KEGG   DRUG: Alpitatug
Entry
D13137                      Drug                                   
Name
Alpitatug (USAN/INN)
Formula
C6560H10154N1706O2106S46
Exact mass
147998.7051
Mol weight
148090.05
Sequence
(Heavy chain)
QVQLQESGPG LVKPSDTLSL TCAVSGNSIT SDYAWNWIRQ PPGKGLEWIG YISYSGSTTY
NPSLKSRVTM SRDTSKNQFS LKLSSVTAVD TAVYYCATGY YYGSGFWGQG TLVTVSSAST
KGPSVFPLAP SSKSTSGGTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF PAVLQSSGLY
SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDKKVEPKSC DKTHTCPPCP APELLGGPSV
FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK PREEQYNSTY
RVVSVLTVLH QDWLNGKEYK CKVSNKALPA PIEKTISKAK GQPREPQVYT LPPSREEMTK
NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSKL TVDKSRWQQG
NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
DIVLTQSPDS LAVSLGERAT INCKASESVE YFGTSLMHWY QQKPGQPPKL LIYAASNRES
GVPDRFSGSG SGTDFTLTIS SLQAEDVAVY YCQQTRKVPY TFGQGTKLEI KRTVAAPSVF
IFPPSDEQLK SGTASVVCLL NNFYPREAKV QWKVDNALQS GNSQESVTEQ DSKDSTYSLS
STLTLSKADY EKHKVYACEV THQGLSSPVT KSFNRGEC
(Disulfide bridge: H22-H6, H144-H200, H220-L218, H226-H'226, H229-H'229, H261-H321, H367-H425, H'22-H'96, H'144-H'200, H'220-L'218, H'261-H'321, H'261-H'321, H'367-H'425, L23-L92, L138-L198, L'23-L'92, L'138-L'198)
  Type
Peptide
Efficacy
Antineoplastic, Anti-kallikrein 2 antibody
  Type
Monoclonal antibody
Comment
Treatment of prostate cancer
Target
KLK2 [HSA:3817] [KO:K01325]
  Pathway
hsa04614  Renin-angiotensin system
hsa04961  Endocrine and other factor-regulated calcium reabsorption
Other DBs
CAS: 2921676-05-1
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