KEGG   DRUG: Imzokitug
Entry
D12849                      Drug                                   
Name
Imzokitug (USAN)
Formula
C6456H10020N1744O2014S48
Exact mass
145740.1853
Mol weight
145830.33
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT DSEMHWVRQA TGQGLEWMGA IQPETGGTAY
NQKFKARVTM TRDTSISTAY MELSSLRSED TAVYYCARRR RNFDYWGQGT LVTVSSASTK
GPSVFPLAPS SKSTSGGTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTQTYICN VNHKPSNTKV DKRVEPKSCD KTHTCPPCPA PELLGGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP REEQYNSTYR
VVSVLTVLHQ DWLNGKEYKC KVSNKALPAP IEKTISKAKG QPREPQVYTL PPSREEMTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPG
(Light chain)
DIVMTQTPLS LSVTPGQPAS ISCRSSQSLF HSSGNTYLHW YLQKPGQPPQ LLIYKVSNRF
SGVPDRFSGS GSGTDFTLKI SRVEAEDVGV YYCSQSTHVP FTFGQGTKLE IKRTVAAPSV
FIFPPSDEQL KSGTASVVCL LNNFYPREAK VQWKVDNALQ SGNSQESVTE QDSKDSTYSL
SSTLTLSKAD YEKHKVYACE VTHQGLSSPV TKSFNRGEC
(Disulfide bridge: H22-H96, H143-H199, H219-L219, H225-H'225, H228-H'228, H260-H320, H366-H424, H'22-H'96, H'143-H'199, H'219-L'219, H'260-H'320, H'366-H'424, L23-L93, L139-L199, L'23-L'93, L'139-L'199)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
CCR8 [HSA:1237] [KO:K04183]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04062  Chemokine signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Chemokine receptors
    CCR8
     D12849  Imzokitug (USAN)
Other DBs
CAS: 2883771-61-5
PubChem: 497621262
LinkDB

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