Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
   Transferases (EC2)
   Hydrolases (EC3)
     Carboxylic-ester hydrolases [EC:3.1.1.-]
     Phosphatases [EC:3.1.3.-]
     Phosphodiesterases [EC:3.1.4.-]
     Sulfatases [EC:3.1.6.-]
     Glycosidases [EC:3.2.1.-]
       AMY [HSA:279 280] [KO:K01176]
       GAA [HSA:2548] [KO:K12316]
       GAA* [HSA_VAR:2548v1] [HSA:2548] [KO:K12316]
       GANC [HSA:2595] [KO:K12317]
       MGAM [HSA:8972] [KO:K12047]
       MAN2B1* [HSA_VAR:4125v1] [HSA:4125] [KO:K12311]
       GUSB [HSA:2990] [KO:K01195]
       GUSB* [HSA_VAR:2990v1] [HSA:2990] [KO:K01195]
       GLA* [HSA_VAR:2717v1] [HSA:2717] [KO:K01189]
       GLA* [HSA_VAR:2717v2] [HSA:2717] [KO:K01189]
       GBA* [HSA_VAR:2629v1] [HSA:2629] [KO:K01201]
       SI [HSA:6476] [KO:K01203]
         D03342  Camiglibose (USAN)
       SI* [HSA_VAR:6476v1] [HSA:6476] [KO:K01203]
       NAGLU* [HSA_VAR:4669v1] [HSA:4669] [KO:K01205]
         D11199  Lesinidase alfa (USAN/INN)
       IDUA* [HSA_VAR:3425v1] [HSA:3425] [KO:K01217]
       HPSE [HSA:10855] [KO:K07964]
     ADP-ribosyl cyclase [EC:3.2.2.6]
     Aminopeptidases [EC:3.4.11.-]
     Dipeptidases [EC:3.4.13.-]
     Peptidyl-peptidases [EC:3.4.14.-]
     Peptidyl-dipeptidases [EC:3.4.15.-]
     Metallocarboxypeptidases [EC:3.4.17.-]
     Serine peptidases [EC:3.4.21.-]
     Cysteine peptidases [EC:3.4.22.-]
     Aspartic peptidases [EC:3.4.23.-]
     Metallo peptidases [EC:3.4.24.- 3.4.17.-]
     Threonine peptidases [EC:3.4.25.-]
     Glutaminase [EC:3.5.1.2]
     Histone deacetylase [EC:3.5.1.98]
     Arginase [EC:3.5.3.1]
     Adenosine deaminase [EC:3.5.4.4]
     Cytidine deaminase [EC:3.5.4.5]
     ATPase [EC:3.6.3.-]
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 19, 2024

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