KEGG   DRUG: Paridiprubart
Entry
D12624                      Drug                                   
Name
Paridiprubart (USAN/INN)
Formula
C6454H9978N1706O2010S40
Exact mass
144821.9837
Mol weight
144911.18
Sequence
(Heavy chain)
XVQLQESGPG LVKPSDTLSL TCAVSGYSIT GGYSWHWIRQ PPGKGLEWMG YIHYSGYTDF
NPSLKTRITI SRDTSKNQFS LKLSSVTAVD TAVYYCARKD PSDAFPYWGQ GTLVTVSSAS
TKGPSVFPLA PSSKSTSGGT AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTQTYI CNVNHKPSNT KVDKRVEPKS CDKTHTCPPC PAPELLGGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSHE DPEVKFNWYV DGVEVHNAKT KPREEQYNST
YRVVSVLTVL HQDWLNGKEY KCKVSSKAFP APIEKTISKA KGQPREPQVY TLPPSREEMT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSK LTVDKSRWQQ
GNVFSCSVMH EALHNHYTQK SLSLSPG
(Light chain)
EIVLTQSPDF QSVTPKEKVT ITCRASQSIS DHLHWYQQKP DQSPKLLIKY ASHAISGVPS
RFSGSGSGTD FTLTINSLEA EDAATYYCQQ GHSFPLTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H145-H201, H221-L214, H227-H'227, H230-H'230, H262-H322, H368-H426, H'22-H'96, H'145-H'201, H'221-L'214, H'262-H'322, H'368-H'426, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Anti-inflammatory
  Type
Monoclonal antibody
Comment
Treatment of pathological inflammatory disorders such as cytokine release syndrome - induced Acute respiratory distress syndrome
Target
TLR4 (CD284) [HSA:7099] [KO:K10160]
  Pathway
hsa04145  Phagosome
hsa04151  PI3K-Akt signaling pathway
hsa04613  Neutrophil extracellular trap formation
hsa04620  Toll-like receptor signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Signaling molecules and receptors
  Pattern recognition receptors
   Toll-like receptors
    TLR4 (CD284)
     D12624  Paridiprubart (USAN/INN)
Other DBs
CAS: 2641646-59-3
PubChem: 497621037
LinkDB

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