KEGG   DRUG: Adakitug
Entry
D12656                      Drug                                   
Name
Adakitug (USAN)
Formula
C6430H9920N1720O2000S42
Exact mass
144575.5678
Mol weight
144664.70
Sequence
(Heavy chain)
QVQLVESGGG VVQPGRSLRL SCTASGFTFS HYGMYWVRQA PGKGLEWVAV IWYDGSYEYN
ADSVKGRFTI SRDNSKNTLY LQMNSLRAED TAVYYCARDR VGLFDYWGQG TLVTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDKRVEPKSC DKTHTCPPCP APELLGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK PREEQYNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKALPA PIEKTISKAK GQPREPQVYT LPPSREEMTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCRASQSIS SSYLAWYQQK PGQAPRLLIY GPSSRATGIP
DRFSGSGSGT DFTLTISRLE PEDFAVYYCQ QYAGSLTFGP GTKVDIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H144-H200, H220-L214, H226-H'226, H229-H'229, H261-H321, H367-H425, H'22-H'96, H'144-H'200, H'220-L'214, H'261-H'321, H'367-H'425, L23-L89, L134-L194, L'23-L'89, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
IL8 [HSA:3576] [KO:K10030]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04062  Chemokine signaling pathway
hsa04064  NF-kappa B signaling pathway
hsa04218  Cellular senescence
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Interleukins
    IL8
     D12656  Adakitug (USAN)
Other DBs
CAS: 2837159-88-1
PubChem: 497621069
LinkDB

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