KEGG   DRUG: Tagmokitug
Entry
D13088                      Drug                                   
Name
Tagmokitug (USAN)
Formula
C6382H9924N1702O2005S46
Exact mass
143959.4067
Mol weight
144048.36
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGASVKV SCKASGYTFT SYYMHWVRQA PGQGLEWMGI INPSGGSTSY
AQKFQGRVTM TRDTSTSTVY MELSSLRSED TAVYYCARAV RNRFRFDYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP CPAPELLGGP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPREEQYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSRDEL
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPGK
(Light chain)
QSALTQPASV SGSPGQSITI SCTGTSSDVG SYNLVSWYQQ HPGKAPKLMI YEVSKRPSGV
SNRFSGSKSG NTASLTISGL QAEDEADYYC SSYAGSSTFV VFGGGTKLTV LGQPKAAPSV
TLFPPSSEEL QANKATLVCL ISDFYPGAVT VAWKADSSPV KAGVETTTPS KQSNNKYAAS
SYLSLTPEQW KSHRSYSCQV THEGSTVEKT VAPTECS
(Disulfide bridge: H22-H96, H146-H202, H222-L216, H228-H'228, H231-H'231, H263-H323, H369-H427, H'22-H'96, H'146-H'202, H'222-L'216, H'263-H'323, H'369-H'427, L22-L90, L139-L198, L'22-L'90, L'139-L'198)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody
Target
CCR8 [HSA:1237] [KO:K04183]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04062  Chemokine signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Chemokine receptors
    CCR8
     D13088  Tagmokitug (USAN)
Other DBs
CAS: 3024486-14-1
PubChem: 508750758
LinkDB

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