KEGG   DRUG: Usilnetug
Entry
D13075                      Drug                                   
Name
Usilnetug (USAN/INN)
Formula
C6478H10068N1708O2022S44
Exact mass
145548.5213
Mol weight
145638.42
Sequence
(Heavy chain)
EVQLQESGPG LVKPSQTLSL TCTFSGFSLS TSGMGVSWIR QPPGKGLEWL AHIYWDDDKR
YNPYMKRRLT ISKDTSKNQV SLKISSVTAA DTAVYYCARR ADDYDVGFAY WGQGTLVTVS
SASTKGPSVF PLAPSSKSTS GGTAALGCLV KDYFPEPVTV SWNSGALTSG VHTFPAVLQS
SGLYSLSSVV TVPSSSLGTQ TYICNVNHKP SNTKVDKKVE PKSCDKTHTC PPCPAPELLG
GPSVFLFPPK PKDTLMISRT PEVTCVVVDV SHEDPEVKFN WYVDGVEVHN AKTKPREEQY
NSTYRVVSVL TVLHQDWLNG KEYKCKVSNK ALPAPIEKTI SKAKGQPREP QVYTLPPSRE
EMTKNQVSLT CLVKGFYPSD IAVEWESNGQ PENNYKTTPP VLDSDGSFFL YSKLTVDKSR
WQQGNVFSCS VMHEALHNHY TQKSLSLSPG K
(Light chain)
DIQMTQSPSS VSASVGDRVT ITCLASQTIG TWLAWYQQKP GKSPKLLIYA ATSLADGVPS
RFSGSGSGTD FTLTISSLQP EDFATYYCQQ LYSSPFTFGQ GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H97, H148-H204, H224-L214, H230-H'230, H233-H'233, H265-H325, H371-H429, H'22-H'97, H'148-H'204, H'224-L'214, H'265-H'325, H'371-H'429, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Dementia therapeutic agent
  Type
Monoclonal antibody
Comment
Treatment of Alzheimer's disease
Target
APP [HSA:351] [KO:K04520]
  Pathway
hsa04726  Serotonergic synapse
hsa05010  Alzheimer disease
Brite
Target-based classification of drugs [BR:br08310]
 Not elsewhere classified
  Organismal systems
   Nervous system
    APP
     D13075  Usilnetug (USAN/INN)
Other DBs
CAS: 2770861-19-1
PubChem: 507530390
LinkDB

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