KEGG   DRUG: Iluzanebart
Entry
D12996                      Drug                                   
Name
Iluzanebart (USAN/INN)
Formula
C6440H9960N1708O2000S50
Exact mass
144823.6205
Mol weight
144913.58
Sequence
(Heavy chain)
EVQLVQSGAE VKKPGESLKI SCKGSGYSFT SYWIGWVRQM PGKGLEWMGI IYPGDADARY
SPSFQGQVTI SADKSISTAY LQWSSLKASD TAMYFCARRR QGIFGDALDF WGQGTLVTVS
SASTKGPSVF PLAPSSKSTS GGTAALGCLV KDYFPEPVTV SWNSGALTSG VHTFPAVLQS
SGLYSLSSVV TVPSSSLGTQ TYICNVNHKP SNTKVDKKVE PKSCDKTHTC PPCPAPELLG
GPSVFLFPPK PKDTLMISRT PEVTCVVVDV SHEDPEVKFN WYVDGVEVHN AKTKPCEEQY
GSTYRCVSVL TVLHQDWLNG KEYKCKVSNK ALPAPIEKTI SKAKGQPREP QVYTLPPSRE
EMTKNQVSLT CLVKGFYPSD IAVEWESNGQ PENNYKTTPP VLDSDGSFFL YSKLTVDKSR
WQQGNVFSCS VMHEALHNHY TQKSLSLSPG K
(Light chain)
EIVMTQSPAT LSVSPGERAT LSCRASQSVS SNLAWFQQKP GQAPRLLIYG ASTRATGIPA
RFSGSGSGTE FTLTISSLQP EDFAVYYCLQ DNNFPPTFGQ GTKVDIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H148-H204, H224-L214, H230-H'230, H233-H'233, H265-H325, H296-H306, H371-H429, H'22-H'96, H'148-H'204, H'224-L'214, H'265-H'325, H'296-H'325, H'371-H'429, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Neuroprotectant
  Type
Monoclonal antibody
Comment
Treatment of adult-onset leukoencephalopathy with axonal spheroids and pigmented glia
Target
TREM2 [HSA:54209] [KO:K14378]
  Pathway
hsa04380  Osteoclast differentiation
Brite
Target-based classification of drugs [BR:br08310]
 Not elsewhere classified
  Organismal systems
   Nervous system
    TREM2
     D12996  Iluzanebart (USAN/INN)
Other DBs
CAS: 2733621-19-5
PubChem: 504099512
LinkDB

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