KEGG   DRUG: Sigvotatug
Entry
D13006                      Drug                                   
Name
Sigvotatug (USAN/INN)
Formula
C6518H10096N1708O2088S40
Exact mass
146984.5165
Mol weight
147074.76
Sequence
(Heavy chain)
QFQLVQSGAE VKKPGASVKV SCKASGYSFT DYNVNWVRQA PGQGLEWIGV INPKYGTTRY
NQKFKGRATL TVDKSTSTAY MELSSLRSED TAVYYCTRGL NAWDYWGQGT LVTVSSASTK
GPSVFPLAPS SKSTSGGTAA LGCLVKDYFP EPVTVSWNSG ALTSGVHTFP AVLQSSGLYS
LSSVVTVPSS SLGTQTYICN VNHKPSNTKV DKKVEPKSCD KTHTCPPCPA PELLGGPSVF
LFPPKPKDTL MISRTPEVTC VVVDVSHEDP EVKFNWYVDG VEVHNAKTKP REEQYNSTYR
VVSVLTVLHQ DWLNGKEYKC KVSNKALPAP IEKTISKAKG QPREPQVYTL PPSRDELTKN
QVSLTCLVKG FYPSDIAVEW ESNGQPENNY KTTPPVLDSD GSFFLYSKLT VDKSRWQQGN
VFSCSVMHEA LHNHYTQKSL SLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCGASENIY GALNWYQQKP GKAPKLLIYG ATNLEDGVPS
RFSGSGSGRD YTFTISSLQP EDIATYYCQN VLTTPYTFGQ GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H143-H199, H219-L214, H225-H'225, H'228-H'228, H260-H320, H366-H424, H'22-H'96, H'143-H'199, H'219-L'214, H'260-H'320, H'366-H'424, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
ITGB6 [HSA:3694] [KO:K06589]
  Pathway
hsa04151  PI3K-Akt signaling pathway
hsa04510  Focal adhesion
hsa04512  ECM-receptor interaction
hsa04810  Regulation of actin cytoskeleton
Brite
Target-based classification of drugs [BR:br08310]
 Cell surface molecules and ligands
  Cell adhesion molecules: other families
   Integrins
    ITGB6
     D13006  Sigvotatug (USAN/INN)
Other DBs
CAS: 2764774-90-3
PubChem: 504099522
LinkDB

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