KEGG   DRUG: Astegolimab
Entry
D11832                      Drug                                   
Name
Astegolimab (USAN/INN)
Formula
C6424H9878N1694O2030S52
Exact mass
144896.7274
Mol weight
144986.78
Sequence
(Heavy chain)
EVQLVQSGAE VKKPGESLKI SCKGSGYSFT NYWIGWVRQM PGKGLEWMGI IYPGNSDTRF
SPSFQGQVTI SADKSITTAY LQWSSLKASD TAMYYCARHG TSSDYYGLDV WGQGTTVTVS
SASTKGPSVF PLAPCSRSTS ESTAALGCLV KDYFPEPVTV SWNSGALTSG VHTFPAVLQS
SGLYSLSSVV TVPSSNFGTQ TYTCNVDHKP SNTKVDKTVE RKCCVECPPC PAPPVAGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVQFNWYVD GVEVHNAKTK PREEQFNSTF
RVVSVLTVVH QDWLNGKEYK CKVSNKGLPA PIEKTISKTK GQPREPQVYT LPPSREEMTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPMLDS DGSFFLYSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCQASQDIS NYLNWYQQKP GKAPKLLIYD ASNLETGVPS
RFSGSGSGTD FTFTISSLQP EDIATYYCQQ DDNFPLTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H135-H'224, H148-H204, H223-L214, H224-H'135, H227-H'227, H230-H'230, H261-H321, H367-H425, H'22-H'96, H'148-H'204, H'223-L'214, H'261-H'321, H'367-H'425, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antiasthmatic, Anti-interleukin 1 receptor-like1 antibody
  Type
Monoclonal antibody
Target
IL1RL1 [HSA:9173] [KO:K05171]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Signaling molecules and receptors
  Cytokine receptors
   Interleukin receptors
    IL1RL1
     D11832  Astegolimab (USAN/INN)
Other DBs
CAS: 2173054-79-8
LinkDB

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