KEGG   DRUG: Falbikitug
Entry
D12810                      Drug                                   
Name
Falbikitug (USAN/INN)
Formula
C6498H10028N1728O2026S48
Exact mass
146220.1377
Mol weight
146310.72
Sequence
(Heavy chain)
QVQLQESGGG LVKPGGSLRL SCAASGFTFS HAWMHWVRQA PGKGLEWVGQ IKAKSDDYAT
YYAESVKGRF TISRDDSKNT LYLQMNSLKT EDTAVYYCTC WEWDLDFWGQ GTMVTVSSAS
TKGPSVFPLA PSSKSTSGGT AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTQTYI CNVNHKPSNT KVDKKVEPKS CDKTHTCPPC PAPELLGGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSHE DPEVKFNWYV DGVEVHNAKT KPREEQYNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKALP APIEKTISKA KGQPREPQVY TLPPSRDELT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSK LTVDKSRWQQ
GNVFSCSVMH EALHNHYTQK SLSLSPGK
(Light chain)
DIVMTQTPLS SPVTLGQPAS ISCRSSQSLL DSDGHTYLNW LQQRPGQPPR LLIYSVSNLE
SGVPDRFSGS GAGTDFTLKI SRVEAEDVGV YYCMQATHAP PYTFGQGTKL EIKRTVAAPS
VFIFPPSDEQ LKSGTASVVC LLNNFYPREA KVQWKVDNAL QSGNSQESVT EQDSKDSTYS
LSSTLTLSKA DYEKHKVYAC EVTHQGLSSP VTKSFNRGEC
(Disulfide bridge: H22-H98, H145-H201, H221-L220, H227-H'227, H'230-H'230, H262-H322, H368-H426, H'22-H'98, H'145-H'201, H'221-L'220, H'262-H'322, H'368-H'426, L23-L93, L140-L200, L'23-L'93, L'140-L'200)
  Type
Peptide
Efficacy
Antineoplastic, Anti-leukemia inhibitory factor antibody
  Type
Monoclonal antibody
Target
LIF [HSA:3976] [KO:K05419]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04550  Signaling pathways regulating pluripotency of stem cells
hsa04630  JAK-STAT signaling pathway
hsa04668  TNF signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   CSF and other factors
    LIF
     D12810  Falbikitug (USAN/INN)
Other DBs
CAS: 2740565-02-8
PubChem: 497621223
LinkDB

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