KEGG   DRUG: Visugromab
Entry
D13004                      Drug                                   
Name
Visugromab (USAN/INN)
Formula
C6434H9922N1686O2012S46
Exact mass
144469.3062
Mol weight
144558.78
Sequence
(Heavy chain)
QITLKESGPT LVKPTQTLTL TCTFSGFSLS TSGMGVSWIR QPPGKGLEWL AHIYWDDDKR
YNPTLKSRLT ITKDPSKNQV VLTMTNMDPV DTATYYCARS SYGAMDYWGQ GTLVTVSSAS
TKGPSVFPLA PCSRSTSEST AALGCLVKDY FPEPVTVSWN SGALTSGVHT FPAVLQSSGL
YSLSSVVTVP SSSLGTKTYT CNVDHKPSNT KVDKRVESKY GPPCPPCPAP EFLGGPSVFL
FPPKPKDTLM ISRTPEVTCV VVDVSQEDPE VQFNWYVDGV EVHNAKTKPR EEQFNSTYRV
VSVLTVLHQD WLNGKEYKCK VSNKGLPSSI EKTISKAKGQ PREPQVYTLP PSQEEMTKNQ
VSLTCLVKGF YPSDIAVEWE SNGQPENNYK TTPPVLDSDG SFFLYSRLTV DKSRWQEGNV
FSCSVMHEAL HNHYTQKSLS LSLG
(Light chain)
DIVLTQSPSF LSASVGDRVT ITCKASQNVG TNVAWFQQKP GKSPKALIYS ASYRYSGVPD
RFTGSGSGTE FTLTISSLQP EDFAAYFCQQ YNNFPYTFGG GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H97, H132-H145, H201-L214, H224-H'224, H227-H'227, H259-H319, H365-H423, H'22-H'97, H'132-H'145, H'201-L'214, H'259-H'319, H'365-H'423, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic, Anti-growth differentiation factor 15 antibody
  Type
Monoclonal antibody
Target
GDF15 [HSA:9518] [KO:K05504]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
Brite
Target-based classification of drugs [BR:br08310]
 Signaling molecules and receptors
  Cytokines
   Transforming growth factors (RSTK-binding)
    GDF15
     D13004  Visugromab (USAN/INN)
Other DBs
CAS: 2556646-63-8
PubChem: 504099520
LinkDB

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