KEGG   DRUG: Tolododekin alfa
Entry
D13096                      Drug                                   
Name
Tolododekin alfa (USAN)
Formula
C2753H4303N751O911S29
Exact mass
63387.5370
Mol weight
63427.06
Sequence
IWELKKDVYV VELDWYPDAP GEMVVLTCDT PEEDGITWTL DQSSEVLGSG KTLTIQVKEF
GDAGQYTCHK GGEVLSHSLL LLHKKEDGIW STDILKDQKE PKNKTFLRCE AKNYSGRFTC
WWLTTISTDL TFSVKSSRGS SDPQGVTCGA ATLSAERVRG DNKEYEYSVE CQEDSACPAA
EESLPIEVMV DAVHKLKYEN YTSSFFIRDI IKPDPPKNLQ LKPLKNSRQV EVSWEYPDTW
STPHSYFSLT FCVQVQGKSK REKKDRVFTD KTSATVICRK NASISVRAQD RYYSSSWSEW
ASVPCSGGGG SGGGGSGGGG SRNLPVATPD PGMFPCLHHS QNLLRAVSNM LQKARQTLEF
YPCTSEEIDH EDITKDKTST VEACLPLELT KNESCLNSRE TSFITNGSCL ASRKTSFMMA
LCLSSIYEDL KMYQVEFKTM NAKLLMDPKR QIFLDQNMLA VIDELMQALN FNSETVPQKS
SLEEPDFYKT KIKLCILLHA FRIRAVTIDR VMSYLNASGG GGEGGGGSEE GGGGSEEGGG
GSEEGGGGSE EGGGGSEEGG GGSEEGGGGS EEGGGGSEEG GGGS
(Disulfide bridge: 177-395)
  Type
Peptide
Efficacy
Antineoplastic
Comment
Single-chain human interlukin-12 fused to phosphorylated aluminum-binding peptide
Target
IL12RB [HSA:3594 3595] [KO:K05063 K05064]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04630  JAK-STAT signaling pathway
hsa04658  Th1 and Th2 cell differentiation
hsa04659  Th17 cell differentiation
Brite
Target-based classification of drugs [BR:br08310]
 Signaling molecules and receptors
  Cytokine receptors
   Interleukin receptors
    IL12RB
     D13096  Tolododekin alfa (USAN)
Other DBs
CAS: 3028474-00-9
PubChem: 508750766
LinkDB

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