KEGG   DRUG: Levilimab
Entry
D12748                      Drug                                   
Name
Levilimab (INN)
Sequence
(Heavy chain)
QVQLVQSGGG LVQPGGSLRL SCAASGFTFS SYYMSWVRQA PGKGLEWVSG IYSDGTTHYG
DSVKGRFTIS RDNAKNTVYL QLNSLRAEDT AMYYCAKGAG PTWWYALDAW GQGTLVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKRVEP KSCDKTHTCP PCPAPPVAGG
PSVFLFPPKP KDTLYITREP EVTCVVVDVS HEDPEVKFNW YVDGVEVHNA KTKPREEQYN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSREE
MTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPGK
(Light chain)
DIQLTQSPSS VSVSVGERVT IDCKSSQSVL SASNTYLNWY QQKPGQAPQL LIYYASTRES
GVPDRFSGSG SGTDFTITIS SLQAEDAAVY YCQQAYRAPV TFGQGTKLEI KRTVAAPSVF
IFPPSDEQLK SGTASVVCLL NNFYPREAKV QWKVDNALQS GNSQESVTEQ DSKDSTYSLS
STLTLSKADY EKHKVYACEV THQGLSSPVT KSFNRGEC
(Disulfide bridge: H22-H95, H147-H203, H223-L218, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'95, H'147-H'203, H'223-L'218, H'264-H'324, H'370-H'428, L23-L92, L138-L198, L'23-L'92, L'138-L'198)
  Type
Peptide
Class
Immunological agent
 DG02019  Interleukin inhibitor
Remark
ATC code: L04AC25
Efficacy
Immunomodulator
  Type
Monoclonal antibody, Anti-IL-6 receptor antibody
Target
IL6R (CD126) [HSA:3570] [KO:K05055]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04630  JAK-STAT signaling pathway
hsa04659  Th17 cell differentiation
Interaction
Brite
Anatomical Therapeutic Chemical (ATC) classification [BR:br08303]
 L ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS
  L04 IMMUNOSUPPRESSANTS
   L04A IMMUNOSUPPRESSANTS
    L04AC Interleukin inhibitors
     L04AC25 Levilimab
      D12748  Levilimab (INN)
Drug groups [BR:br08330]
 Immunological agent
  DG02019  Interleukin inhibitor
   D12748  Levilimab
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    IL6R (CD126)
     D12748  Levilimab (INN)
Other DBs
CAS: 2035008-70-7
PubChem: 497621161
LinkDB

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