Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
   Thyroid hormone like receptors
   Hepatocyte nuclear factor 4 like receptors
   Estrogen like receptors
     Estrogen receptor
     3-Ketosteroid receptor
       NR3C1 (GR) [HSA:2908] [KO:K05771]
       NR3C2 (MR) [HSA:4306] [KO:K08555]
       NR3C3 (PGR) [HSA:5241] [KO:K08556]
       NR3C4 (AR) [HSA:367] [KO:K08557]
         D07456  Androstanolone (INN)
         D00444  Stanozolol (JAN/USP/INN)
         D00389  Metandienone (INN)
         D08193  Metenolone (INN)
         D01301  Methenolone enanthate (USAN)
         D01375  Methenolone acetate (USAN) <JP>
         D00490  Oxymetholone (JP18/USP/INN)
         D05674  Quinbolone (USAN/INN)
         D08409  Prasterone (USAN/INN) <US>
         D01616  Sodium prasterone sulfate hydrate (JP18)
         D00462  Oxandrolone (JAN/USP/INN) <US>
         D07127  Norethandrolone (INN)
         D08250  Nandrolone (INN)
         D00955  Nandrolone decanoate (JAN/USP)
         D00956  Nandrolone phenpropionate (USP)
         D01476  Nandrolone cyclohexylpropionate (JAN)
         D01737  Nandrolone furylpropionate (JAN)
         D05116  Nandrolone cyclotate (USAN)
         D08251  Nandrolone laurate
         D01149  Oxabolone cipionate (JAN/INN)
         D11451  Clascoterone (USAN) <US>
         D00327  Fluoxymesterone (JAN/USP/INN)
         D00408  Methyltestosterone (JP18/USP/INN) <US>
         D00075  Testosterone (JAN/USP) <US>
         D00957  Testosterone cypionate (USP) <US>
         D00958  Testosterone enanthate (JP18/USP) <JP/US>
         D00959  Testosterone propionate (JP18/USP)
         D06085  Testosterone ketolaurate (USAN/INN)
         D06086  Testosterone phenylacetate (USAN)
         D06087  Testosterone undecanoate (USAN) <US>
         D08573  Testosterone decanoate
         D08574  Testosterone phenylpropionate
         D04947  Mesterolone (USAN/INN)
         D07670  Chlormadinone (INN)
         D01299  Chlormadinone acetate (JP18/USAN) <JP>
         D07766  Cyproterone (INN)
         D01368  Cyproterone acetate (JAN/USAN)
         D00289  Danazol (JP18/USP/INN) <JP/US>
         D00586  Flutamide (JP18/USP/INN) <JP/US>
         D00965  Nilutamide (USAN/INN) <US>
         D00961  Bicalutamide (JP18/USP/INN) <JP/US>
         D10218  Enzalutamide (JAN/USAN) <JP/US>
         D11040  Apalutamide (JAN/INN) <JP/US>
         D11045  Darolutamide (JAN/USAN/INN) <JP/US>
         D01329  Oxendolone (JAN/USAN/INN)
         D01533  Mestanolone (JAN/INN)
         D01534  Dromostanolone propionate (USAN)
         D03079  Benorterone (USAN/INN)
         D03144  Bolasterone (USAN/INN)
         D03145  Boldenone undecylenate (USAN)
         D03338  Calusterone (USAN/INN)
         D03515  Cioteronel (USAN/INN)
         D03551  Clometherone (USAN/INN)
         D03675  Delmadinone acetate (USAN)
         D05025  Mibolerone (USP/INN)
         D05174  Nisterime acetate (USAN)
         D05837  Silandrone (USAN/INN)
         D06191  Topterone (USAN/INN)
         D06211  Trenbolone acetate (USP)
         D06357  Zanoterone (USAN/INN)
         D07536  Boldenone (INN)
         D07783  Delmadinone (INN)
         D08196  Methandriol (INN)
         D08197  Methandriol dipropionate
         D08627  Trenbolone (INN)
         D10221  Enobosarm (USAN)
         D11105  Osaterone acetate (JAN)
         D11184  Ralaniten (USAN/INN)
         D11185  Ralaniten acetate (USAN)
         D12303  Deutenzalutamide (USAN)
         D12316  Bavdegalutamide (USAN)
         D12643  Masofaniten (USAN/INN)
         D12866  Gridegalutamide (USAN)
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 19, 2024

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