Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
   Transferases (EC2)
     Methyltransferases [EC:2.1.1.-]
     Acyltransferases [EC:2.3.1.-]
     gamma-Glutamyltransferase [EC:2.3.2.2]
     E3 ubiquitin-protein ligase [EC:2.3.2.27]
     ATP citrate synthase [EC:2.3.3.8]
     Hexosyltransferases [EC:2.4.1.-]
     Pentosyltransferases [EC:2.4.2.-]
       PNP [HSA:4860] [KO:K03783]
       HPRT1 [HSA:3251] [KO:K00760]
         D04931  Mercaptopurine (INN)
         D00161  Mercaptopurine (USP) <JP/US>
         D08603  Tioguanine (INN)
         D06109  Thioguanine (USP) <US>
       NAMPT [HSA:10135] [KO:K03462]
       PARP [HSA:142 10038 10039 143] [KO:K24070 K10798]
       PARP1 [HSA:142] [KO:K24070]
       PARP2 [HSA:10038] [KO:K10798]
       PARP3 [HSA:10039] [KO:K10798]
       TIPARP (PARP7) [HSA:25976] [KO:K15259]
     Alkyl/Aryl transferases [EC:2.5.1.-]
     Aminotransferase [EC:2.6.1.-]
     Phosphotransferase [EC:2.7.1.-]
     DNA polymerase [EC:2.7.7.7]
     Reverse transcriptase [EC:2.7.7.49]
   Hydrolases (EC3)
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 24, 2024

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