KEGG   DRUG: Mipasetamab
Entry
D12279                      Drug                                   
Name
Mipasetamab (USAN/INN)
Formula
C6472H9946N1714O2024S44
Exact mass
145469.5749
Mol weight
145559.43
Sequence
(Heavy chain)
QVQLVESGGG VVQPGRSLRL SCAASGFTFS SYGMSWVRQA PGKGLEWVAT ISSGGSYTYY
PDSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCARHP IYYTYDDTMD YWGQGTTVTV
SSASTKGPSV FPLAPSSKST SGGTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ
SSGLYSLSSV VTVPSSSLGT QTYICNVNHK PSNTKVDKKV EPKSCDKTHT CPPCPAPELL
GGPSVFLFPP KPKDTLMISR TPEVTCVVVD VSHEDPEVKF NWYVDGVEVH NAKTKPREEQ
YNSTYRVVSV LTVLHQDWLN GKEYKCKVSN KALPAPIEKT ISKAKGQPRE PQVYTLPPSR
EEMTKNQVSL TCLVKGFYPS DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSKLTVDKS
RWQQGNVFSC SVMHEALHNH YTQKSLSLSP G
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCSASSSVS SGNFHWYQQK PGLAPRLLIY RTSNLASGIP
ARFSGSGSGT DFTLTISSLE PEDFAVYYCQ QWSGYPWTFG GGTKLEIKRT VAAPSVFIFP
PSDEQLKSGT ASVVCLLNNF YPREAKVQWK VDNALQSGNS QESVTEQDSK DSTYSLSSTL
TLSKADYEKH KVYACEVTHQ GLSSPVTKSF NRGEC
(Disulfide bridge: H22-H96, H149-H205, H225-L215, H231-H'231, H234-H'234, H266-H326, H372-H430, H'22-H'96, H'149-H'205, H'225-L'215, H'266-H'326, H'372-H'430, L23-L89, L135-L195, L'23-L'89, L'135-L'195)
  Type
Peptide
Efficacy
Antineoplastic, Anti-AXL antibody
  Type
Monoclonal antibody
Comment
Treatment of solid tumors
Target
AXL [HSA:558] [KO:K05115]
Brite
Target-based classification of drugs [BR:br08310]
 Protein kinases
  Receptor tyrosine kinases (RTK)
   AXL family
    AXL
     D12279  Mipasetamab (USAN/INN)
Other DBs
CAS: 2361055-48-1
PubChem: 497620692
LinkDB

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