavolisib (USAN/INN)
D PIK3CA* [HSA_VAR:5290v1] [HSA:5290] [KO:K00922]
E D11011 Alpelisib (JAN/USAN/INN) <US>
D PIK3CD [HSA:5293] [KO:K00922]
E D10560 Idelalisib (JAN/USAN/INN) <US>
E D10867 Copanlisib (USAN/INN)
E D10797 Copanlisib hydrochloride (USAN)
E D10798 Copanlisib hydrochloride hydrate (JAN) <US>
E D10555 Duvelisib (USAN/INN)
E D11658 Duvelisib hydrate (JAN) <US>
E D11437 Parsaclisib (USAN/INN)
E D11506 Parsaclisib hydrochloride (JAN/USAN)
E D11322 Umbralisib (USAN/INN)
E D11323 Umbralisib tosylate (USAN) <US>
E D10924 Dezapelisib (USAN)
E D11267 Nemiralisib (USAN/INN)
E D11354 Nemiralisib succinate (USAN)
E D12009 Zandelisib (JAN/USAN/INN)
E D12514 Amdizalisib (USAN/INN)
D PIK3CG [HSA:5294] [KO:K21289]
E D10555 Duvelisib (USAN/INN)
E D11658 Duvelisib hydrate (JAN) <US>
E D11896 Eganelisib (USAN)
D PIK3C [HSA:5290 5291 5293] [KO:K00922]
E D10189 Pictilisib (USAN)
E D10543 Apitolisib (USAN/INN)
E D10552 Dactolisib (USAN/INN)
E D10584 Buparlisib (USAN/INN)
E D10609 Buparlisib hydrochloride (JAN/USAN)
E D10616 Dactolisib tosylate (USAN)
E D10635 Gedatolisib (USAN/INN)
E D10718 Omipalisib (USAN/INN)
E D11158 Leniolisib (USAN/INN)
E D11159 Leniolisib phosphate (USAN)
E D11440 Bimiralisib (USAN/INN)
E D11501 Samotolisib (USAN)
E D11727 Voxtalisib (USAN/INN)
E D11774 Taselisib (USAN/INN)
C DNA polymerase [EC:2.7.7.7]
D POLA [HSA:5422 23649] [KO:K02320 K02321]
E D03546 Clofarabine (JAN/USAN/INN) <JP/US>
C Reverse transcriptase [EC:2.7.7.49]
D TERT [HSA:7015] [KO:K11126]
E D09629 Imetelstat (USAN/INN)
E D09630 Imetelstat sodium (USAN)
B Hydrolases (EC3)
C Carboxylic-ester hydrolases [EC:3.1.1.-]
D LIPF [HSA:8513] [KO:K14452]
E D04028 Orlistat (JAN/USP/INN) <US>
D LIPC [HSA:3990] [KO:K22283]
E D02047 Dextran sulfate sodium (JAN)
E D03343 Dextran sulfate sodium sulfur 5 (JP18) <JP>
D PNLIP [HSA:5406] [KO:K14073]
E D09208 Cetilistat (JAN/USAN/INN) <JP>
D PNLIP [HSA:5406 5407 5408] [KO:K14073 K14074 K14075]
E D04028 Orlistat (JAN/USP/INN) <US>
D PLA2G [HSA:26279 30814 391013 50487 5319 5320 5322 64600 81579 8399 84647] [KO:K01047]
E D06283 Varespladib sodium (USAN)
D PLA2G4A [HSA:5321] [KO:K16342]
E D03938 Ecopladib (USAN/INN)
E D06600 Giripladib (USAN)
E D06674 Efipladib (USAN)
D PLA2G7 (LP-PLA2) [HSA:7941] [KO:K01062]
E D03650 Darapladib (JAN/USAN)
E D04368 Goxalapladib (USAN)
E D05728 Rilapladib (USAN)
E D06283 Varespladib sodium (USAN)
E D08107 Varespladib (USAN/INN)
E D08221 Varespladib methyl (USAN)
D ACHE [HSA:43] [KO:K01049]
E D08094 Itopride (INN)
E D02729 Itopride hydrochloride (JAN) <JP>
E D08838 Acotiamide hydrochloride (USAN) <JP>
E D02292 Gallamine triethiodide (USP)
E D02565 Dimetacrine (INN)
E D08555 Tacrine (INN)
E D02068 Tacrine hydrochloride (USP)
E D07869 Donepezil (JAN/INN) <JP>
E D00670 Donepezil hydrochloride (JP18/USP) <JP/US>
E D03822 Rivastigmine (JAN/USP/INN) <JP/US>
E D02558 Rivastigmine tartrate <US>
E D04292 Galantamine (USAN/INN)
E D02173 Galantamine hydrobromide (JAN/USP) <JP/US>
E D09750 Ipidacrine hydrochloride hydrate (JAN)
E D08261 Neostigmine (BAN)
E D00995 Neostigmine bromide (JAN/USP/INN) <JP>
E D00998 Neostigmine methylsulfate (JP18/USP) <JP/US>
E D00487 Pyridostigmine bromide (JP18/USP/INN) <JP/US>
E D01228 Distigmine bromide (JP18/INN) <JP>
E D01001 Ambenonium chloride (JP18/INN) <JP>
E D02193 Echothiophate iodide (USP) <US>
E D00667 Demecarium bromide (USP/INN)
E D00196 Physostigmine (USP)
E D02418 Physostigmine salicylate (JAN/USP)
E D03826 Physostigmine sulfate (USP)
E D00043 Isoflurophate
E D10529 Paraoxon
E D00469 Pralidoxime chloride (USP) <US>
E D01572 Pralidoxime iodide (JAN/USAN) <JP>
E D05590 Pralidoxime mesylate (USAN)
E D05215 Obidoxime chloride (USAN)
E D00994 Edrophonium chloride (JP18/USP/INN) <JP>
E D03239 Ladostigil tartrate (USAN)
E D03751 Icopezil maleate (USAN)
E D03823 Quilostigmine (USAN/INN)
E D05981 Suronacrine maleate (USAN)
E D06288 Velnacrine maleate (USAN)
E D06365 Zifrosilone (USAN)
E D09835 Zanapezil fumarate (JAN)
E D09917 Latrepirdine (USAN/INN)
E D09918 Latrepirdine dihydrochloride (USAN)
E D12318 Buntanetap (USAN)
E D12319 Buntanetap tartrate (USAN)
D BCHE [HSA:590] [KO:K01050]
E D04435 Hexafluorenium bromide (USAN)
E D03822 Rivastigmine (JAN/USP/INN) <JP/US>
E D02558 Rivastigmine tartrate <US>
E D02193 Echothiophate iodide (USP) <US>
E D00043 Isoflurophate
E D03239 Ladostigil tartrate (USAN)
D LIPA* [HSA_VAR:3988v1] [HSA:3988] [KO:K01052]
E D10377 Sebelipase alfa (USAN) <JP/US>
D LPL [HSA:4023] [KO:K01059]
E D02047 Dextran sulfate sodium (JAN)
E D03343 Dextran sulfate sodium sulfur 5 (JP18) <JP>
E D05255 Omega-3-acid ethyl esters (USP) <JP/US>
E D03747 Ibrolipim (USAN/INN)
E D04268 Elastase ES <JP>
D LPL* [HSA_VAR:4023v1] [HSA:4023] [KO:K01059]
E D10843 Alipogene tiparvovec (INN)
D RPE65 [HSA:6121] [KO:K11158]
E D11008 Voretigene neparvovec (USAN/INN) <US>
D RARRES3 (DDX58, RIG1) [HSA:5920] [KO:K23266]
E D11385 Inarigivir soproxil (USAN)
C Phosphatases [EC:3.1.3.-]
D ALPI (IAP) [HSA:248] [KO:K01077]
E D12277 Ilofotase alfa (USAN)
D ALPL* [HSA_VAR:249v1] [HSA:249] [KO:K01077]
E D10595 Asfotase alfa (USAN/INN) <JP/US>
D NT5E (CD73) [HSA:4907] [KO:K19970]
E D10963 Oleclumab (USAN)
E D12373 Quemliclustat (USAN/INN)
E D12401 Uliledlimab (USAN/INN)
D PPP2C [HSA:5515 5516] [KO:K04382]
E D04262 Fostriecin sodium (USAN)
D PPP3C/PPP3R/CHP [HSA:5530 5532 5533 5534 5535 11261 63928] [KO:K04348 K06268 K17610 K17611]
E D08556 Tacrolimus (INN)
E D00107 Tacrolimus (USP/INN) <JP/US>
E D05480 Pimecrolimus (JAN/USAN/INN) <US>
E D00184 Cyclosporine (USP) <JP/US>
E D09033 Voclosporin (JAN/USAN/INN) <US>
E D10983 Ruclosporin (USAN/INN)
D PPP4C [HSA:5531] [KO:K15423]
E D04262 Fostriecin sodium (USAN)
D PTPN1 [HSA:5770] [KO:K05696]
E D04050 Ertiprotafib (USAN/INN)
E D06252 Trodusquemine (USAN/INN)
D INPP5D (SHIP1) [HSA:3635] [KO:K03084]
E D11275 Rosiptor (USAN/INN)
E D11276 Rosiptor acetate (USAN)
C Phosphodiesterases [EC:3.1.4.-]
D SMPD1* [HSA_VAR:6609v1] [HSA:6609] [KO:K12350]
E D10820 Olipudase alfa (USAN/INN) <JP/US>
D PDE [HSA:10846 27115 50940 5136 5137 5138 5139 5140 5141 5142 5143 5144 5150 5151 5153 8622] [KO:K18438 K18436 K13298 K13755 K18283 K19021 K13296 K13293 K18437]
E D07425 Papaverine (BAN)
E D02218 Papaverine hydrochloride (JP18/USP) <JP>
E D07439 Papaverine sulfate
E D07089 Moxaverine (INN)
E D08238 Moxaverine hydrochloride
E D07546 Bucladesine (INN)
E D01238 Bucladesine sodium (JAN) <JP>
E D01220 Trapidil (JP18/INN) <JP>
E D07961 Flavoxate (INN)
E D00718 Flavoxate hydrochloride (JP18/USP) <JP/US>
E D00691 Dyphylline (USP) <JP>
E D02017 Oxtriphylline (USP)
E D01771 Proxyphylline (JAN/INN) <JP>
E D00371 Theophylline (JP18) <JP/US>
E D01712 Theophylline sodium acetate (JAN)
E D06103 Theophylline (USP)
E D06104 Theophylline sodium glycinate (USP)
E D00227 Aminophylline (USP/INN)
E D05429 Aminophylline hydrate (JP18) <JP>
E D11630 Aminophylline dihydrate <US>
E D03075 Bemoradan (USAN/INN)
E D04006 Enprofylline (USAN/INN)
E D05278 Oxagrelate (USAN/INN)
E D05612 Prinoxodan (USAN/INN)
E D06132 Tibenelast sodium (USAN)
E D09822 Theosalicin (JAN)
D PDE [HSA:5153 5138 5139 5140 5141 5142 5143 5144 8654] [KO:K13755 K18283 K19021 K13296 K13293 K13762]
E D00528 Caffeine (USP) <JP>
E D01453 Caffeine hydrate (JP18) <JP>
E D07603 Caffeine citrate (USP) <US>
D PDE1 [HSA:5136 5153 5137] [KO:K13755]
E D11883 Lenrispodun (USAN)
E D11884 Lenrispodun phosphate (USAN)
D PDE2A [HSA:5138] [KO:K18283]
E D03898 Doxofylline (USAN/INN)
D PDE3 [HSA:5139 5140] [KO:K19021 K13296]
E D01896 Cilostazol (JP18/USP/INN) <JP/US>
E D00231 Inamrinone (USP)
E D02084 Inamrinone ethylenelactate
E D00417 Milrinone (JAN/USP/INN) <JP>
E D02085 Milrinone lactate <US>
E D04004 Enoximone (USAN/INN)
E D04720 Levosimendan (USAN/INN)
E D07455 Anagrelide (INN/BAN)
E D02933 Anagrelide hydrochloride (USP)
E D10255 Anagrelide hydrochloride hydrate (JAN) <JP/US>
E D01385 Ibudilast (JP18/INN) <JP>
E D01133 Pimobendan (JAN/USAN/INN) <JP>
E D01198 Toborinone (JAN/USAN/INN)
E D01690 Vesnarinone (JAN/USAN/INN)
E D02042 Olprinone hydrochloride hydrate (JAN) <JP>
E D04508 Imazodan hydrochloride (USAN)
E D04529 Indolidan (USAN/INN)
E D04628 Isomazole hydrochloride (USAN)
E D04751 Lixazinone sulfate (USAN)
E D05514 Piroximone (USAN)
E D08294 Olprinone (INN)
E D09843 Beradilol monoethyl maleate (JAN)
E D11743 Ensifentrine (USAN/INN)
D PDE4 [HSA:5141 5142 5143 5144] [KO:K13293]
E D07088 Drotaverine (INN)
E D07879 Drotaverine hydrochloride
E D10873 Crisaborole (USAN/INN) <US>
E D08860 Apremilast (JAN/USAN) <JP/US>
E D01630 Propentofylline (JAN/INN)
E D01385 Ibudilast (JP18/INN) <JP>
E D05744 Roflumilast (JAN/USAN/INN) <US>
E D01704 Cilomilast (JAN/USAN/INN)
E D01783 Rolipram (JAN/USAN/INN)
E D02655 Etazolate hydrochloride (USAN)
E D02985 Arofylline (USAN/INN)
E D03516 Cipamfylline (USAN/INN)
E D04185 Filaminast (USAN/INN)
E D05474 Piclamilast (USAN/INN)
E D09020 Tofimilast (INN/USAN)
E D11305 Lotamilast (USAN/INN)
E D11314 Difamilast (JAN/USAN) <JP>
E D11743 Ensifentrine (USAN/INN)
E D12397 Tranimilast (USAN/INN)
D PDE4A [HSA:5141] [KO:K13293]
E D00302 Dipyridamole (JP18/USP/INN) <JP/US>
D PDE4D [HSA:5144] [KO:K13293]
E D12173 Zatolmilast (USAN)
D PDE5 [HSA:8654] [KO:K13762]
E D00302 Dipyridamole (JP18/USP/INN) <JP/US>
E D08514 Sildenafil (INN)
E D02229 Sildenafil citrate (JAN/USP) <JP/US>
E D02008 Tadalafil (JAN/USP/INN) <JP/US>
E D08668 Vardenafil (USAN/INN)
E D02731 Vardenafil dihydrochoride (USAN)
E D03260 Vardenafil hydrochloride hydrate (JAN) <JP/US>
E D09989 Vardenafil hydrochloride (USP)
E D03217 Avanafil (USAN/INN) <US>
E D10027 Udenafil (USAN/INN)
E D03657 Dasantafil (USAN/INN)
E D09621 Gisadenafil (USAN/INN)
E D09622 Gisadenafil besylate (USAN)
D PDE9 [HSA:5152] [KO:K13761]
E D12203 Tovinontrine (USAN/INN)
D PDE10A [HSA:10846] [KO:K18438]
E D11171 Mardepodect (USAN/INN)
E D11245 Balipodect (USAN/INN)
D ENPP2 (ATX) [HSA:5168] [KO:K01122]
E D11844 Ziritaxestat (USAN/INN)
C Sulfatases [EC:3.1.6.-]
D STS [HSA:412] [KO:K01131]
E D09915 Irosustat (USAN/INN)
D GALNS* [HSA_VAR:2588v1] [HSA:2588] [KO:K01132]
E D10333 Elosulfase alfa (USAN) <JP/US>
D ARSA [HSA:410] [KO:K01134]
E D12462 Cebsulfase alfa (USAN)
D ARSB* [HSA_VAR:411v1] [HSA:411] [KO:K01135]
E D06565 Galsulfase (USAN/INN) <JP/US>
D IDS [HSA:3423] [KO:K01136]
E D11812 Pabinafusp alfa (genetical recombination) (JAN) <JP>
D IDS* [HSA_VAR:3423v1] [HSA:3423] [KO:K01136]
E D04499 Idursulfase (USAN/INN) <JP/US>
E D11025 Idursulfase beta (INN) <JP>
C Glycosidases [EC:3.2.1.-]
D AMY [HSA:279 280] [KO:K01176]
E D00216 Acarbose (JAN/USAN/INN) <JP/US>
D GAA [HSA:2548] [KO:K12316]
E D00216 Acarbose (JAN/USAN/INN) <JP/US>
E D00625 Miglitol (JP18/USAN/INN) <JP/US>
E D01665 Voglibose (JP18/USAN/INN) <JP>
E D11798 Cipaglucosidase alfa (USAN)
E D09605 Duvoglustat (USAN/INN)
E D09606 Duvoglustat hydrochloride (USAN)
E D09779 Emiglitate (JAN/INN)
E D11828 Clervonafusp alfa (USAN/INN)
D GAA* [HSA_VAR:2548v1] [HSA:2548] [KO:K12316]
E D03207 Alglucosidase alfa (USAN/INN) <JP/US>
E D11744 Avalglucosidase alfa (USAN/INN) <JP/US>
D GANC [HSA:2595] [KO:K12317]
E D00216 Acarbose (JAN/USAN/INN) <JP/US>
E D00625 Miglitol (JP18/USAN/INN) <JP/US>
E D01665 Voglibose (JP18/USAN/INN) <JP>
E D09779 Emiglitate (JAN/INN)
D MGAM [HSA:8972] [KO:K12047]
E D00216 Acarbose (JAN/USAN/INN) <JP/US>
E D00625 Miglitol (JP18/USAN/INN) <JP/US>
E D01665 Voglibose (JP18/USAN/INN) <JP>
E D09779 Emiglitate (JAN/INN)
D MAN2B1* [HSA_VAR:4125v1] [HSA:4125] [KO:K12311]
E D11024 Velmanase alfa (USAN/INN) <US>
D GUSB [HSA:2990] [KO:K01195]
E D01805 Aceglatone (JAN/INN)
D GUSB* [HSA_VAR:2990v1] [HSA:2990] [KO:K01195]
E D11004 Vestronidase alfa (USAN/INN) <JP/US>
D GLA* [HSA_VAR:2717v1] [HSA:2717] [KO:K01189]
E D02784 Agalsidase alfa (USAN/INN) <JP>
E D03228 Agalsidase beta (INN) <JP/US>
D GLA* [HSA_VAR:2717v2] [HSA:2717] [KO:K01189]
E D05031 Migalastat hydrochloride (JAN/USAN) <JP/US>
D GBA* [HSA_VAR:2629v1] [HSA:2629] [KO:K01201]
E D02810 Alglucerase (JAN/USAN/INN)
E D03020 Imiglucerase (USAN/INN) <JP/US>
E D09029 Velaglucerase alfa (USAN) <JP/US>
E D09675 Taliglucerase alfa (USAN/INN) <US>
D SI [HSA:6476] [KO:K01203]
E D03342 Camiglibose (USAN)
D SI* [HSA_VAR:6476v1] [HSA:6476] [KO:K01203]
E D05782 Sacrosidase (USAN) <US>
D NAGLU* [HSA_VAR:4669v1] [HSA:4669] [KO:K01205]
E D11199 Lesinidase alfa (USAN/INN)
D IDUA* [HSA_VAR:3425v1] [HSA:3425] [KO:K01217]
E D04670 Laronidase (USAN) <JP/US>
D HPSE [HSA:10855] [KO:K07964]
E D11764 Necuparanib (USAN/INN)
E D11765 Necuparanib sodium (USAN)
C ADP-ribosyl cyclase [EC:3.2.2.6]
D CD38 [HSA:952] [KO:K01242]
E D10777 Daratumumab (USAN) <JP/US>
E D11050 Isatuximab (USAN/INN) <JP/US>
E D12315 Ciltacabtagene autoleucel (USAN/INN) <US>
E D11945 Mezagitamab (USAN/INN)
C Aminopeptidases [EC:3.4.11.-]
D ANPEP (CD13) [HSA:290] [KO:K11140]
E D00087 Ubenimex (JP18/INN) <JP>
E D10026 Tosedostat (USAN/INN)
C Dipeptidases [EC:3.4.13.-]
D DPEP1 [HSA:1800] [KO:K01273]
E D02194 Cilastatin sodium (JP18/USP)
E D07698 Cilastatin (INN)
C Peptidyl-peptidases [EC:3.4.14.-]
D CTSC (DPP1) [HSA:1075] [KO:K01275]
E D12120 Brensocatib (USAN/INN)
D DPP4 (CD26) [HSA:1803] [KO:K01278]
E D08516 Sitagliptin (USAN)
E D06645 Sitagliptin phosphate (USAN) <JP/US>
E D12294 Sitagliptin phosphate (JAN)
E D07080 Vildagliptin (JAN/USAN/INN) <JP>
E D08996 Saxagliptin (USAN/INN)
E D09753 Saxagliptin hydrate (JAN) <JP>
E D10262 Saxagliptin hydrochloride <US>
E D06553 Alogliptin benzoate (JAN/USAN) <JP/US>
E D09566 Linagliptin (JAN/USAN/INN) <JP/US>
E D10502 Gemigliptin (prop.INN)
E D11023 Evogliptin (INN)
E D08616 Teneligliptin (INN)
E D09756 Teneligliptin hydrobromide hydrate (JAN) <JP>
E D11968 Teneligliptin hydrobromide (JAN)
E D06578 Denagliptin tosylate (USAN)
E D08631 Carmegliptin (USAN/INN)
E D09326 Carmegliptin dihydrochloride (USAN)
E D09333 Dutogliptin (USAN)
E D09334 Dutogliptin tartrate (USAN)
E D09625 Gosogliptin (USAN/INN)
E D09780 Anagliptin (JAN/INN) <JP>
E D10178 Trelagliptin (USAN)
E D10179 Trelagliptin succinate (JAN/USAN) <JP>
E D10317 Omarigliptin (JAN/USAN/INN) <JP>
D DPP8 [HSA:54878] [KO:K08655]
E D05989 Talabostat (USAN/INN)
E D05990 Talabostat mesylate (USAN)
D DPP9 [HSA:91039] [KO:K08656]
E D05989 Talabostat (USAN/INN)
E D05990 Talabostat mesylate (USAN)
D TPP1* [HSA_VAR:1200v1] [HSA:1200] [KO:K01279]
E D10813 Cerliponase alfa (USAN/INN) <JP/US>
C Peptidyl-dipeptidases [EC:3.4.15.-]
D ACE (CD143) [HSA:1636] [KO:K01283]
E D00251 Captopril (JP18/USP/INN) <JP/US>
E D07892 Enalapril (INN)
E D00621 Enalapril maleate (JP18/USP) <JP/US>
E D08131 Lisinopril (INN)
E D00362 Lisinopril (USP) <JP/US>
E D03753 Perindopril (USAN/INN)
E D00624 Perindopril erbumine (JAN/USP) <JP/US>
E D11580 Perindopril arginine
E D00421 Ramipril (USP/INN) <US>
E D03752 Quinapril (INN)
E D00459 Quinapril hydrochloride (JP18/USP) <US>
E D07499 Benazepril (INN)
E D00620 Benazepril hydrochloride (JAN/USP) <JP/US>
E D07699 Cilazapril (INN)
E D01069 Cilazapril (USAN)
E D07992 Fosinopril (INN)
E D00622 Fosinopril sodium (USP) <US>
E D00383 Trandolapril (JAN/USP/INN) <JP/US>
E D08529 Spirapril (INN)
E D03765 Spirapril hydrochloride (USAN)
E D07781 Delapril (INN)
E D01667 Delapril hydrochloride (JAN/USAN) <JP>
E D08225 Moexipril (INN)
E D00623 Moexipril hydrochloride (USP) <US>
E D08566 Temocapril (INN)
E D01119 Temocapril hydrochloride (JP18/USAN) <JP>
E D08688 Zofenopril (INN)
E D03767 Zofenopril calcium (USAN)
E D08068 Imidapril (INN)
E D01549 Imidapril hydrochloride (JP18) <JP>
E D01900 Alacepril (JP18/INN) <JP>
E D03077 Benazeprilat (USAN/INN)
E D03440 Ceronapril (USAN/INN)
E D03756 Indolapril hydrochloride (USAN)
E D03758 Libenzapril (USAN/INN)
E D03760 Pentopril (USAN/INN)
E D03763 Pivopril (USAN/INN)
E D03769 Enalaprilat (USP) <US>
E D03772 Fosinoprilat (USAN/INN)
E D03773 Quinaprilat (USAN/INN)
E D03775 Spiraprilat (USAN/INN)
E D03776 Zofenoprilat arginine (USAN)
E D04312 Gemopatrilat (USAN/INN)
E D06076 Teprotide (USAN/INN)
C Metallocarboxypeptidases [EC:3.4.17.-]
D FOLH1 (PSMA) [HSA:2346] [KO:K14592]
E D04525 Indium In 111 capromab pendetide (USP)
E D12257 Gallium Ga 68 gozetotide (USAN) <US>
E D12132 Piflufolastat F-18 (USAN) <US>
E D12335 Lutetium Lu 177 vipivotide tetraxetan (USAN) <US>
E D03372 Capromab pendetide (USAN)
E D10070 Iofolastat I 123 (USAN)
E D10683 Technetium Tc99m trofolastat chloride (USAN/INN)
E D12121 Acapatamab (USAN)
E D12566 Nezastomig (USAN)
C Serine peptidases [EC:3.4.21.-]
D CTRB [HSA:1504 440387] [KO:K01310]
E D05183 Ulinastatin (JP18) <JP>
D PRSS [HSA:5644 5645 5646] [KO:K01312]
E D05183 Ulinastatin (JP18) <JP>
D F2 [HSA:2147] [KO:K01313]
E D03692 Desirudin (USAN/INN)
E D06880 Lepirudin (INN)
E D00181 Argatroban (USP) <JP/US>
E D07143 Melagatran (INN)
E D01981 Ximelagatran (JAN/USAN/INN)
E D03136 Bivalirudin (USAN/INN)
E D07144 Dabigatran etexilate (USAN/INN)
E D07082 Dabigatran etexilate mesylate (USAN) <JP/US>
E D03722 Efegatran sulfate (USAN)
E D03728 Napsagatran (USAN)
E D06410 Thrombomodulin alfa (USAN/INN) <JP>
E D09707 Dabigatran (USAN/INN)
E D11280 Bivalirudin trifluoroacetate (USAN) <US>
D F10 [HSA:2159] [KO:K01314]
E D07086 Rivaroxaban (JAN/USAN/INN) <JP/US>
E D03213 Apixaban (JAN/USAN/INN) <JP/US>
E D09710 Edoxaban (USAN/INN)
E D09546 Edoxaban tosilate hydrate (JAN) <JP/US>
E D11568 Edoxaban tosylate (USAN)
E D08873 Betrixaban (USAN)
E D01844 Fondaparinux sodium (JAN/USP/INN) <JP/US>
E D12421 Freeze-dried activated human blood coagulation factor VII concentrate containing factor X <JP>
E D10821 Emicizumab (USAN/INN) <JP/US>
E D11029 Andexanet alfa (USAN/INN) <JP/US>
E D04029 Razaxaban hydrochloride (USAN)
E D04183 Fidexaban (USAN/INN)
E D06142 Tifacogin (USAN/INN)
E D08858 Antithrombin alfa (INN/USAN)
E D08913 Eribaxaban (USAN)
E D09817 Darexaban maleate (JAN)
E D09923 Letaxaban (USAN/INN)
E D10471 Idraparinux sodium (USAN)
D PLG [HSA:5340] [KO:K01315]
E D00160 Aminocaproic acid (USP/INN) <US>
E D01136 Tranexamic acid (JP18/USP/INN) <JP/US>
E D07568 Aminomethylbenzoic acid
E D12149 Plasminogen
D F9 [HSA:2158] [KO:K01321]
E D10821 Emicizumab (USAN/INN) <JP/US>
E D10150 Pegnivacogin sodium (USAN)
E D10484 Pegnivacogin (USAN)
E D12500 Etranacogene dezaparvovec (USAN/INN) <US>
E D12541 Gruticibart (USAN)
D KLKB1 [HSA:3818] [KO:K01324]
E D03931 Ecallantide (USAN/INN) <US>
E D10845 Conestat alfa (INN) <US>
E D11094 Lanadelumab (USAN) <JP/US>
E D11673 Berotralstat (USAN)
E D11674 Berotralstat hydrochloride (JAN/USAN) <JP/US>
E D01672 Gabexate mesilate (JP18) <JP>
E D08004 Gabexate (INN)
E D12396 Sebetralstat (USAN)
D KLK [HSA:3816 3817] [KO:K01325]
E D01672 Gabexate mesilate (JP18) <JP>
E D08004 Gabexate (INN)
D CELA1 [HSA:1990] [KO:K01326]
E D11770 Vonapanitase (USAN/INN)
D ELANE [HSA:1991] [KO:K01327]
E D05183 Ulinastatin (JP18) <JP>
E D01918 Sivelestat sodium (USAN) <JP>
E D03686 Depelestat (USAN/INN)
E D03788 Sivelestat (USAN/INN)
D C1R [HSA:715] [KO:K01330]
E D10845 Conestat alfa (INN) <US>
D C1S [HSA:716] [KO:K01331]
E D10845 Conestat alfa (INN) <US>
E D11530 Sutimlimab (USAN/INN) <JP/US>
D CFB [HSA:629] [KO:K01335]
E D12251 Iptacopan (USAN/INN)
E D12252 Iptacopan hydrochloride (USAN)
D CFD [HSA:1675] [KO:K01334]
E D10440 Lampalizumab (USAN/INN)
E D11641 Danicopan (JAN/USAN/INN)
E D12481 Vemircopan (USAN/INN)
D MASP2 [HSA:10747] [KO:K03993]
E D11531 Narsoplimab (USAN)
D PCSK9 [HSA:255738] [KO:K13050]
E D10557 Evolocumab (USAN/INN) <JP/US>
E D10335 Alirocumab (USAN) <US>
E D11931 Inclisiran (USAN/INN)
E D12293 Inclisiran sodium (JAN) <US>
E D10621 Bococizumab (USAN/INN)
E D11398 Frovocimab (USAN)
D HTRA1 [HSA:5654] [KO:K08784]
E D12379 Galegenimab (USAN)
D LPA [HSA:4018] [KO:K09644]
E D12460 Muvalaplin (USAN)
C Cysteine peptidases [EC:3.4.22.-]
D CASP1 [HSA:834] [KO:K01370]
E D08978 Pralnacasan (USAN/INN)
E D09938 Nivocasan (USAN)
E D10004 Emricasan (USAN/INN)
E D10416 Belnacasan (USAN)
D CASP9 [HSA:842] [KO:K04399]
E D11195 Rimiducid (USAN/INN)
D CTSS [HSA:1520] [KO:K01368]
E D11376 Petesicatib (USAN)
D CTSK [HSA:1513] [KO:K01371]
E D06634 Relacatib (USAN/INN)
E D08955 Odanacatib (JAN/USAN)
C Aspartic peptidases [EC:3.4.23.-]
D REN [HSA:5972] [KO:K01380]
E D09038 Remikiren (INN)
E D03208 Aliskiren (USAN/INN)
E D06412 Aliskiren fumarate (JAN/USAN) <JP/US>
E D03738 Enalkiren (USAN/INN)
E D03741 Ditekiren (USAN)
E D03743 Terlakiren (USAN/INN)
E D03745 Zankiren hydrochloride (USAN)
D BACE [HSA:23621 25825] [KO:K04521 K07747]
E D10739 Verubecestat (JAN/USAN/INN)
E D11509 Elenbecestat (JAN/USAN)
D BACE1 [HSA:23621] [KO:K04521]
E D10946 Lanabecestat (USAN)
E D10947 Lanabecestat camsylate (USAN)
E D11456 Atabecestat (USAN/INN)
E D11690 Umibecestat (USAN/INN)
D PSEN1/PSENEN/NCSTN/APH1A [HSA:5663 55851 23385 51107] [KO:K04505 K06170 K06171 K06172]
E D08869 Begacestat (USAN/INN)
E D09010 Tarenflurbil (USAN/INN)
E D09377 Semagacestat (USAN/INN)
E D09869 Avagacestat (USAN)
E D10960 Nirogacestat (USAN/INN)
E D11151 Crenigacestat (USAN/INN)
E D11453 Nirogacestat hydrobromide (USAN)
E D12235 Osugacestat (USAN)
C Metallo peptidases [EC:3.4.24.- 3.4.17.-]
D MME (CD10) [HSA:4311] [KO:K01389]
E D08464 Racecadotril (INN)
E D01070 Candoxatril (JAN/USAN/INN)
E D01970 Omapatrilat (JAN/USAN/INN)
E D03349 Candoxatrilat (USAN/INN)
E D03929 Ecadotril (USAN/INN)
E D10225 Sacubitril (JAN/USAN/INN)
D MMP1 [HSA:4312] [KO:K01388]
E D03517 Cipemastat (USAN/INN)
E D03795 Marimastat (USAN/INN)
E D03800 Rebimastat (USAN/INN)
E D03802 Tanomastat (USAN/INN)
E D11020 Diclofenac etalhyaluronate sodium (JAN) <JP>
D MMP2 [HSA:4313] [KO:K01398]
E D03061 Batimastat (USAN/INN)
E D03793 Ilomastat (USAN/INN)
E D03795 Marimastat (USAN/INN)
E D03797 Prinomastat (USAN/INN)
E D03800 Rebimastat (USAN/INN)
E D03802 Tanomastat (USAN/INN)
D MMP3 [HSA:4314] [KO:K01394]
E D03795 Marimastat (USAN/INN)
E D03797 Prinomastat (USAN/INN)
D MMP7 [HSA:4316] [KO:K01397]
E D03795 Marimastat (USAN/INN)
D MMP8 [HSA:4317] [KO:K01402]
E D03517 Cipemastat (USAN/INN)
E D03800 Rebimastat (USAN/INN)
D MMP9 [HSA:4318] [KO:K01403]
E D03061 Batimastat (USAN/INN)
E D03517 Cipemastat (USAN/INN)
E D03793 Ilomastat (USAN/INN)
E D03795 Marimastat (USAN/INN)
E D03797 Prinomastat (USAN/INN)
E D03800 Rebimastat (USAN/INN)
E D03802 Tanomastat (USAN/INN)
E D11262 Andecaliximab (USAN/INN)
D MMP12 [HSA:4321] [KO:K01413]
E D03795 Marimastat (USAN/INN)
D MMP13 [HSA:4322] [KO:K07994]
E D03517 Cipemastat (USAN/INN)
E D03797 Prinomastat (USAN/INN)
E D08859 Apratastat (USAN/INN)
D MMP14 [HSA:4323] [KO:K07763]
E D03797 Prinomastat (USAN/INN)
E D03800 Rebimastat (USAN/INN)
D ADAM10 [HSA:102] [KO:K06704]
E D09320 Aderbasib (USAN/INN)
D ADAM17 [HSA:6868] [KO:K06059]
E D08859 Apratastat (USAN/INN)
E D09320 Aderbasib (USAN/INN)
D ADAMTS5 [HSA:11096] [KO:K08620]
E D11995 Aldumastat (USAN)
C Threonine peptidases [EC:3.4.25.-]
D PSMB1 [HSA:5689] [KO:K02732]
E D09640 Marizomib (USAN/INN)
E D10110 Delanzomib (USAN)
D PSMB2 [HSA:5690] [KO:K02734]
E D09640 Marizomib (USAN/INN)
D PSMB5 [HSA:5693] [KO:K02737]
E D03150 Bortezomib (JAN/USAN/INN) <JP/US>
E D12311 Bortezomib hydrate (JAN) <JP/US>
E D08880 Carfilzomib (JAN/USAN/INN) <JP/US>
E D10130 Ixazomib (USAN)
E D10131 Ixazomib citrate (JAN/USAN) <JP/US>
E D09640 Marizomib (USAN/INN)
E D10110 Delanzomib (USAN)
E D10318 Oprozomib (USAN/INN)
D PSMB8 [HSA:5696] [KO:K02740]
E D12512 Zetomipzomib (USAN/INN)
E D12513 Zetomipzomib maleate (USAN)
D PSMB9 [HSA:5698] [KO:K02741]
E D12512 Zetomipzomib (USAN/INN)
E D12513 Zetomipzomib maleate (USAN)
C Glutaminase [EC:3.5.1.2]
D GLS [HSA:2744] [KO:K01425]
E D11738 Telaglenastat (USAN/INN)
E D11739 Telaglenastat hydrochloride (USAN)
C Histone deacetylase [EC:3.5.1.98]
D HDAC [HSA:3065 3066 8841 9759 10014 10013 51564 55869 9734 83933 79885] [KO:K06067 K11404 K11406 K11407 K11408 K11405 K11409 K18671 K11418]
E D06320 Vorinostat (JAN/USAN) <JP/US>
E D06637 Romidepsin (JAN/USAN/INN) <JP/US>
E D10319 Panobinostat (USAN/INN)
E D10019 Panobinostat lactate (JAN) <JP>
E D08870 Belinostat (USAN/INN) <US>
E D09338 Entinostat (JAN/USAN/INN)
E D10060 Abexinostat (USAN)
E D10084 Abexinostat hydrochloride (USAN)
E D10321 Quisinostat (USAN/INN)
E D10322 Quisinostat hydrochloride (USAN)
E D10977 Remetinostat (USAN/INN)
E D12551 Bocodepsin (USAN)
E D12552 Bocodepsin besylate (USAN)
D HDAC1 [HSA:3065] [KO:K06067]
E D05988 Tacedinaline (USAN/INN)
E D09357 Mocetinostat dihydrobromide (USAN)
E D09641 Mocetinostat (USAN/INN)
E D10993 Tucidinostat (JAN/USAN/INN) <JP>
E D11182 Tinostamustine (USAN/INN)
E D11319 Fimepinostat (USAN/INN)
E D11442 Nanatinostat (USAN)
D HDAC2 [HSA:3066] [KO:K06067]
E D09357 Mocetinostat dihydrobromide (USAN)
E D09641 Mocetinostat (USAN/INN)
E D10993 Tucidinostat (JAN/USAN/INN) <JP>
E D11182 Tinostamustine (USAN/INN)
E D11319 Fimepinostat (USAN/INN)
E D11442 Nanatinostat (USAN)
D HDAC3 [HSA:8841] [KO:K11404]
E D09357 Mocetinostat dihydrobromide (USAN)
E D09641 Mocetinostat (USAN/INN)
E D10993 Tucidinostat (JAN/USAN/INN) <JP>
E D11182 Tinostamustine (USAN/INN)
E D11319 Fimepinostat (USAN/INN)
E D11442 Nanatinostat (USAN)
D HDAC4 [HSA:9759] [KO:K11406]
E D11319 Fimepinostat (USAN/INN)
D HDAC5 [HSA:10014] [KO:K11406]
E D11319 Fimepinostat (USAN/INN)
D HDAC6 [HSA:10013] [KO:K11407]
E D10661 Ricolinostat (USAN/INN)
E D10918 Citarinostat (USAN)
E D11182 Tinostamustine (USAN/INN)
E D11319 Fimepinostat (USAN/INN)
D HDAC7 [HSA:51564] [KO:K11408]
E D11319 Fimepinostat (USAN/INN)
D HDAC8 [HSA:55869] [KO:K11405]
E D09357 Mocetinostat dihydrobromide (USAN)
E D09641 Mocetinostat (USAN/INN)
E D11319 Fimepinostat (USAN/INN)
E D11442 Nanatinostat (USAN)
D HDAC9 [HSA:9734] [KO:K11409]
E D11319 Fimepinostat (USAN/INN)
D HDAC10 [HSA:83933] [KO:K18671]
E D10993 Tucidinostat (JAN/USAN/INN) <JP>
E D11319 Fimepinostat (USAN/INN)
D HDAC11 [HSA:79885] [KO:K11418]
E D09357 Mocetinostat dihydrobromide (USAN)
E D09641 Mocetinostat (USAN/INN)
C Arginase [EC:3.5.3.1]
D ARG1 [HSA:383] [KO:K01476]
E D11792 Numidargistat (USAN)
D ARG1* [HSA_VAR:383v1] [HSA:383] [KO:K01476]
E D11695 Pegzilarginase (USAN/INN)
C Adenosine deaminase [EC:3.5.4.4]
D ADA [HSA:100] [KO:K01488]
E D00155 Pentostatin (JAN/USAN/INN) <JP/US>
D ADA* [HSA_VAR:100v1] [HSA:100] [KO:K01488]
E D11017 Elapegademase (USAN/INN) <JP/US>
C Cytidine deaminase [EC:3.5.4.5]
D CDA [HSA:978] [KO:K01489]
E D11679 Cedazuridine (USAN/INN)
C ATPase [EC:3.6.3.-]
D ATP1A [HSA:476 477 478 480] [KO:K01539]
E D06881 Acetyldigitoxin (INN)
E D07555 Acetyldigoxin
E D00297 Digitoxin (JAN/USP/INN)
E D00298 Digoxin (JP18/USP) <JP/US>
E D01972 Lanatoside C (JAN/INN)
E D01240 Deslanoside (JP18/USP/INN) <JP>
E D09847 Metildigoxin (INN)
E D02587 Metildigoxin (JP18) <JP>
E D07147 Gitoformate (INN)
E D01379 Proscillaridin (JAN/USAN/INN)
E D00112 G-Strophanthin (JAN)
E D00645 Bretylium tosylate (USP)
E D07520 Bepridil (INN)
E D00631 Bepridil hydrochloride (USAN) <JP>
E D07556 beta-Acetyldigoxin
D ATP2A [HSA:487 488 489] [KO:K05853]
E D10715 Mipsagargin (USAN/INN)
D ATP4 [HSA:495 496] [KO:K01542 K01543]
E D00455 Omeprazole (JP18/USP/INN) <JP/US>
E D01207 Omeprazole sodium (USAN)
E D05261 Omeprazole sodium injection (JAN) <JP>
E D05259 Omeprazole magnesium (USP) <US>
E D05353 Pantoprazole (USAN/INN)
E D02593 Pantoprazole sodium (USP) <US>
E D00355 Lansoprazole (JP18/USP/INN) <JP/US>
E D08463 Rabeprazole (INN)
E D00724 Rabeprazole sodium (JP18/USP) <JP/US>
E D07917 Esomeprazole (INN)
E D01984 Esomeprazole magnesium (USP) <JP/US>
E D04056 Esomeprazole sodium (USAN) <US>
E D09339 Esomeprazole potassium (USAN)
E D10120 Esomeprazole strontium (USAN) <US>
E D11114 Esomeprazole magnesium dihydrate <US>
E D08903 Dexlansoprazole (INN/USAN) <US>
E D11784 Vonoprazan (USAN/INN)
E D10466 Vonoprazan fumarate (JAN/USAN) <JP>
E D12246 Tegoprazan (INN)
E D01920 Tenatoprazole (JAN/INN)
E D05722 Revaprazan hydrochloride (USAN)
E D05900 Timoprazole (INN)
E D05901 Picoprazole (INN)
E D05906 Leminoprazole (INN)
E D09837 Penaprazole sodium hydrate (JAN)
D ABCB1 (CD243) [HSA:5243] [KO:K05658]
E D03128 Biricodar dicitrate (USAN)
E D03968 Elacridar hydrochloride (USAN)
E D06008 Tariquidar (USAN/INN)
E D06084 Tesmilifene hydrochloride (USAN)
E D06277 Valspodar (USAN/INN)
E D06387 Zosuquidar trihydrochloride (USAN)
E D11782 Encequidar (USAN/INN)
E D11783 Encequidar mesylate (USAN)
B Lyases (EC4)
C Carboxy-lyases [EC:4.1.1.-]
D GAD [HSA:2571 2572] [KO:K01580]
E D00399 Valproic acid (USP) <US>
E D00304 Divalproex sodium (USP) <US>
E D00710 Valproate sodium (USAN) <JP/US>
E D08667 Calcium valproate
D ODC1 [HSA:4953] [KO:K01581]
E D07883 Eflornithine (INN)
E D00829 Eflornithine hydrochloride (USAN) <US>
D HDC [HSA:3067] [KO:K01590]
E D07405 Tritoqualine (INN)
E D03158 Brocresine (USAN/INN)
D DDC [HSA:1644] [KO:K01593]
E D00558 Carbidopa (USP) <US>
E D01653 Benserazide hydrochloride (JP18)
E D03082 Benserazide (USAN/INN)
E D04997 Methyldopate hydrochloride (USP)
D DDC* [HSA_VAR:1644v1] [HSA:1644] [KO:K01593]
E D12407 Eladocagene exuparvovec (USAN/INN)
D AMD1 [HSA:262] [KO:K01611]
E D07258 Mitoguazone (INN)
D GGCX [HSA:2677] [KO:K10106]
E D07457 Anisindione (INN)
C Aldehyde-lyases [EC:4.1.2.-]
D CA [HSA:759 760 761 762 763 11238 765 766 767 768 771 377677 23632] [KO:K01672 K18245 K18246]
E D01822 Clofenamide (JAN/INN)
E D00218 Acetazolamide (JP18/USP/INN) <JP/US>
E D01196 Acetazolamide sodium (JAN) <JP/US>
E D00518 Dichlorphenamide (USP) <US>
E D07871 Dorzolamide (INN)
E D00653 Dorzolamide hydrochloride (JP18/USP) <JP/US>
E D00655 Methazolamide (JAN/USP/INN) <US>
E D02441 Ethoxzolamide
E D03845 Sezolamide hydrochloride (USAN)
D CA2 [HSA:760] [KO:K18245]
E D00537 Topiramate (JAN/USP/INN) <JP/US>
E D00652 Brinzolamide (JAN/USP/INN) <JP/US>
D CA4 [HSA:762] [KO:K18246]
E D00537 Topiramate (JAN/USP/INN) <JP/US>
D CA9 [HSA:768] [KO:K01672]
E D09593 Girentuximab (USAN/INN)
E D09632 Iodine I 124 girentuximab (USAN/INN)
C Hydro-lyases [EC:4.2.1.-]
D CBS [HSA:875] [KO:K01697]
E D12197 Pegtibatinase (USAN)
C Phosphorus-oxygen lyases [EC:4.6.1.-]
D ADCY [HSA:107 108 109 196883 111 112 113 114 115 55811] [KO:K08041 K08042 K08043 K08044 K08045 K08046 K08047 K08048 K08049 K11265]
E D01697 Colforsin daropate hydrochloride (JAN) <JP>
E D03584 Colforsin (USAN/INN)
D NPR [HSA:4881 4882] [KO:K12323 K12324]
E D04051 Erythrityl tetranitrate (USAN)
E D02935 Anaritide acetate (USAN)
E D10063 Cenderitide (USAN)
D NPR1 [HSA:4881] [KO:K12323]
E D05147 Nesiritide (USAN/INN)
E D05148 Nesiritide citrate (USAN)
E D03328 Carperitide (USAN/INN) <JP>
D NPR2 [HSA:4882] [KO:K12324]
E D11190 Vosoritide (USAN/INN) <JP/US>
D GUCY1A [HSA:2977 2982] [KO:K12318]
E D01810 Nicorandil (JP18/USAN/INN) <JP>
E D11051 Vericiguat (JAN/USAN/INN) <JP/US>
E D09572 Riociguat (JAN/USAN/INN) <JP/US>
E D00517 Amyl nitrite (JP18/USP) <JP>
E D07577 Cinaciguat (JAN/INN)
E D11274 Praliciguat (USAN/INN)
E D11475 Olinciguat (USAN/INN)
E D12516 Zagociguat (USAN/INN)
D GUCY1B [HSA:2983] [KO:K12319]
E D01810 Nicorandil (JP18/USAN/INN) <JP>
E D11051 Vericiguat (JAN/USAN/INN) <JP/US>
E D09572 Riociguat (JAN/USAN/INN) <JP/US>
E D00517 Amyl nitrite (JP18/USP) <JP>
E D07577 Cinaciguat (JAN/INN)
E D11274 Praliciguat (USAN/INN)
E D11475 Olinciguat (USAN/INN)
E D12516 Zagociguat (USAN/INN)
D GUCY2C [HSA:2984] [KO:K12320]
E D09355 Linaclotide (JAN/USAN) <JP/US>
E D06612 Linaclotide acetate (USAN)
E D09948 Plecanatide (USAN/INN) <US>
E D10976 Recanaclotide (USAN/INN)
E D11233 Dolcanatide (USAN/INN)
C Moco biosynthesis enzyme [EC:4.1.99.2 4.6.1.17]
D MOCS1* [HSA_VAR:4337v1] [HSA:4337] [KO:K20967]
E D11779 Fosdenopterin (USAN)
E D11780 Fosdenopterin hydrobromide (USAN) <US>
B Isomerases (EC5)
C Peptidylprolyl isomerase [EC:5.2.1.8]
D PPIA [HSA:5478] [KO:K03767]
E D10087 Alisporivir (USAN)
C Prostaglandin-E synthase [EC:5.3.99.3]
D PTGES [HSA:9536] [KO:K15729]
E D01545 Aceclofenac (JAN/INN)
C Thromboxane-A synthase [EC:5.3.99.5]
D TBXAS1 (CYP5A1) [HSA:6916] [KO:K01832]
E D07140 Picotamide (BAN)
E D01220 Trapidil (JP18/INN) <JP>
E D01683 Ozagrel hydrochloride hydrate (JAN) <JP>
E D01684 Ozagrel sodium (JP18) <JP>
E D03661 Dazmegrel (USAN/INN)
E D03663 Dazoxiben hydrochloride (USAN)
E D04276 Furegrelate sodium (USAN)
E D05502 Pirmagrel (USAN/INN)
E D05727 Ridogrel (USAN/INN)
E D06077 Terbogrel (USAN/INN)
E D08327 Ozagrel (INN)
C DNA topoisomerase [EC:5.99.1.-]
D TOP1 [HSA:7150] [KO:K03163]
E D08618 Topotecan (BAN)
E D02168 Topotecan hydrochloride (USAN) <JP/US>
E D08086 Irinotecan (INN)
E D01061 Irinotecan hydrochloride (USP) <JP/US>
E D10642 Irinotecan sucrosofate (USAN)
E D10367 Etirinotecan pegol (USAN/INN)
E D10422 Etirinotecan pegol tetrahydrochloride (USAN)
E D10427 Etirinotecan pegol tetratriflutate (USAN)
E D03225 Belotecan hydrochloride (USAN)
E D02756 Aclarubicin (USAN/INN)
E D01911 Aclarubicin hydrochloride (JP18) <JP>
E D11529 Trastuzumab deruxtecan (USAN/INN) <JP/US>
E D10985 Sacituzumab govitecan (USAN/INN) <US>
E D01432 Exatecan mesylate (USAN)
E D03954 Edotecarin (USAN/INN)
E D03977 Elsamitrucin (USAN/INN)
E D04031 Rubitecan (USAN/INN)
E D04822 Lurtotecan dihydrochloride (USAN)
E D05385 Pegamotecan (USAN)
E D09327 Cositecan (USAN)
E D09679 Tenifatecan (USAN/INN)
E D10464 Firtecan pegol (USAN/INN)
E D12184 Patritumab deruxtecan (USAN/INN)
E D12359 Datopotamab deruxtecan (USAN/INN)
D TOP2 [HSA:7153 7155] [KO:K03164]
E D00125 Etoposide (JP18/USP/INN) <JP/US>
E D04107 Etoposide phosphate (USAN) <US>
E D02698 Teniposide (USP/INN)
E D03899 Doxorubicin (USAN/INN)
E D01275 Doxorubicin hydrochloride (JP18/USP) <JP/US>
E D07776 Daunorubicin (INN)
E D01264 Daunorubicin hydrochloride (JP18/USP) <JP/US>
E D10787 Daunorubicin citrate
E D07901 Epirubicin (INN)
E D02214 Epirubicin hydrochloride (JP18/USP) <JP/US>
E D02756 Aclarubicin (USAN/INN)
E D01911 Aclarubicin hydrochloride (JP18) <JP>
E D06386 Zorubicin hydrochloride (USAN)
E D08062 Idarubicin (INN)
E D01747 Idarubicin hydrochloride (JP18/USP) <JP/US>
E D08224 Mitoxantrone (INN)
E D02166 Mitoxantrone hydrochloride (JAN/USP) <JP/US>
E D01885 Pirarubicin (JP18/INN)
E D08386 Pirarubicin hydrochloride <JP>
E D02697 Valrubicin (USP/INN) <US>
E D08854 Amrubicin (USAN/INN)
E D07100 Amrubicin hydrochloride (JAN/USAN) <JP>
E D05522 Pixantrone (USAN/INN)
E D09654 Pixantrone dimaleate (USAN)
E D02321 Amsacrine (USAN/INN)
E D08024 Vosaroxin (USAN)
E D03730 Dexrazoxane (JAN/USAN/INN) <JP/US>
E D07807 Dexrazoxane hydrochloride <US>
E D01404 Sobuzoxane (JAN) <JP>
E D03220 Becatecarin (USAN/INN)
E D03602 Crisnatol mesylate (USAN)
E D03977 Elsamitrucin (USAN/INN)
E D04262 Fostriecin sodium (USAN)
E D04498 Idronoxil (USAN/INN)
E D04685 Ledoxantrone trihydrochloride (USAN)
E D04783 Losoxantrone hydrochloride (USAN)
E D04914 Menogaril (USAN/INN)
E D05054 Mitindomide (USAN/INN)
E D05510 Piroxantrone hydrochloride (USAN)
E D06059 Teloxantrone hydrochloride (USAN)
E D06167 Tirapazamine (USAN/INN)
E D06190 Topixantrone (USAN/INN)
E D08871 Berubicin hydrochloride (USAN)
E D08981 Quarfloxin (USAN)
E D10090 Amonafide (USAN)
E D10091 Amonafide l-malate (USAN)
E D10383 Aldoxorubicin (USAN)
E D10384 Aldoxorubicin Hydrochloride (USAN)
B Ligases (EC6)
C Ubiquitin activating enzyme [EC:6.2.1.45]
D UBLE1 [HSA:10055 10054] [KO:K10684 K10685]
E D12268 Subasumstat (USAN)
C GART [EC:6.3.4.13 2.1.2.2 6.3.3.1]
D GART [HSA:2618] [KO:K11787]
E D07472 Pemetrexed (INN) <US>
E D03828 Pemetrexed disodium (USAN) <US>
E D06503 Pemetrexed sodium hydrate (JAN) <JP/US>
E D10596 Pemetrexed sodium hemipentahydrate (JAN) <JP/US>
E D04766 Lometrexol sodium (USAN)
E D05400 Pelitrexol (USAN/INN)
E D11352 Pemetrexed tromethamine (USAN) <US>
C Carbamoyl-phosphate synthase [EC:6.3.4.16]
D CPS1 [HSA:1373] [KO:K01948]
E D07130 Carglumic acid (JAN/USAN/INN) <JP/US>
C Acetyl-CoA carboxylase [EC:6.4.1.2]
D ACACA [HSA:31] [KO:K11262]
E D11186 Olumacostat glasaretil (USAN/INN)
E D11640 Firsocostat (USAN/INN)
E D11902 Clesacostat (USAN)
E D11903 Clesacostat tromethamine (USAN)
D ACACB [HSA:32] [KO:K01946]
E D11186 Olumacostat glasaretil (USAN/INN)
E D11640 Firsocostat (USAN/INN)
E D11902 Clesacostat (USAN)
E D11903 Clesacostat tromethamine (USAN)
#
ANucleic acids
B RNAs
C MicroRNAs
D MIR155 [HSA:406947] [KO:K17009]
E D11163 Cobomarsen (USAN/INN)
E D11164 Cobomarsen sodium (USAN)
#
ANot elsewhere classified
B Signaling molecules
C Transcription factor
D NFE2L2 [HSA:4780] [KO:K05638]
E D10964 Omaveloxolone (USAN/INN) <US>
D AHR [HSA:196] [KO:K09093]
E D11365 Tapinarof (JAN/USAN) <US>
D HIF1A [HSA:3091] [KO:K08268]
E D10464 Firtecan pegol (USAN/INN)
D HIF2A [HSA:2034] [KO:K09095]
E D11954 Belzutifan (JAN/USAN/INN) <US>
D MYC [HSA:4609] [KO:K04377]
E D08956 Omacetaxine mepesuccinate (USAN) <US>
D SP1 [HSA:6667] [KO:K04684]
E D09014 Terameprocol (INN/USAN)
D EGR1 [HSA:1958] [KO:K09203]
E D11286 Brivoligide sodium (USAN)
E D11341 Brivoligide (USAN)
D NANOG [HSA:79923] [KO:K10164]
E D10903 Amcasertib (USAN/INN)
D NFKB1 [HSA:4790] [KO:K02580]
E D01146 Iguratimod (JAN/INN) <JP>
D STAT3 [HSA:6774] [KO:K04692]
E D10717 Napabucasin (JAN/USAN/INN)
D TP53 (p53) [HSA:7157] [KO:K04451]
E D08887 Cenersen sodium (USAN)
D RELA (NKFB3, p65) [HSA:5970] [KO:K04735]
E D12181 Edasalonexent (USAN/INN)
C Translation factor
D EIF4A3 [HSA:9775] [KO:K13025]
E D11837 Zotatifin (USAN/INN)
D EIF4E [HSA:1977] [KO:K03259]
E D10614 Briciclib (USAN/INN)
E D10694 Briciclib sodium (USAN)
C Chaperone and folding catalyst
D HSP90 [HSA:3320 3326 7184] [KO:K04079 K09487]
E D06554 Alvespimycin hydrochloride (USAN)
E D06650 Tanespimycin (USAN)
E D09375 Retaspimycin (USAN/INN)
E D09376 Retaspimycin hydrochloride (USAN)
E D10126 Ganetespib (USAN)
E D10646 Luminespib (USAN/INN)
E D10647 Luminespib mesylate (USAN)
E D10719 Onalespib (USAN/INN)
E D11766 Onalespib lactate (USAN)
E D11920 Pimitespib (JAN) <JP>
D HSP90B1 (GP96) [HSA:7184] [KO:K09487]
E D06667 Vitespen (USAN)
D CLU [HSA:1191] [KO:K17252]
E D09403 Custirsen sodium (USAN)
D APCS (SAP) [HSA:325] [KO:K23267]
E D11464 Miridesap (USAN/INN)
E D11471 Dezamizumab (USAN/INN)
E D12402 Zinpentraxin alfa (USAN)
C Spliceosome
D NCBP [HSA:4686 22916 392517] [KO:K12882 K12883]
E D12345 Obefazimod (USAN)
D SMN1 [HSA:6606] [KO:K13129]
E D11559 Onasemnogene abeparvovec (USAN/INN) <US>
D SMN2 [HSA:6607] [KO:K13129]
E D10881 Nusinersen (USAN/INN)
E D10791 Nusinersen sodium (JAN) <JP/US>
E D11406 Risdiplam (JAN/USAN/INN) <JP/US>
E D12272 Branaplam (USAN/INN)
E D12273 Branaplam hydrochloride (USAN)
C G protein
D RAC1 [HSA:5879] [KO:K04392]
E D11032 Plitidepsin (INN)
D KRAS* [HSA_VAR:3845v1] [HSA:3845] [KO:K07827]
E D12055 Sotorasib (JAN/USAN) <JP/US>
E D12301 Adagrasib (USAN) <US>
C Signaling adaptor
D ARRB [HSA:408 409] [KO:K04439]
E D11214 Oliceridine (USAN/INN)
D GRB2 [HSA:2885] [KO:K04364]
E D11165 Prexigebersen (USAN/INN)
C mTOR signaling
D CASTOR [HSA:652968 729438] [KO:K23080 K23081]
E D11183 Sapanisertib (USAN/INN)
C Wnt signaling
D SOST [HSA:50964] [KO:K16834]
E D10156 Romosozumab (USAN) <JP/US>
E D10094 Blosozumab (USAN)
D RSPO3 [HSA:84870] [KO:K23098]
E D11369 Rosmantuzumab (USAN)
D CTNNB1 [HSA:1499] [KO:K02105]
E D12445 Foscenvivint (JAN/INN)
C Notch signaling
D NOTCH1 [HSA:4851] [KO:K02599]
E D11151 Crenigacestat (USAN/INN)
E D11229 Brontictuzumab (USAN/INN)
D NOTCH2 [HSA:4853] [KO:K20994]
E D11775 Tarextumab (USAN/INN)
D NOTCH3 [HSA:4854] [KO:K20995]
E D11775 Tarextumab (USAN/INN)
D DLL3 [HSA:10683] [KO:K06051]
E D10981 Rovalpituzumab tesirine (USAN/INN)
E D11117 Rovalpituzumab (USAN)
E D12234 Tarlatamab (USAN)
D DLL4 [HSA:54567] [KO:K06051]
E D10353 Demcizumab (USAN/INN)
E D10460 Enoticumab (USAN/INN)
E D11126 Navicixizumab (USAN/INN)
E D11642 Dilpacimab (USAN/INN)
C TGF-beta signaling
D SMAD7 [HSA:4092] [KO:K19631]
E D10955 Mongersen sodium (USAN)
E D10956 Mongersen (INN)
C Calcium signaling
D CALM [HSA:801 805 808 810 91860 51806 163688] [KO:K02183]
E D04789 Lubeluzole (USAN/INN)
C cAMP signaling
D ADCYAP [HSA:116] [KO:K05262]
E D12459 Vipalanebart (USAN)
B Cellular process
C Cell cycle
D CCND1 [HSA:595] [KO:K04503]
E D08956 Omacetaxine mepesuccinate (USAN) <US>
D CDC7 [HSA:8317] [KO:K02214]
E D12176 Simurosertib (USAN/INN)
C Apoptosis
D BCL2 [HSA:596] [KO:K02161]
E D08290 Oblimersen (INN)
E D05216 Oblimersen sodium (USAN)
E D08954 Obatoclax mesylate (USAN)
D BCL2* [HSA_VAR:596v1] [HSA:596] [KO:K02161]
E D10679 Venetoclax (JAN/USAN/INN) <JP/US>
D BCL2L [HSA:598 599 4170 597] [KO:K04570 K02163 K02539 K02162]
E D09935 Navitoclax (JAN/USAN/INN)
E D09936 Navitoclax dihydrochloride (USAN)
D MCL1 [HSA:4170] [KO:K02539]
E D08956 Omacetaxine mepesuccinate (USAN) <US>
E D11962 Murizatoclax (USAN/INN)
E D11963 Tapotoclax (USAN/INN)
D BIRC5 [HSA:332] [KO:K08731]
E D09909 Gataparsen (USAN/INN)
E D09910 Gataparsen sodium (USAN)
E D10164 Sepantronium bromide (JAN/USAN)
C Membrane trafficking
D GPNMB [HSA:10457] [KO:K20732]
E D09623 Glembatumumab (USAN/INN)
E D09912 Glembatumumab vedotin (USAN)
D MSLN [HSA:10232] [KO:K20733]
E D09767 Amatuximab (USAN)
D RTN4 [HSA:57142] [KO:K20720]
E D10331 Ozanezumab (USAN)
D SNCA [HSA:6622] [KO:K04528]
E D11420 Prasinezumab (USAN/INN)
E D11467 Cinpanemab (USAN)
D LINGO1 [HSA:84894] [KO:K23533]
E D11767 Opicinumab (USAN/INN)
D SORT1 [HSA:6272] [KO:K12388]
E D12427 Latozinemab (USAN/INN)
C Cytoskeleton
D MYL2 [HSA:4633] [KO:K10351]
E D12253 Aficamten (USAN)
D MYL3 [HSA:4634] [KO:K12749]
E D12253 Aficamten (USAN)
D MYL4 [HSA:4635] [KO:K12750]
E D12253 Aficamten (USAN)
D MYH6_7 [HSA:4624 4625] [KO:K17751]
E D04510 Imciromab pentetate (USAN)
E D12253 Aficamten (USAN)
D MYH7 [HSA:4625] [KO:K17751]
E D12265 Mavacamten (USAN/INN) <US>
D TNNC2 [HSA:7125] [KO:K12042]
E D11363 Reldesemtiv (USAN)
D TNNI2 [HSA:7136] [KO:K12043]
E D11363 Reldesemtiv (USAN)
D TNNT3 [HSA:7140] [KO:K12046]
E D11363 Reldesemtiv (USAN)
D DMD [HSA:1756] [KO:K10366]
E D10114 Drisapersen (USAN)
E D10115 Drisapersen sodium (JAN/USAN)
E D11918 Renadirsen sodium (JAN)
D DMD* [HSA_VAR:1756v1] [HSA:1756] [KO:K10366]
E D09900 Eteplirsen (USAN/INN) <US>
E D11707 Golodirsen (USAN/INN) <US>
E D11528 Viltolarsen (JAN/USAN) <JP/US>
E D11988 Casimersen (USAN/INN) <US>
D TUBB [HSA:10381 10382 10383 203068 347688 347733 7280 81027 84617] [KO:K07375]
E D11691 Tirbanibulin (USAN/INN) <US>
E D11692 Tirbanibulin mesylate (USAN)
E D08675 Vinblastine (INN)
E D01068 Vinblastine sulfate (JP18/USP) <JP/US>
E D08679 Vincristine (INN)
E D02197 Vincristine sulfate (JP18/USP) <JP/US>
E D06304 Vindesine (USAN/INN)
E D01769 Vindesine sulfate (JAN/USAN) <JP>
E D08680 Vinorelbine (INN)
E D01935 Vinorelbine tartrate (USP) <JP/US>
E D09032 Vinflunine ditartrate (USAN)
E D00491 Paclitaxel (JAN/USP/INN) <JP/US>
E D07866 Docetaxel (JAN/INN) <JP/US>
E D02165 Docetaxel (USP) <JP/US>
E D05333 Paclitaxel poliglumex (USAN/INN)
E D09755 Cabazitaxel (USAN/INN)
E D10452 Cabazitaxel acetonate (JAN) <JP/US>
E D04645 Ixabepilone (JAN/USAN/INN) <US>
E D09980 Trastuzumab emtansine (USAN/INN) <JP/US>
E D09587 Brentuximab vedotin (USAN) <JP/US>
E D11525 Enfortumab vedotin (USAN) <JP/US>
E D11595 Belantamab mafodotin (USAN) <US>
E D11814 Tisotumab vedotin (USAN/INN) <US>
E D04066 Estramustine (USAN/INN)
E D02398 Estramustine phosphate sodium (USAN)
E D06397 Estramustine phosphate sodium hydrate (JAN) <JP/US>
E D08914 Eribulin mesylate (USAN) <JP/US>
E D00570 Colchicine (JP18/USP) <JP/US>
E D01919 Soblidotin (JAN/INN)
E D03059 Batabulin sodium (USAN)
E D03364 Cantuzumab mertansine (USAN)
E D04864 Maytansine (USAN)
E D05062 Mivobulin isethionate (USAN)
E D06001 Taltobulin (USAN/INN)
E D06009 Tasidotin hydrochloride (USAN)
E D06305 Vinepidine sulfate (USAN)
E D06306 Vinglycinate sulfate (USAN)
E D06307 Vinleurosine sulfate (USAN)
E D06308 Vinrosidine sulfate (USAN)
E D06309 Vinzolidine sulfate (USAN)
E D06560 Batabulin (USAN/INN)
E D06576 Cevipabulin fumarate (USAN)
E D08889 Cevipabulin succinate (USAN)
E D09691 Vedotin (USAN)
E D09912 Glembatumumab vedotin (USAN)
E D09927 Lorvotuzumab mertansine (USAN/INN)
E D10013 Indibulin (USAN/INN)
E D10029 Verubulin (USAN/INN)
E D10030 Verubulin hydrochloride (USAN)
E D10073 Lexibulin (USAN)
E D10454 Cantuzumab ravtansine (USAN)
E D10954 Mirvetuximab soravtansine (USAN/INN) <US>
E D11228 Soravtansine (USAN)
E D11232 Denintuzumab mafodotin (USAN/INN)
E D11238 Lifastuzumab vedotin (USAN/INN)
E D11494 Lisavanbulin (USAN/INN)
E D11681 Avanbulin (USAN/INN)
E D12183 Farletuzumab ecteribulin (USAN)
E D12210 Ozuriftmab vedotin (USAN)
E D12220 Mecbotamab vedotin
E D12310 Tusamitamab ravtansine (USAN/INN)
E D12519 Sabizabulin (USAN/INN)
E D12520 Sabizabulin hydrochloride (USAN)
D KIF11 [HSA:3832] [KO:K10398]
E D04640 Ispinesib mesylate (USAN)
E D09636 Litronesib (USAN/INN)
D MAPT (TAU) [HSA:4137] [KO:K04380]
E D11210 Flortaucipir F 18 (USAN) <US>
E D11293 Gosuranemab (USAN)
E D11384 Hydromethylthionine mesylate (USAN)
E D11427 Hydromethylthionine (USAN)
E D11533 Zagotenemab (USAN)
E D11687 Semorinemab (USAN/INN)
E D11840 Tilavonemab (USAN/INN)
E D12228 Bepranemab (USAN/INN)
D FLNA [HSA:2316] [KO:K04437]
E D12003 Simufilam (USAN)
E D12004 Simufilam hydrochloride (USAN)
C Ubiquitin system
D NAE1 [HSA:8883] [KO:K04532]
E D10413 Pevonedistat (USAN)
E D10654 Pevonedistat hydrochloride (JAN/USAN)
D KEAP1 [HSA:9817] [KO:K10456]
E D03846 Dimethyl fumarate (JAN/USAN) <JP/US>
D DIABLO (SMAC) [HSA:56616] [KO:K10522]
E D12565 Xevinapant (USAN/INN)
D CRBN [HSA:51185] [KO:K11793]
E D12000 Mezigdomide (USAN)
D RAD51 [HSA:5888] [KO:K04482]
E D12558 Emzadirib (USAN)
C Chromatin
D BMI1 [HSA:648] [KO:K11459]
E D11889 Unesblin (USAN)
D MEN1 [HSA:4221] [KO:K14970]
E D12419 Ziftomenib (USAN/INN)
C Cilia formation
D CEP290 [HSA:80184] [KO:K16533]
E D12488 Sepofarsen (USAN/INN)
B Organismal systems
C Complement and coagulation
D F8 [HSA:2157] [KO:K03899]
E D00291 Desmopressin (INN)
E D02235 Desmopressin acetate (USP) <JP/US>
D F8* [HSA_VAR:2157v1] [HSA:2157] [KO:K03899]
E D12434 Valoctocogene roxaparvovec (USAN/INN)
D F11 [HSA:2160] [KO:K01323]
E D11802 Milvexian (USAN)
E D12563 Frunexian (USAN
E D12564 Frunexian hydrochloride (USAN)
D VWF [HSA:7450] [KO:K03900]
E D11160 Caplacizumab (USAN/INN) <JP/US>
E D10758 Turoctocog alfa pegol (genetical recombination) (JAN) <JP>
D KNG1 [HSA:3827] [KO:K03898]
E D03330 Kallidinogenase (JP18/INN) <JP>
D C3 (C3b) [HSA:718] [KO:K03990]
E D11613 Pegcetacoplan (JAN/USAN/INN) <US>
D C5 [HSA:727] [KO:K03994]
E D03940 Eculizumab (USAN/INN) <JP/US>
E D11054 Ravulizumab (USAN) <JP/US>
E D10023 Pexelizumab (USAN/INN)
E D11473 Nomacopan (USAN)
E D11477 Pozelimab (USAN)
E D11696 Crovalimab (USAN/INN)
E D11748 Avacincaptad pegol sodium (USAN)
E D12208 Gefurulimab (USAN)
E D12356 Zilucoplan sodium (JAN)
E D12357 Zilucoplan (USAN/INN)
D C5 (C5a) [HSA:727] [KO:K03994]
E D11331 Olendalizumab (USAN)
E D11838 Vilobelimab (USAN)
D SERPINA1 [HSA:5265] [KO:K03984]
E D11965 alpha 1-Antitrypsin <JP>
D SERPINC1 (AT3) [HSA:462] [KO:K03911]
E D07510 Adomiparin (USAN)
E D02112 Heparin sodium (JP18/USP/INN) <JP/US>
E D04427 Heparin calcium (JP18) <JP>
E D03353 Dalteparin sodium (JAN/USP/INN) <JP/US>
E D03674 Enoxaparin sodium (JAN/USP/INN) <JP/US>
E D04977 Parnaparin sodium (JP18) <JP>
E D03337 Reviparin sodium (JAN)
E D03644 Danaparoid sodium (JAN/USAN) <JP>
E D06398 Tinzaparin sodium (USAN)
E D08547 Sulodexide (INN)
E D01844 Fondaparinux sodium (JAN/USP/INN) <JP/US>
E D02956 Anticoagulant heparin (USP)
E D02980 Adomiparin sodium (USAN)
E D03673 Deligoparin sodium (USAN/INN)
E D10418 Delparantag pentahydrochloride (USAN)
E D11810 Fitusiran sodium (JAN)
D SERPIND1 [HSA:3053] [KO:K03912]
E D08547 Sulodexide (INN)
E D02980 Adomiparin sodium (USAN)
D SERPINE1 (PAI1) [HSA:5054] [KO:K03982]
E D03766 Diaplasinin (USAN)
E D06160 Tiplasinin (USAN)
E D08656 Aleplasinin (USAN/INN)
D TFPI [HSA:7035] [KO:K03909]
E D11261 Marstacimab (USAN)
E D11847 Concizumab (USAN)
D GP6 [HSA:51206] [KO:K06264]
E D12413 Glenzocimab (USAN/INN)
C Acute phase protein
D SAA [HSA:6288 6289] [KO:K17310]
E D12482 Anselamimab (INN)
C Immune system
D FCGRT [HSA:2217] [KO:K24019]
E D11876 Efgartigimod alfa (USAN/INN) <JP/US>
E D11666 Nipocalimab (USAN)
E D11983 Batoclimab (USAN/INN)
E D12144 Orilanolimab (USAN/INN)
E D12182 Rozanolixizumab (INN)
D FCGR2B (CD32) [HSA:2213] [KO:K12560]
E D11339 Valziflocept (USAN)
D FCER1A [HSA:2205] [KO:K08089]
E D05251 Omalizumab (USAN/INN) <JP/US>
E D03095 Benzylpenicilloyl polylysine (USP) <US>
D FCER1G [HSA:2207] [KO:K07983]
E D03095 Benzylpenicilloyl polylysine (USP) <US>
D FCRL5 [HSA:83416] [KO:K06727]
E D11984 Cevostamab (USAN/INN)
D ALOX5AP [HSA:241] [KO:K20735]
E D05671 Quiflapon sodium (USAN)
E D06664 Veliflapon (USAN/INN)
E D10069 Fiboflapon (USAN)
E D10122 Fiboflapon sodium (USAN)
D LGALS3 [HSA:3958] [KO:K06831]
E D11495 Belapectin (USAN)
E D12221 Olitigaltin (USAN)
C Endocrine system
D GNRH1 (LHRH) [HSA:2796] [KO:K05252]
E D03701 Detirelix acetate (USAN)
C Circulatory system
D CALCA (CGRP) [HSA:796] [KO:K12332]
E D10936 Galcanezumab (USAN/INN) <JP/US>
E D11055 Fremanezumab (USAN/INN) <JP/US>
E D11303 Eptinezumab (USAN) <US>
D HBA [HSA:3039 3040] [KO:K13822]
E D03436 Cellulose, oxidized (JAN/USP) <JP>
E D06456 Cellulose, oxidized regenerated (USP)
D HBB [HSA:3043] [KO:K13823]
E D03436 Cellulose, oxidized (JAN/USP) <JP>
E D06456 Cellulose, oxidized regenerated (USP)
C Digestive system
D MTTP [HSA:4547] [KO:K14463]
E D09637 Lomitapide (USAN/INN)
E D09638 Lomitapide mesylate (USAN) <JP/US>
E D05060 Mitratapide (USAN/INN)
D APOB [HSA:338] [KO:K14462]
E D08946 Mipomersen sodium (USAN)
D APOC3 [HSA:345] [KO:K08759]
E D11648 Volanesorsen (USAN/INN)
E D11650 Volanesorsen sodium (USAN)
C Nervous system
D SNAP25 [HSA:6616] [KO:K18211]
E D00783 Botulinum toxin type A (JAN) <JP/US>
E D02735 Rimabotulinumtoxin B (USAN) <JP/US>
E D11405 Prabotulinumtoxin A (USAN) <US>
E D10012 Incobotulinumtoxin A (JAN/USAN) <JP/US>
E D10921 Daxibotulinumtoxin A (USAN)
D RGMA [HSA:56963] [KO:K23096]
E D11355 Elezanumab (USAN/INN)
D HTT* [HSA_VAR:3064v1] [HSA:3064] [KO:K04533]
E D12012 Tominersen sodium (JAN)
E D12013 Tominersen (USAN/INN)
C Sensory system
D RBP4 [HSA:5950] [KO:K18271]
E D12351 Tinlarebant (USAN)
!
#
#[ DRUG | BRITE | KEGG2 | KEGG ]
#Last updated: March 25, 2023
#
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