KEGG   DRUG: Rilogrotug
Entry
D12852                      Drug                                   
Name
Rilogrotug (USAN)
Formula
C6452H9972N1712O2024S48
Exact mass
145355.6605
Mol weight
145445.68
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGSSVKV SCKASGYTFS DYNMDWVRQA PGQGLEWMGQ INPNNGLIFF
NQKFKGRVTL TADKSTSTAY MELSSLRSED TAVYYCAREA ITTVGAMDYW GQGTLVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKRVEP KSCDKTHTCP PCPAPELLGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS HEDPEVKFNW YVDGVEVHNA KTKPREEQYN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSREE
MTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRTSENLH NYLAWYQQKP GKAPKLLIYD AKTLADGVPS
RFSGSGSGTD YTLTISSLQP EDFATYYCQH FWSSPYTFGQ GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H147-H203, H223-L214, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'96, H'147-H'203, H'223-L'214, H'264-H'324, H'370-H'428, L23-L88, L134-L194 L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Anti-growth differentiation factor 15 antibody
  Type
Monoclonal antibody
Comment
Treatment of cachexia in cancer patients with elevated GDF-15 levels
Target
GDF15 [HSA:9518] [KO:K05504]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Transforming growth factors (RSTK-binding)
    GDF15
     D12852  Rilogrotug (USAN)
Other DBs
CAS: 2894138-72-6
PubChem: 497621265
LinkDB

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