Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
   Transferases (EC2)
   Hydrolases (EC3)
     Carboxylic-ester hydrolases [EC:3.1.1.-]
     Phosphatases [EC:3.1.3.-]
     Phosphodiesterases [EC:3.1.4.-]
     Sulfatases [EC:3.1.6.-]
     Glycosidases [EC:3.2.1.-]
     ADP-ribosyl cyclase [EC:3.2.2.6]
     Aminopeptidases [EC:3.4.11.-]
     Dipeptidases [EC:3.4.13.-]
     Peptidyl-peptidases [EC:3.4.14.-]
     Peptidyl-dipeptidases [EC:3.4.15.-]
     Metallocarboxypeptidases [EC:3.4.17.-]
     Serine peptidases [EC:3.4.21.-]
     Cysteine peptidases [EC:3.4.22.-]
     Aspartic peptidases [EC:3.4.23.-]
     Metallo peptidases [EC:3.4.24.- 3.4.17.-]
     Threonine peptidases [EC:3.4.25.-]
     Glutaminase [EC:3.5.1.2]
     Histone deacetylase [EC:3.5.1.98]
     Arginase [EC:3.5.3.1]
     Adenosine deaminase [EC:3.5.4.4]
     Cytidine deaminase [EC:3.5.4.5]
     ATPase [EC:3.6.3.-]
       ATP1A [HSA:476 477 478 480] [KO:K01539]
       ATP2A [HSA:487 488 489] [KO:K05853]
       ATP4 [HSA:495 496] [KO:K01542 K01543]
         D00455  Omeprazole (JP18/USP/INN) <JP/US>
         D01207  Omeprazole sodium (USAN)
         D05261  Omeprazole sodium injection (JAN) <JP>
         D05259  Omeprazole magnesium (USP) <US>
         D05353  Pantoprazole (USAN/INN)
         D02593  Pantoprazole sodium (USP) <US>
         D00355  Lansoprazole (JP18/USP/INN) <JP/US>
         D08463  Rabeprazole (INN)
         D00724  Rabeprazole sodium (JP18/USP) <JP/US>
         D07917  Esomeprazole (INN)
         D01984  Esomeprazole magnesium (USP) <JP/US>
         D04056  Esomeprazole sodium (USAN) <US>
         D09339  Esomeprazole potassium (USAN)
         D10120  Esomeprazole strontium (USAN) <US>
         D11114  Esomeprazole magnesium dihydrate <US>
         D08903  Dexlansoprazole (INN/USAN) <US>
         D12816  Dexlansoprazole sesquihydrate <US>
         D11784  Vonoprazan (USAN/INN)
         D10466  Vonoprazan fumarate (JAN/USAN) <JP/US>
         D12246  Tegoprazan (INN)
         D01920  Tenatoprazole (JAN/INN)
         D05722  Revaprazan hydrochloride (USAN)
         D05900  Timoprazole (INN)
         D05901  Picoprazole (INN)
         D05906  Leminoprazole (INN)
         D09837  Penaprazole sodium hydrate (JAN)
       ABCB1 (CD243) [HSA:5243] [KO:K05658]
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 20, 2024

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