Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
   Serine/threonine kinases
   Receptor serine/threonine kinases (RSTK)
   Receptor tyrosine kinases (RTK)
   Non-receptor tyrosine kinases
     SRC family
     ABL family
     SYK family
     JAK family
       JAK [HSA:3716 3717 3718] [KO:K11217 K04447 K11218]
       JAK1 [HSA:3716] [KO:K11217]
       JAK2 [HSA:3717] [KO:K04447]
         D09959  Ruxolitinib (USAN/INN)
         D09960  Ruxolitinib phosphate (JAN/USAN) <JP/US>
         D11046  Delgocitinib (JAN/USAN/INN) <JP>
         D10630  Fedratinib (USAN/INN)
         D11296  Fedratinib hydrochloride (USAN) <US>
         D11768  Pacritinib (USAN/INN) <US>
         D10315  Momelotinib (USAN/INN)
         D10358  Momelotinib dihydrochloride (USAN)
         D10889  Momelotinib hydrochloride hydrate (JAN) <US>
         D09970  Tofacitinib (USAN)
         D09783  Tofacitinib citrate (JAN/USAN) <JP/US>
         D10308  Baricitinib (JAN/USAN/INN) <JP/US>
         D11106  Filgotinib maleate (JAN/USAN) <JP>
         D10653  Peficitinib (USAN/INN)
         D10721  Peficitinib hydrobromide (JAN/USAN) <JP>
         D10365  Gandotinib (USAN/INN)
         D11599  Zotiraciclib (USAN)
         D11600  Zotiraciclib citrate (USAN)
         D11676  Gusacitinib (USAN/INN)
         D11677  Gusacitinib hydrochloride (USAN)
         D11866  Deuruxolitinib (USAN)
         D11867  Deuruxolitinib phosphate (USAN)
         D12118  Nezulcitinib (USAN)
         D12545  Tinengotinib (USAN/INN)
       JAK2* [HSA_VAR:3717v1] [HSA:3717] [KO:K04447]
       JAK3 [HSA:3718] [KO:K11218]
       TYK2 [HSA:7297] [KO:K11219]
     FAK family
     TEC family
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: March 29, 2024

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