KEGG   DRUG: Lirentelimab
Entry
D11906                      Drug                                   
Name
Lirentelimab (USAN)
Formula
C6408H9884N1700O2006S46
Exact mass
144219.0824
Mol weight
144308.30
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFSLT IYGAHWVRQA PGKGLEWVGV IWAGGSTNYN
SALMSRFTIS KDNSKNTVYL QMNSLRAEDT AVYYCARDGS SPYYYSMEYW GQGTTVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKRVEP KSCDKTHTCP PCPAPELLGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS HEDPEVKFNW YVDGVEVHNA KTKPREEQYN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSREE
MTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPGK
(Light chain)
EIVLTQSPAT LSLSPGERAT LSCSATSSVS YMHWFQQKPG QAPRLLIYST SNLASGIPAR
FSGSGSGTDF TLTISSLEPE DFAVYYCQQR SSYPFTFGPG TKLDIKRTVA APSVFIFPPS
DEQLKSGTAS VVCLLNNFYP REAKVQWKVD NALQSGNSQE SVTEQDSKDS TYSLSSTLTL
SKADYEKHKV YACEVTHQGL SSPVTKSFNR GEC
(Disulfide bride: H22-H95, H147-H203, H223-L213, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'95, H'147-H'203, H'223-L'213, H'264-H'324, H'370-H'428, L23-L87, L133-L193, L'23-L'87, L'133-L'193)
  Type
Peptide
Efficacy
Anti-inflammatory, Anti-Siglec-8 antibody
  Type
Monoclonal antibody
Comment
Treatment of eosinophilic gastrointestinal diseases, systemic mastocytosis, chronic urticaria, and/or severe allergic conjunctivitis
Target
SIGLEC8 [HSA:27181] [KO:K06748]
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Cell adhesion molecules: Ig superfamiy
   SIGLEC family
    SIGLEC8
     D11906  Lirentelimab (USAN)
Other DBs
CAS: 2283348-97-8
PubChem: 497620319
LinkDB

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