KEGG   DRUG: Lemzoparlimab
Entry
D12385                      Drug                                   
Name
Lemzoparlimab (USAN/INN)
Formula
C6444H10042N1732O2019S46
Exact mass
145466.3510
Mol weight
145556.16
Sequence
(Heavy chain)
EVQLVESGGG LVKPGGSLRL SCAASGLTFE RAWMNWVRQA PGKGLEWVGR IKRKTDGETT
DYAAPVKGRF SISRDDSKNT LYLQMNSLKT EDTAVYYCAG SNRAFDIWGQ GTMVTVSSAS
TKGPSVFPLA PCSRSTSEST AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTKTYT CNVDHKPSNT KVDKRVESKY GPPCPPCPAP EFLGGPSVFL
FPPKPKDTLM ISRTPEVTCV VVDVSQEDPE VQFNWYVDGV EVHNAKTKPR EEQFNSTYRV
VSVLTVLHQD WLNGKEYKCK VSNKGLPSSI EKTISKAKGQ PREPQVYTLP PSQEEMTKNQ
VSLTCLVKGF YPSDIAVEWE SNGQPENNYK TTPPVLDSDG SFFLYSRLTV DKSRWQEGNV
FSCSVMHEAL HNHYTQKSLS LSLGK
(Light chain)
DIVMTQSPDS LAVSLGERAT INCKSSQSVL YAGNNRNYLA WYQQKPGQPP KLLINQASTR
ASGVPDRFSG SGSGTEFTLI ISSLQAEDVA IYYCQQYYTP PLAFGGGTKL EIKRTVAAPS
VFIFPPSDEQ LKSGTASVVC LLNNFYPREA KVQWKVDNAL QSGNSQESVT EQDSKDSTYS
LSSTLTLSKA DYEKHKVYAC EVTHQGLSSP VTKSFNRGEC
(Disulfide bridge: H22-H98, H132-L220, H145-H201, H224-H'224, H227-H'227, H259-H319, H365-H423, H'22-H'98, H'132-L'220, H'145-H'201 H'259-H'319, H'365-H'423, L23-L94, L140-L200, L'23-L'94, L'140-L'200)
  Type
Peptide
Efficacy
Antineoplastic, Anti-CD47 antibody
  Type
Monoclonal antibody
Target
CD47 [HSA:961] [KO:K06266]
  Pathway
hsa04512  ECM-receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   CD molecules
    CD47
     D12385  Lemzoparlimab (USAN/INN)
Other DBs
CAS: 2377483-71-9
PubChem: 497620798
LinkDB

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