KEGG   DRUG: Gruticibart
Entry
D12541                      Drug                                   
Name
Gruticibart (USAN)
Formula
C6388H9908N1690O2013S42
Exact mass
143847.3156
Mol weight
143935.94
Sequence
(Heavy chain)
QVQLQESGPG LVKPSETLSI TCTVSGFSLT GYGIYWVRQP PGKGLEWLGM IWGDGRTDYN
SALKSRVTIS KDNSKSQVSL KLSSVTAADT ARYYCARDYY GSKDYWGQGT TVTVSSASTK
GPSVFPLAPC SRSTSESTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTKTYTCN VDHKPSNTKV DKRVESKYGP PCPPCPAPEF LGGPSVFLFP
PKPKDTLMIS RTPEVTCVVV DVSQEDPEVQ FNWYVDGVEV HNAKTKPREE QFNSTYRVVS
VLTVLHQDWL NGKEYKCKVS NKGLPSSIEK TISKAKGQPR EPQVYTLPPS QEEMTKNQVS
LTCLVKGFYP SDIAVEWESN GQPENNYKTT PPVLDSDGSF FLYSRLTVDK SRWQEGNVFS
CSVMHEALHN HYTQKSLSLS LGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCKASQDVS TAVAWYQQKP GKAPKLLIYL TSYRNTGVPD
RFSGSGSGTD FTFTISSLQP EDIAVYYCQQ HYKTPYSFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H95, H130-L214, H143-H199, H222-H'222, H225-H'225, H257-H317, H363-H421, H'22-H'95, H'130-L'214, H'143-H'199, H'257-H'317, H'363-H'421, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Contact activation inhibitor
  Type
Monoclonal antibody
Comment
Treatment of thrombosis and thromboembolism
Target
F9 [HSA:2158] [KO:K01321]
  Pathway
hsa04610  Complement and coagulation cascades
Brite
Target-based classification of drugs [BR:br08310]
 Peptidases and inhibitors
  Serine peptidases
   Chymotrypsin family
    F9
     D12541  Gruticibart (USAN)
Other DBs
CAS: 2704554-77-6
PubChem: 497620954
LinkDB

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