Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
     Dehydrogenases [EC:1.1.1.-]
     Oxidases [EC:1.1.3.-]
     Dehydrogenases [EC:1.2.1.-]
     Dehydrogenases [EC:1.3.-.-]
     Amine oxidases [EC:1.4.3.-]
     Dihydrofolate reductase [EC:1.5.1.3]
     NAD(P)H dehydrogenase [EC:1.6.5.2]
     Peroxidase [EC:1.11.1.-]
     Peroxygenase [EC:1.11.2.-]
     Dioxygenases [EC:1.13.11.-]
     Prolyl 4-hydroxylase [EC:1.14.11.2]
     HIF hydroxylase [EC:1.14.11.29]
     Nitic oxide synthase [EC:1.14.13.39]
     Cytochrome P450 [EC:1.14.14.-]
       CYP3A [HSA:1551 1576 1577 64816] [KO:K17691 K17689 K17690 K17692]
       CYP19A1 (ARO) [HSA:1588] [KO:K07434]
       CYP17A1 [HSA:1586] [KO:K00512]
       CYP46A1 [HSA:10858] [KO:K07440]
       CYP51A1 [HSA:1595] [KO:K05917]
       CYP11B1 [HSA:1584] [KO:K00497]
       CYP11B2 [HSA:1585] [KO:K07433]
         D11061  Osilodrostat (USAN/INN)
         D11062  Osilodrostat phosphate (JAN/USAN) <JP/US>
         D12773  Lorundrostat (USAN/INN)
         D12774  Lorundrostat hydrobromide (USAN)
         D12789  Baxdrostat (USAN/INN)
       CYP11A1 [HSA:1583] [KO:K00498]
       CYP26 [HSA:1592 56603 340665] [KO:K07437 K12664 K12665]
     Other monooxygenases [EC:1.14.16.- 1.14.17.- 1.14.18.-]
     Prostaglandin synthase [EC:1.14.99.1]
     Histone demethylase [EC:1.14.99.66]
     Superoxide dismutase [EC:1.15.1.1]
     Xanthine dehydrogenase/oxidase [EC:1.17.1.4 1.17.3.2]
     Ribonucleoside-diphosphate reductase [EC:1.17.4.1]
     Vitamin-K-epoxide reductase [EC:1.17.4.4]
     Thyroxine 5'-deiodinase [EC:1.21.99.4]
   Transferases (EC2)
   Hydrolases (EC3)
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: March 29, 2024

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