Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
     Dehydrogenases [EC:1.1.1.-]
     Oxidases [EC:1.1.3.-]
     Dehydrogenases [EC:1.2.1.-]
     Dehydrogenases [EC:1.3.-.-]
     Amine oxidases [EC:1.4.3.-]
     Dihydrofolate reductase [EC:1.5.1.3]
     NAD(P)H dehydrogenase [EC:1.6.5.2]
       NQO1 [HSA:1728] [KO:K00355]
         D08682  Warfarin (INN)
         D00564  Warfarin sodium (USP) <US>
         D01280  Warfarin potassium (JP18) <JP>
         D07064  Acenocoumarol (INN)
     Peroxidase [EC:1.11.1.-]
     Peroxygenase [EC:1.11.2.-]
     Dioxygenases [EC:1.13.11.-]
     Prolyl 4-hydroxylase [EC:1.14.11.2]
     HIF hydroxylase [EC:1.14.11.29]
     Nitic oxide synthase [EC:1.14.13.39]
     Cytochrome P450 [EC:1.14.14.-]
     Other monooxygenases [EC:1.14.16.- 1.14.17.- 1.14.18.-]
     Prostaglandin synthase [EC:1.14.99.1]
     Histone demethylase [EC:1.14.99.66]
     Superoxide dismutase [EC:1.15.1.1]
     Xanthine dehydrogenase/oxidase [EC:1.17.1.4 1.17.3.2]
     Ribonucleoside-diphosphate reductase [EC:1.17.4.1]
     Vitamin-K-epoxide reductase [EC:1.17.4.4]
       VKORC1 [HSA:79001] [KO:K05357]
         D03798  Dicumarol (USAN)
         D08354  Phenindione (INN)
         D08682  Warfarin (INN)
         D00564  Warfarin sodium (USP) <US>
         D01280  Warfarin potassium (JP18) <JP>
         D05457  Phenprocoumon (USAN/INN)
         D07064  Acenocoumarol (INN)
         D07131  Ethyl biscoumacetate (INN)
         D07135  Clorindione (INN)
         D07136  Diphenadione (INN)
         D07137  Tioclomarol (INN)
         D07969  Fluindione (INN)
         D07134  Flocoumafen (JAN)
         D09676  Tecarfarin (USAN/INN)
         D09677  Tecarfarin sodium (USAN)
     Thyroxine 5'-deiodinase [EC:1.21.99.4]
   Transferases (EC2)
   Hydrolases (EC3)
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 20, 2024

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