G Protein-coupled receptors
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Rhodopsin family
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Acetylcholine (muscarinic)
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Adrenaline
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Dopamine
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Histamine
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Serotonin
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Trace amine
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Angiotensin
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Bradykinin
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Cholecystokinin
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Endothelin
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Follicle stimulating hormone
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Ghrelin
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Gonadotropin-releasing hormone
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Lutropin-choriogonadotropic hormone
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Melanocortin
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Motilin
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Neuropeptide Y
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Opioid
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OPRM1 [HSA:4988] [KO:K04215]
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D08639 Trimebutine (INN)
D01500 Trimebutine maleate (JP18) <JP>
D06618 Methylnaltrexone bromide (JAN/USAN) <US>
D02878 Alvimopan (USAN) <US>
D10479 Naloxegol (USAN/INN)
D10375 Naloxegol oxalate (USAN) <US>
D08249 Naloxone (INN)
D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
D11620 Naloxone hydrochloride dihydrate <US>
D10188 Naldemedine (USAN/INN)
D10478 Naldemedine tosylate (JAN/USAN) <JP/US>
D07861 Diphenoxylate (INN)
D03860 Diphenoxylate hydrochloride (USP)
D08144 Loperamide (INN)
D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
D03809 Difenoxin (USAN/INN)
D11583 Difenoxin hydrochloride
D07113 Loperamide oxide (INN)
D10403 Eluxadoline (USAN/INN) <US>
D00320 Fentanyl (JAN/USP/INN) <JP/US>
D01399 Fentanyl citrate (JP18/USP) <JP/US>
D10811 Fentanyl hydrochloride (JAN)
D07122 Alfentanil (INN)
D00835 Alfentanil hydrochloride (USP) <US>
D05938 Sufentanil (USAN/INN)
D00845 Sufentanil citrate (USP) <US>
D02941 Anileridine (USP/INN)
D02942 Anileridine hydrochloride (USP)
D08473 Remifentanil (INN)
D01177 Remifentanil hydrochloride (JAN/USAN) <JP/US>
D08233 Morphine (BAN)
D00842 Morphine sulfate (USP) <JP/US>
D02271 Morphine hydrochloride hydrate (JP18) <JP>
D08234 Morphine tartrate
D08047 Hydromorphone (INN)
D00839 Hydromorphone hydrochloride (JAN/USP) <JP/US>
D07285 Nicomorphine (INN)
D08273 Nicomorphine hydrochloride
D05312 Oxycodone (USAN/INN) <US>
D00847 Oxycodone hydrochloride (USP) <US>
D03783 Oxycodone terephthalate (USP)
D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
D07831 Dihydrocodeine (INN)
D01481 Dihydrocodeine phosphate (JP18) <JP>
D03825 Dihydrocodeine bitartrate (USP)
D07832 Dihydrocodeine thiocyanate
D08323 Oxymorphone (INN)
D00844 Oxymorphone hydrochloride (USP) <US>
D08100 Ketobemidone (INN)
D08101 Ketobemidone hydrochloride
D08343 Pethidine (INN)
D01383 Meperidine hydrochloride (USP) <JP/US>
D07809 Dextropropoxyphene (INN)
D00482 Propoxyphene hydrochloride (USAN) <US>
D05632 Propoxyphene napsylate (USAN)
D00498 Pentazocine (JP18/USP/INN) <JP>
D02111 Pentazocine lactate (USP)
D02227 Pentazocine hydrochloride (JAN/USP) <JP>
D07132 Buprenorphine (JAN/INN) <JP/US>
D00836 Buprenorphine hydrochloride (JP18/USP) <JP/US>
D03197 Butorphanol (USAN/INN)
D00837 Butorphanol tartrate (JAN/USP) <US>
D08246 Nalbuphine (INN)
D00843 Nalbuphine hydrochloride (USAN) <US>
D08597 Tilidine (INN)
D06147 Tilidine hydrochloride (USAN)
D08623 Tramadol (INN)
D01355 Tramadol hydrochloride (JP18/USP) <JP/US>
D00838 Dezocine (USAN)
D08182 Meptazinol (INN)
D04924 Meptazinol hydrochloride (USAN)
D06007 Tapentadol (USAN/INN)
D10199 Tapentadol hydrochloride (JAN) <JP/US>
D11214 Oliceridine (USAN/INN) <US>
D05113 Naltrexone (USAN/INN) <US>
D02095 Naltrexone hydrochloride (USP) <US>
D05111 Nalmefene (USAN/INN)
D02104 Nalmefene hydrochloride <US>
D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
D08195 Methadone (BAN)
D02102 Methadone hydrochloride (JAN/USP) <JP/US>
D04716 Levomethadyl acetate (USAN)
D00840 Levomethadyl acetate hydrochloride (USAN)
D08121 Levomethadone (INN)
D08122 Levomethadone hydrochloride
D07286 Diamorphine (BAN)
D07810 Diacetylmorphine hydrochloride
D07929 Ethylmorphine (BAN)
D02205 Ethylmorphine hydrochloride hydrate (JP18)
D08045 Hydrocodone (INN)
D03725 Hydrocodone bitartrate (USP) <US>
D04461 Hydrocodone polistirex (USAN)
D08046 Hydrocodone hydrochloride
D00195 Codeine (USP)
D02101 Codeine phosphate (USP) <JP>
D03579 Codeine polistirex (USAN)
D03580 Codeine sulfate (USP) <US>
D07740 Codeine hydrochloride
D07385 Pholcodine (INN)
D07557 O-Acetyldihydrocodeine hydrochloride
D08247 Nalorphine (INN)
D08248 Nalorphine hydrochloride (USP)
D00841 Levorphanol tartrate (USP) <US>
D01435 Ethoheptazine citrate (JAN)
D02238 Levallorphan tartrate (JP18) <JP>
D03156 Brifentanil hydrochloride (USAN)
D03405 Carfentanil citrate (USAN)
D03618 Cyclazocine (USAN/INN)
D04764 Lofentanil oxalate (USAN)
D04973 Methadyl acetate (USAN)
D05048 Mirfentanil hydrochloride (USAN)
D05217 Ocfentanil hydrochloride (USAN)
D05631 Propiram fumarate (USAN)
D05667 Quadazocine mesylate (USAN)
D06189 Tonazocine mesylate (USAN)
D06208 Trefentanil hydrochloride (USAN)
D06268 Trimeperidine (INN)
D06342 Xorphanol mesylate (USAN)
D07620 Carfentanil (INN)
D07863 Diprenorphine (INN)
D07864 Diprenorphine hydrochloride
D07937 Etorphine (INN)
D08123 Levorphanol (INN)
D10162 Samidorphan (USAN)
D10163 Samidorphan l-malate (USAN)
D10349 Bevenopran (USAN/INN)
D10371 Methylsamidorphan (USAN)
D10436 Cebranopadol (USAN/INN)
D10612 Benzhydrocodone (USAN/INN)
D10648 Methylsamidorphan chloride (USAN/INN)
D10690 Axelopran sulfate (USAN)
D10692 Benzhydrocodone hydrochloride (USAN)
D10740 Axelopran (USAN/INN)
D11291 Asalhydromorphone (USAN)
D11292 Asalhydromorphone hydrochloride (USAN)
D11424 Oxycodegol (USAN/INN)
D11425 Oxycodegol phosphate (USAN)
D12660 Alphacetylmethadol (INN)
D12661 Betacetylmethadol (INN)
D12662 Allylprodine (INN)
D12666 Alphameprodine (INN)
D12667 Betameprodine (INN)
D12668 Clonitazene (INN)
D12669 Etonitazene (INN)
D12674 Alphamethadol (INN)
D12675 Betamethadol (INN)
D12676 Isomethadone (INN)
D12678 Alphaprodine (INN)
D12679 Betaprodine (INN)
D12680 Etoxeridine (INN)
D12681 Hydroxypethidine (INN)
D12682 Furethidine (INN)
D12683 Piminodine (INN)
D12685 Benzethidine (INN)
D12686 Hydromorphinol (INN)
D12687 Levophenacylmorphan (INN)
D12688 Phenomorphan (INN)
D12689 Methyldihydromorphine (INN)
D12690 Metopon (BAN)
D12691 Methyldesorphine (INN)
D12692 Norlevorphanol (INN)
D12693 Phenampromide (INN)
D12694 Diampromide (INN)
D12696 Levomethorphan (INN)
D12697 Morpheridin (INN)
D12700 Acetorphine (INN)
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OPRK1 [HSA:4986] [KO:K04214]
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D08639 Trimebutine (INN)
D01500 Trimebutine maleate (JP18) <JP>
D08249 Naloxone (INN)
D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
D11620 Naloxone hydrochloride dihydrate <US>
D08144 Loperamide (INN)
D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
D07113 Loperamide oxide (INN)
D10403 Eluxadoline (USAN/INN) <US>
D05312 Oxycodone (USAN/INN) <US>
D00847 Oxycodone hydrochloride (USP) <US>
D03783 Oxycodone terephthalate (USP)
D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
D08100 Ketobemidone (INN)
D08101 Ketobemidone hydrochloride
D00498 Pentazocine (JP18/USP/INN) <JP>
D02111 Pentazocine lactate (USP)
D02227 Pentazocine hydrochloride (JAN/USP) <JP>
D07132 Buprenorphine (JAN/INN) <JP/US>
D00836 Buprenorphine hydrochloride (JP18/USP) <JP/US>
D03197 Butorphanol (USAN/INN)
D00837 Butorphanol tartrate (JAN/USP) <US>
D08246 Nalbuphine (INN)
D00843 Nalbuphine hydrochloride (USAN) <US>
D00838 Dezocine (USAN)
D05113 Naltrexone (USAN/INN) <US>
D02095 Naltrexone hydrochloride (USP) <US>
D05111 Nalmefene (USAN/INN)
D02104 Nalmefene hydrochloride <US>
D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
D08247 Nalorphine (INN)
D08248 Nalorphine hydrochloride (USP)
D06405 Nalfurafine hydrochloride (JAN/USAN) <JP>
D11111 Difelikefalin (USAN/INN)
D10890 Difelikefalin acetate (JAN) <JP/US>
D01879 Eptazocine hydrobromide (JAN)
D02238 Levallorphan tartrate (JP18) <JP>
D03618 Cyclazocine (USAN/INN)
D04649 Ketazocine (USAN/INN)
D05299 Oxilorphan (USAN/INN)
D05646 Proxorphan tartrate (USAN)
D05667 Quadazocine mesylate (USAN)
D05907 Spiradoline mesylate (USAN)
D06189 Tonazocine mesylate (USAN)
D06342 Xorphanol mesylate (USAN)
D06395 Enadoline hydrochloride (USAN)
D07863 Diprenorphine (INN)
D07864 Diprenorphine hydrochloride
D07904 Eptazocine (INN)
D07937 Etorphine (INN)
D11831 Aticaprant (USAN/INN)
D12700 Acetorphine (INN)
D12869 Navacaprant (USAN/INN)
D12870 Navacaprant hydrochloride (USAN)
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OPRD1 [HSA:4985] [KO:K04213]
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OPRL1 [HSA:4987] [KO:K04216]
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Orexin
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Oxytocin
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Relaxin
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Somatostatin
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Tachykinin
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Thrombin
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Thyrotropin-releasing hormone
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Vasopressin
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Purine / pyrimidine
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Adenosine
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Cysteinyl leukotriene
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Free fatty acid
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Leukotriene
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Lysophosphatidic acid
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Prostaglandin
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Prostacyclin
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Sphingolipid
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Thromboxane
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Cannabinoid
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Melatonin
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Platelet activating factor
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R-spondin
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Secretin receptor family
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Metabotropic glutamate receptor family
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Frizzled / Smoothened family
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Others
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Ion channels
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Nuclear receptors
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Protein kinases
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Cytokines and receptors
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Cell surface molecules and ligands
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Transporters
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Enzymes
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Nucleic acids
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Not elsewhere classified
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