KEGG   DRUG: Flotetuzumab
Entry
D11306                      Drug                                   
Name
Flotetuzumab (USAN/INN)
Formula
C2618H4040N704O813S16
Exact mass
58861.1959
Mol weight
58897.3592
Sequence
(A chain)
DFVMTQSPDS LAVSLGERVT MSCKSSQSLL NSGNQKNYLT WYQQKPGQPP KLLIYWASTR
ESGVPDRFSG SGSGTDFTLT ISSLQAEDVA VYYCQNDYSY PYTFGQGTKL EIKGGGSGGG
GEVQLVESGG GLVQPGGSLR LSCAASGFTF STYAMNWVRQ APGKGLEWVG RIRSKYNNYA
TYYADSVKDR FTISRDDSKN SLYLQMNSLK TEDTAVYYCV RHGNFGNSYV SWFAYWGQGT
LVTVSSGGCG GGKVAALKEK VAALKEKVAA LKEKVAALKE
(B chain)
XAVVTQEPSL TVSPGGTVTL TCRSSTGAVT TSNYANWVQQ KPGQAPRGLI GGTNKRAPWT
PARFSGSLLG GKAALTITGA QAEDEADYYC ALWYSNLWVF GGGTKLTVLG GGGSGGGGEV
QLVQSGAELK KPGASVKVSC KASGYTFTDY YMKWVRQAPG QGLEWIGDII PSNGATFYNQ
KFKGRVTITV DKSTSTAYME LSSLRSEDTA VYYCARSHLL RASWFAYWGQ GTLVTVSSGG
CGGGEVAALE KEVAALEKEV AALEKEVAAL EK
(Disulfide bridge: A23-A94, A143-A219, A249-B241, B22-B90, B140-B214)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody, bispecific antibody
Comment
Treatment of hematologic malignancies
Target
IL3RA (CD123) [HSA:3563] [KO:K04737]
CD3 [HSA:915 916 917] [KO:K06450 K06451 K06452]
  Pathway
hsa04640  Hematopoietic cell lineage
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    IL3RA (CD123)
     D11306  Flotetuzumab (USAN/INN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3
     D11306  Flotetuzumab (USAN/INN)
Other DBs
CAS: 1664355-28-5
PubChem: 384585284
LinkDB

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