Target-based Classification of Drugs

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 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
     Adrenaline
       ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
       ADRA1A [HSA:148] [KO:K04135]
       ADRA1D [HSA:146] [KO:K04137]
       ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
       ADRA2A [HSA:150] [KO:K04138]
       ADRA2B [HSA:151] [KO:K04139]
       ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
         D00095  Epinephrine (USP/INN) <JP/US>
         D00996  Epinephrine hydrochloride (JAN)
         D02149  Epinephrine bitartrate (JAN/USP)
         D07931  Etilefrine (INN)
         D01573  Etilefrine hydrochloride (JP18) <JP>
         D08090  Isoprenaline (INN)
         D01390  Isoproterenol hydrochloride (USP) <JP/US>
         D02066  Isoproterenol sulfate (USP)
         D02150  l-Isoprenaline hydrochloride (JP18) <JP>
         D00076  Noradrenaline (JP18) <JP>
         D05206  Norepinephrine bitartrate (USP) <US>
         D08284  Norepinephrine hydrochoride
         D09794  Norepinephrine hydrochloride (JAN)
         D02976  Arbutamine hydrochloride (USAN)
         D00124  Ephedrine (USP)
         D01386  Ephedrine hydrochloride (JP18/USP) <JP/US>
         D04018  Ephedrine sulfate (USP) <US>
         D01277  Droxidopa (JP18/USAN/INN) <JP/US>
         D07156  Alprenolol (INN)
         D01182  Alprenolol hydrochloride (JP18/USAN)
         D08318  Oxprenolol (INN)
         D01806  Oxprenolol hydrochloride (JP18/USP)
         D00513  Pindolol (JP18/USP/INN) <JP/US>
         D08443  Propranolol (INN)
         D00483  Propranolol hydrochloride (JP18/USP) <JP/US>
         D07181  Mepindolol (INN)
         D07624  Carteolol (INN)
         D00599  Carteolol hydrochloride (JP18/USP) <JP/US>
         D07182  Tertatolol (INN)
         D08572  Tertatolol hydrochloride
         D07537  Bopindolol (INN)
         D01794  Bopindolol malonate (JAN)
         D07590  Bupranolol (INN)
         D01454  Bupranolol hydrochloride (JP18)
         D08074  Penbutolol (INN)
         D00602  Penbutolol sulfate (JP18/USP)
         D07183  Cloranolol (INN)
         D07184  Talinolol (INN)
         D08368  Phenylpropanolamine (INN)
         D01224  Phenylpropanolamine hydrochloride (JAN/USP)
         D05466  Phenylpropanolamine polistirex (USAN)
         D08449  Pseudoephedrine (INN)
         D00485  Pseudoephedrine hydrochloride (USP)
         D05648  Pseudoephedrine polistirex (USAN)
         D05649  Pseudoephedrine sulfate (USP)
         D02349  Dipivefrin (USAN)
         D01017  Dipivefrin hydrochloride (USP)
         D08115  Levobunolol (INN)
         D01025  Levobunolol hydrochloride (JAN/USP) <JP/US>
         D02374  Metipranolol (USAN/INN)
         D02081  Metipranolol hydrochloride
         D07496  Befunolol (INN)
         D01512  Befunolol hydrochloride (JAN)
         D01444  Bunitrolol hydrochloride (JAN)
         D01504  Bufetolol hydrochloride (JP18) <JP>
         D01691  Nipradilol (JAN/INN) <JP>
         D01795  Tilisolol hydrochloride (JAN)
         D01906  Dilevalol hydrochloride (JAN/USAN)
         D01952  L-Methylephedrine hydrochloride (JAN)
         D02109  dl-Methylephedrine hydrochloride (JP18) <JP>
         D02765  Adaprolol maleate (USAN)
         D02834  Alprenoxime hydrochloride (USAN)
         D03502  Cimaterol (USAN/INN)
         D03729  Dexpropranolol hydrochloride (USAN)
         D03759  Diacetolol hydrochloride (USAN)
         D04026  Epinephryl borate (USP)
         D04120  Exaprolol hydrochloride (USAN)
         D04190  Flestolol sulfate (USAN)
         D04888  Medroxalol (USAN/INN)
         D04889  Medroxalol hydrochloride (USAN)
         D05228  Octodrine (USAN/INN)
         D05345  Pamatolol sulfate (USAN)
         D05688  Racepinephrine (USP/INN)
         D05689  Racepinephrine hydrochloride (USP)
         D06014  Tazolol hydrochloride (USAN)
         D06162  Tiprenolol hydrochloride (USAN)
         D06176  Tolamolol (USAN/INN)
         D08206  Methylephedrine (BAN)
         D08598  Tilisolol (INN)
         D08982  Racephedrine hydrochloride (USAN)
         D09842  dl-Methylephedrine saccharinate (JAN)
         D09843  Beradilol monoethyl maleate (JAN)
       ADRB1 [HSA:153] [KO:K04141]
       ADRB2 [HSA:154] [KO:K04142]
       ADRB3 [HSA:155] [KO:K04143]
     Dopamine
     Histamine
     Serotonin
     Trace amine
     Angiotensin
     Bradykinin
     Cholecystokinin
     Endothelin
     Follicle stimulating hormone
     Ghrelin
     Gonadotropin-releasing hormone
     Lutropin-choriogonadotropic hormone
     Melanocortin
     Motilin
     Neuropeptide Y
     Opioid
     Orexin
     Oxytocin
     Relaxin
     Somatostatin
     Tachykinin
     Thrombin
     Thyrotropin-releasing hormone
     Vasopressin
     Purine / pyrimidine
     Adenosine
     Cysteinyl leukotriene
     Free fatty acid
     Leukotriene
     Lysophosphatidic acid
     Prostaglandin
     Prostacyclin
     Sphingolipid
     Thromboxane
     Cannabinoid
     Melatonin
     Platelet activating factor
     R-spondin
   Secretin receptor family
   Metabotropic glutamate receptor family
   Frizzled / Smoothened family
   Others
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 18, 2024

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