KEGG   DRUG: Efpixileukin alfa
Entry
D13094                      Drug                                   
Name
Efpixileukin alfa (USAN)
Formula
C3018H4712N792O905S22
Exact mass
67234.0895
Mol weight
67275.94
Sequence
(Heavy chain)
APASSSTKKT QLQLEHLLLN LQMILNGINN YKNPKLTRML TFKFYMPKKA TELKHLQCLE
EELKPLEEVL KLAQSKNFHL RPRDLISNIN VIVLELKGSE TTFMCEYADE TATIVEFLNR
WITFSQSIIS TLTEPKSSDK THTCPPCPAP PVAGPSVFLF PPKPKDTLMI SRTPEVTCVV
VDVKHEDPEV KFNWYVDGVE VHNAKTKPRE EQYNSTYRVV SVLTVLHQDW LNGKEYKCKV
SNKALPAPIE KTISKAKGQP REPQVYTLPP SREQMTKNQV KLTCLVKGFY PSDIAVEWES
NGQPENNYKT TPPVLDSDGS FFLYSKLTVD KSRWQQGNVF SCSVLHEALH SHYTQKSLSL
SPGK
(Light chain)
EPKSSDKTHT CPPCPAPPVA GPSVFLFPPK PKDTLMISRT PEVTCVVVDV KHEDPEVKFN
WYVDGVEVHN AKTKPREEEY NSTYRVVSVL TVLHQDWLNG KEYKCKVSNK ALPAPIEKTI
SKAKGQPREP QVYTLPPSRE EMTKNQVSLT CDVSGFYPSD IAVEWESDGQ PENNYKTTPP
VLDSDGSFFL YSKLTVDKSR WEQGDVFSCS VLHEALHSHY TQKSLSLSPG K
(Disulfide bridge: H58-H105, H144-L11, H147-L14, H178-H238, H284-H342, L45-L105, L151-L209)
  Type
Peptide
Efficacy
Anti-inflammatory disease
Comment
Treatment of atopic dermatitis and psoriasis
Target
IL2RA (CD25) [HSA:3559] [KO:K05068]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04630  JAK-STAT signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokine receptors
   Interleukin receptors
    IL2RA (CD25)
     D13094  Efpixileukin alfa (USAN)
Other DBs
CAS: 2996895-52-2
PubChem: 508750764
LinkDB

» Japanese version   » Back

DBGET integrated database retrieval system