Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
   Transferases (EC2)
   Hydrolases (EC3)
     Carboxylic-ester hydrolases [EC:3.1.1.-]
     Phosphatases [EC:3.1.3.-]
     Phosphodiesterases [EC:3.1.4.-]
     Sulfatases [EC:3.1.6.-]
     Glycosidases [EC:3.2.1.-]
     ADP-ribosyl cyclase [EC:3.2.2.6]
     Aminopeptidases [EC:3.4.11.-]
     Dipeptidases [EC:3.4.13.-]
     Peptidyl-peptidases [EC:3.4.14.-]
     Peptidyl-dipeptidases [EC:3.4.15.-]
     Metallocarboxypeptidases [EC:3.4.17.-]
     Serine peptidases [EC:3.4.21.-]
     Cysteine peptidases [EC:3.4.22.-]
     Aspartic peptidases [EC:3.4.23.-]
     Metallo peptidases [EC:3.4.24.- 3.4.17.-]
     Threonine peptidases [EC:3.4.25.-]
     Glutaminase [EC:3.5.1.2]
     Histone deacetylase [EC:3.5.1.98]
       HDAC [HSA:3065 3066 8841 9759 10014 10013 51564 55869 9734 83933 79885] [KO:K06067 K11404 K11406 K11407 K11408 K11405 K11409 K18671 K11418]
       HDAC1 [HSA:3065] [KO:K06067]
         D05988  Tacedinaline (USAN/INN)
         D09357  Mocetinostat dihydrobromide (USAN)
         D09641  Mocetinostat (USAN/INN)
         D10993  Tucidinostat (JAN/USAN/INN) <JP>
         D11182  Tinostamustine (USAN/INN)
         D11319  Fimepinostat (USAN/INN)
         D11442  Nanatinostat (USAN)
       HDAC2 [HSA:3066] [KO:K06067]
         D09357  Mocetinostat dihydrobromide (USAN)
         D09641  Mocetinostat (USAN/INN)
         D10993  Tucidinostat (JAN/USAN/INN) <JP>
         D11182  Tinostamustine (USAN/INN)
         D11319  Fimepinostat (USAN/INN)
         D11442  Nanatinostat (USAN)
       HDAC3 [HSA:8841] [KO:K11404]
         D09357  Mocetinostat dihydrobromide (USAN)
         D09641  Mocetinostat (USAN/INN)
         D10993  Tucidinostat (JAN/USAN/INN) <JP>
         D11182  Tinostamustine (USAN/INN)
         D11319  Fimepinostat (USAN/INN)
         D11442  Nanatinostat (USAN)
       HDAC4 [HSA:9759] [KO:K11406]
       HDAC5 [HSA:10014] [KO:K11406]
       HDAC6 [HSA:10013] [KO:K11407]
       HDAC7 [HSA:51564] [KO:K11408]
       HDAC8 [HSA:55869] [KO:K11405]
         D09357  Mocetinostat dihydrobromide (USAN)
         D09641  Mocetinostat (USAN/INN)
         D11319  Fimepinostat (USAN/INN)
         D11442  Nanatinostat (USAN)
       HDAC9 [HSA:9734] [KO:K11409]
       HDAC10 [HSA:83933] [KO:K18671]
       HDAC11 [HSA:79885] [KO:K11418]
         D09357  Mocetinostat dihydrobromide (USAN)
         D09641  Mocetinostat (USAN/INN)
     Arginase [EC:3.5.3.1]
     Adenosine deaminase [EC:3.5.4.4]
     Cytidine deaminase [EC:3.5.4.5]
     ATPase [EC:3.6.3.-]
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 17, 2024

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