KEGG   DRUG: Solrikitug
Entry
D13085                      Drug                                   
Name
Solrikitug (USAN/INN)
Formula
C6466H10022N1714O2010S48
Exact mass
145378.1291
Mol weight
145468.25
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYIFT DYAMHWVRQA PGQGLEWMGT FIPLLDTSDY
AQKFQGRVTM TADTSTSTAY MELRSLRSDD TAVYYCARMG VTHSYVMDAW GQGTLVTVSS
ASTKGPSVFP LAPSSKSTSG GTAALGCLVK DYFPEPVTVS WNSGALTSGV HTFPAVLQSS
GLYSLSSVVT VPSSSLGTQT YICNVNHKPS NTKVDKKVEP KSCDKTHTCP PCPAPELLGG
PSVFLFPPKP KDTLMISRTP EVTCVVVDVS HEDPEVKFNW YVDGVEVHNA KTKPREEQYN
STYRVVSVLT VLHQDWLNGK EYKCKVSNKA LPAPIEKTIS KAKGQPREPQ VYTLPPSRDE
LTKNQVSLTC LVKGFYPSDI AVEWESNGQP ENNYKTTPPV LDSDGSFFLY SKLTVDKSRW
QQGNVFSCSV MHEALHNHYT QKSLSLSPGK
(Light chain)
EIVLTQSPGT LSLSPGERAT LSCRASQPIS ISVHWYQQKP GQAPRLLIYF ASQSISGIPD
RFSGSGSGTD FTLTISRLEP EDFAVYYCQQ TFSLPYTFGQ GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H147-H203, H223-L214, H229-H'229, H232-H'232, H264-H324, H370-H428, H'22-H'96, H'147-H'203, H'223-L'214, H'264-H'324, H'370-H'428, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Anti-inlammatory, Immunomodulator
  Type
Monoclonal antibody
Comment
Treatment of immunologic conditions
Target
CRLF2 (TSLPR) [HSA:64109] [KO:K05078]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04630  JAK-STAT signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    CRLF2 (TSLPR)
     D13085  Solrikitug (USAN/INN)
Other DBs
CAS: 2768721-24-8
PubChem: 507530400
LinkDB

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