KEGG   DRUG: Davutamig
Entry
D12424                      Drug                                   
Name
Davutamig (USAN)
Formula
C6427H9906N1700O2030S45
Exact mass
144821.1605
Mol weight
144910.60
Sequence
(Heavy chain)
EVQLVESGGG LVQPGTSLRL SCAASGFTFD DYAMHWVRQA PGKGLEWVSG ITWNSYNIDY
ADSVKGRFTI SRDNAKNSLY LQMNSLRAED TALYYCAKDD DYSNYVYFDY WGQGTLVTVS
SASTKGPSVF PLAPCSRSTS ESTAALGCLV KDYFPEPVTV SWNSGALTSG VHTFPAVLQS
SGLYSLSSVV TVPSSSLGTK TYTCNVDHKP SNTKVDKRVE SKYGPPCPPC PAPEFLGGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSQE DPEVQFNWYV DGVEVHNAKT KPREEQFNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKGLP SSIEKTISKA KGQPREPQVY TLPPSQEEMT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSR LTVDKSRWQE
GNVFSCSVMH EALHNHYTQK SLSLSLGK
(heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFIVT TNYMTWLRQA PGKGLEWVSL IYSSGHTYYA
DSVKGRFTIS RHNSKNTLYL QMDSLRAEDT AVYYCASAFA ADVFDIWGQG TMVTVSSAST
KGPSVFPLAP CSRSTSESTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTKTYTC NVDHKPSNTK VDKRVESKYG PPCPPCPAPE FLGGPSVFLF
PPKPKDTLMI SRTPEVTCVV VDVSQEDPEV QFNWYVDGVE VHNAKTKPRE EQFNSTYRVV
SVLTVLHQDW LNGKEYKCKV SNKGLPSSIE KTISKAKGQP REPQVYTLPP SQEEMTKNQV
SLTCLVKGFY PSDIAVEWES NGQPENNYKT TPPVLDSDGS FFLYSRLTVD KSRWQEGNVF
SCSVMHEALH NRFTQKSLSL SPGK
(Lihgt chain)
DIQMTQSPSS LSASVGDRVT ITCRASQSIS SYLNWYQQKP GKAPKLLIYA ASSLQSGVPS
RFSGSGSGTD FTLTISSLQP EDFATYYCQQ SYSTPPITFG QGTRLEIKRT VAAPSVFIFP
PSDEQLKSGT ASVVCLLNNF YPREAKVQWK VDNALQSGNS QESVTEQDSK DSTYSLSSTL
TLSKADYEKH KVYACEVTHQ GLSSPVTKSF NRGEC
(Disulfide bridge: H22-H96, H135-L215, H148-H204, H227-h223, H230-h226, H262-H322, H368-H426, h22-h95, h131-L'215, h114-h200, h258-h318, h364-h422, L23-L88, L135-L195, L'23-L'88, L'135-L'195)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Bispecific antibody
Comment
Biparatopic antibody
Target
MET [HSA:4233] [KO:K05099]
  Pathway
hsa04014  Ras signaling pathway
hsa04151  PI3K-Akt signaling pathway
hsa05200  Pathways in cancer
Brite
Target-based classification of drugs [BR:br08310]
 Protein kinases
  Receptor tyrosine kinases (RTK)
   MET family
    MET
     D12424  Davutamig (USAN)
Other DBs
CAS: 2648058-48-2
PubChem: 497620837
LinkDB

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