KEGG   DRUG: Melrilimab
Entry
D11796                      Drug                                   
Name
Melrilimab (USAN)
Formula
C6522H10080N1712O2106S48
Exact mass
147616.0886
Mol weight
147707.23
Sequence
(Heavy chain)
EVQLLESGGG LVQPGGSLRL SCAASGFTFS IYDMIWVRQA PGKGLEWVSS IRGEGGGTYY
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCARDP WSTEGSFFVL DYWGQGTLVT
VSSASTKGPS VFPLAPCSRS TSESTAALGC LVKDYFPEPV TVSWNSGALT SGVHTFPAVL
QSSGLYSLSS VVTVTSSNFG TQTYTCNVDH KPSNTKVDKT VERKCCVECP PCPAPPAAAS
SVFLFPPKPK DTLMISRTPE VTCVVVDVSA EDPEVQFNWY VDGVEVHNAK TKPREEQFNS
TFRVVSVLTV LHQDWLNGKE YKCKVSNKGL PSSIEKTISK TKGQPREPQV YTLPPSREEM
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPML DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPGK
(Light chain)
EIVLTQSPAT LSLSPGERAT LSCRASQSVD DDLAWYQQKP GQAPRLLIYD ASNRATGIPA
RFSGSGSGTD FTLTISSLEP EDFAVYYCQQ YITAPLTFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H137-H'226, H150-H206, H225-L214, H226-H'137, H229-H'229, H232-H'232, H263-H323, H369-H427, H'22-H'96, H'150-H'206, H'225-L'214, H'369-H'427, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antiasthmatic, Anti-interleukin 1 receptor-like 1 protein antibody
  Type
Monoclonal antibody
Target
IL1RL1 [HSA:9173] [KO:K05171]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    IL1RL1
     D11796  Melrilimab (USAN)
Other DBs
CAS: 2222865-46-3
PubChem: 405226662
LinkDB

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