KEGG   DRUG: Ulviprubart
Entry
D12825                      Drug                                   
Name
Ulviprubart (USAN/INN)
Formula
C6550H10086N1730O2034S42
Exact mass
146866.7246
Mol weight
146957.34
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT DHNMHWVKQA TGQGLEWFGF INPNTGVTRY
NQKFQGRVTL TINKAISTAY LELSSLRSED TAVYYCARDY YGSAWFAYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP CPAPELLGGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPREEQYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSREEM
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPGK
(Light chain)
DIVMTQSPDS LAVSLGERAT INCKSSQTLL YSSDQKNYLA WYQQKPGQPP KLLIYWASTR
ESGVPDRFSG SGSGTDFTLT ISSLQAEDVA VYYCQQYYNY PTFGGGTKVE IKRTVAAPSV
FIFPPSDEQL KSGTASVVCL LNNFYPREAK VQWKVDNALQ SGNSQESVTE QDSKDSTYSL
SSTLTLSKAD YEKHKVYACE VTHQGLSSPV TKSFNRGEC
(Disulfide bridge: H22-H96, H146-H202, H222-L219, H228-H'228, H231-H'231, H263-H323, H369-H427, H'22-H'96, H'146-H'202, H'222-L'219, H'263-H'323, H'369-H'427, L23-L94, L139-L199, L'23-L'94, L'139-L'199)
  Type
Peptide
Efficacy
Antineoplastic, Immunosuppressant
  Type
Monoclonal antibody
Comment
Treatment of inclusion body myositis and T cell large granular lymphocytic leukemia
Target
KLRG1 [HSA:10219] [KO:K10076]
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Other cell surface molecules
   Other
    KLRG1
     D12825  Ulviprubart (USAN/INN)
Other DBs
CAS: 2569434-60-0
PubChem: 497621238
LinkDB

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