KEGG   DRUG: Tulisokibart
Entry
D12760                      Drug                                   
Name
Tulisokibart (USAN/INN)
Formula
C6476H10054N1718O2078S42
Exact mass
146482.2136
Mol weight
146572.19
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGFDIQ DTYMHWVKQR PGQGLEWMGR IDPASGHTKY
DPKFQVRVTI TRDTSTSTVY LELSSLRSED TAVYYCARSG GLPDVWGQGT TVTVSSASTK
GPSVFPLAPS SKSTSGGTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTQTYICN VNHKPSNTKV DKKVEPKSCD KTHTCPPCPA PEAAGGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP REEQYNSTYR
VVSVLTVLHQ DWLNGKEYKC KVSNKALAAP IEKTISKAKG QPREPQVYTL PPSRDELTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPGK
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCRASSSVS YMYWYQQKPG QAPRPLIYAT SNLASGIPDR
FSGSGSGTDF TLTISRLEPE DFAVYYCQQW EGNPRTFGGG TKLEIKRTVA APSVFIFPPS
DEQLKSGTAS VVCLLNNFYP REAKVQWKVD NALQSGNSQE SVTEQDSKDS TYSLSSTLTL
SKADYEKHKV YACEVTHQGL SSPVTKSFNR GEC
(Disulfide bridge: H22-H96, H143-H199, H219-L213, H225-H'225, H228-H'228, H260-H320, H366-H424, H'22-H'96, H'143-H'199, H'219-L'213, H'260-H'320, H'366-H'424, L23-L87, L133-L193, L'23-L'87, L'133-L'193)
  Type
Peptide
Efficacy
Anti-inflammatory
  Type
Monoclonal antibody
Comment
Treatment of Crohn's disease, ulcerative colitis, and scleroderma-associated interstitial lung disease
Target
TNFSF15 [HSA:9966] [KO:K05478]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Tumor necrosis factors
    TNFSF15
     D12760  Tulisokibart (USAN/INN)
Other DBs
CAS: 2648504-55-4
PubChem: 497621173
LinkDB

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