KEGG   DRUG: Verekitug
Entry
D12973                      Drug                                   
Name
Verekitug (USAN/INN)
Formula
C6390H9904N1708O2004S42
Exact mass
143975.3854
Mol weight
144064.06
Sequence
(Heavy chain)
EVQLLESGGG LVQPGGSLRL SCAASGFTFR SSAMHWVRQA PGKGLKWVSS VSGSGAGTYY
ADSVKGRFTI SRDNPKNTLY LQMNSLRAED TAVYYCVKEG GSRGFDYWGQ GTLVTVSSAS
TKGPSVFPLA PSSKSTSGGT AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTQTYI CNVNHKPSNT KVDKKVEPKS CDKTHTCPPC PAPELLGGPS
VFLFPPKPKD TLMISRTPEV TCVVVDVSHE DPEVKFNWYV DGVEVHNAKT KPREEQYNST
YRVVSVLTVL HQDWLNGKEY KCKVSNKALP APIEKTISKA KGQPREPQVY TLPPSRDELT
KNQVSLTCLV KGFYPSDIAV EWESNGQPEN NYKTTPPVLD SDGSFFLYSK LTVDKSRWQQ
GNVFSCSVMH EALHNHYTQK SLSLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRASQDIS NYLAWFQQKP GKAPKSLIYT ASSLQSGVPS
KFSGSGSGTD FTLTISSLQP EDFATYYCQQ YNLYPPTFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H145-H201, H221-L214, H227-H'227, H230-H'230, H262-H322, H'22-H'96, H'221-L'214, H'262-H'322, H'145-H'201, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Anti-inflammatory
  Type
Monoclonal antibody
Comment
Treatment of asthma and inflammatory diseases
Target
CRLF2 (TSLPR) [HSA:64109] [KO:K05078]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04630  JAK-STAT signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    CRLF2 (TSLPR)
     D12973  Verekitug (USAN/INN)
Other DBs
CAS: 2768386-15-6
PubChem: 503268993
LinkDB

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