KEGG   DRUG: Emirodatamab
Entry
D12641                      Drug                                   
Name
Emirodatamab (USAN/INN)
Formula
C4684H7200N1270O1461S37
Exact mass
105799.7811
Mol weight
105865.3242
Sequence
QVTLKESGPT LVKPTETLTL TCTLSGFSLN NARMGVSWIR QPPGKCLEWL AHIFSNDEKS
YSTSLKNRLT ISKDSSKTQV VLTMTNVDPV DTATYYCARI VGYGSGWYGF FDYWGQGTLV
TVSSGGGGSG GGGSGGGGSD IQMTQSPSSL SASVGDRVTI TCRASQGIRN DLGWYQQKPG
KAPKRLIYAA STLQSGVPSR FSGSGSGTEF TLTISSLQPE DFATYYCLQH NSYPLTFGCG
TKVEIKSGGG GSEVQLVESG GGLVQPGGSL KLSCAASGFT FNKYAMNWVR QAPGKGLEWV
ARIRSKYNNY ATYYADSVKD RFTISRDDSK NTAYLQMNNL KTEDTAVYYC VRHGNFGNSY
ISYWAYWGQG TLVTVSSGGG GSGGGGSGGG GSQTVVTQEP SLTVSPGGTV TLTCGSSTGA
VTSGNYPNWV QQKPGQAPRG LIGGTKFLAP GTPARFSGSL LGGKAALTLS GVQPEDEAEY
YCVLWYSNRW VFGGGTKLTV LGGGGDKTHT CPPCPAPELL GGPSVFLFPP KPKDTLMISR
TPEVTCVVVD VSHEDPEVKF NWYVDGVEVH NAKTKPCEEQ YGSTYRCVSV LTVLHQDWLN
GKEYKCKVSN KALPAPIEKT ISKAKGQPRE PQVYTLPPSR EEMTKNQVSL TCLVKGFYPS
DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSKLTVDKS RWQQGNVFSC SVMHEALHNH
YTQKSLSLSP GKGGGGSGGG GSGGGGSGGG GSGGGGSGGG GSDKTHTCPP CPAPELLGGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPCEEQYGS
TYRCVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSREEM
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPGK
(Disulfide bridge: 22-97, 46-239, 162-227, 274-350, 414-482, 511-768, 514-771, 546-606, 577-587, 652-710, 803-863, 834-844, 909-967)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody, bispecific antibody
Comment
Treatment of acute myeloid leukemia
Target
FLT3 (CD135) [HSA:2322] [KO:K05092]
CD3E [HSA:916] [KO:K06451]
  Pathway
hsa04640  Hematopoietic cell lineage
hsa05200  Pathways in cancer
Brite
Target-based classification of drugs [BR:br08310]
 Protein kinases
  Receptor tyrosine kinases (RTK)
   PDGFR family
    FLT3 (CD135)
     D12641  Emirodatamab (USAN/INN)
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD3E
     D12641  Emirodatamab (USAN/INN)
Other DBs
CAS: 2449199-61-3
LinkDB

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