KEGG   DRUG: Baminercept
Entry
D08866                      Drug                                   
Name
Baminercept (USAN/INN);
Baminercept alfa (USAN)
Formula
C4074H6282N1134O1274S68
Exact mass
93650.2648
Mol weight
93710.88
Sequence
AVPPYASENQ TCRDQEKEYY EPQHRICCSR CPPGTYVSAK CSRIRDTVCA TCAENSYNEH
WNYLTICQLC RPCDPVMGLE EIAPCTSKRK TQCRCQPGMF CAAWALECTH CELLSDCPPG
TEAELKDEVG KGNNHCVPCK AGHFQNTSSP SARCQPHTRC ENQGLVEAAP GTAQSDTTCK
NPLEPLPPEM SGTMVDKTHT CPPCPAPELL GGPSVFLFPP KPKDTLMISR TPEVTCVVVD
VSHEDPEVKF NWYVDGVEVH NAKTKPREEQ YNSTYRVVSV LTVLHQDWLN GKEYKCKVSN
KALPAPIEKT ISKAKGQPRE PQVYTLPPSR DELTKNQVSL TCLVKGFYPS DIAVEWESNG
QPENNYKTTP PVLDSDGSFF LYSKLTVDKS RWQQGNVFSC SVMHEALHNH YTQKSLSLSP
G
(Disulfide bridge: 12-27, 28-41, 31-49, 52-67, 70-85, 73-93, 95-101, 108-117, 111-136, 139-154, 160-179, 236-296, 342-400, 201-201', 204-204')
  Type
Peptide
Efficacy
Anti-inflammatory, TNF inhibitor
Comment
Fusion protein
Treatment of rheumatoid arthritis
Target
LTB (TNFC, TNFSF3) [HSA:4050] [KO:K03157]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04064  NF-kappa B signaling pathway
hsa05323  Rheumatoid arthritis
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Tumor necrosis factors
    LTB (TNFC, TNFSF3)
     D08866  Baminercept (USAN/INN)
Other DBs
CAS: 909110-25-4
PubChem: 96025549
LinkDB

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