KEGG   DRUG: Boserolimab
Entry
D12256                      Drug                                   
Name
Boserolimab (USAN)
Formula
C6426H9908N1686O2013S46
Exact mass
144375.1916
Mol weight
144464.59
Sequence
(Heavy chain)
EIQLVQSGAE VKKPGASVKV SCKASGYTFT NYGMNWVKQA PGQGLKWMGW INTNTGEPTY
AEEFKGRFTF TLDTSISTAY MELSSLRSED TAVYYCAREG DAMDYWGQGT TVTVSSASTK
GPSVFPLAPS SKSTSGGTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTQTYICN VNHKPSNTKV DKKVEPKSCD KTHTCPPCPA PELLGGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP REEQYNSTYR
VVSVLTVLHQ DWLNGKEYKC KVSNKALPAP IEKTISKAKG QPREPQVYTL PPSRDELTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPGK
(Light chain)
EIVLTQSPAT LSLSPGERAT LSCSASSSVS YMHWYQQKPG QAPKRWIYDT SKLASGVPAR
FSGSGSGTDY SLTISSLEPE DFAVYYCQQW NSYPFTFGQG TKLEIKRTVA APSVFIFPPS
DEQLKSGTAS VVCLLNNFYP REAKVQWKVD NALQSGNSQE SVTEQDSKDS TYSLSSTLTL
SKADYEKHKV YACEVTHQGL SSPVTKSFNR GEC
(Disulfide bridge: H22-H96, H143-H199, H219-L213, H225-H'225, H228-H'228, H260'H320, H366-H424, H'22-H'96, H'143-H'199, H'219-L'213, H'260-H'320, H'366-H'424, L23-L87, L133-L193, L'23-L'87, L'133-L'193)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
TNFRSF7 (CD27) [HSA:939] [KO:K05144]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Tumor necrosis factor receptors
    TNFRSF7 (CD27)
     D12256  Boserolimab (USAN)
Other DBs
CAS: 2209116-30-1
PubChem: 497620669
LinkDB

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