KEGG   DRUG: Amlitelimab
Entry
D12550                      Drug                                   
Name
Amlitelimab (USAN/INN)
Formula
C6648H9976N1728O2046S48
Exact mass
148287.6291
Mol weight
148379.89
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFS NYAMNWVRQA PGKGLEWVST ISGSGGATRY
ADSVKGRFTI SRDNSRNTVY LQMNSLRVED TAVFYCTKDR LIMATVRGPY YYGMDVWGQG
TTVTVSSAST KGPSVFPLAP CSRSTSESTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF
PAVLQSSGLY SLSSVVTVPS SSLGTKTYTC NVDHKPSNTK VDKRVESKYG PPCPPCPAPE
FEGGPSVFLF PPKPKDTLMI SRTPEVTCVV VDVSQEDPEV QFNWYVDGVE VHNAKTKPRE
EQFNSTYRVV SVLTVLHQDW LNGKEYKCKV SNKGLPSSIE KTISKAKGQP REPQVYTLPP
SQEEMTKNQV SLTCLVKGFY PSDIAVEWES NGQPENNYKT TPPVLDSDGS FFLYSRLTVD
KSRWQEGNVF SCSVMHEALH NHYTQKSLSL SLGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRASQSIS SYLNWYQQKP GKAPNLLIYA ASSLQSGVPS
RFSGSGSETD FTLTISSLQP EDFATYYCQQ SHSVSFTFGP GTKVDIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H154-H210, H141-L214, H233-H'233, H236-H'236, H268-H328, H374-H432, H'22-H'96, H'154-H'210, H'141-L'214, H'268-H'328, H'374-H'432, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Immunomodulator
  Type
Monoclonal antibody
Comment
Treatment of immune mediated diseases
Target
TNFSF4 (CD252, OX40L) [HSA:7292] [KO:K05469]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Tumor necrosis factors
    TNFSF4 (CD252, OX40L)
     D12550  Amlitelimab (USAN/INN)
Other DBs
CAS: 2378692-15-8
PubChem: 497620963
LinkDB

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